| Cimetidine | IC50 | 140.0 [1], 270.0 [2], 781.0 [3], 1000.0 [4] |
| Cimetidine | Ki | 70.0 [1], 170.0 [2], 490.0 [3], 5431.0 [4] |
| Histamine | Ki | 5000.0 [1], 50118.72 [2], 25118900000000.0 [3] |
| Burimamide | Ki | 3981.07 [1] |
| Immepip | Ki | 1000.0 [1], 10000.0 [2] |
| 2-(2-(4-Tert-Butylphenylthio)ethyl)-1H-imidazole | Ki | 1000.0 [1] |
| 3-Ethyl-1-[5-(1H-imidazol-4-yl)pentyl]thiourea | Ki | 10000.0 [1] |
| (8S)-N-[(3-Fluorophenyl)methyl]pentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 2148.0 [1] |
| (8S)-N-[2-(3-Fluorophenyl)ethyl]pentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 4423.0 [1] |
| (8S)-N-[2-(3-Fluorophenyl)ethyl]-N-methylpentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 4450.0 [1] |
| 5-[(3,4-Dimethoxyphenyl)methyl]-5-azahexacyclo[5.4.1.02,6.03,10.04,8.09,12]dodecan-4-ol | Ki | 3581.0 [1] |
| 7-[2-[2-(3-Chlorophenyl)ethylamino]ethyl]quinolin-2-Amine | Ki | 100.0 [1] |
| 1-[(4-Chlorophenyl)methyl]-3-[5-(1H-imidazol-4-yl)pentyl]thiourea | Ki | 1584.89 [1] |
| 1-{4-[3-((S)-3-Amino-pyrrolidin-1-yl)-propoxy]-phenyl}-ethanone | Ki | 31000.0 [1], 50000.0 [2] |
| Verapamil | Ki | 2547.0 [1] |
| Imatinib | Ki | 1930.0 [1] |
| Tamoxifen | Ki | 9240.0 [1] |
| Chlorpromazine | Ki | 2582.0 [1] |
| Haloperidol | Ki | 1147.0 [1] |
| Clozapine | Ki | 3550.0 [1] |
| Risperidone | Ki | 1458.0 [1] |
| Amiodarone | Ki | 10379.0 [1] |
| Amitriptyline | Ki | 718.0 [1] |
| Ketoconazole | Ki | 21507.0 [1] |
| Medroxyprogesterone acetate | Ki | 27453.0 [1] |
| Imiquimod | Ki | 1481.0 [1] |
| Clomipramine | Ki | 2015.0 [1] |
| Quinacrine | Ki | 3476.0 [1] |
| Promethazine | Ki | 1146.0 [1] |
| Mianserin | Ki | 992.0 [1] |
| Miconazole | Ki | 6637.0 [1] |
| Clotrimazole | Ki | 5079.0 [1] |
| Thioridazine | Ki | 934.0 [1] |
| Fluphenazine | Ki | 1205.0 [1] |
| Gentian violet | Ki | 1136.0 [1] |
| Nortriptyline | Ki | 2295.0 [1] |
| Cyproheptadine | Ki | 195.0 [1] |
| Loperamide | Ki | 3030.0 [1] |
| Pepcid | Ki | 41.0 [1] |
| Ketotifen | Ki | 4060.0 [1] |
| Promazine | Ki | 2810.0 [1] |
| Doxepin | Ki | 1836.0 [1] |
| Maprotiline | Ki | 393.0 [1] |
| Lisuride | Ki | 1022.0 [1] |
| Desloratadine | Ki | 1080.0 [1] |
| Astemizole | Ki | 1654.0 [1] |
| Econazole | Ki | 1565.0 [1] |
| Benztropine | Ki | 1185.0 [1] |
| Thioperamide | Ki | 10000.0 [1] |
| Metergoline | Ki | 959.0 [1] |
| Orphenadrine | Ki | 6845.0 [1] |
| Dimaprit | Ki | 25118.86 [1] |
| Dicyclomine | Ki | 1598.0 [1] |
| Clemastine | Ki | 364.0 [1] |
| Tirilazad | Ki | 13884.0 [1] |
| Ebastine | Ki | 2867.1 [1] |
| Dexchlorpheniramine | Ki | 8228.0 [1] |
| Impromidine | Ki | 501.19 [1] |
| Penfluridol | Ki | 1000.0 [1] |
| 1-[(5-Chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazine | Ki | 8511.38 [1] |
| Ciproxifan | Ki | 10000.0 [1] |
| 4-Methylhistamine | Ki | 7943.28 [1] |
| Tiotidine | IC50 | 22.0 [1] |
| (1S,2R)-2-(Octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol | Ki | 88.5 [1] |
| Conessine | Ki | 10000.0 [1] |
| alpha-Methyltryptamine | Ki | 10000.0 [1] |
| Amthamine | Ki | 6309.57 [1] |
| 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide | IC50 | 10000.0 [1] |
| 6-((3-Cyclobutyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)oxy)-N-methyl-3-pyridinecarboxamide | Ki | 3162.28 [1] |
| Cipargamin | IC50 | 10000.0 [1] |
| 4-(4-Butylpiperidin-1-yl)-1-o-tolylbutan-1-one | Ki | 1000.0 [1] |
| N-Desmethyl loperamide | Ki | 1.7 [1] |
| 2-Methyl-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]-5-(trifluoromethyl)quinazolin-4-one | IC50 | 10000.0 [1] |
| Impentamine | Ki | 3981070000000.0 [1] |
| Benzonitrile, 3-fluoro-5-(2-(2-(fluoromethyl)-4-thiazolyl)ethynyl)- | Ki | 10000.0 [1] |
| N,N-Diallyl-5-methoxytryptamine | Ki | 4265.8 [1] |
| (2R)-2-Amino-1-[4-[3-[4-(cyclopropanecarbonyl)phenoxy]propyl]piperazin-1-yl]propan-1-one | Ki | 70794.58 [1] |
| 4'-(3-((3R)-3-(Dimethylamino)pyrrolidinyl)propoxy)(1,1'-biphenyl)-4-carbonitrile | Ki | 10000.0 [1] |
| Methimepip | Ki | 10000.0 [1] |
| N4-(2,6-Dichlorobenzyl)-6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine | Ki | 1000.0 [1] |
| 2,4-Pyrimidinediamine, 5-[5-iodo-4-methoxy-2-(1-methylethyl)phenoxy]- | Ki | 100000000.0 [1] |
| 4-(1H-Imidazol-5-yl)butan-1-amine | Ki | 794328.23 [1] |
| Unii-N4Y2V13I7F | Ki | 2126.0 [1] |
| 1-(6-((3-Cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[D]azepin-7-YL)oxy)pyridin-3-YL)pyrrolidin-2-one | Ki | 3162.28 [1] |
| 5-[(3-Cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-methylpyrazine-2-carboxamide | Ki | 3162.28 [1] |
| 3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]-5,6,7,8-tetrahydroquinazolin-4-one | IC50 | 1000.0 [1] |
| 2-[[(2R)-1-[4-[4-[3-(Azepan-1-yl)propoxy]phenyl]butyl]pyrrolidin-2-yl]methyl]-4-[(4-chlorophenyl)methyl]phthalazin-1-one | IC50 | 10000.0 [1] |
| Thalictruberine | Ki | 672.0 [1] |
| CID 11496610 | Ki | 850.0 [1] |
| 2-Chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzoxazepine | Ki | 8709.64 [1] |
| (Z)-But-2-enedioic acid;9-chloro-4-methyl-13-oxa-4-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaene | Ki | 5.7 [1] |
| 1-Cyano-2-[4-(1H-imidazol-5-yl)butyl]-3-(2-phenylsulfanylethyl)guanidine | Ki | 4073.8 [1] |
| (4S,5S)-4-(3,4-Difluorophenyl)-N-[3-[4-(4-fluorophenyl)piperidin-1-yl]propyl]-5-methyl-2-oxo-1,3-oxazolidine-3-carboxamide | Ki | 1000.0 [1] |
| 1H-Imidazole-4-propanamine | Ki | 1000000000000.0 [1] |
| (7As,11aS)-4-piperazin-1-yl-5,6,7a,8,9,10,11,11a-octahydro-[1]benzofuro[2,3-h]quinazolin-2-amine | Ki | 9120.11 [1] |
| 1-[(1-Benzyl-1H-tetrazol-5-yl)-phenyl-methyl]-4-methyl-piperazine | IC50 | 20000.0 [1] |
| Ethyl 4-[3-(4-hexanoylphenoxy)propyl]piperazine-1-carboxylate | Ki | 12589.25 [1] |
| [4-[4-[3-[(2S,5S)-2,5-Dimethylpyrrolidin-1-yl]propoxy]phenyl]phenyl]-morpholin-4-ylmethanone | Ki | 10000.0 [1] |
| N-[1-[3-(3-Oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide | Ki | 1000.0 [1] |
| 6-(1H-Imidazol-5-yl)hexan-1-amine | Ki | 5011870000000.0 [1] |