 | Gly-arg-gly-asp-ser | IC50 | 100000.0 [1] |
 | (S)-2-(2,6-Dichlorobenzamido)-3-(2',6'-dimethoxy-[1,1'-biphenyl]-4-yl)propanoic acid | IC50 | 414.0 [1] |
 | 2-[(9S)-14-[3-(Pyridin-2-ylamino)propoxy]-9-tricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaenyl]acetic acid | Ki | 18000.0 [1] |
 | CID 53340771 | IC50 | 1.3 [1] |
 | CID 72949858 | IC50 | 1.8 [1] |
 | (2S)-3-[[(5S,8S)-8-[(1H-Imidazol-2-ylamino)methyl]-7-(pyridin-3-ylmethoxycarbonyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 32.0 [1] |
 | (3S)-3-[3-(3,5-Dimethylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 50.12 [1] |
 | (2S)-2-[[2-(Diethylamino)-5-[(4-fluorophenyl)sulfonyl-prop-2-ynylamino]pyrimidin-4-yl]amino]-3-[4-(pyrrolidine-1-carbonyloxy)phenyl]propanoic acid | IC50 | 500.0 [1] |
 | (2-{4-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid | IC50 | 64.0 [1] |
 | (3S)-3-(1,3-Benzodioxol-5-yl)-4-[3-[3-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)propyl]-1,2,4-oxadiazol-5-yl]butanoic acid | IC50 | 2.6 [1] |
 | (2S)-3-[[(5S,8S)-7-Phenylmethoxycarbonyl-8-[(pyridin-2-ylamino)methyl]-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 49.0 [1] |
 | (2S)-3-[[(5S,8S)-8-[(1H-Imidazol-2-ylamino)methyl]-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 180.0 [1] |
 | (2S)-3-[[(5S,8S)-8-[(1H-Imidazol-2-ylamino)methyl]-7-phenylmethoxycarbonyl-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 41.0 [1] |
 | (2S)-3-[[(5S,8S)-8-[(1H-Benzimidazol-2-ylamino)methyl]-7-butoxycarbonyl-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 87.0 [1] |
 | (2S)-3-[[(5S,8S)-8-[(1H-Imidazol-2-ylamino)methyl]-7-methoxycarbonyl-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 57.0 [1] |
 | (2S)-3-[[(5S,8S)-7-Butoxycarbonyl-8-[(1H-imidazol-2-ylamino)methyl]-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 130.0 [1] |
 | (2S)-3-[[(5S,8S)-8-[(1H-Benzimidazol-2-ylamino)methyl]-7-methoxycarbonyl-1-oxa-2,7-diazaspiro[4.4]non-2-ene-3-carbonyl]amino]-2-[(2,4,6-trimethylphenyl)sulfonylamino]propanoic acid | IC50 | 34.0 [1] |
 | (3S)-3-(3-Bromo-5-chloro-2-hydroxyphenyl)-3-[[2-[[5-[(5-hydroxy-1,4,5,6-tetrahydropyrimidin-2-yl)amino]pyridine-3-carbonyl]amino]acetyl]amino]propanoic acid | IC50 | 1.59 [1] |
 | (3S)-3-(3-Bromo-5-chloro-2-hydroxyphenyl)-3-[[2-[[3-hydroxy-5-[(5-hydroxy-1,4,5,6-tetrahydropyrimidin-2-yl)amino]benzoyl]amino]acetyl]amino]propanoic acid | IC50 | 10.4 [1] |
 | 3-Phenyl-4-[4-[3-(2-pyridinylamino)propoxy]phenyl]butanoic acid | IC50 | 96.0 [1] |
 | 3-(1,3-Benzoxazol-6-yl)-4-[3-[3-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)propyl]-1,2,4-oxadiazol-5-yl]butanoic acid | IC50 | 2.7 [1] |
 | 3-(2,3-Dihydro-1-benzofuran-6-yl)-4-[3-[3-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)propyl]-1,2,4-oxadiazol-5-yl]butanoic acid | IC50 | 9.7 [1] |
 | {2-Methoxy-4-[3-(1,4,5,6-tetrahydro-pyrimidin-2-ylamino)-benzoylamino]-phenoxy}-acetic acid | IC50 | 82.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[4-[(6-methylpyridin-2-yl)amino]butanoylamino]phenyl]propanoic acid | IC50 | 199.53 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[4-[(5-methylpyridin-2-yl)amino]butanoylamino]phenyl]propanoic acid | IC50 | 316.23 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[[3-(diaminomethylideneamino)benzoyl]amino]phenyl]propanoic acid | IC50 | 0.06 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[[4-(diaminomethylideneamino)benzoyl]amino]phenyl]propanoic acid | IC50 | 794.33 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 0.63 [1] |
 | (3S)-3-(3-Morpholin-4-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 251.19 [1] |
 | (3S)-3-(3-Cyclopropyl-5-morpholin-4-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 63.1 [1] |
 | (3S)-3-[3-(3,5-Dimethylpyrazol-1-yl)-5-morpholin-4-ylphenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 100.0 [1] |
 | (3R)-3-(3-Morpholin-4-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 794.33 [1] |
 | (3S)-3-[3-(2,5-Dimethyl-1H-imidazol-4-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 100.0 [1] |
 | (3S)-4-[(3R)-3-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]-3-[3-(1,2,4-triazol-4-yl)phenyl]butanoic acid | IC50 | 63.1 [1] |
 | (3S)-3-[3-(5-Methyl-1H-pyrazol-3-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 63.1 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[[4-(diaminomethylideneamino)cyclohexanecarbonyl]amino]phenyl]propanoic acid | IC50 | 2.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[5-(4,5-dihydro-1H-imidazol-2-ylamino)pentanoylamino]phenyl]propanoic acid | IC50 | 0.31 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[4-(4,5-dihydro-1H-imidazol-2-ylamino)butanoylamino]phenyl]propanoic acid | IC50 | 0.13 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[4-(diaminomethylideneamino)butanoylamino]phenyl]propanoic acid | IC50 | 0.02 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-(3,5-difluorophenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 40.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)-2-methylpyrrolidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 10000.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[5-(1,4,5,6-tetrahydropyrimidin-2-ylamino)pentanoylamino]phenyl]propanoic acid | IC50 | 2.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[4-(pyridin-2-ylamino)butanoylamino]phenyl]propanoic acid | IC50 | 0.2 [1] |
 | (2S)-2-[[(4R)-3-(Benzenesulfonyl)-1,3-thiazolidine-4-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 16.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[5-(pyridin-2-ylamino)pentanoylamino]phenyl]propanoic acid | IC50 | 2.0 [1] |
 | (2S)-2-[[(4R)-3-(Benzenesulfonyl)-5,5-dimethyl-1,3-thiazolidine-4-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 2000.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)piperidine-2-carbonyl]amino]-3-[4-[4-(diaminomethylideneamino)butanoylamino]phenyl]propanoic acid | IC50 | 0.25 [1] |
 | (2S)-3-[4-[4-(Diaminomethylideneamino)butanoylamino]phenyl]-2-[[(2S)-1-(3,5-dimethylphenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 790.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)piperidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 0.31 [1] |
 | (3S)-3-[3-[(3S)-Oxolan-3-yl]oxyphenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 50.12 [1] |
 | (3S)-3-[3-(Oxan-4-yloxy)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 100.0 [1] |
 | (3S)-3-[3-(Oxetan-3-yloxy)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 100.0 [1] |
 | (3S)-3-[3-[(3R)-Oxolan-3-yl]oxyphenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 125.89 [1] |
 | (3S)-3-[3-(Oxolan-3-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 63.1 [1] |
 | (3S)-4-[(3R)-3-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]-3-[3-(1,2,4-triazol-1-yl)phenyl]butanoic acid | IC50 | 100.0 [1] |
 | (3S)-3-[3-(2,4-Dimethylpyrazol-3-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 39.81 [1] |
 | (3S)-4-[(3R)-3-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]-3-[3-(triazol-1-yl)phenyl]butanoic acid | IC50 | 63.1 [1] |
 | (3S)-3-[3-(3-Methyl-1,2,4-triazol-4-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 100.0 [1] |
 | (3S)-3-[3-(1,4-Dimethylimidazol-2-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 100.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)azetidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 160.0 [1] |
 | (2S)-2-[[(2S,4S)-1-(Benzenesulfonyl)-4-fluoropyrrolidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 0.5 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-(2,4,6-trimethylphenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 10000.0 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-pyridin-3-ylsulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 32.0 [1] |
 | (2S)-2-[[(2S,4R)-1-(Benzenesulfonyl)-4-fluoropyrrolidine-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 0.5 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-thiophen-2-ylsulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 50.0 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-(2-nitrophenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 630.0 [1] |
 | (2S)-3-[4-[4-(Diaminomethylideneamino)butanoylamino]phenyl]-2-[[(2S)-1-(4-methylphenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 630.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[[2-[4-(diaminomethylideneamino)phenyl]acetyl]amino]phenyl]propanoic acid | IC50 | 50.12 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)-2,5-dihydropyrrole-2-carbonyl]amino]-3-[4-[5-(diaminomethylideneamino)pentanoylamino]phenyl]propanoic acid | IC50 | 800.0 [1] |
 | (2S)-2-[[(2S)-1-(Benzenesulfonyl)pyrrolidine-2-carbonyl]amino]-3-[4-[[3-(diaminomethylideneamino)adamantane-1-carbonyl]amino]phenyl]propanoic acid | IC50 | 2511.89 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-(4-fluoro-2-methylphenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 500.0 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-(3-nitrophenyl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 13.0 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-[5-(dimethylamino)naphthalen-1-yl]sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 79.0 [1] |
 | (2S)-3-[4-[5-(Diaminomethylideneamino)pentanoylamino]phenyl]-2-[[(2S)-1-(4-methylnaphthalen-1-yl)sulfonylpyrrolidine-2-carbonyl]amino]propanoic acid | IC50 | 6300.0 [1] |
 | (3S)-3-[3-(3,5-Dimethyl-1,2,4-triazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 50.12 [1] |
 | (3S)-3-[3-(3-Methylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 158.49 [1] |
 | (3S)-3-(3-Pyrazol-1-ylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 125.89 [1] |
 | (3S)-3-[3-(5-Methylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 50.12 [1] |
 | (3S)-3-(3-Cyclopropylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 158.49 [1] |
 | (3S)-3-[3-(4-Methylpyrazol-1-yl)phenyl]-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 1995.26 [1] |
 | (3R)-3-(3-Cyclopropylphenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 3981.07 [1] |
 | (3S)-3-(3-Bromophenyl)-4-[(3R)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]pyrrolidin-1-yl]butanoic acid | IC50 | 199.53 [1] |
 | 3-[4-[[3-[(5-Oxo-1,4-dihydroimidazol-2-yl)amino]benzoyl]amino]phenyl]-2-(propan-2-yloxycarbonylamino)propanoic acid | IC50 | 17.7 [1] |
 | 2-{4-[3-(1,4,5,6-Tetrahydro-pyrimidin-2-ylamino)-benzoylamino]-phenyl}-cyclopropanecarboxylic acid | IC50 | 320.0 [1] |
 | [4-(3-Guanidino-benzoylamino)-2-methoxy-phenoxy]-acetic acid | IC50 | 222.0 [1] |
 | [4-(3-Guanidino-benzoylamino)-phenoxy]-acetic acid | IC50 | 351.0 [1] |
 | 2-Acetylamino-3-[4-(3-guanidino-benzoylamino)-phenyl]-propionic acid | IC50 | 16.0 [1] |
 | 3-[4-(3-Guanidino-benzoylamino)-2-methoxy-phenyl]-2-isopropoxycarbonylamino-propionic acid | IC50 | 1.1 [1] |
 | 3-[4-(3-Guanidino-benzoylamino)-phenyl]-2-isopropoxycarbonylamino-propionic acid | IC50 | 0.47 [1] |
 | 2-(3-Tert-Butyl-ureido)-3-[4-(3-guanidino-benzoylamino)-phenyl]-propionic acid | IC50 | 4.8 [1] |
 | 2-Tert-Butoxycarbonylamino-3-[4-(3-guanidino-benzoylamino)-phenyl]-propionic acid | IC50 | 6.7 [1] |
 | 3-[2-Methoxy-4-[[3-(1,4,5,6-tetrahydropyrimidin-2-ylamino)benzoyl]amino]phenyl]-2-(propan-2-yloxycarbonylamino)propanoic acid | IC50 | 0.68 [1] |
 | 3-[4-(3-Guanidino-benzoylamino)-phenyl]-propionic acid | IC50 | 758.0 [1] |
 | 3-{2-Methoxy-4-[3-(1,4,5,6-tetrahydro-pyrimidin-2-ylamino)-benzoylamino]-phenyl}-propionic acid | IC50 | 162.0 [1] |
 | 2-(Benzenesulfonamido)-3-[4-[[3-(1,4,5,6-tetrahydropyrimidin-2-ylamino)benzoyl]amino]phenyl]propanoic acid | IC50 | 10.4 [1] |
 | 3-{4-[3-(4,5-Dihydro-1H-imidazol-2-ylamino)-benzoylamino]-3,5-dimethyl-phenyl}-acrylic acid | IC50 | 264.0 [1] |
 | 3-[4-(3-Guanidino-benzoylamino)-3,5-dimethyl-phenyl]-acrylic acid | IC50 | 2070.0 [1] |
 | 3-[3-Fluoro-4-(3-guanidino-benzoylamino)-phenyl]-acrylic acid | IC50 | 426.0 [1] |
 | 3-[4-[[3-(Diaminomethylideneamino)benzoyl]amino]phenyl]-2-(methanesulfonamido)propanoic acid | IC50 | 29.0 [1] |
 | 3-{3-Chloro-4-[3-(1,4,5,6-tetrahydro-pyrimidin-2-ylamino)-benzoylamino]-phenyl}-acrylic acid | IC50 | 85.0 [1] |