![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_5c4226cb830a715d78c0e812b3dc9cdd.svg) | BMS-345541 free base | IC50 | 4000.0 [1], 7000.0 [2], 7400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_cda2c0d4fb3e64d2d833b7a45de09f97.svg) | N,12-Dimethyl-4-phenyl-5-thia-3,7,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-8-amine | IC50 | 3500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 39.0 [1], 233.0 [2] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_1ed2abe58887dc0b39d0a378921ec617.svg) | N-(6-Chloro-9h-pyrido[3,4-b]indol-8-yl)-3-pyridinecarboxamide | IC50 | 100.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_8234c79ad4f66a353350852beb5c645b.svg) | IKK-3 Inhibitor | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_5eb7c0a7cacc81912401d61a086270ec.svg) | 2-Amino-6-(2-hydroxyphenyl)-4-(piperidin-3-yl)nicotinonitrile | IC50 | 25.0 [1], 640.0 [2] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_c6db1d6dcee6e175b3f267c444b82bcb.svg) | N-(2-Hydroxyethyl)-N-methyl-4-(2-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)benzenesulfonamide | IC50 | 3162.28 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_911177fa2869dc2bdbb469ec8bdbe1ad.svg) | Ikk-IN-3 | IC50 | 400.0 [1], 910.0 [2] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_4cbaf293bcef43bb19d8e103e811b548.svg) | N,12-Dimethyl-4-phenyl-5-oxa-3,7,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-8-amine | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_865746d835583d88973389664b06f06d.svg) | N-[[3-[12-Methyl-8-(methylamino)-5-thia-3,7,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-4-yl]phenyl]methyl]acetamide | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_efd1fd77db1b4aa2a203a649ccf609c0.svg) | N-(2-Hydroxyethyl)-4-(2-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)benzenesulfonamide | IC50 | 316.23 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_e96387ed7bf7bcc63fa4871d4bd704d2.svg) | N-(1,1-Dioxothian-4-yl)-4-(2-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)benzenesulfonamide | IC50 | 12.59 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_9f8d90734fbd076d0f69a0cd2f3a2e8d.svg) | N,5,12-Trimethyl-4-phenyl-3,5,7,10,12-pentazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-8-amine | IC50 | 4280.0 [1], 4300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_74c6bfc2119f396001686553946f1e5a.svg) | N-(5-(4-(Cyclopropylamino)-1-methyl-1H-pyrazolo[5,1-b]purin-7-yl)-2-fluorobenzyl)acetamide | IC50 | 9700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_c9ce605e2e26d2116e0266ed92c933bb.svg) | 9H-Pyrido[3,4-B]indole | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ac3e480be97d6b6b37a55fb286e12989.svg) | Wedelolactone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_e02f47dfecdec520aa0e453d4d995fe9.svg) | N-[3,5-Bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ef10bad63b05c4d3b58fc3fdd89dd3bf.svg) | Bms-345541 | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_01ee52814ec477c7ff5398120cd01839.svg) | CID 46215815 | IC50 | 25118.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ef3bb5e9eebea0a564c792421c9ebf1b.svg) | 1-(5-Methoxy-2-(thiophen-2-yl)quinazolin-4-ylamino)-3-methyl-1H-pyrrole-2,5-dione | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_395eadb5c11749508e849fc6f2ebcb7c.svg) | CID 22291652 | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_4e8b5202a71aafe003ab207cc4576058.svg) | 3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 591.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_fa6bb23d0a45b7ba93e3c09b9d34e672.svg) | A-770041 | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_27d3a5b4d06517b7e7f7d0e79a2b07e5.svg) | CID 44219749 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_dad0aaa048ebcd00eb20a880841bc7cd.svg) | 2-Amino-6-(2-(cyclopropylmethoxy)-6-hydroxyphenyl)-4-(4-piperidinyl)-3-pyridinecarbonitrile | IC50 | 250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_991f4eb39853d679b1b738198f628b67.svg) | IKK Inhibitor VII | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_bed5906fd28416c909277c96cfa5f5b2.svg) | 2-Amino-3-phenyl-5-(pyridin-4-yl)benzamide | IC50 | 3162.28 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_d08c8df6e94005871234961fea54ad8e.svg) | 3-Methyl-4-phenyl-1H-pyrazol-5-amine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_5f9d90b38bf8a433ad98aef5d1ac5970.svg) | Unii-BL7xsd8R7B | IC50 | 4960.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ae731e7b3444ffc61b7ea08d4dd4951a.svg) | 4-(4-Chlorophenyl)-3-methyl-1H-pyrazol-5-amine | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_a854ddb6bfde0a9a88ce4fa095d11537.svg) | N-[3-[2-Amino-3-cyano-6-(2-hydroxyphenyl)pyridin-4-yl]phenyl]-5-oxooxolane-2-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_aa699795408b1b00afa26249ca5e9dbd.svg) | 2-Amino-3-(4-methanesulfonamidophenyl)-5-phenylbenzamide | IC50 | 12589.25 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_83e14a15872fce09dfb2e4b93eefacb5.svg) | 2-Amino-5-(4-fluorophenyl)-3-(pyridin-4-yl)benzamide | IC50 | 5011.87 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_116c2ff6beb0da8839daf2834956e6c9.svg) | [3-[8-(2-Aminoethylamino)-12-methyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-4-yl]phenyl]methanol | IC50 | 450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_4979de01cec63dc317ddaf322908a334.svg) | 2-Amino-5-(4-fluorophenyl)-N-methyl-3-[4-(pyrrolidine-1-sulfonyl)phenyl]benzamide | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_58857746bb908d8c0eb627e1af46c827.svg) | 2-Methoxy-5-(pyridin-4-yl)benzamide | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_c4a66428e90180ce5b8319a155ab9ea9.svg) | 5-(4-Chlorophenyl)-2-methoxy-3-(4-sulfamoylphenyl)benzamide | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_427ee039f6e369ae814c5c04966e3265.svg) | 3-(7-Phenylmethoxyisoquinolin-6-yl)benzenesulfonamide | IC50 | 25118.86 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_bcf12368507eeccd7f86ac00660c194b.svg) | 4-(7-Phenylmethoxyisoquinolin-6-yl)benzenesulfonamide | IC50 | 25118.86 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_072558bb7e4832c547f06adbdb6ef1c3.svg) | 3-Amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide | IC50 | 2800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_edc84196e7f0496a1c21e674ea92f53d.svg) | Unii-8FX9DP2Y1W | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_54032e356f0dad22a2a869fb4dfc0293.svg) | 2-Amino-5-phenylbenzamide | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_011012aa587558b4e20ee47ffe2c3743.svg) | 2-Amino-4-[4-(hydroxymethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Ki | 650.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_04d49d855dd5892ba8b5cb3954595ac2.svg) | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-yl]-phenyl}-3-piperidin-1-yl-propionamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 3800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_7a12f170a7cb55113185f3edf40ef06b.svg) | Eudistomin N | IC50 | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_12d0c9d9f1ade6d62c787628d2ab32af.svg) | 4-Phenyl-1H-pyrrolo[2,3-b]pyridine | IC50 | 3981.07 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_27a9235a7b74fa5070f9aa22f372cd33.svg) | 4-[6-(Cyclopropylmethylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[2-(dimethylamino)ethyl]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ddf2ef993e10f80b25ae8a5e90a83b7c.svg) | N'-[4-(Furan-3-yl)-12-methyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl]ethane-1,2-diamine | IC50 | 940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_713995c7ccd1129582528680e8b10197.svg) | 4-[3-(Aminomethyl)phenyl]-N,12-dimethyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-amine | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_d65f66d741190614a9b10e8b233e09ef.svg) | 12-Methyl-8-(methylamino)-4-[3-[2-(sulfamoylamino)ethyl]phenyl]-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene | IC50 | 440.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_1d6fbc0ce6a61ce9f033613ce761fe81.svg) | 2-Amino-N-methyl-3-[3-[12-methyl-8-(methylamino)-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-4-yl]phenyl]propanamide | IC50 | 330.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_a43afe770910d7255dc852906b37081d.svg) | 3-Amino-5-phenylthiophene-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_5a3c1d6e40b3918454ee189e5585b0e8.svg) | 3-Methoxy-N-[[3-[3-methyl-7-(methylamino)-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-11-yl]phenyl]methyl]propanamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_551b37c8962221992a8c5bea6362e8c9.svg) | 4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-ylamino}-benzonitrile | IC50 | 3802.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 3750.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_b8951a39a47a63540209bede3aab488e.svg) | N-[[3-[3-Methyl-7-(methylamino)-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-11-yl]phenyl]methyl]acetamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_f74ea2c48f2b4e50135c587236d3a254.svg) | 4-[6-(Cyclopropylmethylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S)-pyrrolidin-2-yl]methyl]benzamide | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ca8ca0342d4f6b2933de76a0905d2d71.svg) | 6-Methoxy-9H-pyrido[3,4-b]indole | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_71e3109f3d1e43ea2fb3f86fd66dba86.svg) | 12-Methyl-N-(2-piperidin-1-ylethyl)-11,14,17-triazatetracyclo[8.7.0.03,8.011,15]heptadeca-1,3,5,7,9,12,14,16-octaen-16-amine | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_228981ea27c5ff48225817203e22270d.svg) | N'-(12-Methyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl)ethane-1,2-diamine | IC50 | 12100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_9e83be4e9496db28d66d4a37a1d40aab.svg) | 6,8-Dichloro-9h-pyrido[3,4-b]indole | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_f8d4088ea7069f315c39533f6b9d791f.svg) | 5-Pyrimidin-5-yl-1H-indole-7-carboxamide | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_0731e513dda8b4631f904dc8f0082e8c.svg) | 7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_8a1dd344b4c05cae661cf29886a18d50.svg) | 5-Phenyl-3-(1-propan-2-ylsulfonylpiperidin-4-yl)-1H-indole-7-carboxamide | IC50 | 3162.28 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_8c4c1555fc78fd0be2a6f8ec77ba4b46.svg) | 3-[1-(Ethanesulfonyl)-4-piperidinyl]-5-phenyl-1H-indole-7-carboxamide | IC50 | 1995.26 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_1fe60e6d13674f8cf1dfc82fac3410b2.svg) | 7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_029f5b4cad89a2c59efa869fd9853874.svg) | N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_9410f28bb188cd1db519c68d1040508e.svg) | 5-Bromo-6-methoxy-beta-carboline | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_1b9322978d45fe964261288bf8881ebf.svg) | 5-Phenyl-3-[1-(propylsulfonyl)-4-piperidinyl]-1H-indole-7-carboxamide | IC50 | 1995.26 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_c2aa7e0fb640ea7529d7330460976868.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamide | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_98598461b658b3f77425e67c797f8e2d.svg) | N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_a3bd9a5a28d4f4d2890ccf5cdf08d883.svg) | N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_cde4e83180955e4849d8daba0837480d.svg) | N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamide | Ki | 970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_10421e3bbd509c83a1b664e2a591f506.svg) | 5-Amino-2-phenyloxazole-4-carboxylic acid amide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_b9553da9dcbbc9585dbd2fa6949060a8.svg) | N,3-Dimethyl-11-phenyl-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaen-7-amine | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_f64ae507fb96828f441cbfe1c221da9b.svg) | 1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_2d6824ed4663109c98dca83443bd727c.svg) | 3-{[(1R)-1-Phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_d0daa255fc95cccc7e01f58b87cfb70e.svg) | 2-Amino-5-phenyl-3-[4-(sulfamoylmethyl)phenyl]benzamide | IC50 | 7943.28 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_81a2dd658141e00f3859db5f67b4914b.svg) | N,12-Dimethyl-11,14,17-triazatetracyclo[8.7.0.03,8.011,15]heptadeca-1,3,5,7,9,12,14,16-octaen-16-amine | IC50 | 230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_a46d58badfcb15b9bf73f8726e9edc93.svg) | N,12-Dimethyl-14,15,17-triazatetracyclo[8.7.0.03,8.011,15]heptadeca-1,3,5,7,9,11,13,16-octaen-16-amine | IC50 | 670.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_ddc6d45656bb4e58e59b8ae9e6b6eda9.svg) | 2-[(12-Methyl-4-phenyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl)amino]acetamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_33b36dfb02b851021d6fe9c727e46608.svg) | 8-Methoxy-12-methyl-4-phenyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_780cd4700a8c5d56c7291fd7b216f81e.svg) | 4-(4-Fluorophenyl)-N,12-dimethyl-5-thia-3,7,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-8-amine | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_d10ba231151fa36e68b70e74b70b0f87.svg) | N-[[3-[12-Methyl-8-(methylamino)-5-thia-3,7,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-4-yl]phenyl]methyl]methanesulfonamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_e9512b16a73fd4b61045d8befd5edc43.svg) | N-Ethyl-4-(4-fluorophenyl)-12-methyl-5-thia-3,7,10,12-tetrazatricyclo[7.3.0.02,6]dodeca-1(9),2(6),3,7,10-pentaen-8-amine | IC50 | 3400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_47e82c9176c94bdbb785311cfa0311d0.svg) | N-(2-Aminoethyl)-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzenesulfonamide | IC50 | 251.19 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_25108dbced460f76f8afebcc49e1beb2.svg) | 4-(4-Pyrrolidin-1-ylsulfonylphenyl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 1258.93 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_482cb49acab4cd308def9ac164616570.svg) | 2-[2-[3-[12-Methyl-8-(methylamino)-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-4-yl]phenyl]ethylamino]acetamide | IC50 | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_45efe077f02067d660e6a6778d72d1d6.svg) | N-(2-Aminoethyl)-4-(2-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)benzenesulfonamide | IC50 | 125.89 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_5cb40431a5aadc9ee836d291db983599.svg) | 2-[4-[4-(2-Aminoethylsulfamoyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-2-yl]acetamide | IC50 | 158.49 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_dc9a854464a2b3e274880f8c66484aad.svg) | N'-[12-Methyl-4-(1H-pyrrol-2-yl)-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl]ethane-1,2-diamine | IC50 | 1260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_75e6f8a53efabfcf1c268c66807f93e9.svg) | N'-(12-Methyl-4-pyridin-2-yl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl)ethane-1,2-diamine | IC50 | 1240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_cc6f9969423897c78a05854b15216216.svg) | N'-[4-(2-Methoxyphenyl)-12-methyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl]ethane-1,2-diamine | IC50 | 13000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_b6d1f7a9d0d6e8360279810178025aa9.svg) | N'-[4-(3-Methoxyphenyl)-12-methyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl]ethane-1,2-diamine | IC50 | 690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/inhibitor-of-nuclear-factor-kappa-b-kinase-alpha-subunit_f7f574fa2e7118ab8513d6f10ed1d62e.svg) | N'-[4-(4-Methoxyphenyl)-12-methyl-3-thia-1,7,10-triazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl]ethane-1,2-diamine | IC50 | 2800.0 [1] |