![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_db73eda68e8c605bf06d779827ec4e13.svg) | Strychnine | IC50 | 58.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_0f5cd07e2b17ea29d8b3cbe20c56e54a.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-propoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 116.0 [1], 354.81 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_43e5d4e643c28e71b28b5c5ba84420b0.svg) | (4Ar,5aS,8aS,13aS,15aS,15bR)-6-propyl-4a,5,5a,7,8,13a,15,15a,15b,16-decahydro-2H-4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-6-ium-14-one;bromide | IC50 | 6530.0 [1], 13489.63 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_8505e3cd29263b2d445518ddcbe8d9a8.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-prop-2-enoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 46.0 [1], 158.49 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_35dd254a0e48b7e3d03a671c576fddbb.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-methoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 56.0 [1], 213.8 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_284bd02637e8ba4b95e69f32ca9d0887.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-prop-2-ynoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 43.0 [1], 239.88 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_f5b2a0e58614baf403ab132db806a5ff.svg) | Strychnine, 2-propionamido- | IC50 | 311.0 [1], 940.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_106778d948900a936e8c84395fce6848.svg) | 2-Aminostrychnine | IC50 | 97.0 [1], 270.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_c20897cfd4dbb225127b86869d37fea5.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-hydroxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 80.0 [1], 210.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_ee06d3ae246907e6fa353ed24314c407.svg) | Gelsemine | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_591f03e288d5c25c4c37deb1ec6a4010.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-(2-phenylethoxyimino)-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 776.25 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_2d874e8b42c3b99b1c6349e5a656da9b.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-(2-methylpropoxyimino)-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 1122.02 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_1581287077a1d478b0199c96926bec6e.svg) | Methyl 5-[(E)-[(4aR,5aS,8aR,13aS,15aR,15bR)-14-oxo-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-15-ylidene]amino]oxypentanoate | IC50 | 1479.11 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_ab514f4e1c3f79d12c517bf2371312d0.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-phenylmethoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 309.03 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_c2548254104babd4a7b9c5ec5a4618a8.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-pentoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 707.95 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_c49458bab6906d913241d64c27c7bd85.svg) | Methyl 2-[(E)-[(4aR,5aS,8aR,13aS,15aR,15bR)-14-oxo-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-15-ylidene]amino]oxyacetate | IC50 | 660.69 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_97e7b517e6adc42c322326b37bf16072.svg) | (4Ar,5aS,8aR,13aS,15E,15aR,15bR)-15-butoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one | IC50 | 870.96 [1] |
![](https://images.aatbio.com/dataset/ic50/glycine-receptor-alpha-1-beta_e673745608671528c2ca9bc2db706f97.svg) | (4Ar,5aS,8aR,13aS,15aS,15bR)-2,4a,5,5a,8,13a,15,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinoline-7,14-dione | IC50 | 10000.0 [1] |