Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1/gamma-2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	2-(4,5,6-Trihydroxy-3-oxo-3H-xanthen-9-yl)-cyclohexane-1-carboxylic acid	IC50	100.0 [1], 3000.0 [2], 8000.0 [3]
	1-Amino-4-[4-(4-amino-2-sulfophenyl)anilino]-9,10-dioxoanthracene-2-sulfonic acid	IC50	16000.0 [1], 18000.0 [2], 30000.0 [3], 62000.0 [4]
	1-Amino-4-(3-aminoanilino)-9,10-dioxoanthracene-2-sulfonic acid	IC50	6000.0 [1], 14000.0 [2], 15000.0 [3], 19000.0 [4]
	2-Anthracenesulfonic acid, 1-amino-4-[(4-aminophenyl)amino]-9,10-dihydro-9,10-dioxo-	IC50	2500.0 [1], 12000.0 [2], 75000.0 [3]
	1-Amino-9,10-dioxo-4-(3-sulfamoylphenylamino)-9,10-dihydroanthracene-2-sulfonic acid	IC50	10000.0 [1], 43000.0 [2], 58000.0 [3]
	30,34-Bis[(9,10-dioxoanthracen-1-yl)amino]nonacyclo[18.10.2.22,5.03,16.04,13.06,11.017,31.022,27.028,32]tetratriaconta-1(30),2(34),3(16),4(13),5(33),6,8,10,14,17(31),18,20(32),22,24,26,28-hexadecaene-12,21-dione	IC50	13500.0 [1], 16000.0 [2], 167000.0 [3]
	8-Iodo-N-(8-iodo-10-phenyl-5H-phenazin-2-yl)-10-phenylphenazin-10-ium-2-amine	IC50	2000.0 [1], 12000.0 [2]
	Fluorone black	IC50	300000.0 [1]
	Aminoquinuride	IC50	24000.0 [1]
	(E)-3-(3,4,5-Trihydroxy-6-oxoxanthen-9-yl)prop-2-enoic acid	IC50	200.0 [1]
	7-Methyl-3-(4,5,6-trihydroxy-3-oxo-3H-xanthen-9-yl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid	IC50	700.0 [1]
	8-(3,4,5-Trihydroxy-6-oxoxanthen-9-yl)naphthalene-1-carboxylic acid	IC50	130.0 [1]
	3-(3,4,5-Trihydroxy-6-oxoxanthen-9-yl)propanoic acid	IC50	2500.0 [1]
	6-Hydroxy-3-oxo-3H-xanthene-9-propionic acid	IC50	300000.0 [1]
	Benzoic acid, 3-(6-hydroxy-3-oxo-3H-xanthen-9-yl)-	IC50	300000.0 [1]
	2-(6-Hydroxy-3-oxo-3H-xanthen-9-yl)cyclohexanecarboxylic acid	IC50	300000.0 [1]
	3-(3-Hydroxy-6-oxoxanthen-9-yl)-7-methylbicyclo[2.2.1]hept-5-ene-2-carboxylic acid	IC50	14000.0 [1]
	6-Hydroxy-9-(2-hydroxyphenyl)xanthen-3-one	IC50	300000.0 [1]
	(E)-3-(3-Hydroxy-6-oxo-xanthen-9-yl)prop-2-enoic acid	IC50	300000.0 [1]
	1-(4-Amino-2-methylquinolin-6-yl)-3-(4-amino-2-methylquinolin-7-yl)urea	IC50	13000.0 [1]
	6-(3,4-Dihydroxy-6-oxoxanthen-9-yl)cyclohex-3-ene-1-carboxylic acid	IC50	700.0 [1]
	2-Bromo-1-(10-ethyl-5,6,7,8-tetrahydrophenanthren-2-yl)ethanone	IC50	100.0 [1]
	8-Iodo-N-(8-iodo-10-phenyl-5H-phenazin-2-yl)-10-phenyl-5H-phenazin-2-amine	IC50	2000.0 [1]
	1-Amino-4-{[4-(methylamino)phenyl]amino}-9,10-dioxo-9,10-dihydroanthracene-2-sulfonic acid	IC50	59000.0 [1]
	3-(4,5,6-Trihydroxy-3-oxo-3h-xanthen-9-yl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid	IC50	30000.0 [1]
	2-(4,5,6-Trihydroxy-3-oxo-3h-xanthen-9-yl)benzoic acid	IC50	200.0 [1]
	1,4,5,6,7,7-Hexachloro-3-(3,4,5-trihydroxy-6-oxoxanthen-9-yl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid	IC50	5000.0 [1]
	7,8,9,10,11,11-Hexachloro-4-(3,4,5-trihydroxy-6-oxoxanthen-9-yl)tricyclo[4.4.1.01,6]undecane-3-carboxylic acid	IC50	200.0 [1]
	(9Z)-9-(3,3-Dihydroxyprop-2-enylidene)-4,5,6-trihydroxy-9aH-xanthen-3-one	IC50	200.0 [1]
	N,4-Bis(4-amino-2-methylquinolin-6-yl)-2,2-dimethyl-3-oxobutanamide	IC50	74000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 30 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/guanine-nucleotide-binding-protein-g-i-g-s-g-t-subunit-beta-1-gamma-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 20). Quest Database™ Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/guanine-nucleotide-binding-protein-g-i-g-s-g-t-subunit-beta-1-gamma-2-inhibitors-ic50-ki.
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