Histone acetyltransferase KAT8 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	4-Amino-1-naphthol	IC50	1100.0 [1], 1600.0 [2], 1800.0 [3], 9700.0 [4]
	4-Amino-1-naphthol	Ki	17.0 [1], 2600.0 [2]
	2-(4-Heptylphenethyl)-6-hydroxybenzoic acid	IC50	15000.0 [1], 27000.0 [2], 47000.0 [3]
	Phenylhydrazine	IC50	1000000.0 [1]
	1-Naphthylamine	IC50	181000.0 [1]
	Phenylhydrazine hydrochloride	IC50	1000000.0 [1]
	4-Aminophenol	IC50	500000.0 [1]
	4-Chloroaniline	IC50	1000000.0 [1]
	Anacardic acid	IC50	43000.0 [1]
	4-Hydroxyquinoline	IC50	500000.0 [1]
	1-Nitronaphthalene	IC50	1000000.0 [1]
	4-Fluoroaniline	IC50	1000000.0 [1]
	2-Hydroxy-6-((8Z,11Z)-pentadeca-8,11,14-trienyl)benzoic acid	IC50	43000.0 [1]
	4-Fluorobenzylamine	IC50	1000000.0 [1]
	8-Amino-2-naphthalenesulfonic acid	IC50	940000.0 [1]
	4-Nitro-1-naphthol	IC50	141000.0 [1]
	(4-Fluorophenyl)hydrazine	IC50	310000.0 [1]
	2,8-Bis(5-methyl-2-furyl)pyrido[3,2-g]quinoline-4,6-dicarboxylic acid	IC50	17000.0 [1]
	2-(1-Naphthyl)-N-(2-{[2-oxo-2-(1-pyrrolidinyl)ethyl]sulfanyl}-1,3-benzothiazol-6-yl)acetamide	IC50	14000.0 [1]
	4-[2-(1,3-Benzothiazol-2-yl)vinyl]-N,N-diethylbenzenesulfonamide	IC50	6000.0 [1]
	(4-Aminonaphthalen-1-yl)methanol	IC50	500000.0 [1]
	4-(Dimethylamino)naphthalen-1-ol hydrochloride	IC50	23000.0 [1]
	8-Aminoisoquinolin-5-ol	IC50	7600.0 [1]
	4-(Aminomethyl)naphthalen-1-ol;hydrochloride	IC50	500000.0 [1]
	4-Amino-3-methoxynaphthalen-1-ol	IC50	177000.0 [1]
	N-(4-Hydroxynaphthalen-1-yl)decanamide	IC50	250000.0 [1]
	N-(4-Hydroxynaphthalen-1-yl)-2-phenylacetamide	IC50	365000.0 [1]
	4-[(E)-2-(5-Chloro-1,3-benzothiazol-2-yl)ethenyl]-N,N-diethylbenzenesulfonamide	IC50	30000.0 [1]
	4-[(E)-2-(5,6-Dimethyl-1,3-benzothiazol-2-yl)ethenyl]-N,N-diethylbenzenesulfonamide	IC50	7700.0 [1]
	N,N-Diethyl-4-[(E)-2-(5-fluoro-1,3-benzothiazol-2-yl)ethenyl]benzenesulfonamide	IC50	40000.0 [1]
	N,N-Diethyl-4-[(E)-2-(6-fluoro-1,3-benzothiazol-2-yl)ethenyl]benzenesulfonamide	IC50	6600.0 [1]
	4-[(E)-2-(5-Bromo-1,3-benzothiazol-2-yl)ethenyl]-N,N-diethylbenzenesulfonamide	IC50	30000.0 [1]
	N-(5-Ethyl-1,3,4-thiadiazol-2-yl)-3-[3-[(5-ethyl-1,3,4-thiadiazol-2-yl)amino]-3-oxopropyl]sulfanylpropanamide	IC50	18000.0 [1]
	4-Hydroxynaphthalene-1-carboxamide	IC50	500000.0 [1]
	4-Methoxynaphthalen-1-amine hydrochloride	IC50	89000.0 [1]
	4-(Benzyloxy)naphthalen-1-amine	IC50	500000.0 [1]
	N-(4-Hydroxynaphthalen-1-yl)acetamide	IC50	500000.0 [1]
	N-(4-Hydroxynaphthalen-1-yl)propanamide	IC50	500000.0 [1]
	4-Methoxyphenylhydrazine hydrochloride	IC50	680000.0 [1]
	2,4-Dichlorophenylhydrazine hydrochloride	IC50	1000000.0 [1]
	2-(7-Methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-3-yl)-N-naphthalen-1-ylacetamide	IC50	25000.0 [1]
	3-(1-Benzofuran-2-carbonyl)-1-(furan-2-ylmethyl)-4-hydroxy-2-(4-methylphenyl)-2H-pyrrol-5-one	IC50	29000.0 [1]
	4-Amino-1-naphthalenecarbonitrile	IC50	500000.0 [1]
	7,9-Di(thiophen-2-yl)thieno[2,3-b:4,5-b']dipyridine-2,4-diol	IC50	23000.0 [1]
	Chembl4172065	IC50	66000.0 [1]
	N-(4-Hydroxynaphthalen-1-yl)-4-methylbenzenesulfonamide	IC50	37000.0 [1]
	[({[3-Cyano-4-phenyl-6-(2-thienyl)-2-pyridinyl]sulfanyl}acetyl)amino]acetic acid	IC50	74000.0 [1]
	4-Aminonaphthalen-1-yl acetate	IC50	500000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 48 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Histone acetyltransferase KAT8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/histone-acetyltransferase-kat8-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 20). Quest Database™ Histone acetyltransferase KAT8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-acetyltransferase-kat8-inhibitors-ic50-ki.
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