 | 1-(3,4-Dihydroxybenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 5.6 [1] |
 | 1-(1,3-Benzodioxole-5-ylcarbonyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 70.0 [1] |
 | 1-(3,4-Dihydroxybenzoyl)isoquinoline-3,6,7-triol | Ki | 28.0 [1] |
 | 1-(3,4-Dihydroxybenzyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 7.5 [1] |
 | 1-(3-Hydroxy-4-methoxy-benzoyl)-6,7-dimethoxy-isoquinoline-3-carboxylic Acid | Ki | 10000.0 [1] |
 | 1-(3,4-Dihydroxybenzyl)isoquinoline-3,6,7-triol | Ki | 29.0 [1] |
 | 6,7-Dimethoxy-1-(3,4-dimethoxybenzoyl)isoquinoline-3-ol | Ki | 10000.0 [1] |
 | 7-Hydroxy-1-(3-hydroxy-4-methoxy-benzoyl)-6-methoxy-isoquinoline-3-carboxylic Acid | Ki | 320.0 [1] |
 | 6,7-Dimethoxy-1-(3,4-dimethoxybenzoyl)isoquinoline-3-carboxylic acid ethyl ester | Ki | 10000.0 [1] |
 | 1-(3,4-Dihydroxybenzoyl)isoquinoline-6,7-diol | Ki | 58.0 [1] |
 | 1-[3-Fluoro-4-(3,5-dichlorophenoxy)benzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 9.0 [1] |
 | 6,7-Dihydroxy-1-(1-naphthylcarbonyl)isoquinoline-3-carboxylic acid | Ki | 27.0 [1] |
 | 6,7-Dimethoxy-1-(3,4-dihydroxybenzoyl)isoquinoline-3-carboxylic acid | Ki | 10000.0 [1] |
 | 8-Bromo-6-methoxy-7-hydroxy-1-(3,4-dihydroxybenzoyl)isoquinoline-3-carboxylic acid | Ki | 140.0 [1] |
 | 6,7-Dihydroxy-1-(2,4-dichlorobenzoyl)isoquinoline-3-carboxylic acid | Ki | 44.0 [1] |
 | 5-Bromo-7-methoxy-6-hydroxy-1-(3,4-dihydroxybenzoyl)isoquinoline-3-carboxylic acid | Ki | 70.0 [1] |
 | 4-(3,4-Dihydroxybenzyl)-6,7-dihydroxy-2-quinolinecarboxylic acid | Ki | 8.0 [1] |
 | 6,7-Dihydroxy-1-(2-naphthylcarbonyl)isoquinoline-3-carboxylic acid | Ki | 13.0 [1] |
 | 1-(3-Fluoro-4-p-tolyloxy-benzoyl)-6,7-dihydroxy-isoquinoline-3-carboxylic acid | Ki | 9.4 [1] |
 | 1-[4-(Trifluoromethyl)benzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 38.0 [1] |
 | 1-[3-Fluoro-4-[4-(trifluoromethyl)phenoxy]benzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 32.0 [1] |
 | 1-(3,4-Dichlorobenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 29.0 [1] |
 | 1-(4-Aminobenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 130.0 [1] |
 | 6-Amino-1-(3,4-dihydroxy-benzoyl)-7-hydroxy-isoquinoline-3-carboxylic acid | Ki | 60.0 [1] |
 | 1-[4-(2-Ethylhexylamino)-3-fluorobenzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 62.0 [1] |
 | 1-[4-(4-Chlorophenyl)sulfanyl-3-fluorobenzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 31.0 [1] |
 | 1-[3-Fluoro-4-(4-phenylphenoxy)benzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 32.0 [1] |
 | 1-[4-(3,4-Dichlorophenoxy)-3-fluorobenzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 12.0 [1] |
 | 1-[4-(4-Chlorophenoxy)-3-fluorobenzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 20.0 [1] |
 | 1-[4-(Methylsulfonylamino)benzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 110.0 [1] |
 | 1-(4-Nitrobenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 32.0 [1] |
 | 1-(3-Fluorobenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 110.0 [1] |
 | 1-(alpha-Hydroxy-3-fluorobenzyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 24.0 [1] |
 | 1-(alpha-Hydroxy-2-chlorobenzyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 25.0 [1] |
 | 1-(alpha-Hydroxy-2,4,6-trimethylbenzyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 11.0 [1] |
 | 1-(3,4-Difluorobenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 51.0 [1] |
 | 1-(alpha-Hydroxy-4-phenoxybenzyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 32.0 [1] |
 | 1-[3-Fluoro-4-(3-chlorophenoxy)benzoyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 11.0 [1] |
 | 1-[alpha-Hydroxy-4-(trifluoromethyl)benzyl]-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 18.0 [1] |
 | 1-(2,4,6-Trimethylbenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 100.0 [1] |
 | 1-(2-Chlorobenzoyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 110.0 [1] |
 | 1-(1,3-Benzodioxole-5-ylmethyl)-6,7-dihydroxyisoquinoline-3-carboxylic acid | Ki | 72.0 [1] |
 | 6-Amino-1-(1,3-benzodioxole-5-carbonyl)-7-hydroxyisoquinoline-3-carboxylic acid | Ki | 850.0 [1] |
 | 1-(1,3-Benzodioxole-5-carbonyl)-7-hydroxy-6-(methanesulfonamido)isoquinoline-3-carboxylic acid | Ki | 10000.0 [1] |