 | Staurosporine | IC50 | 2639.0 [1] |
 | Doramapimod | IC50 | 30000.0 [1] |
 | Bisindolylmaleimide IX mesylate | IC50 | 0.37 [1] |
 | N-(Pyridin-4-yl)-3-[1-(4-chlorobenzyl)indol-3-yl]-propanamide | IC50 | 100000.0 [1] |
 | 1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanone | IC50 | 100000.0 [1] |
 | 3-[1-[(4-Chlorophenyl)methyl]indol-3-yl]-N-(4-nitrophenyl)propanamide | IC50 | 100000.0 [1] |
 | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
 | N-[2-[2-Aminoethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]acetamide | IC50 | 40.0 [1] |
 | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
 | Tilfrinib | IC50 | 10000.0 [1] |
 | 1-Tert-butyl-3-[7-(4-hydroxy-3-methoxyphenyl)-1,5-naphthyridin-2-yl]urea | IC50 | 100000.0 [1] |
 | 4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium | IC50 | 10000.0 [1] |
 | N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amine | Ki | 1000000.0 [1] |
 | 1-Benzyl-3-[7-(1-methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]urea | IC50 | 100000.0 [1] |
 | 1-Tert-butyl-3-[7-(1-methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]urea | IC50 | 100000.0 [1] |
 | 1-[7-(1-Methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]-3-phenylurea | IC50 | 100000.0 [1] |
 | 1-Ethyl-3-[7-(4-methoxyphenyl)-1,5-naphthyridin-2-yl]urea | IC50 | 100000.0 [1] |
 | 1-[7-(3,4-Dimethoxyphenyl)-1,5-naphthyridin-2-yl]-3-ethylurea | IC50 | 13600.0 [1] |
 | 1-Tert-butyl-3-[7-(3,4-dimethoxyphenyl)-1,5-naphthyridin-2-yl]urea | IC50 | 100000.0 [1] |
 | 1-[7-(1-Methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]-3-(2-phenylethyl)urea | IC50 | 100000.0 [1] |
 | 1-(4-Methoxyphenyl)-3-(3-phenylpyrido[3,4-b]pyrazin-8-yl)urea | IC50 | 20430.0 [1] |
 | N-(3-Chloro-4-fluorophenyl)-3-phenylpyrido[3,4-b]pyrazin-8-amine | IC50 | 100000.0 [1] |
 | 3-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 2730.0 [1] |
 | N-Phenyl-3-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 100000.0 [1] |
 | N-(3-Methoxyphenyl)-3-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 100000.0 [1] |
 | 1-(3-Methoxyphenyl)-3-(2-phenylpyrido[3,4-b]pyrazin-5-yl)urea | IC50 | 100000.0 [1] |
 | 1-Ethyl-3-(2-phenylpyrido[3,4-b]pyrazin-5-yl)urea | IC50 | 100000.0 [1] |
 | N-(3-Ethynylphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine | IC50 | 100000.0 [1] |
 | 3-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-7-amine | IC50 | 100000.0 [1] |
 | N-(2-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine | IC50 | 100000.0 [1] |
 | N-(4-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine | IC50 | 100000.0 [1] |
 | 2-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-5-amine | IC50 | 922.0 [1] |
 | N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine | IC50 | 100000.0 [1] |
 | 2-(4-Methoxyphenyl)-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-5-amine | IC50 | 7250.0 [1] |
 | 2-(4-Methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-5-amine | IC50 | 100000.0 [1] |
 | 2-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-7-amine | IC50 | 30510.0 [1] |
 | N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-7-amine | IC50 | 100000.0 [1] |
 | 1-(3-Phenylpyrido[3,4-b]pyrazin-8-yl)-3-prop-2-enylurea | IC50 | 100000.0 [1] |
 | N-(3-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-7-amine | IC50 | 100000.0 [1] |
 | N-(3-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine | IC50 | 100000.0 [1] |
 | 1-(3-Methoxyphenyl)-3-(3-phenylpyrido[3,4-b]pyrazin-8-yl)urea | IC50 | 100000.0 [1] |
 | 2-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 2590.0 [1] |
 | N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-8-amine | IC50 | 8150.0 [1] |
 | 2-(4-Methoxyphenyl)-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 3210.0 [1] |
 | 2-(4-Methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 4020.0 [1] |
 | N-(2,5-Dimethoxyphenyl)-2-(4-methoxyphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 13100.0 [1] |
 | N-Phenyl-2-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 11850.0 [1] |
 | N-(3-Methoxyphenyl)-2-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine | IC50 | 12650.0 [1] |