Glutathione S-transferase A2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	2-[2-(4-Amino-4-carboxybutyrylamino)-3-oxo-3-(carboxymethylamino)propylthio]succinic acid	IC50	19100.0 [1]
	(4S)-4-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]amino]-2-methylpropanoyl]amino]-3-[4-(phosphonomethyl)phenyl]propanoyl]amino]-3-(6-chloro-1H-indol-3-yl)propanoyl]amino]-5-[[1-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]cyclopropyl]amino]-5-oxopentanoic acid	IC50	5.0 [1]
	[(3S,4S,5R)-3,4,5-Trihydroxy-6-oxocyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	[(4R,5S,6R)-4,5,6-Trihydroxy-3-oxocyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-3-(1,4-dimethoxy-1,4-dioxobutan-2-yl)sulfanyl-1-oxopropan-2-yl]amino]-5-oxopentanoic acid	IC50	250000.0 [1]
	[(3S,4R,5R)-4,5-Dihydroxy-3-methoxy-6-oxocyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-1-oxo-3-(4-oxohexan-2-ylsulfanyl)propan-2-yl]amino]-5-oxopentanoic acid	IC50	90000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-1-oxo-3-(3-oxocyclohexyl)sulfanylpropan-2-yl]amino]-5-oxopentanoic acid	IC50	220000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-1-oxo-3-(5-oxohexan-3-ylsulfanyl)propan-2-yl]amino]-5-oxopentanoic acid	IC50	4100.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-3-(2-methyl-5-oxohexan-3-yl)sulfanyl-1-oxopropan-2-yl]amino]-5-oxopentanoic acid	IC50	66000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-1-oxo-3-(3-oxo-1-phenylbutyl)sulfanylpropan-2-yl]amino]-5-oxopentanoic acid	IC50	41000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-1-oxo-3-(2-oxoheptan-4-ylsulfanyl)propan-2-yl]amino]-5-oxopentanoic acid	IC50	8400.0 [1]
	2-Amino-5-[[3-(3-butoxy-1-carboxy-3-oxopropyl)sulfanyl-1-(carboxymethylamino)-1-oxopropan-2-yl]amino]-5-oxopentanoic acid	IC50	48000.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-3-(1,4-dioxo-1,4-dipropoxybutan-2-yl)sulfanyl-1-oxopropan-2-yl]amino]-5-oxopentanoic acid	IC50	143300.0 [1]
	2-Amino-5-[[1-(carboxymethylamino)-3-(4-methyl-3-oxo-1-phenylpentyl)sulfanyl-1-oxopropan-2-yl]amino]-5-oxopentanoic acid	IC50	31900.0 [1]
	(6Ar,8R,9R,10aS,10bR)-8,9-dimethoxy-2,2,8,9-tetramethyl-4,6a,10a,10b-tetrahydro-[1,4]dioxino[2,3-h][1,3]benzodioxin-6-one	IC50	100000.0 [1]
	[(3S,4R,5R)-3-Decoxy-4,5-dihydroxy-6-oxocyclohexen-1-yl]methyl acetate	IC50	37800.0 [1]
	[(3R,4S,5R)-3,4,5-Trihydroxy-6-oxocyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	(2R,3R,4Ar,8R,8aS)-8-hydroxy-7-(hydroxymethyl)-2,3-dimethoxy-2,3-dimethyl-8,8a-dihydro-4aH-1,4-benzodioxin-5-one	IC50	100000.0 [1]
	[(2R,3R,4Ar,8R,8aS)-8-hydroxy-2,3-dimethoxy-2,3-dimethyl-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-7-yl]methyl acetate	IC50	100000.0 [1]
	[(3R,4R,5R)-4,5-Dihydroxy-3-methoxy-6-oxocyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	[(3R,4R,5R)-4,5-Dihydroxy-6-oxo-3-phenylmethoxycyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	[(2R,3R,4Ar,8R,8aS)-8-hydroxy-2,3-dimethoxy-2,3-dimethyl-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	100000.0 [1]
	[(2R,3R,4Ar,8R,8aS)-2,3,8-trimethoxy-2,3-dimethyl-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	100000.0 [1]
	[(3S,4R,5R)-4,5-Dihydroxy-6-oxo-3-phenylmethoxycyclohexen-1-yl]methyl acetate	IC50	100000.0 [1]
	[(2R,3R,4Ar,8S,8aS)-2,3-dimethoxy-2,3-dimethyl-5-oxo-8-phenylmethoxy-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	100000.0 [1]
	[(2R,3R,4Ar,8S,8aS)-2,3-dimethoxy-2,3-dimethyl-8-(naphthalen-2-ylmethoxy)-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	77600.0 [1]
	[(2R,3R,4Ar,8S,8aS)-2,3-dimethoxy-2,3-dimethyl-8-(3-methylbut-2-enoxy)-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	96300.0 [1]
	[(2R,3R,4Ar,8S,8aS)-8-hexoxy-2,3-dimethoxy-2,3-dimethyl-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	93000.0 [1]
	[(2R,3R,4Ar,8S,8aS)-8-[(2E)-3,7-dimethylocta-2,6-dienoxy]-2,3-dimethoxy-2,3-dimethyl-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	178600.0 [1]
	[(2R,3R,4Ar,8S,8aS)-2,3-dimethoxy-2,3-dimethyl-5-oxo-8-[(E)-3-phenylprop-2-enoxy]-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	94200.0 [1]
	[(2R,3R,4Ar,8S,8aS)-2,3-dimethoxy-2,3-dimethyl-5-oxo-8-[(4-phenylphenyl)methoxy]-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	66300.0 [1]
	[(2R,3R,4Ar,8S,8aS)-8-decoxy-2,3-dimethoxy-2,3-dimethyl-5-oxo-8,8a-dihydro-4aH-1,4-benzodioxin-6-yl]methyl acetate	IC50	33100.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 33 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Glutathione S-transferase A2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/glutathione-s-transferase-a2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Glutathione S-transferase A2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutathione-s-transferase-a2-inhibitors-ic50-ki.
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