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Growth factor receptor-bound protein 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-[[(2S)-1-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-1-oxo-3-[4-(phosphonomethyl)phenyl]propan-2-yl]amino]-2-oxoacetic acidIC5020.0 [1], 50.0 [2], 500.0 [3], 3000.0 [4]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5020.0 [1], 42.9 [2], 55.0 [3], 80.0 [4], 500.0 [5]
2-[(9S,10S,11E,14R,18S)-18-(2-Amino-2-oxoethyl)-14-[(5-methylindol-1-yl)methyl]-8,17,20-trioxo-10-[4-(phosphonomethyl)phenyl]-7,16,19-triazaspiro[5.14]icos-11-en-9-yl]acetic acidIC5010.0 [1], 15.0 [2], 630.0 [3], 10000.0 [4]
2-[4-[(2S)-3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-(oxaloamino)-3-oxopropyl]phenyl]propanedioic acidIC5022.1 [1], 70.0 [2]
2-[[(2S)-1-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-[4-(carboxymethyl)phenyl]-1-oxopropan-2-yl]amino]-2-oxoacetic acidIC50600.0 [1], 1000.0 [2]
3-[(5S,8S,11S,14S,17S,20S,26S,29S,32R)-17-(2-Amino-2-oxoethyl)-32-carbamoyl-14-(2-carboxyethyl)-11,29-bis[(4-hydroxyphenyl)methyl]-8-(2-methylpropyl)-26-(2-methylsulfanylethyl)-3,6,9,12,15,18,21,24,27,30-decaoxo-20-propan-2-yl-1-thia-4,7,10,13,16,19,22,25,28,31-decazacyclotritriacont-5-yl]propanoic acidIC5015000.0 [1], 20000.0 [2], 100000.0 [3], 100000000.0 [4]
[4-[(10R,11E,14S,18S)-18-(2-Amino-2-oxoethyl)-14-(naphthalen-1-ylmethyl)-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-10-yl]phenyl]methylphosphonic acidIC5020.0 [1], 26.0 [2], 10000.0 [3]
(3-Aminophenyl)methyl N-[(2S)-1-[[1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC501.0 [1], 120.0 [2]
2-[(9S,10S,11E,14S,18S)-18-(2-Amino-2-oxoethyl)-14-(naphthalen-1-ylmethyl)-8,17,20-trioxo-10-[4-(phosphonomethyl)phenyl]-7,16,19-triazaspiro[5.14]icos-11-en-9-yl]acetic acidIC502.0 [1], 12.1 [2], 1000.0 [3]
5-[(2S)-3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-(oxaloamino)-3-oxopropyl]-2-(carboxymethoxy)benzoic acidIC50500.0 [1], 1300.0 [2]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(5-methylindol-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC500.4 [1], 4.0 [2]
(3-Aminophenyl)methyl N-[(2S)-1-[[(2S,3S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC5065.0 [1]
2-[4-[(2S)-3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-(oxaloamino)-3-oxopropyl]phenyl]-2-fluoropropanedioic acidIC50170.0 [1]
2-[4-[(2S)-3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-(oxaloamino)-3-oxopropyl]phenoxy]propanedioic acidIC501100.0 [1]
[4-[(2S)-2-Acetamido-3-[[(2S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC504320.0 [1]
[4-[(2S)-2-Acetamido-3-[[2-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-2-oxoethyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC5067000.0 [1]
2-[[(2S)-1-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-[4-(carboxymethoxy)phenyl]-1-oxopropan-2-yl]amino]-2-oxoacetic acidIC5015000.0 [1], 19000.0 [2]
1,2,4-Oxadiazole Analogue 12dIC50500000.0 [1]
2-[4-[(2S)-3-[[1-[[(2S)-4-Amino-1-[3-(5-methylindol-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-(oxaloamino)-3-oxopropyl]phenyl]propanedioic acidIC508.0 [1]
(3R)-4-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-4-oxo-3-[[4-(phosphonomethyl)phenyl]methyl]butanoic acidIC508.0 [1], 10000.0 [2]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC5047.0 [1], 70.0 [2]
[[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]-difluoromethyl]phosphonic acidIC5080.0 [1], 500.0 [2]
Disodium;2-[4-[(9S,10S,11E,14S,18S)-18-(2-amino-2-oxoethyl)-9-(carboxymethyl)-14-(naphthalen-1-ylmethyl)-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-10-yl]phenyl]propanedioateIC504.3 [1], 12.1 [2]
[4-[(2S)-3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-azido-3-oxopropyl]phenyl]methylphosphonic acidIC505000.0 [1], 30000.0 [2]
2-[[10-Amino-11-(4-diacetyloxyphosphoryloxyphenyl)-7,9-dioxoundecyl]amino]-4-(3-naphthalen-1-ylpropylamino)-4-oxobutanoic acidIC5047.0 [1], 64.0 [2]
(2S)-2-[[(2S,3S)-2-[[(2S)-2-Amino-3-(4-diacetyloxyphosphoryloxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-(3-naphthalen-1-ylpropylamino)-4-oxobutanoic acidIC50330.0 [1], 580.0 [2]
[2-Amino-4-[(2S)-2-amino-3-[[1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC500.0 [1], 1.0 [2]
DactinomycinIC505000.0 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(2-hydroxynaphthalen-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5043.0 [1]
Actinomycin C3IC507600.0 [1]
8-O-MethylsclerotiorinamineIC505300.0 [1]
1,2,4-Oxadiazole Analogue 4aIC50456000.0 [1]
1,2,4-Oxadiazole Analogue 5dIC50500000.0 [1]
1,2,4-Oxadiazole Analogue 12bIC50500000.0 [1]
1,2,4-Oxadiazole Analogue 5fIC50500000.0 [1]
[4-[(2S)-2-Acetamido-3-[[(1S)-4-amino-1-[3-(carbamoylamino)phenyl]-4-oxobutyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC506500.0 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(8-hydroxynaphthalen-2-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5011.1 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(5-hydroxyindol-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC500.3 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(1R,2S)-2-carbamoylcyclohexyl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methyl-[hydroxy(phenyl)methyl]phosphinic acidIC50530.0 [1]
[4-[2-(4-Aminopyrimidin-2-yl)-5-methyl-1,3-thiazol-4-yl]phenyl] dihydrogen phosphateIC5025900.0 [1]
[4-[(2S)-2-Acetamido-3-[[(1S)-1-[3-(carbamoylamino)phenyl]-2-methylpropyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC506190.0 [1]
[4-[(10S,14R,18S)-18-(2-Amino-2-oxoethyl)-14-(naphthalen-1-ylmethyl)-8,12,17,20-tetraoxo-7,11,16,19-tetrazaspiro[5.14]icosan-10-yl]phenyl]methylphosphonic acidIC507900.0 [1]
(4S)-4-Amino-5-[[(2S)-1-[[(2S,3S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]amino]-5-oxopentanoic acidIC507900.0 [1]
(3-Aminophenyl)methyl N-[(2S)-1-[[(2S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC50497.0 [1]
(4S)-4-[(2-Aminobenzoyl)amino]-5-[[(2S)-1-[[(2S,3S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]amino]-5-oxopentanoic acidIC5022.0 [1]
[4-[(2S)-2-Amino-3-[[(2S,3S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC5056900.0 [1]
Benzyl N-[(2S)-1-[[(2S,3S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC506350.0 [1]
2-[4-[(2S)-2-[[(2S)-2-[(3-Aminophenyl)methoxycarbonylamino]-3-(4-phosphonooxyphenyl)propanoyl]amino]-3-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-2-methyl-3-oxopropyl]phenyl]acetic acidIC50198.0 [1]
(2S)-2-[[1-[[(2S)-2-Acetamido-3-(4-hydroxyphenyl)propanoyl]amino]cyclohexanecarbonyl]amino]-N-(3-naphthalen-1-ylpropyl)butanediamideIC5050000.0 [1]
[4-[(2S)-3-[[(2S)-1-[[(2S)-4-Amino-1-[[(2S)-1-[(2S)-2-(butylcarbamoyl)pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-oxo-2-(propanoylamino)propyl]phenyl] dihydrogen phosphateIC501630.0 [1]
4-[(2S)-2-[[(2S)-2-[(3-Aminophenyl)methoxycarbonylamino]-3-(4-phosphonooxyphenyl)propanoyl]amino]-3-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-2-methyl-3-oxopropyl]benzoic acidIC50153.0 [1]
(3-Aminophenyl)methyl N-[(2S)-1-[[(2S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC50235.0 [1]
(3-Aminophenyl)methyl N-[(2S)-1-[[(2S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-(4-hydroxyphenyl)-2-methyl-1-oxopropan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC501098.0 [1]
5-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]-2-(carboxymethoxy)benzoic acidIC506700.0 [1]
2-[4-[(2S)-2-[[(2S)-2-Acetamido-4-amino-4-oxobutanoyl]amino]-3-[[(2S)-1-[[(2S)-4-amino-1-[[(2S,3S)-1-[[(2S)-1-amino-4-carboxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-oxopropyl]phenoxy]propanedioic acidIC50120000.0 [1]
[4-[(2S)-2-Acetamido-3-[[(2S,3S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphateIC508640.0 [1]
2-[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]-2-(carboxymethoxy)phenoxy]acetic acidIC50100000.0 [1]
2-[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenoxy]propanedioic acidIC502750.0 [1]
[4-[3-[[1-[[(2S)-1,4-Diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5052500.0 [1]
[4-[(10S,12E,15S,19S)-19-(2-Amino-2-oxoethyl)-15-(naphthalen-1-ylmethyl)-8,18,21-trioxo-7,17,20-triazaspiro[5.15]henicos-12-en-10-yl]phenyl]methylphosphonic acidIC5010000.0 [1]
(3R)-4-[[1-[[(2S)-4-Amino-1-[2-[(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]ethylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-4-oxo-3-[[4-(phosphonomethyl)phenyl]methyl]butanoic acidIC50167.0 [1]
2-[(9S,10S,11E,14R,18S)-18-(2-Amino-2-oxoethyl)-10-[4-[[hydroxy(methyl)phosphoryl]methyl]phenyl]-14-[(5-methylindol-1-yl)methyl]-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-9-yl]acetic acidIC506.3 [1]
2-[4-[(9S,10S,11E,14R,18S)-18-(2-Amino-2-oxoethyl)-9-(carboxymethyl)-14-[(5-methylindol-1-yl)methyl]-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-10-yl]anilino]-2-oxoacetic acidIC508.8 [1]
2-[4-[(9S,10S,11E,14R,18S)-18-(2-Amino-2-oxoethyl)-9-(carboxymethyl)-14-[(5-methylindol-1-yl)methyl]-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-10-yl]phenyl]propanedioic acidIC503.3 [1]
2-[(9S,10S,11E,14R,18S)-18-(2-Amino-2-oxoethyl)-10-[4-[[benzyl(hydroxy)phosphoryl]methyl]phenyl]-14-[(5-methylindol-1-yl)methyl]-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-9-yl]acetic acidIC508.4 [1]
2-[(9S,10S,11E,14R,18S)-18-(2-Amino-2-oxoethyl)-10-[4-(carboxymethyl)phenyl]-14-[(5-methylindol-1-yl)methyl]-8,17,20-trioxo-7,16,19-triazaspiro[5.14]icos-11-en-9-yl]acetic acidIC5022.5 [1]
2-[[(9S,12S,15S,21R,30S)-9-[(3-Amino-4-hydroxyphenyl)methyl]-30-(2-amino-2-oxoethyl)-21-carbamoyl-12-(2-methylpropyl)-8,11,14,17,19,23,29,32-octaoxo-19lambda4-thia-7,10,13,16,22,28,31-heptazaspiro[5.26]dotriacontan-15-yl]methyl]propanedioic acidIC5058.0 [1]
4-[(9S,12S,15S,19S,21R,30S)-30-(2-Amino-2-oxoethyl)-21-carbamoyl-9-[(4-hydroxyphenyl)methyl]-12-(2-methylpropyl)-8,11,14,17,19,23,29,32-octaoxo-19lambda4-thia-7,10,13,16,22,28,31-heptazaspiro[5.26]dotriacontan-15-yl]butanoic acidIC5077000.0 [1]
2-[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]-2-fluoropropanedioic acidIC50680.0 [1]
(3-Aminophenyl)methyl N-[(2S)-1-[[(2R)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-1-oxo-2-(4-phosphonooxyphenyl)propan-2-yl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC5013.0 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(1R,2S)-2-carbamoylcyclohexyl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methyl-(hydroxymethyl)phosphinic acidIC507600.0 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(1R,2S)-2-carbamoylcyclohexyl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methyl-(2-hydroxyethyl)phosphinic acidIC501600.0 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(1R,2S)-2-carbamoylcyclohexyl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methyl-benzylphosphinic acidIC501200.0 [1]
[4-[3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-1-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC502000.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-(4-Carbamimidoylcyclohexyl)-2-[[(2S)-1-[(2S)-2-[[6-(carbamothioylamino)-3',6'-dihydroxyspiro[1H-2-benzofuran-3,9'-xanthene]-1-carbonyl]amino]-2-piperidin-4-ylacetyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3,3-dimethylbutanoyl]amino]-4-methylpentanoic acidIC50700.0 [1]
Phosphoric acid 4-[2-(4-amino-2-pyrimidinylamino)ethyl]phenyl esterIC50200000.0 [1]
1-[3-[4-(3-Aminophenyl)butyl]phenyl]-6,6-dimethyl-1,3,5-triazine-2,4-diamine;hydrochlorideIC505700000.0 [1]
4-[(5S,8S,11S,14S,17S,26R)-17-(2-Amino-2-oxoethyl)-26-carbamoyl-14-(3-carboxypropyl)-11-[(4-hydroxyphenyl)methyl]-14-methyl-8-(2-methylpropyl)-3,6,9,12,15,18,24-heptaoxo-1-thia-4,7,10,13,16,19,25-heptazacycloheptacos-5-yl]butanoic acidIC5060700.0 [1]
4-[(5S,8S,11S,14R,17S,26R)-17-(2-Amino-2-oxoethyl)-26-carbamoyl-14-(2-carboxyethyl)-11-[(4-hydroxyphenyl)methyl]-14-methyl-8-(2-methylpropyl)-3,6,9,12,15,18,24-heptaoxo-1-thia-4,7,10,13,16,19,25-heptazacycloheptacos-5-yl]butanoic acidIC5060500.0 [1]
4-[(5S,8S,11S,14S,17S,26R)-11-[(3-Amino-4-hydroxyphenyl)methyl]-17-(2-amino-2-oxoethyl)-26-carbamoyl-14-(2-carboxyethyl)-14-methyl-8-(2-methylpropyl)-3,6,9,12,15,18,24-heptaoxo-1-thia-4,7,10,13,16,19,25-heptazacycloheptacos-5-yl]butanoic acidIC5017000.0 [1]
4-[(5S,8S,11S,14S,17S,26R)-17-(2-Amino-2-oxoethyl)-26-carbamoyl-14-(2-carboxyethyl)-11-[(4-hydroxyphenyl)methyl]-14-methyl-8-(2-methylpropyl)-3,6,9,12,15,18,24-heptaoxo-1-thia-4,7,10,13,16,19,25-heptazacycloheptacos-5-yl]butanoic acidIC5070000.0 [1]
2-[[(5S,8S,11S,14S,17S,26R)-11-[(3-Amino-4-hydroxyphenyl)methyl]-17-(2-amino-2-oxoethyl)-26-carbamoyl-14-(3-carboxypropyl)-14-methyl-8-(2-methylpropyl)-3,6,9,12,15,18,24-heptaoxo-1-thia-4,7,10,13,16,19,25-heptazacycloheptacos-5-yl]methyl]propanedioic acidIC509500.0 [1]
(4S)-4-[[(2S)-3-[3-(2-Carboxyethyl)-4-hydroxyphenyl]-2-[[(2S)-2-[[(2S)-5-carboxy-2-(9H-fluoren-9-ylmethoxycarbonylamino)pentanoyl]amino]-4-methylpentanoyl]amino]propanoyl]amino]-5-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-4-methyl-5-oxopentanoic acidIC505600.0 [1]
(4S)-4-[[(2S)-3-[3-(2-Carboxyethyl)-4-hydroxyphenyl]-2-(9H-fluoren-9-ylmethoxycarbonylamino)propanoyl]amino]-5-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-4-methyl-5-oxopentanoic acidIC50168000.0 [1]
(5S)-6-[[(2S)-1-[[(2S)-3-(3-Amino-4-hydroxyphenyl)-1-[[1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(9H-fluoren-9-ylmethoxycarbonylamino)-6-oxohexanoic acidIC505800.0 [1]
2-[(2S)-2-Amino-3-[[(2S)-1-[[(2S)-3-(3-amino-4-hydroxyphenyl)-1-[[(2S)-4-carboxy-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-2-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]propanedioic acidIC5019000.0 [1]
(5R)-6-[[(2S)-1-[[(2S)-1-[[1-[[(2S)-1,4-Diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(9H-fluoren-9-ylmethoxycarbonylamino)-5-methyl-6-oxohexanoic acidIC501000000.0 [1]
(5R)-6-[[(2S)-1-[[(2S)-3-(3-Amino-4-hydroxyphenyl)-1-[[1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(9H-fluoren-9-ylmethoxycarbonylamino)-5-methyl-6-oxohexanoic acidIC50700000.0 [1]
2-[(2S)-3-[[(2S)-1-[[(2S)-3-(3-Amino-4-hydroxyphenyl)-1-[[(2S)-4-carboxy-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-2-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-(9H-fluoren-9-ylmethoxycarbonylamino)-3-oxopropyl]propanedioic acidIC504400.0 [1]
2-[(2S)-3-[[(2S)-1-[[(2S)-3-(3-Amino-4-hydroxyphenyl)-1-[[1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-(9H-fluoren-9-ylmethoxycarbonylamino)-3-oxopropyl]propanedioic acidIC502500.0 [1]
(5S)-6-[[(2S)-1-[[(2S)-3-(3-Amino-4-hydroxyphenyl)-1-[[1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(9H-fluoren-9-ylmethoxycarbonylamino)-5-methyl-6-oxohexanoic acidIC503900.0 [1]
(5S)-6-[[(2S)-1-[[(2S)-1-[[1-[[(2S)-1,4-Diamino-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-(9H-fluoren-9-ylmethoxycarbonylamino)-5-methyl-6-oxohexanoic acidIC50117700.0 [1]
4-[(5S,8S,11S,14S,17S,26R)-17-(2-Amino-2-oxoethyl)-26-carbamoyl-14-(carboxymethyl)-11-[(4-hydroxyphenyl)methyl]-14-methyl-8-(2-methylpropyl)-3,6,9,12,15,18,24-heptaoxo-1-thia-4,7,10,13,16,19,25-heptazacycloheptacos-5-yl]butanoic acidIC50108000.0 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(6,7-dimethoxynaphthalen-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5084.4 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(6-methoxynaphthalen-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC50129.9 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(6-hydroxynaphthalen-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5042.7 [1]
[4-[(2S)-2-Acetamido-3-[[1-[[(2S)-4-amino-1-[3-(7-hydroxynaphthalen-1-yl)propylamino]-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-3-oxopropyl]phenyl]methylphosphonic acidIC5024.6 [1]
2-[4-[(2S)-3-[[1-[[(2S)-4-Amino-1-(3-naphthalen-2-ylpropylamino)-1,4-dioxobutan-2-yl]carbamoyl]cyclohexyl]amino]-2-(oxaloamino)-3-oxopropyl]phenyl]propanedioic acidIC5050.0 [1]
(3-Aminophenyl)methyl N-[(2S)-1-[[1-[[(6S)-6-carbamoylcyclohex-2-en-1-yl]carbamoyl]cyclohexyl]amino]-1-oxo-3-(4-phosphonooxyphenyl)propan-2-yl]carbamateIC501.6 [1]
2-[[(5S,8R,11S,14R,17S,20R,26R,29S,32R)-17-(2-Amino-2-oxoethyl)-32-carbamoyl-14-(3-carboxypropyl)-11,29-bis[(4-hydroxyphenyl)methyl]-8-(2-methylpropyl)-26-(2-methylsulfanylethyl)-3,6,9,12,15,18,21,24,27,30-decaoxo-20-propan-2-yl-1-thia-4,7,10,13,16,19,22,25,28,31-decazacyclotritriacont-5-yl]methyl]propanedioic acidIC501510.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Growth factor receptor-bound protein 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/growth-factor-receptor-bound-protein-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Growth factor receptor-bound protein 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/growth-factor-receptor-bound-protein-2-inhibitors-ic50-ki.
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