| Ethyl 3-[8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanoylamino]benzoate | IC50 | 800.0 [1], 57000.0 [2] |
| CID 2821848 | IC50 | 17300.0 [1], 9110000.0 [2] |
| N-(1-Adamantyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1600.0 [1], 210000.0 [2] |
| N-(2,4-Dibromophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1500.0 [1], 92000.0 [2] |
| N-(2-Chloro-4-methylphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 2300.0 [1], 76000.0 [2] |
| N-(2,4-Dichlorophenyl)-11-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]undecanamide | IC50 | 3300.0 [1], 142000.0 [2] |
| N-(2,4-Dichlorophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1900.0 [1], 153000.0 [2] |
| N-(2-Hydroxy-4-methoxyphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1300.0 [1], 360000.0 [2] |
| N-(4-Azidophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1800.0 [1], 100000.0 [2] |
| N-(2,4-Difluorophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 2300.0 [1], 110000.0 [2] |
| N-(1-Adamantyl)-11-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]undecanamide | IC50 | 3800.0 [1], 124000.0 [2] |
| N-(2,4-Dimethoxyphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1100.0 [1], 205000.0 [2] |
| 8-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-yloxyphenyl)octanamide | IC50 | 1100.0 [1], 93000.0 [2] |
| 8-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(2-methylpropoxy)phenyl]octanamide | IC50 | 4800.0 [1], 55000.0 [2] |
| N-(4-Methoxyphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 3900.0 [1], 201000.0 [2] |
| 8-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propoxyphenyl)octanamide | IC50 | 1600.0 [1], 40000.0 [2] |
| N-(2,4-Dichlorophenyl)-6-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]hexanamide | IC50 | 4100.0 [1] |
| N-(1-Adamantyl)-2-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide | IC50 | 30000000.0 [1] |
| N-(2,4-Dichlorophenyl)-4-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]butanamide | IC50 | 9800.0 [1] |
| N-(2-Hydroxyphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 27000.0 [1] |
| 11-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-naphthalen-1-ylundecanamide | IC50 | 6600.0 [1] |
| N-(2,4-Dihydroxyphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 17000.0 [1] |
| N-(4-Iodophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 1300.0 [1] |
| N-(2,4-Dibromophenyl)-2-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide | IC50 | 30000.0 [1] |
| N-(4-Hydroxyphenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 30000.0 [1] |
| N-(2,4-Dibromophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfonyl]octanamide | IC50 | 1400.0 [1] |
| N-(2,4-Dichlorophenyl)-N-methyl-2-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide | IC50 | 30000.0 [1] |
| 4-[[5-[[1-(1-Adamantyl)triazol-4-yl]methylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]methyl]-2-methylphthalazin-1-one | IC50 | 30000.0 [1] |
| N-(2,4-Dichlorophenyl)-N-methyl-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 11900.0 [1] |
| (2,4-Dichlorophenyl) 8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanoate | IC50 | 800.0 [1] |
| (2,4-Dichlorophenyl) 11-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]undecanoate | IC50 | 8700.0 [1] |
| 4-[(5-Decylsulfanyl-4-methyl-1,2,4-triazol-3-yl)methyl]-2-methylphthalazin-1-one | IC50 | 7600.0 [1] |
| N-(2,4-Dichlorophenyl)-16-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]hexadecanamide | IC50 | 7300.0 [1] |
| N-(4-Chlorophenyl)-11-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]undecanamide | IC50 | 20000.0 [1] |
| 3-[8-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanoylamino]benzoic acid | IC50 | 30000.0 [1] |
| N-(2,4-Dichlorophenyl)-10-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]decanamide | IC50 | 2300.0 [1] |
| 2-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propan-2-yloxyphenyl)acetamide | IC50 | 30000.0 [1] |
| N-(4-Chlorophenyl)-8-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]octanamide | IC50 | 800.0 [1] |
| 8-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-naphthalen-1-yloctanamide | IC50 | 1900.0 [1] |
| 2-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(2-methylpropoxy)phenyl]acetamide | IC50 | 30000.0 [1] |
| N-(2-Chlorophenyl)-11-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]undecanamide | IC50 | 15000.0 [1] |
| 2-[[4-Methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propoxyphenyl)acetamide | IC50 | 30000.0 [1] |
| N-(2,4-Dichlorophenyl)-5-[4-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]triazol-1-yl]pentanamide | IC50 | 30000.0 [1] |
| Ethyl 2-[[2-[[4-methyl-5-[(3-methyl-4-oxophthalazin-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate | IC50 | 30000.0 [1] |