![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_d46cc932d50b832fdfbed630dfd214d3.svg) | Navarixin | IC50 | 0.05 [1], 1.0 [2], 2.6 [3], 450.0 [4], 680.0 [5] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_d46cc932d50b832fdfbed630dfd214d3.svg) | Navarixin | Ki | 4.0 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_700e85fe5d74c80286817c52365902d5.svg) | CID 46897162 | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_07cce337763e2d596beba2ccea809992.svg) | (R)-3-(3,4-Dioxo-2-(1-phenylpropylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide | IC50 | 6.8 [1], 48.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_07cce337763e2d596beba2ccea809992.svg) | (R)-3-(3,4-Dioxo-2-(1-phenylpropylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide | Ki | 4.0 [1], 4.4 [2], 4.7 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_9eda49f5d915d61d452cd1a2f00f841b.svg) | 1-(2-Bromophenyl)-3-(2-hydroxy-4-nitrophenyl)urea | IC50 | 22.0 [1], 30.0 [2], 40.0 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b7d63d2332bd54bde4709f0409848f55.svg) | [2-[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]sulfanylmethyl]-4-(trifluoromethoxy)phenyl]boronic acid | IC50 | 21.0 [1], 22.0 [2], 130.0 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_e16bc42236611f42ff667093cdc953b8.svg) | Elubrixin | IC50 | 5.1 [1], 260.7 [2], 310.5 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5cacdd2c27d8a0c06e4e728435e1da30.svg) | (2R)-2-[[2-Amino-5-[[(2,3-difluorophenyl)methyl]thio]thiazolo[4,5-d]pyrimidin-7-yl]amino]-1-propanol | IC50 | 3.98 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_fd05eb3a6ad16b452b93713084b04d63.svg) | 2-(5-(2,3-Difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)-2-methylpropan-1-ol | IC50 | 14.0 [1], 15.85 [2], 25.12 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b9fe439652eaf6b2764d7d88806a5885.svg) | 1-(2-Chloro-3-fluorophenyl)-3-(4-chloro-2-hydroxy-3-propan-2-ylsulfonylphenyl)urea | IC50 | 0.4 [1], 0.5 [2], 10.0 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b430288d4c9d47b29521fc3ddd6156e5.svg) | 3-[[3,4-Dioxo-2-(pentan-3-ylamino)cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | IC50 | 5.0 [1], 15.0 [2], 19.1 [3] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_2cd3b2e5fbf8ce0dbb4064a5681bf1a1.svg) | Reparixin | IC50 | 1.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_fcbc952e7ada188268cff63cc6d3ade6.svg) | Danirixin | IC50 | 5.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_45f6b360171a5fbc7e74390b471d0466.svg) | N-[6,7-Dichloro-3-(5-thiophen-2-ylthiophen-2-yl)quinoxalin-2-yl]-N',N'-diethylbutane-1,4-diamine | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_0bebf069fe449121ddb7ec4ae63405fa.svg) | 2-Methyl-5-[(phenylsulfanyl)methyl]pyrazolo[1,5-a]pyrimidin-7-ol | IC50 | 2000.0 [1], 10300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_f5550a9ad6696789b5eee84b5ee69848.svg) | 1-(2-Hydroxy-4-nitrophenyl)-3-phenylurea | IC50 | 320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_e0cae9ed6ec7432021b307eca6717d8f.svg) | [5-(4-Fluorophenylcarbamoyl)pyridin-2-ylsulfanyl]acetic acid | IC50 | 1200.0 [1], 5000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_42ee789698c96428048789e33b180a7a.svg) | 3-[[2-[[(1R)-1-(3-Fluorophenyl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | IC50 | 4.9 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_42ee789698c96428048789e33b180a7a.svg) | 3-[[2-[[(1R)-1-(3-Fluorophenyl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | Ki | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5132d51cf974f32cc7bbee80374ddd4e.svg) | 3-[[3,4-Dioxo-2-[[(1R)-1-thiophen-2-ylpropyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5132d51cf974f32cc7bbee80374ddd4e.svg) | 3-[[3,4-Dioxo-2-[[(1R)-1-thiophen-2-ylpropyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | Ki | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_bbd17ee5e826675f45477ee937df88ba.svg) | 1-(4-Cyano-2-hydroxyphenyl)-3-phenylurea | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_a3fd64392855301754612ed82f06b86e.svg) | (2R)-2-[[2-Amino-5-[(phenylmethyl)thio]thiazolo[4,5-d]pyrimidin-7-yl]amino]-1-propanol | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_f2845bf784958ac2fda1ea9a31157da0.svg) | 5-Benzylsulfanyl-7-[[(2R)-1-hydroxypropan-2-yl]amino]-3H-[1,3]thiazolo[4,5-d]pyrimidin-2-one | IC50 | 4.5 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5f95e55d4d7cd47abc2e5a78ab8b5f93.svg) | 5-[(2,3-Difluorophenyl)methylsulfanyl]-7-[[(2R)-1-hydroxypropan-2-yl]amino]-3H-[1,3]thiazolo[4,5-d]pyrimidin-2-one | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_aba94a3f15c3cacc97f2ffab5247af1e.svg) | 2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-(5-methylthiophen-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamide | IC50 | 5.3 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_aba94a3f15c3cacc97f2ffab5247af1e.svg) | 2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-(5-methylthiophen-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamide | Ki | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_a4ca6d6f62495052780644e36b7d8a3b.svg) | 3-(2-Hydroxyphenylamino)-4-(phenylamino)cyclobut-3-ene-1,2-dione | IC50 | 235.0 [1], 476.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_7ab56a61397baeac8a957f03fb493ee7.svg) | 2-[[2-Amino-5-[[(2-fluorophenyl)methyl]thio]thiazolo[4,5-d]pyrimidin-7-yl]amino]-(2R)-1-propanol | IC50 | 12.59 [1], 13.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_ddb117df5512d3b7a7ac0d238e5add10.svg) | CID 24879232 | IC50 | 5.0 [1], 50.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_1fe881b01e08ad304d7d08bb23c78051.svg) | (R)-2-(5-(2,3-Difluorobenzylthio)-2-aminothiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol | IC50 | 9.5 [1], 25.12 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_3c8ea510d272e0c330ed5b60d8bff1af.svg) | (2R)-2-[[2-Amino-5-[(3-chloro-2-fluorophenyl)methylsulfanyl]-[1,3]thiazolo[4,5-d]pyrimidin-7-yl]amino]propan-1-ol | IC50 | 3.0 [1], 3.98 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_1070d427b4778e4ddb4cf15a28ae0736.svg) | (2R)-2-[[2-Amino-5-(furan-2-ylmethylsulfanyl)-[1,3]thiazolo[4,5-d]pyrimidin-7-yl]amino]propan-1-ol | IC50 | 31.62 [1], 35.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_ad5fd6cef7b3a981acaaa87961f3d0e9.svg) | 4-(3,4-Dioxo-2-(phenylamino)cyclobut-1-enylamino)-3-hydroxybenzonitrile | IC50 | 3.0 [1], 15.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_3ab93b2479613d2e9d30735a45f1ed85.svg) | 3-(2-Hydroxy-4-nitrophenylamino)-4-(phenylamino)cyclobut-3-ene-1,2-dione | IC50 | 22.0 [1], 36.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_ce0f8fe0ba6ca7ce2a63799ce5322a61.svg) | (R)-2-(2-Amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_ce0f8fe0ba6ca7ce2a63799ce5322a61.svg) | (R)-2-(2-Amino-5-(benzylthio)thiazolo[4,5-d]pyrimidin-7-ylamino)butan-1-ol | Ki | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5ae0ca58effdda80d2f1dd6be22609a9.svg) | 1-(4-Chloro-2-hydroxy-3-sulfamoyl-phenyl)-3-(2,3-dichlorophenyl)urea | IC50 | 2.0 [1], 316.23 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_381467146180cf9a8d7f4ff4b5e0cf62.svg) | 1-(2-Bromophenyl)-3-(4-cyano-2-hydroxyphenyl)urea | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_0cfe94d7e899cab9b613d95f7f85e9f9.svg) | (2R)-2-[[2-Amino-5-[(2-methyl-1,3-thiazol-4-yl)methylsulfanyl]-[1,3]thiazolo[4,5-d]pyrimidin-7-yl]amino]propan-1-ol | IC50 | 120.0 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_4ffbb578f85bc75b90b9dde56fe3f9a1.svg) | 1-[4-Chloro-2-hydroxy-3-[(3S)-3-methyloxolan-3-yl]sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 5.2 [1], 39.81 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_d8efe42ea899a5b77d237d51015c36f4.svg) | 3-(2-(Cyclopentylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamide | IC50 | 8.0 [1], 144.8 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_f04932fff17ceef5f56b1690dd0b68bb.svg) | 3-[(2-Chlorophenyl)amino]-7-nitro-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxide | IC50 | 81.0 [1], 1100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_aead188f3b3f54c8556c8e4fc38b8619.svg) | 7-Nitro-3-{[2-(phenyloxy)phenyl]amino}-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxide | IC50 | 54.0 [1], 490.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_ea5616f1cf5624cbf61b1ee8eb473a2e.svg) | 7-Chloro-3-(2-chloroanilino)-1,1-dioxo-4H-1lambda6,2,4-benzothiadiazin-5-ol | IC50 | 92.0 [1], 520.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_11b227323180c94bc5655aa542e7db7f.svg) | 1-(4-Chloro-2-hydroxy-3-piperazin-1-ylsulfonylphenyl)-3-(2,3-dichlorophenyl)urea | IC50 | 0.63 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_d13c1f78dc23f7cc99564ae2001dc1bf.svg) | 3-[(2-Bromophenyl)amino]-7-nitro-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxide | IC50 | 26.0 [1], 600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_929f223081e8b21b3772694a4a7e210d.svg) | 1-[4-Chloro-2-hydroxy-3-(3-pyrrolidin-1-ylcyclobutyl)sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_1be2c134de1b567015ef8485dc45dc73.svg) | 1-[4-Chloro-2-hydroxy-3-[(3R)-3-methyloxolan-3-yl]sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.0 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_0a32ed530e898ccf2f729f5db6948b72.svg) | 1-[4-Chloro-2-hydroxy-3-(3-methyloxolan-3-yl)sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.26 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_8450262767be8064ee94985b91fae713.svg) | 1-[4-Chloro-3-[3-(dimethylamino)cyclobutyl]sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.0 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_4a3cd2cba6d80025663599b5757dbe62.svg) | 1-[4-Chloro-3-(1,1-difluoroethylsulfonyl)-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.4 [1], 630.96 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_cc4a9f30564eddd0e89469f21ca9c9d5.svg) | 1-(3-Tert-butylsulfonyl-4-cyano-2-hydroxyphenyl)-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.2 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b8ffbf78fd993a274d88aef05111cb36.svg) | 1-[4-Chloro-2-hydroxy-3-[2-(oxan-4-yl)propan-2-ylsulfonyl]phenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.5 [1], 398.11 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5a777d4d07bacbc2734c51260bc0c9cb.svg) | 1-[4-Chloro-3-[4-(fluoromethyl)oxan-4-yl]sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.26 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_e82893d9daf57ee3f09bb4942f492195.svg) | 1-[4-Chloro-3-[1-(2-fluoroethyl)piperidin-4-yl]sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.63 [1], 199.53 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_3f4164842f7d906eaf3b8da19c88e793.svg) | 1-[4-Chloro-2-hydroxy-3-(4-methyloxan-4-yl)sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.5 [1], 199.53 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_a2d817c1a06c6867ddd8ecad0c31a289.svg) | 1-[4-Chloro-3-(4-fluorooxan-4-yl)sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.2 [1], 63.1 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_e4d365ba67be37efba960679925b218c.svg) | Cxcr2-IN-1 | IC50 | 0.5 [1], 25.12 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_e3e605bc82ef71c5c069a3df26171afa.svg) | 1-[4-Chloro-2-hydroxy-3-(oxolan-3-ylsulfonyl)phenyl]-3-(2,3-dichlorophenyl)urea | IC50 | 0.5 [1], 7.94 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_c3232948cb785adf83e01ee9a80ffb15.svg) | 1-[4-Chloro-2-hydroxy-3-(1-methylpiperidin-4-yl)sulfonylphenyl]-3-(2,3-dichlorophenyl)urea | IC50 | 1.58 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_6a986399fcbfc156a04f4ea909ec7be5.svg) | 1-[4-Chloro-3-(1-ethylpiperidin-4-yl)sulfonyl-2-hydroxyphenyl]-3-(2-chloro-3-fluorophenyl)urea | IC50 | 1.26 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_65983d3684adb78be586d498452d72fb.svg) | 1-[4-Chloro-2-hydroxy-3-[(3S)-1-methylpyrrolidin-3-yl]sulfonylphenyl]-3-(2,3-dichlorophenyl)urea | IC50 | 1.26 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_984821bce866ebf5c2d8cb0abdcbfa19.svg) | 1-[4-Chloro-3-(4-ethylpiperazin-1-yl)sulfonyl-2-hydroxyphenyl]-3-(2-chloro-3-fluorophenyl)urea | IC50 | 1.0 [1], 1995.26 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_3afbaa77a2656983c97d8077c18aa9b0.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-[(3S)-1-methylpyrrolidin-3-yl]sulfonylphenyl]urea | IC50 | 0.5 [1], 79.43 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_437f95a2c2486ac96117d3de01c52443.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-[(4S)-1-methylazepan-4-yl]sulfonylphenyl]urea | IC50 | 0.5 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_17331477230384e961daaabe8132b011.svg) | 1-[4-Chloro-2-hydroxy-3-(4-methylpiperazin-1-yl)sulfonylphenyl]-3-(2,3-dichlorophenyl)urea | IC50 | 0.79 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b907889860b3d059f95ccf28307ae02c.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-(4-propan-2-ylpiperazin-1-yl)sulfonylphenyl]urea | IC50 | 1.58 [1], 1995.26 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_69c6a312bfe61facdb2c7a5e622fbdd0.svg) | 1-[4-Chloro-3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl-2-hydroxyphenyl]-3-(2-chloro-3-fluorophenyl)urea | IC50 | 3.98 [1], 3162.28 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_3dadec0d8dd7bb86a7454a487dc5f82f.svg) | 1-[4-Chloro-3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl-2-hydroxyphenyl]-3-(2,3-dichlorophenyl)urea | IC50 | 10.0 [1], 15848.93 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_34de7cc5dd60e868603877029e491635.svg) | 1-(4-Chloro-3-ethylsulfonyl-2-hydroxyphenyl)-3-(2,3-dichlorophenyl)urea | IC50 | 0.5 [1], 6309.57 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_104428891a2eda2a7cc14cb63866a06a.svg) | 1-(4-Chloro-2-hydroxy-3-propan-2-ylsulfonylphenyl)-3-(2,3-dichlorophenyl)urea | IC50 | 0.63 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5401bf44d87719dfcb65e49aeac02ba6.svg) | 1-[4-Chloro-2-hydroxy-3-(oxan-4-ylsulfonyl)phenyl]-3-(2,3-dichlorophenyl)urea | IC50 | 0.79 [1], 6.31 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_dff378dccc104df094d21bebce387c3c.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-(piperidine-1-carbonyl)phenyl]urea | IC50 | 0.5 [1], 6.31 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_9fc14ec6339058d07de9fd5cb6e1c3de.svg) | 1-(3-Tert-butylsulfonyl-4-chloro-2-hydroxyphenyl)-3-(2-chloro-3-fluorophenyl)urea | IC50 | 0.5 [1], 39.81 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_7021468e103377c871d0f8f9de6e4af1.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-[(2-methyl-2-azaspiro[3.3]heptan-6-yl)sulfonyl]phenyl]urea | IC50 | 0.4 [1], 630.96 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_2ce6a62610c05a8588f60974b2330c9d.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-[(7-methyl-7-azaspiro[3.5]nonan-2-yl)sulfonyl]phenyl]urea | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_8bf756c60359aa7e42b0c087fc47c0e1.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-[(3-methyl-3-azaspiro[5.5]undecan-9-yl)sulfonyl]phenyl]urea | IC50 | 0.4 [1], 25.12 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_e154f3cf3f6cc581062ebfc1e22a040f.svg) | 1-(2-Chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-(pyrrolidine-1-carbonyl)phenyl]urea | IC50 | 1.0 [1], 7.94 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b947a9948740d9218ab9ac28f9d545e2.svg) | 1-[4-Chloro-3-(1-fluoro-2-methylpropan-2-yl)sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.63 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_5f5a7f265888e07da0fac12549c63350.svg) | 1-[4-Chloro-2-hydroxy-3-(1-methoxypropan-2-ylsulfonyl)phenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.26 [1], 398.11 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_23d978a4d9ae89670e2ef80fa7f27d3d.svg) | 1-[4-Chloro-2-hydroxy-3-[2-[(3S)-oxolan-3-yl]propan-2-ylsulfonyl]phenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.58 [1], 316.23 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_a2d24d0032fcae01e18e8bea1f5b1479.svg) | 1-[4-Chloro-3-(1-cyclobutylpiperidin-4-yl)sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.4 [1], 501.19 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_fca1140ec8faa2e9b44ae12967117da7.svg) | 1-[4-Chloro-3-[2-(dimethylamino)-1,1-difluoroethyl]sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 2.0 [1], 630.96 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_7f6596b58f78e886cfafa31c1a9e5f2c.svg) | 1-[4-Chloro-3-(4-ethyloxan-4-yl)sulfonyl-2-hydroxyphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.32 [1], 398.11 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_65cda9c28f5380d493bf673c78e3349e.svg) | 1-[4-Chloro-2-hydroxy-3-(oxan-3-ylsulfonyl)phenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.58 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_ea6da7f3dd86e0961a830800c37a6340.svg) | 1-[4-Chloro-2-hydroxy-3-(3-methyloxan-3-yl)sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 2.0 [1], 199.53 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_1a9fe3e825cf632836b549dad71e8b69.svg) | 1-(3-Tert-butylsulfonyl-4-chloro-2-hydroxyphenyl)-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 1.0 [1], 316.23 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_18e8c0a7b5b70bc99a20fe68bc7c469b.svg) | 3-[[4-[[(1R)-2,2-Dimethyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_18e8c0a7b5b70bc99a20fe68bc7c469b.svg) | 3-[[4-[[(1R)-2,2-Dimethyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | Ki | 91.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_f274f4dbe281aa7475414e67f4d09dc9.svg) | 2-[(2,6-Dichlorobenzyl)sulfanyl]-4-hydroxy-6-phenyl-5-pyrimidinecarbonitrile | IC50 | 4300.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_496b8a6e0d600300235a3c8ade08ea7c.svg) | Nvp cxcr2 20 | IC50 | 40.0 [1], 140.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_9040f8a30a4a5e8ae441d55cc3e4e909.svg) | 2-Hydroxy-N,N-dimethyl-3-[[4-[[(1R)-2-methyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]benzamide | IC50 | 36.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_9040f8a30a4a5e8ae441d55cc3e4e909.svg) | 2-Hydroxy-N,N-dimethyl-3-[[4-[[(1R)-2-methyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]benzamide | Ki | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_8554fb84defbbd2f31a0260d7af46767.svg) | 4-Tert-butyl-2-(4-chloro-2-hydroxy-3-propan-2-ylsulfonylanilino)-1H-pyrimidin-6-one | IC50 | 6.31 [1], 580.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_d9c295dc96eafe7a7db196bf20d8f01f.svg) | 1-[4-Cyano-2-hydroxy-3-(4,4,4-trifluoro-2-methylbutan-2-yl)sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]urea | IC50 | 0.16 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_443189ff3f3cddac878ab2d965248db2.svg) | 2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-(5-methylfuran-2-yl)ethyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamide | IC50 | 2.4 [1], 5.4 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_b7b58eb71ca82dde986bfcf3cb7943fe.svg) | 2-Benzyl-5-(2,3-difluorophenylsulfanylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol | IC50 | 330.0 [1], 350.0 [2] |
![](https://images.aatbio.com/dataset/ic50/interleukin-8-receptor-b_150bf93ac37c802126565bcdb9f2e68b.svg) | 3-[[2-[[(1R)-1-(4-Bromofuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamide | IC50 | 2.0 [1], 3.5 [2] |