![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_1762def150dc40530698249fb914660e.svg) | CID 53340771 | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_1137659560ccde6568e277be476a7ef5.svg) | CID 72949858 | IC50 | 0.2 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_faddca7ec5c5558b4e725d0abd59963a.svg) | (3S)-3-[3-(3,5-Dimethylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 15.85 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_9ae8e4e8f86ac2b952ac2dfcfc96bc62.svg) | (3S)-3-(3-Bromo-5-chloro-2-hydroxyphenyl)-3-[[2-[[5-[(5-hydroxy-1,4,5,6-tetrahydropyrimidin-2-yl)amino]pyridine-3-carbonyl]amino]acetyl]amino]propanoic acid | IC50 | 0.65 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_49563cb292c93bfd5f9ef2023c4cb25b.svg) | (3S)-3-(3-Bromo-5-chloro-2-hydroxyphenyl)-3-[[2-[[3-hydroxy-5-[(5-hydroxy-1,4,5,6-tetrahydropyrimidin-2-yl)amino]benzoyl]amino]acetyl]amino]propanoic acid | IC50 | 1.71 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_af90f11653ad4fe9324cbeda96c05608.svg) | 3-(3-Fluorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 1584.89 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_7a0141fe7ecd6a2db5e7f3766dd5682c.svg) | 3-(1,3-Benzodioxol-5-yl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_27b24d0775dd274b019158788df747f0.svg) | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[[3-(diaminomethylideneamino)benzoyl]amino]phenyl]propanoic acid | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_c39fc1c5846704efb67b74424a24c08f.svg) | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_3085ab33b4697b976a0b208c1e71c0ce.svg) | 3-(2-Fluorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 3981.07 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_639756b99f4a558b8f22cac1b22ebcbb.svg) | 3-(2-Chlorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_cc540e59f2c4f10bcc09dbdaa6ae1ff2.svg) | 3-(2-Methylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 1258.93 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_f2d2227522ed6e614febd7b38940a3f4.svg) | 3-(2-Methoxyphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_20b3430f57e29583adb2cf7156f194b3.svg) | 3-(3-Chlorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_0772d1d12bae18cf9f10c72828537776.svg) | 3-(3-Methylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 630.96 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_e9ba9dc0b80d198c56f5139271c614e4.svg) | 3-(3-Methoxyphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_c0f345c01adc137a6fc39e64c7b1727b.svg) | 3-(4-Fluorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_e0ae050a9950fc07dce00125737e5c3b.svg) | 3-(4-Chlorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 630.96 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_2768d0d5aceac8ed22e44483d9c3e2f6.svg) | 3-(4-Methylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_6e545a926a702a4e7610fe30aa8fe599.svg) | 3-(4-Methoxyphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_86a77e50bd0703ad60a543af1ff27db0.svg) | 3-(4-Cyanophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_cdd3ac3565125030c8ed3d88b08ce674.svg) | 3-[5-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]-3-[4-(trifluoromethyl)phenyl]propanoic acid | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_0398be91f421b223f2f94dfa509f0d30.svg) | 3-[5-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]-3-[4-(trifluoromethoxy)phenyl]propanoic acid | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_87c920fa46e7fed25431ff6292dfd0f1.svg) | 3-(4-Methylsulfonylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_ebef66e37d118583c1a98ea368679d17.svg) | 3-(4-Phenylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 316.23 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_3ae4c31a1f69416f7964a94e27e9f7b9.svg) | 3-(3-Cyanophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_c17cbfd29897340a773b4f4bb15125fa.svg) | 3-[5-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]-3-[3-(trifluoromethyl)phenyl]propanoic acid | IC50 | 158.49 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_2528eebe15ac929a8d55f40f636fb8e1.svg) | (3S)-3-[5-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]-3-[3-(trifluoromethyl)phenyl]propanoic acid | IC50 | 125.89 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_16863ee99749237a66635ea236126444.svg) | (3R)-3-[5-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]-3-[3-(trifluoromethyl)phenyl]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_e7a8ba13be2cc8a115e37fd6503ef8b1.svg) | 3-[5-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]-3-[3-(trifluoromethoxy)phenyl]propanoic acid | IC50 | 251.19 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_d0827f16cb1583f0c568361f90188dee.svg) | 3-(2,3-Dichlorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_c7430f4c065777846f20c96aa7bed4a0.svg) | 3-(3,4-Dichlorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 199.53 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_aa0aefcd1a8d5dd644fbe87d2db7608c.svg) | 3-(3,5-Dichlorophenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_0a62522864fcc803f4abba0519d500b0.svg) | 3-(3,4-Dimethylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_0fb490dddca5fd4588b1cd7a8a0ea708.svg) | 3-(2,3-Dihydro-1H-inden-5-yl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 398.11 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_a7c86581c648033c7258adca4bc7ecd3.svg) | 3-(3,5-Dimethylphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 630.96 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_88518508e1ec5f5053d0a48625a22238.svg) | 3-(3,4-Dimethoxyphenyl)-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 398.11 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_11f14a26ed67a8ab6f927868ae60a36e.svg) | 3-[4-Chloro-3-(trifluoromethyl)phenyl]-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_cca53e47ce48e8a9f860de4532b9786a.svg) | (3S)-3-(3-Morpholin-4-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 15.85 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_f6d21c9c7eecd0d6865979b65d1f545d.svg) | (3S)-3-(3-Cyclopropyl-5-morpholin-4-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 15.85 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_6255039ac215e8e24ba3263fa13290cc.svg) | (3S)-3-[3-(3,5-Dimethylpyrazol-1-yl)-5-morpholin-4-ylphenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_87e0afe9fad08c34605f502c3835604b.svg) | (3R)-3-(3-Morpholin-4-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_eea64d6777e256d463c277af5eeea7ad.svg) | (3S)-3-[3-(2,5-Dimethyl-1H-imidazol-4-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_ba1dfc42752ad79a69fe0b889c70bfe6.svg) | (3S)-4-[(3R)-3-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]-3-[3-(1,2,4-triazol-4-yl)phenyl]butanoic acid | IC50 | 6.31 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_1d282ddbeed228fb80abc65c27aee416.svg) | 3-(3-Imidazol-1-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 25.12 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_b2b956d26f7d59ffac189529f165b6c9.svg) | (3S)-3-[3-(5-Methyl-1H-pyrazol-3-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 3.98 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_a46be915162075d186b7e9d69ede84ca.svg) | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[5-(4,5-dihydro-1H-imidazol-2-ylamino)pentanoylamino]phenyl]propanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_b86f4a28a587b074d945149ac93b3de3.svg) | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[4-(pyridin-2-ylamino)butanoylamino]phenyl]propanoic acid | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_b17c2e31c6d798cdeebbc21f65e8b523.svg) | (2S)-2-[[(2S)-1-(Benzenesulfonyl)piperidine-2-carbonyl]amino]-3-[4-[4-(diaminomethylideneamino)butanoylamino]phenyl]propanoic acid | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_71411d8d399775af2c5ebf23d6246b73.svg) | (2S)-2-[[(2S)-1-(Benzenesulfonyl)piperidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_588b934b5787fe3751fff2fce68e5a91.svg) | (3S)-3-[3-[(3S)-Oxolan-3-yl]oxyphenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 6.31 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_876277cad7cd7a3d7544d271de7464ac.svg) | (3S)-3-[3-(Oxan-4-yloxy)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 6.31 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_2da2a6c72743551e74c2b9576b3e80d0.svg) | (3S)-3-[3-(Oxetan-3-yloxy)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 2.51 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_e700cf861fbf2a44df5871053b04b03a.svg) | (3S)-3-[3-[(3R)-Oxolan-3-yl]oxyphenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_a05478b4b0b49fe1aa382826ad6d2976.svg) | (3S)-3-[3-(Oxolan-3-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_7a6ca2517f25aa479168162579ec5242.svg) | (3S)-4-[(3R)-3-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]-3-[3-(1,2,4-triazol-1-yl)phenyl]butanoic acid | IC50 | 6.31 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_6edca9563d70e60197f9c1d0791896c4.svg) | (3S)-3-[3-(2,4-Dimethylpyrazol-3-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 7.94 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_00bb6b1c0b55ce9431c2bd2604044edf.svg) | (3S)-4-[(3R)-3-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]-3-[3-(triazol-1-yl)phenyl]butanoic acid | IC50 | 5.01 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_fca8956a3f32a30968bb120143476aea.svg) | (3S)-3-[3-(3-Methyl-1,2,4-triazol-4-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_811bb7d60be6eb049847319c186acb99.svg) | (3S)-3-[3-(1,4-Dimethylimidazol-2-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 7.94 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_bbe2eabc2fd493b79ff2fa48ac35f062.svg) | (3R)-3-[3-(3,5-Dimethylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 398.11 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_cfee6ce011b6d7ac2191db6fdaeaa970.svg) | (3S)-3-[3-(3,5-Dimethyl-1,2,4-triazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_55129fc59311c91fccdeb970979e595b.svg) | (3S)-3-[3-(3-Methylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 31.62 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_d90ab9b69b305331896d8e5116a4e9d8.svg) | (3S)-3-(3-Pyrazol-1-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_2261c1f7e92f5c90130e998c6d97a8e3.svg) | (3S)-3-[3-(5-Methylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_f2dd149d1322367b4366dd695e81a99f.svg) | (3S)-3-(3-Cyclopropylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 6.31 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_ba0838c6cf052c3c61ac40aeaa3ff62f.svg) | (3S)-3-[3-(4-Methylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 39.81 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_61b73395058153934f57e2e9f4d5f319.svg) | (3R)-3-(3-Cyclopropylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 125.89 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_d810e8f01e87f38be84cc3d7267a39ba.svg) | (3S)-3-(3-Bromophenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 3.16 [1] |
![](https://images.aatbio.com/dataset/ic50/integrin-alpha-v-beta-8_c5896b24d68e24f172b6be4280db2cd1.svg) | 3-Phenyl-3-[5-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)pentanoylamino]propanoic acid | IC50 | 794.33 [1] |