| Arg-gly-asp-ser | IC50 | 13000.0 [1], 31000.0 [2] |
| 3-(3-(Carbamoyl)benzamido)-3-(4-methoxyphenyl)propanoic acid | IC50 | 0.8 [1], 17.0 [2] |
| 3-(3-(Carbamoyl)benzamido)-3-(3,4-dimethoxyphenyl)propanoic acid | IC50 | 0.7 [1], 11.6 [2] |
| 3-(3-(Carbamoyl)benzamido)-3-phenylpropanoic acid | IC50 | 1.0 [1], 25.0 [2] |
| 3-[3-(2,3-Dihydro-1H-isoindol-5-ylcarbamoyl)-propionylamino]-3-phenyl-propionic acid; hydrochloride | IC50 | 8.3 [1], 860.0 [2] |
| 3-[[4-(2,3-Dihydro-1H-isoindol-5-ylamino)-4-oxobutanoyl]amino]-3-(4-propan-2-yloxyphenyl)propanoic acid | IC50 | 6.0 [1], 105.0 [2] |
| 3-[[4-(2,3-Dihydro-1H-isoindol-5-ylamino)-4-oxobutanoyl]amino]-3-(3,4-dimethoxyphenyl)propanoic acid | IC50 | 9.0 [1], 890.0 [2] |
| 3-(1,3-Benzodioxol-5-yl)-3-[[4-(2,3-dihydro-1H-isoindol-5-ylamino)-4-oxobutanoyl]amino]propanoic acid | IC50 | 0.22 [1], 31.0 [2] |
| 3-[[4-(2,3-Dihydro-1H-isoindol-5-ylamino)-4-oxobutanoyl]amino]-3-(4-methoxyphenyl)propanoic acid | IC50 | 2.6 [1], 160.0 [2] |
| 3-(4-Fluorophenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 1.0 [1], 8.9 [2] |
| 3-(1,3-Benzodioxol-5-yl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 0.4 [1], 90.0 [2] |
| 3-(4-Methylphenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 0.9 [1], 96.0 [2] |
| 3-(4-Methoxyphenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 3.5 [1], 310.0 [2] |
| 3-(3,4-Dimethoxyphenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 0.63 [1], 64.0 [2] |
| 3-(4-Methoxyphenyl)-3-[[5-oxo-5-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)pentanoyl]amino]propanoic acid | IC50 | 18.0 [1], 4200.0 [2] |
| 3-(3,4-Dimethoxyphenyl)-3-[[5-oxo-5-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)pentanoyl]amino]propanoic acid | IC50 | 5.0 [1], 127.0 [2] |
| 3-(1,3-Benzodioxol-5-yl)-3-[[5-oxo-5-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)pentanoyl]amino]propanoic acid | IC50 | 0.78 [1], 53.0 [2] |
| 3-[[4-Oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 1.21 [1], 30.01 [2] |
| 3-[[4-Oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]-3-phenylpropanoic acid | IC50 | 1.01 [1], 13.01 [2] |
| 3-(3-Fluorophenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 1100.0 [1], 10000.0 [2] |
| 3-(2-Fluorophenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 5.0 [1], 570.0 [2] |
| 3-(4-Chlorophenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 65.0 [1], 2000.0 [2] |
| 3-[[4-Oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]-3-(4-propan-2-yloxyphenyl)propanoic acid | IC50 | 87.0 [1] |
| 3-(4-Ethoxy-3-methoxyphenyl)-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 510.0 [1] |
| 3-Naphthalen-1-yl-3-[[4-oxo-4-(1,2,3,4-tetrahydroisoquinolin-7-ylamino)butanoyl]amino]propanoic acid | IC50 | 5200.0 [1] |