![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_173905a1d8206fe6271a8ee9486c99d9.svg) | Foretinib | IC50 | 1.48 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 2.93 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | Ki | 2.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_34ec291e290db2e13648ccc8dee7e3a5.svg) | Cabozantinib | IC50 | 3.2 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_179888a64edb35ddee0be2a16e245b3a.svg) | MK-2461 | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_76787d25691f7fba9b30cd2607d2cf7e.svg) | N-[4-[2-(Cyclopropanecarbonylamino)imidazo[1,2-a]pyridin-6-yl]oxy-3-fluorophenyl]-6-methyl-2-oxo-1-phenyl-3H-pyridin-1-ium-3-carboxamide;hydrochloride | IC50 | 1.8 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_13756c608c557f48b9b323793aa85ae2.svg) | MGCD-265 analog | IC50 | 37.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_c1834625131d0c2ad0228dc67b109c54.svg) | MK-8033 | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_6218d7660845b31fc510a0466313fd99.svg) | Amg-458 | IC50 | 60.0 [1], 60.1 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_6218d7660845b31fc510a0466313fd99.svg) | Amg-458 | Ki | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_bfd85af270caa82a688349ad39ce47ce.svg) | 3-{4-[(6,7-Dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1-(2-phenylacetyl)thiourea | IC50 | 80.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_bfd85af270caa82a688349ad39ce47ce.svg) | 3-{4-[(6,7-Dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1-(2-phenylacetyl)thiourea | Ki | 1.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_e7ecb06887875f4d78baf892d82c33a5.svg) | Bms-777607 | IC50 | 3.9 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_14411dd3120773160cc07f6ade4c2560.svg) | 2-(4-(1-(Quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyrazol-1-yl)ethanol | IC50 | 4.0 [1], 4.8 [2], 50.12 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_14411dd3120773160cc07f6ade4c2560.svg) | 2-(4-(1-(Quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyrazol-1-yl)ethanol | Ki | 5.0 [1], 3900.0 [2], 9400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_0d9863ed59ccd1ba92b866d4ff4460aa.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-2-oxo-3-phenylimidazolidine-1-carboxamide | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_996164250bbde43ee54714faae2ca9dc.svg) | Met Kinase Inhibitor | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_11549cc58762e998db6ef36098510dec.svg) | 7-Methoxy-4-((6-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy)quinoline | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_008b82bfee0baa55c0bab6b3c3e488d2.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_829d9468648eaacd7ae7ad912dac6a2f.svg) | N-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_829d9468648eaacd7ae7ad912dac6a2f.svg) | N-[4-(6,7-Dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_088eb7e3c0fbd58f12adde928af7d44f.svg) | Pha-665752 | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_3ca463911c10f9e6fd157255477b222e.svg) | Jnj-38877605 | IC50 | 0.95 [1], 1.0 [2], 4.0 [3], 5.5 [4], 9.5 [5] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a97274caafef70d6423d3784397e9e54.svg) | Pyrimidone, 22 | IC50 | 8.9 [1], 10.0 [2], 17.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a97274caafef70d6423d3784397e9e54.svg) | Pyrimidone, 22 | Ki | 8.9 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_d003396626f828bad7bbc0670df7974b.svg) | 7-Methoxy-N-[[6-(3-methyl-1,2-thiazol-5-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methyl]-1,5-naphthyridin-4-amine | IC50 | 3.0 [1], 5.0 [2], 6.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_d003396626f828bad7bbc0670df7974b.svg) | 7-Methoxy-N-[[6-(3-methyl-1,2-thiazol-5-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methyl]-1,5-naphthyridin-4-amine | Ki | 3.2 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_3675ea77fc19d393771a33a213dcb993.svg) | Exelixis | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_891690896eeff1c78d6c3aa623867591.svg) | 7-Methoxy-4-[[6-(3,4,5-trifluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methoxy]quinoline | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_3c87ee505c56c8f66f423c9499af032e.svg) | 6-[[5-(1-Methylpyrazol-4-yl)triazolo[4,5-b]pyrazin-3-yl]methyl]quinoline | IC50 | 1.0 [1], 5.0 [2], 6.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_3c87ee505c56c8f66f423c9499af032e.svg) | 6-[[5-(1-Methylpyrazol-4-yl)triazolo[4,5-b]pyrazin-3-yl]methyl]quinoline | Ki | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_4007905bf1b83417ff849df1a48deeff.svg) | N-(4-(6,7-Dimethoxyquinolin-4-yloxy)-3-fluorophenyl)-2-oxo-3-phenylimidazolidine-1-carboxamide | IC50 | 30.0 [1], 53.0 [2], 80.0 [3], 90.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_4007905bf1b83417ff849df1a48deeff.svg) | N-(4-(6,7-Dimethoxyquinolin-4-yloxy)-3-fluorophenyl)-2-oxo-3-phenylimidazolidine-1-carboxamide | Ki | 1.7 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 2000.0 [1], 5000.0 [2], 10000.0 [3], 20000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_0b26d99558edb7945fcd4dd139772b8b.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 2.7 [1], 50.0 [2], 50.5 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_0b26d99558edb7945fcd4dd139772b8b.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 2.7 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_ce7820b1774232cc857645e5c91d9722.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-3-methyl-5-oxo-1-phenyl-2-propylpyrazole-4-carboxamide | IC50 | 1.0 [1], 48.8 [2], 49.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_ce7820b1774232cc857645e5c91d9722.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-3-methyl-5-oxo-1-phenyl-2-propylpyrazole-4-carboxamide | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_299f60fa01ae06e7e6754a7708ea764c.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 1.0 [1], 37.0 [2], 37.1 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_299f60fa01ae06e7e6754a7708ea764c.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1,5-dimethyl-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 1.0 [1], 1.1 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_2a2660d026243688162755690ee4d31f.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-5-methyl-1-(2-methylpropyl)-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 8.0 [1], 204.0 [2], 205.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_2a2660d026243688162755690ee4d31f.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-5-methyl-1-(2-methylpropyl)-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 7.9 [1], 8.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_5d18b5d269298b34df700590b02c098e.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1-[(2R)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 1.0 [1], 23.9 [2], 24.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_5d18b5d269298b34df700590b02c098e.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1-[(2R)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_5d9c6aa4b003cacfe953a92f8749cba7.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1-[(2S)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenylpyrazole-4-carboxamide | IC50 | 1.1 [1], 23.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_5d9c6aa4b003cacfe953a92f8749cba7.svg) | N-[3-Fluoro-4-(7-methoxyquinolin-4-yl)oxyphenyl]-1-[(2S)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenylpyrazole-4-carboxamide | Ki | 1.1 [1], 1.2 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_fb688c8844d3beb9acf7e66723fed7f2.svg) | N-[4-[2-(1-Ethylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-3-(4-fluorophenyl)-2-oxoimidazolidine-1-carboxamide | IC50 | 27.0 [1], 50.0 [2], 80.0 [3], 240.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_3967f1261f1958810b393b6f50ce9b27.svg) | 14-(Dimethylsulfamoylamino)-5-(1-methylpyrazol-4-yl)-2-oxo-7-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,9,12,14-heptaene | IC50 | 4.0 [1], 80.0 [2], 2300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_95a0bd49e8f0995cb52a25e6fd825622.svg) | 4,4,4-Trifluoro-3-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyanilino]-N-phenylbutanamide | IC50 | 120.0 [1], 600.0 [2], 2000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a40095a79a599a6cda5c4729587e3d26.svg) | 6-[6-(1-Methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-ylmethyl]-quinoline | IC50 | 44.0 [1], 69.0 [2], 210.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a40095a79a599a6cda5c4729587e3d26.svg) | 6-[6-(1-Methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-ylmethyl]-quinoline | Ki | 9.1 [1], 74.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_44aa3a6da7f2767bb07774343291b239.svg) | 4-[6-Amino-7-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]furo[3,2-c]pyridin-3-yl]-3,6-dihydro-2H-pyridine-1-carboxamide | IC50 | 26.0 [1], 42.0 [2], 72.0 [3], 110.0 [4], 600.0 [5] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_295456cbf7462dfb1eaccb88d6610904.svg) | Ceritinib | IC50 | 1000.0 [1], 1339.0 [2], 3170.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_aba28ba585d470d0fb1d160136f20f63.svg) | Sgx-523 | IC50 | 3.1 [1], 4.0 [2], 10.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_148d73a3c69ad2442b2ff4fa96bdd7d2.svg) | Tepotinib | IC50 | 1.0 [1], 3.0 [2], 12.0 [3], 100.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_21d6e904e32e34e781ccc6fa674af808.svg) | 2-Anilino-5-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-3-methylpyrimidin-4-one | IC50 | 63.0 [1], 204.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_21d6e904e32e34e781ccc6fa674af808.svg) | 2-Anilino-5-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-3-methylpyrimidin-4-one | Ki | 14.0 [1], 63.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_f2cc18ad5e660107226d8ffcd618f049.svg) | 4-[[6-(3,4-Difluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methoxy]-7-methoxyquinoline | IC50 | 9.0 [1], 26.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_31834f3b299fabd311c318495f3a11c2.svg) | 4-[[6-(3,5-Difluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methoxy]-7-methoxyquinoline | IC50 | 7.0 [1], 14.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_0867a4b23aa1261f5cb0270b8bc6fbc1.svg) | 4-((6-Phenyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl)methyl)phenol | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_0867a4b23aa1261f5cb0270b8bc6fbc1.svg) | 4-((6-Phenyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl)methyl)phenol | Ki | 1231.2 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_4ea34da568b591c3e564c159dc82da53.svg) | N'-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-N-phenylpropanediamide | IC50 | 28.0 [1], 30.0 [2], 310.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_877302b8970932e44cb0ebb834e06ea9.svg) | N-[3-Fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-N'-methyl-N'-phenylpropanediamide | IC50 | 40.0 [1], 43.0 [2], 160.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_32c42f09aed37667ccd6db596b95de84.svg) | CID 50942314 | IC50 | 10.0 [1], 44.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_d18f629912511ec170cadb0abc53b05d.svg) | 5-[8-Fluoro-3-[(1S)-1-[3-(2-methoxyethoxy)quinolin-6-yl]ethyl]-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-3-methyl-1,2-oxazole | IC50 | 1.0 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_4a442f939c39e8e80f3a090313130005.svg) | 4-((6-(3-Fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy)-7-methoxyquinoline | IC50 | 7.0 [1], 20.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_4a442f939c39e8e80f3a090313130005.svg) | 4-((6-(3-Fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy)-7-methoxyquinoline | Ki | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_96fd26ce57ec5417926f25dd1a0d5133.svg) | 4-[6-(1-Piperidin-4-ylpyrazol-4-yl)pyrrolo[3,2-b]pyridin-1-yl]sulfonyl-2,1,3-benzoxadiazole | IC50 | 9.0 [1], 130.0 [2], 200.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_351dca11b0978ed72c57335a69174e49.svg) | 3-[(1S)-1-[3-(2-Methoxyethoxy)quinolin-6-yl]ethyl]-5-(3-methyl-1,2-thiazol-5-yl)triazolo[4,5-c]pyridin-4-one | IC50 | 0.6 [1], 1.0 [2], 2.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_e9da0f3b0f4f977e5ba9003068778a84.svg) | 1-(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonylpyrrolo[3,2-b]pyridin-6-ol | IC50 | 15.0 [1], 35.0 [2], 2810.0 [3], 3600.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_244a570dc1f43136597a5cc7147a8e97.svg) | 1-(2,1,3-Benzoxadiazol-4-ylsulfonyl)pyrrolo[3,2-b]pyridin-6-amine | IC50 | 16.0 [1], 1300.0 [2], 2200.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_f1ba9a3fcaddc2ebc1359d0e7a75f4fa.svg) | Tert-butyl 4-[4-[1-(2,1,3-benzoxadiazol-4-ylmethyl)pyrrolo[3,2-b]pyridin-6-yl]pyrazol-1-yl]piperidine-1-carboxylate | IC50 | 33.0 [1], 3080.0 [2], 3280.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a4b82563b5c8d541158097f7f1008790.svg) | 1-[4-[1-(2,1,3-Benzoxadiazol-4-ylsulfonyl)pyrrolo[3,2-b]pyridin-6-yl]piperazin-1-yl]ethanone | IC50 | 12.0 [1], 370.0 [2], 500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_e6580d7656dd721eb8eda370b4e264d1.svg) | 4-[6-[6-(4-Methylpiperazin-1-yl)pyridin-3-yl]pyrrolo[3,2-b]pyridin-1-yl]sulfonyl-2,1,3-benzoxadiazole | IC50 | 15.0 [1], 820.0 [2], 1310.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_cbb8d928d759c4e4cfb35b77102a0e61.svg) | [4-[1-(2,1,3-Benzoxadiazol-4-ylsulfonyl)pyrrolo[3,2-b]pyridin-6-yl]piperazin-1-yl]-pyridin-3-ylmethanone | IC50 | 11.0 [1], 430.0 [2], 480.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_1fe4e53ad12c0c4bc19eb8378ed59a3b.svg) | 6-Chloro-5-[6-(1-piperidin-4-ylpyrazol-4-yl)pyrrolo[3,2-b]pyridin-1-yl]sulfonylimidazo[2,1-b][1,3]thiazole | IC50 | 9.0 [1], 90.0 [2], 110.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_f24b23344aac718bfa0d5b0e07b4d324.svg) | Tert-butyl 4-[1-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonylpyrrolo[3,2-b]pyridin-6-yl]piperazine-1-carboxylate | IC50 | 15.0 [1], 27.0 [2], 110.0 [3], 1946.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_74b84d7e0465e7f1ad19a538545a3596.svg) | 4-[[6-(1-Piperidin-4-ylpyrazol-4-yl)pyrrolo[3,2-b]pyridin-1-yl]methyl]-2,1,3-benzoxadiazole | IC50 | 19.0 [1], 1800.0 [2], 1880.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_6fa595e8b492cbab08f08d586e6f06cd.svg) | 1-[4-[1-(2,1,3-Benzoxadiazol-4-ylsulfonyl)pyrrolo[3,2-b]pyridin-6-yl]piperazin-1-yl]-2-(methylamino)ethanone | IC50 | 14.0 [1], 570.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_807fa90a349e3687875d50fb3955dcaa.svg) | 1-(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonylpyrrolo[3,2-b]pyridin-6-amine | IC50 | 10.0 [1], 490.0 [2], 580.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_b49bbce538d3961a014ba30c1faf7566.svg) | Tert-butyl 4-[4-[1-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonylpyrrolo[3,2-b]pyridin-6-yl]pyrazol-1-yl]piperidine-1-carboxylate | IC50 | 19.0 [1], 27.0 [2], 147.0 [3], 450.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_7484802d00d8ba1db697df4d12364e90.svg) | 2-[[5-Chloro-2-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-8-yl)amino]pyrimidin-4-yl]amino]-3-fluoro-N-methylbenzamide | IC50 | 30.0 [1], 99.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_3b63168436801b607ec3eed609d3e1b7.svg) | 2-[[5-Chloro-2-[(5,5-dimethyl-2-oxo-3,4-dihydro-1H-1-benzazepin-8-yl)amino]pyrimidin-4-yl]amino]-3-fluoro-N-methylbenzamide | IC50 | 10.0 [1], 54.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_60a34a7bd0583832a77a26655d54f194.svg) | 3-(Quinolin-6-ylmethyl)triazolo[4,5-b]pyrazin-5-amine | IC50 | 34.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_60a34a7bd0583832a77a26655d54f194.svg) | 3-(Quinolin-6-ylmethyl)triazolo[4,5-b]pyrazin-5-amine | Ki | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_717a437add2d881c7d58aabccef74086.svg) | N-(2-Oxo-5-phenyl-7-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,9,12,14-heptaen-14-yl)methanesulfonamide | IC50 | 31.0 [1], 220.0 [2], 2500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a663b46fb97c88a3cf92243ddd32af41.svg) | 4,4,4-Trifluoro-3-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyanilino]-N-(4-fluorophenyl)butanamide | IC50 | 90.0 [1], 370.0 [2], 400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_4920bb9b2f00a1d540791d3fedf9429d.svg) | 4,4,4-Trifluoro-3-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyanilino]-N-(2-methoxyphenyl)butanamide | IC50 | 840.0 [1], 1800.0 [2], 2000.0 [3], 10000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_02d01ae48d323b0125be350e64bb0d1d.svg) | 4,4,4-Trifluoro-N-(4-fluorophenyl)-3-[4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyanilino]butanamide | IC50 | 180.0 [1], 880.0 [2], 2000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_e9817a68180fd27b8be3cb9779f8d759.svg) | Golvatinib | IC50 | 14.0 [1], 20.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_83f168413fde213ed776ff4e7cbe23cf.svg) | CID 21081761 | IC50 | 1.8 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_9e48bc4412b7047b44e1bb0572185347.svg) | N'-[3-Fluoro-4-(5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)oxyphenyl]-N-(4-fluorophenyl)propanediamide | IC50 | 780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_cd8853b99c351008c76e4c1c29a4d1cc.svg) | 2-(4-Fluorophenyl)-N-[[3-fluoro-4-[(3-pyridin-3-yl-1H-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]carbamoyl]acetamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_788f22c2c87790d1ecdd3374502555ed.svg) | 1-(4-(2-(Thiazol-2-yl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenyl)-3-(2-phenylacetyl)thiourea | IC50 | 28.0 [1], 65.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_2a303891fe450819ba7d463a5d0e526e.svg) | N-[[3-Fluoro-4-[2-(1-methylimidazol-2-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]carbamothioyl]-2-phenylacetamide | IC50 | 2.0 [1], 51.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_611d32bbba5ae97b3dce29adff5bb851.svg) | N-[4-[2-(1-Ethylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-2-oxo-3-phenylimidazolidine-1-carboxamide | IC50 | 25.0 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_509439e0101ceccb37543ff9b81734ba.svg) | N-[4-[2-(1-Ethylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-3-(2-fluorophenyl)-2-oxoimidazolidine-1-carboxamide | IC50 | 21.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_e811822b1f7f507b091ad4050d0318bb.svg) | N-[4-[2-(1-Ethylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-3-(2-methoxyphenyl)-2-oxoimidazolidine-1-carboxamide | IC50 | 26.0 [1], 60.0 [2] |
![](https://images.aatbio.com/dataset/ic50/hepatocyte-growth-factor-receptor_a95022143674b2ed06807d6d51834deb.svg) | N-[4-[2-[1-[2-(Dimethylamino)ethyl]imidazol-4-yl]thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-2-oxo-3-phenylimidazolidine-1-carboxamide | IC50 | 34.0 [1], 60.0 [2] |