![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_56beacecb5834864d949ff03a7a1da24.svg) | Anacardic acid | IC50 | 5000.0 [1], 33900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_648e324896787c42a6531032172f0920.svg) | N-(3-Aminopropyl)-4-methyl-2-nitrobenzenamine | IC50 | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_3e79293baa6554a056f207112eab907b.svg) | 2-(4-Fluorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-one | IC50 | 720.0 [1], 1640.0 [2], 9700.0 [3], 9740.0 [4] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_9620a896d267a8560eca00146db2c982.svg) | 2-Hydroxy-6-((8Z,11Z)-pentadeca-8,11,14-trienyl)benzoic acid | IC50 | 8500.0 [1], 667050.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_d3a96a92333cc20d419ac7fe4adaf7db.svg) | 4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 39.81 [1], 60.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_d3a96a92333cc20d419ac7fe4adaf7db.svg) | 4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one | Ki | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_9a9f99ea10bcd1869a049becf440923a.svg) | 2-[[4-(Trifluoromethyl)phenyl]methyl]-[1,2]thiazolo[5,4-b]pyridin-3-one | IC50 | 25500.0 [1], 130000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_fc353e516c40c5531708a17449b3a20b.svg) | Garcinol | IC50 | 5000.0 [1], 6000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_1f3bdc53bb07828a1afc1b805b9cd03e.svg) | 2-Phenyl-isothiazolo[5,4-b]pyridin-3-one | IC50 | 6100.0 [1], 7850.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_2d5e0d7c97ae5abfa7dd0cc62562dcbd.svg) | [[(3R)-4-[[3-[2-[2-[[(5S)-5-Acetamido-6-amino-6-oxohexyl]amino]-2-oxoethyl]sulfanylethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphate | IC50 | 108300.0 [1], 200000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ca17b639eb2f18a80f6af45f61bb708e.svg) | 5-Chloro-2-ethylisothiazol-3(2H)-one | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_9359ff17716b5b48acbb00f2ec71bd0e.svg) | 2-(4-Chlorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-one | IC50 | 3530.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_24323f14d187649b1fe4a891552e4627.svg) | 4-Bromo-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 10000.0 [1], 12589.25 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_c2a51d822a776f16002ddf5174849eea.svg) | 2-(4-Nitrophenyl)isothiazolo[5,4-b]pyridin-3-one | IC50 | 2990.0 [1], 4100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_a3224f27ecf144bd47ec996361838fbc.svg) | Methyl 3-(5-chloro-3-oxoisothiazol-2(3H)-yl)propanoate | IC50 | 1800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_5394dfe34c9b79f83ed97a63810886b3.svg) | Methyl 3-(5-chloro-1-oxido-3-oxoisothiazol-2(3H)-yl)propanoate | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_35a9f63c35e488863740f7b08b990dd1.svg) | (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-aminohexanoyl]amino]-5-amino-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]-6-aminohexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[2-[2-[3-[[(2R)-4-[[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-2-hydroxy-3,3-dimethylbutanoyl]amino]propanoylamino]ethylsulfanyl]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]-6-aminohexanoyl]amino]-5-amino-5-oxopentanoyl]amino]-4-methylpentanoic acid | IC50 | 300.0 [1], 2270.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ea73a4dbdcb8fa4fe6e36f0c85773a4e.svg) | 4-Chloro-2-methyl-5-[[(3R,5S)-1-methyl-5-(2-methylpropyl)piperidin-3-yl]amino]pyridazin-3-one | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_4a8bdf050c4fb270fcdbed83e052b18e.svg) | 2-[(4-Chlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-one | IC50 | 17450.0 [1], 17500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_c986b6031ee0af764d6d9e490fbaf18a.svg) | 6-[[(1S,2S)-1-[4-(Benzenesulfonyl)phenyl]-1-(dimethylamino)propan-2-yl]amino]-2,4-dimethyl-1,2,4-triazine-3,5-dione | IC50 | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_423bc00274fd1433a1fa05ce3714df77.svg) | N-(3-Aminopropyl)-2-nitrobenzenamine | IC50 | 5000.0 [1], 5600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_1b132512f1a80d34849fb3ed83dd99c3.svg) | 2-(4-Bromophenyl)-5-nitro-isothiazolo[5,4-b]pyridin-3-one | IC50 | 860.0 [1], 4910.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_1072bdd96b6c297cc64ee7143fbf403b.svg) | 5-Nitro-2-(4-nitrophenyl)isothiazolo[5,4-b]pyridin-3-one | IC50 | 11800.0 [1], 15800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_e523ec84d3e93289adb4d78b2263c2c9.svg) | 2-(4-Methoxyphenyl)-5-nitro-isothiazolo[5,4-b]pyridin-3-one | IC50 | 1830.0 [1], 3420.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_cecbec94af63b09f4d37df1fad93ab95.svg) | 2-(4-Nitrophenyl)-5-methylisothiazolo[5,4-b]pyridin-3(2H)-one | IC50 | 2720.0 [1], 15300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_98de2c55f84c20aa2c7ffa40e9544426.svg) | 2-[(3,4-Dichlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-one | IC50 | 6940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_770e62b0bb0883604f5a34ec1e9b13eb.svg) | 2-Benzyl-6-nitro-1,2-benzothiazol-3-one | IC50 | 7660.0 [1], 51300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_d15856481b9992c531af28acfd2c0838.svg) | N'-[[6-(3-Aminopropylimino)-1-hydroxypyridin-3-yl]methyl]propane-1,3-diamine | IC50 | 900.0 [1], 930.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_00ce96e83ec5386509794ab61b224ccf.svg) | [[(3S)-4-[[3-[2-[[1-[(5S)-5-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-aminohexanoyl]amino]-3-phosphonooxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[(2S)-1-[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-6-oxohexyl]triazol-4-yl]methylsulfanyl]ethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphate | IC50 | 1700.0 [1], 33000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_b435cd00363f22e88f8a3d51577b10bc.svg) | [[(3S)-4-[[3-[2-[[1-[(5S)-5-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-aminohexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[(2S)-1-[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-6-oxohexyl]triazol-4-yl]methylsulfanyl]ethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphate | IC50 | 2800.0 [1], 117000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_673d3c0cb8b81fd6e89698690668b3f1.svg) | (-)-Epigallocatechin gallate | IC50 | 60000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_4ae967bda795520e140f94070aba735c.svg) | Coenzyme A | IC50 | 41910.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ee5e134a0f9db83ed684beb97013f149.svg) | Plumbagin | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_0bcab5d8647f968734b5b9966bb4ff42.svg) | 4-Aminophenol | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_2a98362ac4d9ba93f4199fc9675599bc.svg) | Embelin | IC50 | 7200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_aeaebb397e7f5522eed6a8a7d6cb8719.svg) | 1-Methyl-2-quinolone | IC50 | 70000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_44d1a6e5980820d01a8d1ca3b47b75c3.svg) | Sgc-cbp30 | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_cc13628645c821a4d949b6b2e0576a37.svg) | 4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic Acid | IC50 | 7943.28 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_6fbc55e8605e89175bbb018ffc78f33d.svg) | Guttiferone E | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_16c2d85ba0302e7e1e14e3c14e1b9e5f.svg) | 4-Amino-1-naphthol | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_956917942ed65243d452c57283629da0.svg) | CID 72201043 | IC50 | 35000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_706b94c9e6ddb96fa5f00a1e011bdd19.svg) | 4-[(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamide | Ki | 5520.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_d9590244f2cccf1c183559f251d3e34a.svg) | 2-(4-Methylpyrimidin-2-yl)-1,2-benzothiazol-3-one | IC50 | 13600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_655ca0b7debd175337b550410e8c6b74.svg) | 3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_863c28a3a55f4953997b5a88219b4eb9.svg) | 2-(4-Pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiazol-3-one | IC50 | 6190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_21229a1ebcbeb2f41d2320f22e49f178.svg) | 2-(1,3-Thiazol-2-yl)-1,2-benzothiazol-3-one | IC50 | 5770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_8f587be957e90cc2349e65e06e0e83b1.svg) | Ethyl 4-(3-oxo-1,2-benzisothiazol-2(3H)-yl)benzoate | IC50 | 6950.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_e681a4fa3a5554771b16010a9723bfbb.svg) | 2-(1,3-Benzothiazol-2-yl)-1,2-benzothiazol-3-one | IC50 | 4550.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_c4f5353328a5926d5b3e06c851dafef3.svg) | 4,6-Dimethyl-2-(thiophene-2-carbonyl)-[1,2]thiazolo[5,4-b]pyridin-3-one | IC50 | 9300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ba6ac7b31d925c9fad92516bf3db4916.svg) | 4-Nitro-1-naphthol | IC50 | 221000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ed91c1f4ab0ca474a4cfc4a7a11c55f3.svg) | 2-(3-Chloro-4-fluorophenyl)-3(2H)-isothiazolone | IC50 | 4200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ccda26fa3c6ef148fc4af2021f4aec91.svg) | 2-(3-Chloro-2-fluorophenyl)-3(2H)-isothiazolone | IC50 | 5400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_83b67f6960aacb2e3d50fc7c13d45f5b.svg) | 2-(3-Methoxyphenyl)isothiazolo[5,4-b]pyridin-3(2H)-one | IC50 | 5030.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_3b2db7e956c8f5e782a66018a23382bd.svg) | 2-Phenylisothiazol-3(2H)-one | IC50 | 28000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_20a5468b26c48166284cfe2bfe6dfcdb.svg) | 4-[(2-Amino-3-chloro-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamide | Ki | 3340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_7672efe17e797eb419ee4a28137dfb48.svg) | 4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_6990fcbf87d98742eab4fabf34e6d217.svg) | [(3,5-Dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)amino] 4-methoxybenzenesulfonate | IC50 | 34700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_bdc572ed6528ad5cd07ad6a998837c32.svg) | 2-(4-Bromophenyl)isothiazolo[5,4-b]pyridin-3(2H)-one | IC50 | 4430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_f4264875efa098337df06f940867fce5.svg) | 2-(4-Methoxyphenyl)isothiazolo[5,4-b]pyridin-3(2H)-one | IC50 | 5710.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_1f9b7e5bdfbdf8ba81949e8cc4bf7c26.svg) | 2-(2-Pyridyl)-isothiazol-3(2H)-one | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_a807de320ed0ba7e36bac6b6aa1c553c.svg) | Ethyl 2-(4,6-dimethyl-3-oxoisothiazolo[5,4-b]pyridin-2(3H)-yl)acetate | IC50 | 13600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_005ddc0fafb4624ed704d74aa7a9896c.svg) | (Z)-2-Hydroxy-6-(4-(pentyloxy)styryl)benzoic acid | IC50 | 662000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_cbdf19229d5baac2dcbceba45a9008cd.svg) | Isothiazolo[5,4-b]pyridin-3(2H)-one, 2-(phenylmethyl)- | IC50 | 22960.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ba6c458cef44ebde344a4c0e58953eb6.svg) | N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_88d123e25c79c23e380ea61e9c6d6f3a.svg) | 1-(3-Phenylazanyl-1,4,6,7-Tetrahydropyrazolo[4,3-C]pyridin-5-Yl)ethanone | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_0bee2ef5aed0b70eca4c36306b6cc435.svg) | 2-Ethylisothiazol-3(2H)-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_0ebf8c19b2229f8e32287e670568e8ea.svg) | 4-Chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-one | IC50 | 19952.62 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_f1cb6c5cb09ef33ea524bd4dd020fe36.svg) | 2-[4-(Dimethylamino)phenyl]-1,2-thiazol-3-one | IC50 | 5400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_891670cb641dacb39fd161b766023487.svg) | 4-Chloro-2-methyl-5-[(1-methylpiperidin-4-yl)amino]pyridazin-3-one | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_65bf800f24f6d3c6068ae41533f41430.svg) | 4-Chloro-2-methyl-5-[(4-methyl-1,3-thiazol-5-yl)methylamino]pyridazin-3-one | IC50 | 7943.28 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_5f4e813cd4f6543a8874faca0afa2ac6.svg) | 4-Chloro-2-methyl-5-(propan-2-ylamino)pyridazin-3-one | IC50 | 31622.78 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_96e4655bd63a3aedbf69519cabe6b686.svg) | 4-Chloro-2-methyl-5-[(1-methylpiperidin-3-yl)amino]pyridazin-3-one | IC50 | 1258.93 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_dc3b42398a058d294057b59a1cdb668c.svg) | 4-Chloro-2-methyl-5-[(1-methylpyrrolidin-3-yl)amino]pyridazin-3-one | IC50 | 15848.93 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_e1cf76121bde5a9d946852bbd8796eaa.svg) | 8-[[(1R,2R)-1-(Dimethylamino)-1-phenylpropan-2-yl]amino]-6-methylpyrido[2,3-d]pyridazin-5-one | IC50 | 19.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_7bae080063e1125ada0207d815a479a7.svg) | 1-[3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_07f19120049570c4c459cbb4a2216ebe.svg) | 1-[3-[2-Fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3R)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_94507d1eee9085deec878ddd85994d54.svg) | 4-Chloro-2-methyl-5-[[(3S)-1-methylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 6309.57 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_d127bb06496e3fb32b5aec9e3f9a3b1e.svg) | 4-Chloro-2-methyl-5-[[(3R)-1-methylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_2cd428cba788bf0b8e77726b85df7b01.svg) | 4-(Dimethylamino)naphthalen-1-ol hydrochloride | IC50 | 4200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_6bd97c31313d7af50bc03add5bbc72ca.svg) | (1S,3E,5R,7S)-3-[(3,4-Dihydroxyphenyl)-hydroxymethylidene]-6,6-dimethyl-7-[(Z)-3-methylbut-1-enyl]-5-(3-methylbut-2-enyl)-1-[(E,2R)-5-methyl-2-prop-1-en-2-ylhex-3-enyl]bicyclo[3.3.1]nonane-2,4,9-trione | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_0df77083856582d763d57e4615171346.svg) | 4,5-Dichloro-2-ethylisothiazol-3(2H)-one | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_723688d46bf63ca9bb35a4c7319de2a1.svg) | Methyl 3-(3-Oxo-2-isothiazolyl)propanoate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_3a89fdd8ac9527ebdb74d9789546dc97.svg) | 2-Pentylisothiazol-3(2H)-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_978bea7426d80ec34af98e9a9f0c26c1.svg) | 5-(N-Benzylamino)-4-chloro-2-methyl-3(2H)-pyridazinone | IC50 | 12589.25 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_8bec80b24a452bf18731584f2b220e0c.svg) | 4-Chloro-2-methyl-5-[(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)amino]pyridazin-3-one | IC50 | 316.23 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_603635930d35098c33486345ffaea029.svg) | 8-Aminoisoquinolin-5-ol | IC50 | 7100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_86f8da538faf67dc1a5d459ac5ff8d81.svg) | 2-p-Tolylisothiazolo[5,4-b]pyridine-3(2H)-one | IC50 | 4630.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_5986419096142a2bb95e35881e46f18f.svg) | 4-[(E)-(2-Amino-4-Hydroxy-3,5-Dimethylphenyl)diazenyl]-N-(Pyridin-2-Yl)benzenesulfonamide | Ki | 3340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_fb69094f67a7eebad12c30b087b0230e.svg) | 5-Anilino-4-chloro-2-methylpyridazin-3-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_22339fd40a77c4d6b94a16c0b7b562ec.svg) | 4-Chloro-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 25118.86 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_8b217bb333a37ccc3d5c8c889fa5af5e.svg) | 4-Chloro-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 79.43 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_df2edad8f4139c115b485e35eafabb0e.svg) | 4-Chloro-2-methyl-5-[[(3R,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one | IC50 | 39810.72 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_3e24a735f9f05cc193a1846e7d5ec6f3.svg) | 4-Chloro-2-methyl-5-(3-methylanilino)pyridazin-3-one | IC50 | 6309.57 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_c087bf851c1cc54136b033e04682d937.svg) | 5-[2-(Aminomethyl)anilino]-4-chloro-2-methylpyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_fcf2ce514f07459050b4e8676eb35a45.svg) | 3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_ee19c44fe23cd63eeebe483bf602cc25.svg) | 3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-4-fluoro-5-(1-methylpyrazol-4-yl)benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_66f36cdb1c212ba2ae9ef53075c29058.svg) | CID 145948689 | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_fa44b72275df2582692739dd72425d01.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]-4-fluorobenzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_85a2956dc90c939e22fb6420e5725771.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]benzoic acid | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/histone-acetyltransferase-pcaf_56ee0082ae60186b992a0a052290c2c2.svg) | 3-[(1-Acetylindole-3-carbonyl)amino]-5-(oxan-2-yloxymethyl)benzoic acid | IC50 | 20000.0 [1] |