 | Pyrilamine | IC50 | 1.3 [1], 1.8 [2], 3.0 [3], 12.59 [4], 46.77 [5] |
| Pyrilamine | Ki | 5.01e+17 [1] |
 | Histamine | IC50 | 158.49 [1], 1000.0 [2] |
| Histamine | Ki | 15848900000000.0 [1] |
 | Cetirizine | Ki | 14.0 [1] |
 | Risperidone | IC50 | 454.0 [1], 868.0 [2] |
| Risperidone | Ki | 33.0 [1] |
 | Clozapine | Ki | 1.0 [1], 1.1 [2] |
 | Olanzapine | Ki | 1.2 [1], 2.0 [2] |
 | Loratadine | IC50 | 290.0 [1], 1500000.0 [2] |
| Loratadine | Ki | 20.0 [1], 37.0 [2], 311.0 [3], 414.0 [4] |
 | Haloperidol | Ki | 323.0 [1], 440.0 [2], 730.0 [3] |
 | Quetiapine | Ki | 4.6 [1], 8.7 [2], 10.0 [3], 19.0 [4], 21.0 [5] |
 | Aripiprazole | IC50 | 420.0 [1] |
| Aripiprazole | Ki | 25.1 [1], 100.0 [2] |
 | Terfenadine | IC50 | 1.0 [1], 563.0 [2] |
| Terfenadine | Ki | 2.59 [1], 40.0 [2], 58.0 [3] |
 | Ketotifen | IC50 | 1.0 [1], 2300.0 [2] |
| Ketotifen | Ki | 0.14 [1], 0.16 [2] |
 | Fexofenadine | IC50 | 15.0 [1], 78.0 [2] |
| Fexofenadine | Ki | 27.0 [1] |
 | Diphenhydramine | IC50 | 84000.0 [1] |
| Diphenhydramine | Ki | 14.79 [1], 20.0 [2] |
 | Desloratadine | IC50 | 16000.0 [1] |
| Desloratadine | Ki | 0.97 [1], 1.16 [2] |
 | Latrepirdine | IC50 | 158.0 [1], 160.0 [2], 1580.0 [3] |
 | 2-[[(2R)-1-[4-[4-[3-(Azepan-1-yl)propoxy]phenyl]butyl]pyrrolidin-2-yl]methyl]-4-[(4-chlorophenyl)methyl]phthalazin-1-one | Ki | 10.0 [1], 15.85 [2] |
 | (-)-Dimethyl-{2-[3-((R)-1-pyrazin-2-yl-ethyl)-1H-inden-2-yl]-ethyl}-amine | Ki | 1.3 [1], 1.5 [2] |
 | Chlorpromazine | IC50 | 12.0 [1] |
| Chlorpromazine | Ki | 1.96 [1], 4.25 [2] |
 | Mianserin | IC50 | 3.39 [1] |
| Mianserin | Ki | 0.17 [1], 1.7 [2] |
 | Ziprasidone | Ki | 5.3 [1], 47.0 [2], 510.0 [3] |
 | Chlorpheniramine | IC50 | 66.0 [1] |
| Chlorpheniramine | Ki | 0.92 [1], 7.0 [2] |
 | Doxepin | Ki | 0.07 [1], 0.18 [2], 0.25 [3] |
 | Astemizole | Ki | 1.61 [1], 2.09 [2], 3.0 [3] |
 | Azelastine | Ki | 1.2 [1], 1.26 [2] |
 | 2-Chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzoxazepine | Ki | 7.76 [1], 8.32 [2] |
 | 4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)butan-1-one | Ki | 8780.0 [1] |
 | CID 11753159 | IC50 | 40.0 [1] |
| CID 11753159 | Ki | 31.62 [1] |
 | N,N-Dimethyl-2-[3-(pyrazin-2-ylmethyl)-1H-inden-2-yl]ethanamine | Ki | 4.0 [1] |
 | N,N-Dimethyl-1-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)methanamine | IC50 | 6.76 [1], 1000.0 [2] |
 | Benzo[B]thiophene-2-ethanamine, N,N-dimethyl-3-[(1R)-1-(2-pyridinyl)ethyl]- | Ki | 4.0 [1], 4000.0 [2] |
 | 1-[1-[(4-Fluorophenyl)methyl]benzimidazol-2-yl]-N-methyl-N-(oxan-4-ylmethyl)piperidin-4-amine | Ki | 3.9 [1] |
 | Antihistamine-1 | Ki | 6.9 [1] |
 | [1-[(4-Fluorophenyl)methyl]benzimidazol-2-yl]-[1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl]methanone | IC50 | 7.23 [1], 59.0 [2] |
 | [1-[2-[3-(3,4-Dimethoxyphenyl)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-3-yl]ethyl]piperidin-4-yl]-[1-[(4-fluorophenyl)methyl]benzimidazol-2-yl]methanone | IC50 | 6.48 [1], 309.0 [2] |
 | Amitriptyline | Ki | 0.56 [1], 1.12 [2] |
 | Promethazine | IC50 | 5.4 [1] |
| Promethazine | Ki | 0.33 [1] |
 | Fluphenazine | Ki | 4.66 [1], 40.0 [2] |
 | Promazine | IC50 | 2454.71 [1] |
| Promazine | Ki | 0.4 [1] |
 | Maprotiline | Ki | 1.02 [1], 1.67 [2] |
 | Thioperamide | Ki | 10000.0 [1] |
 | Tripelennamine | IC50 | 39.81 [1] |
| Tripelennamine | Ki | 1e+17 [1] |
 | Chlorprothixene | IC50 | 870.96 [1] |
| Chlorprothixene | Ki | 3.75 [1] |
 | Orphenadrine | IC50 | 97723.72 [1] |
| Orphenadrine | Ki | 144.0 [1] |
 | Sertindole | Ki | 0.51 [1], 570.0 [2] |
 | Zotepine | Ki | 0.62 [1], 3.4 [2] |
 | 2-(2-Aminoethyl)pyridine | IC50 | 1258.93 [1] |
| 2-(2-Aminoethyl)pyridine | Ki | 6309570000000.0 [1] |
 | 1-[(5-Chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazine | Ki | 977.24 [1], 46773.51 [2] |
 | Ciproxifan | Ki | 2511.89 [1], 10000.0 [2] |
 | N-[4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclohexyl]quinoline-4-carboxamide | Ki | 630.96 [1] |
 | Histaprodifen | IC50 | 794.33 [1] |
| Histaprodifen | Ki | 501187000000000.0 [1] |
 | 2-(3-Trifluoromethylphenyl)histamine | IC50 | 1000.0 [1] |
| 2-(3-Trifluoromethylphenyl)histamine | Ki | 251189000000000.0 [1] |
 | N,N-Diallyl-5-methoxytryptamine | Ki | 1258.93 [1], 10000.0 [2] |
 | 2,6,3,5-Ethanediylidenepentaleno(1,6-bc)pyrrol-2(1H)-ol, octahydro-1-(phenylmethyl)- | Ki | 10000.0 [1] |
 | 2-(3-Chlorophenyl)histamine | IC50 | 1995.26 [1] |
| 2-(3-Chlorophenyl)histamine | Ki | 158489000000000.0 [1] |
 | 4-(3-(4-Chlorophenyl)-3-hydroxypyrrolidin-1-yl)-1-(4-fluorophenyl)butan-1-one | Ki | 259.6 [1], 1467.0 [2] |
 | 2-(2-(4-Tert-Butylphenylthio)ethyl)-1H-imidazole | Ki | 1000.0 [1] |
 | R-Dimethindene | Ki | 0.4 [1], 0.44 [2] |
 | 2-[(11E)-11-[2-(Dimethylamino)ethylidene]-6H-benzo[c][1]benzoxepin-2-yl]acetic acid | Ki | 11.0 [1] |
 | 6-Chloro-2-(4-methylpiperazin-1-yl)-N-(thiophen-2-ylmethyl)quinazolin-4-amine | Ki | 19.95 [1], 549.54 [2] |
 | 1-(4-Fluorophenyl)-4-[4-[pyrimidin-2-yl]piperazin-1-yl]butan-1-one | Ki | 911.8 [1], 912.0 [2] |
 | [3-(4-Chloro-phenyl)-3-pyridin-2-yl-propyl]-[4-(1H-imidazol-4-yl)-butyl]-methyl-amine | Ki | 7.0 [1] |
 | 2,8-Dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole | IC50 | 40.0 [1], 146.0 [2] |
 | Norketotifen | IC50 | 11000.0 [1] |
 | 1H-Imidazole-5-decanamine | IC50 | 501.19 [1] |
| 1H-Imidazole-5-decanamine | Ki | 199526000000000.0 [1] |
 | 1-(17-Chloro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine | IC50 | 2.34 [1] |
 | 8-(1H-Imidazol-5-yl)octan-1-amine | IC50 | 3162.28 [1] |
| 8-(1H-Imidazol-5-yl)octan-1-amine | Ki | 25118900000000.0 [1] |
 | 2-(6-Fluoro-3-(pyridazin-3-ylmethyl)-1H-inden-2-yl)-N,N-dimethylethanamine | Ki | 1.7 [1] |
 | N-(1-(3-Ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine | Ki | 624.0 [1] |
 | 4-[(4-Chlorophenyl)methyl]-2-[[(2R)-1-methylpyrrolidin-2-yl]methyl]phthalazin-1-one | Ki | 0.16 [1] |
 | 3-((E)-3-Carboxy-3-phenyl-allyl)-4,6-dichloro-1H-indole-2-carboxylic acid | IC50 | 3.0 [1], 10000.0 [2] |
 | 2-[10-[3-[4-(1,3-Dimethyl-2,6-dioxopyrimidin-4-yl)piperazin-1-yl]propyl]phenothiazin-2-yl]acetic acid | IC50 | 40.0 [1] |
 | 2-[3-[(1R)-1-(3-Methoxypyrazin-2-yl)ethyl]-6-methyl-1H-inden-2-yl]-N,N-dimethylethanamine | Ki | 2.7 [1] |
 | 2-[6-Fluoro-3-[(1R)-1-(3-methoxypyrazin-2-yl)ethyl]-1H-inden-2-yl]-N,N-dimethylethanamine | Ki | 0.7 [1] |
 | (8S)-N-[2-(3-Fluorophenyl)ethyl]pentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 2376.0 [1] |
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