![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_7ace065e00b56633701011ddaac397d8.svg) | (1R,3R,6R,7S,8S,9S,11S,12S,13S,16S,17S)-8-Tert-butyl-6,9,12,17-tetrahydroxy-13-methyl-2,4,15,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.012,16]nonadecane-5,14,18-trione | IC50 | 1700.0 [1], 2400.0 [2], 2511.89 [3], 5011.87 [4], 5900.0 [5] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_db73eda68e8c605bf06d779827ec4e13.svg) | Strychnine | IC50 | 51.0 [1], 93.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_db73eda68e8c605bf06d779827ec4e13.svg) | Strychnine | Ki | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_bfa92afabe22373d293e574beb10dd93.svg) | Ginkgolide-B | IC50 | 1700.0 [1], 1995.26 [2], 3162.28 [3] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_7fde918ee0ca858da3cc942a4b123d8a.svg) | Ginkgolide A | IC50 | 630.96 [1], 1995.26 [2], 3800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_991f8bf2dced6087558dde1cd2619ca0.svg) | Ginkgolide M | IC50 | 501.19 [1], 650.0 [2], 794.33 [3] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_0f5cd07e2b17ea29d8b3cbe20c56e54a.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-propoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 109.0 [1], 110.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_0f5cd07e2b17ea29d8b3cbe20c56e54a.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-propoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | Ki | 241.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_8505e3cd29263b2d445518ddcbe8d9a8.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-prop-2-enoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 49.0 [1], 95.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_8505e3cd29263b2d445518ddcbe8d9a8.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-prop-2-enoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | Ki | 370.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_35dd254a0e48b7e3d03a671c576fddbb.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-methoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 75.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_35dd254a0e48b7e3d03a671c576fddbb.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-methoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | Ki | 189.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_f5b2a0e58614baf403ab132db806a5ff.svg) | Strychnine, 2-propionamido- | IC50 | 201.0 [1], 540.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_f5b2a0e58614baf403ab132db806a5ff.svg) | Strychnine, 2-propionamido- | Ki | 67.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_bb045330d73cb5a93223075190112571.svg) | (1S,3R,6R,7S,8S,9S,11S,12S,13S,16S)-8-Tert-butyl-6,9,12-trihydroxy-13-methyl-2,4,15,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.012,16]nonadecane-5,14,18-trione | IC50 | 3981.07 [1], 6400.0 [2], 7943.28 [3] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_c20897cfd4dbb225127b86869d37fea5.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-hydroxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 82.0 [1], 97.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_c20897cfd4dbb225127b86869d37fea5.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-hydroxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | Ki | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_43e5d4e643c28e71b28b5c5ba84420b0.svg) | (4Ar,5aS,8aS,13aS,15aS,15bR)-6-propyl-4a,5,5a,7,8,13a,15,15a,15b,16-decahydro-2H-4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-6-ium-14-one;bromide | IC50 | 4590.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_284bd02637e8ba4b95e69f32ca9d0887.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-prop-2-ynoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 52.0 [1], 59.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_6436358c772c335c71530d93cf2513bf.svg) | (1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-Tert-butyl-9-chloro-6,12,17-trihydroxy-16-methyl-2,4,14,18-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,19-trione | IC50 | 3162.28 [1], 7943.28 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_7e62d0a08eee5cd69cc1397ffd917913.svg) | (1R,3R,6R,7S,8S,9S,10S,11R,12R,13S,16S,17R)-9-Azido-8-tert-butyl-6,12,17-trihydroxy-16-methyl-2,4,14,18-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,19-trione | IC50 | 7943.28 [1], 15848.93 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_cddf23420671c4a0cc1f13c910c3c473.svg) | (6R,8S,11S,16R,17S)-8-Tert-butyl-6,16,17-trihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_64200ede9ce59228c492ee8be424e848.svg) | (1S,8S,11S,13S,16S,17R)-8-Tert-butyl-17-hydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,6,15,18-tetrone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_b915c0b906975d11f4395dc759837c13.svg) | 10-Acetoxy-ginkgolide B | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e58a0080f3c56abcf896ae38de2777ff.svg) | [(1R,6R,8S,11S,13S,16R,17S)-8-Tert-butyl-16-methyl-5,15,18-trioxo-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecan-6-yl] acetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e69e5115c9517a470650fafa8888761b.svg) | 10-Methoxymethyloxy-ginkgolide A | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_b4c5a0a2673de519b705c27bd44b3fb5.svg) | (1S,6R,8S,9R,11S)-8-Tert-butyl-6,9-dihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadeca-12,16-diene-5,15,18-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_268e62f429ff3640b3397ad043866bd9.svg) | Methyl (2R)-2-[(1S,2R,3S,6S,8S,10S)-10-tert-butyl-2-hydroxy-16-methoxy-3-methyl-4,14-dioxo-5,13,15-trioxapentacyclo[7.5.2.01,8.02,6.08,12]hexadecan-9-yl]-2-methoxyacetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_152525d15cb3175fcca45682527c587e.svg) | (1R,2R,3S,6S,8S,10R,11R)-10-Tert-butyl-2,11,16-trihydroxy-3-methyl-5,13,15-trioxapentacyclo[7.5.2.01,8.02,6.08,12]hexadecane-4,14-dione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_f2b58ebf4c06005424b60e9a2e576e72.svg) | (1S,2R,3S,6S,8S,10R)-10-Tert-butyl-2-hydroxy-3-methyl-5,13,15-trioxapentacyclo[7.5.2.01,8.02,6.08,12]hexadecane-4,14,16-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_4fa53b55fe6f57d3c41c99791b4101c1.svg) | [(1R,6R,8S,11R)-8-Tert-butyl-13-methoxy-5,15,16-trioxo-2,4,14,17-tetraoxapentacyclo[8.5.2.01,11.03,7.07,11]heptadecan-6-yl] acetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_22c7f53412269d1c4f97e219238c6aac.svg) | (1R,6R,8S,11S)-8-Tert-butyl-6,13-dimethoxy-2,4,14,17-tetraoxapentacyclo[8.5.2.01,11.03,7.07,11]heptadecane-5,15,16-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_5b53c7426ad41b7fa290c04f638b09e6.svg) | Methyl (2E)-2-[(1R,6R,8S,11S)-8-tert-butyl-6-hydroxy-5,15-dioxo-2,4,16-trioxapentacyclo[8.4.2.01,11.03,7.07,11]hexadecan-14-ylidene]propanoate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_d5d2a994e8b88983f28d84ec47c61f70.svg) | Methyl 2-[(1R,6R,8S,11S,14R)-8-tert-butyl-6-hydroxy-5,15-dioxo-2,4,16-trioxapentacyclo[8.4.2.01,11.03,7.07,11]hexadecan-14-yl]propanoate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_a5991b4d85f95c9356fa4b3859ddea6b.svg) | (1S,6R,8S,11S,13R,16R,17R)-8-Tert-butyl-6,17-dihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,18-dione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_3da738e29025e25bae911d77d19be689.svg) | (1S,6R,8S,11S,13S,16R,17R)-8-Tert-butyl-6,17-dihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecan-18-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e5b45c1df4c99499a96b181111c415eb.svg) | (1R,6R,8S,11S,13S,16R,17R)-8-Tert-butyl-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-6,17-diol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_8175a2eb06f02ea2f2f660bc7efbd6cc.svg) | (1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-Tert-butyl-6,12,17-trihydroxy-16-methyl-9-(methylamino)-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_3351c946fe7ceeea8a826e7e90a1e346.svg) | (1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-Tert-butyl-9-(ethylamino)-6,12,17-trihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_436e4fadc03bbbe3ff786e7e35f5e1da.svg) | [(1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-Tert-butyl-6,12,17-trihydroxy-16-methyl-5,15,18-trioxo-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecan-9-yl] 2-phenylacetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_0087e92321e8086449dfd259d956bee7.svg) | (1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-Tert-butyl-6,9,12,17-tetrahydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_5260a85faf99f706cc3f1e417b8deee1.svg) | [(1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-Tert-butyl-6,12,17-trihydroxy-16-methyl-5,15,18-trioxo-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecan-9-yl] acetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_272869fa4f0efe9aa72b38e7617a9870.svg) | (1S,6R,8S,11R,12R,13S,16S,17R)-8-Tert-butyl-6,12,17-trihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,9,15,18-tetrone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_9a8d77b10f78787243cd54e1576defed.svg) | [(1S,6R,8S,9R,11S,12R,13S,16S,17R)-8-Tert-butyl-6,12,17-trihydroxy-16-methyl-5,15,18-trioxo-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecan-9-yl] trifluoromethanesulfonate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_58ac21ed0baaa5f9c83d1d0512adcdb0.svg) | (3S,8R,12R,16S,17R,21S)-3-Tert-butyl-17-hydroxy-16-methyl-6,9,11,14,20,22-hexaoxaheptacyclo[10.8.1.15,18.04,8.04,21.013,17.018,21]docosane-7,15,19-trione | IC50 | 7943.28 [1], 12589.25 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_08e811e8dceecd92694fa205c1c6be57.svg) | 3,14-Didehydroginkgolide A | IC50 | 3162.28 [1], 6309.57 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e9d560f17a996444fc025afcd892d16e.svg) | 10-Methoxy-ginkgolide C | IC50 | 5011.87 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_2549bd97dcdc42b86b8c41cdcbb8e4e9.svg) | (1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-Tert-butyl-9-fluoro-6,12,17-trihydroxy-16-methyl-2,4,14,18-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,19-trione | IC50 | 3162.28 [1], 7943.28 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_106778d948900a936e8c84395fce6848.svg) | 2-Aminostrychnine | IC50 | 76.0 [1], 77.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_804b8f0d63e25d5aef7540aa573a24f3.svg) | Alcuronium | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_279cd9f3d71067192157e557364f96b4.svg) | Trimethyl-[[20-[(trimethylazaniumyl)methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl]azanium;diiodide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_05057bee5ac208928570dc1c1a9c1278.svg) | 5-Hydroxy-4-[(Z)-indol-3-ylidenemethyl]-3-methyl-1H-imidazol-2-one | IC50 | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e6e95de1349eafed7021889f0bd60f49.svg) | 5-[(1H-Indol-3-yl)methylidene]-1,3-dimethylimidazolidine-2,4-dione | IC50 | 200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_591f03e288d5c25c4c37deb1ec6a4010.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-(2-phenylethoxyimino)-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_2d874e8b42c3b99b1c6349e5a656da9b.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-(2-methylpropoxyimino)-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_1581287077a1d478b0199c96926bec6e.svg) | Methyl 5-[(E)-[(4aR,5aS,8aR,13aS,15aR,15bR)-14-oxo-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-15-ylidene]amino]oxypentanoate | IC50 | 720.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_ab514f4e1c3f79d12c517bf2371312d0.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-phenylmethoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_c2548254104babd4a7b9c5ec5a4618a8.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-pentoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_c49458bab6906d913241d64c27c7bd85.svg) | Methyl 2-[(E)-[(4aR,5aS,8aR,13aS,15aR,15bR)-14-oxo-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-15-ylidene]amino]oxyacetate | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_97e7b517e6adc42c322326b37bf16072.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-butoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 370.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_4c3dc1e81a9b3c0d77c04471331329a9.svg) | CID 145948364 | IC50 | 25900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_f6bcb23a4a93c7adfa01cb345ef50622.svg) | (1R,9R,18S,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-10,26-dioxa-8,15,24,31-tetrazaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e324179bfc273aa69989ec5fda2c810b.svg) | (2E)-2-[(1R,9Z,11S,13S,17S,18R,20R,27S,29R,30R,31S)-19-Phenyl-21-oxa-8,14,19,26-tetrazadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e673745608671528c2ca9bc2db706f97.svg) | (4Ar,5aS,8aR,13aS,15aS,15bR)-2,4a,5,5a,8,13a,15,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinoline-7,14-dione | IC50 | 6900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_511b3b7e244ef3f68521a3cbc9ac96ba.svg) | [20-[[Dimethyl-[(4-nitrophenyl)methyl]azaniumyl]methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl-dimethyl-[(4-nitrophenyl)methyl]azanium | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_3ead7fb679101aaf33d6e2a54ccc7d72.svg) | [20-[[Dimethyl(prop-2-enyl)azaniumyl]methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl-dimethyl-prop-2-enylazanium | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_79e71b2be09a917594a3bb0d2fefa638.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Dimethyl-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_d185a33820dee9bc6bb606934b382a4b.svg) | (1R,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-15-prop-2-enyl-10,26-dioxa-8,24,31-triaza-15-azoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_fc760627b8b7f6e6b69d2cfbba879ad7.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-15,31-bis(prop-2-enyl)-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_45e84370034d041781d795e0c6fad817.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(E)-but-2-enyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_b497587a5df2afce9b1c595689fb4905.svg) | 2-[(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-31-(2-Acetyloxyethyl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaen-15-yl]ethyl acetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_ba84f513713bbc009d8b861611798728.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Di(cyclohex-2-en-1-yl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_bb2363dae4b783e026690b1856b45afc.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Dibenzyl-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_42032f9797e51bda0be07b15022bb6f6.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(3,4-dimethoxyphenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_bb025f4bb375ccf3ddd31af7edf3a119.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(4-bromophenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_41a881d57c901f61e2dd774f395b900f.svg) | (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(4-nitrophenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_c37b36a62657ac35e260b8c1f89d80e7.svg) | (2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Dimethyl-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_68ea088121db41e0938a00248b939461.svg) | (2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Di(cyclohex-2-en-1-yl)-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_e06b6ed9efe6ebf85878c95166429e25.svg) | (2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Bis[(3,4-dimethoxyphenyl)methyl]-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_7bbfcd3f651109bbf0e030aebc660936.svg) | (2E)-2-[(1S,9Z,11S,13S,18R,20R,27S,29R,30R,31S)-14,26-Bis[(4-nitrophenyl)methyl]-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-subunit-alpha-1_7d238473806ba5b2db9ea4bde1ea66bc.svg) | (2E)-2-[(1S,9Z,11S,13S,25Z,27S,33S,35S,36S,38E)-38-(2-Hydroxyethylidene)-14,30-dimethyl-8,24-diaza-14,30-diazoniaundecacyclo[25.5.2.211,14.11,26.110,17.02,7.013,17.018,23.030,33.08,35.024,36]octatriaconta-2,4,6,9,18,20,22,25-octaen-28-ylidene]ethanol | IC50 | 100000.0 [1] |