Glutamate receptor ionotropic kainate 3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Glutamic acid	Ki	789.0 [1]
	Kainic acid	Ki	10.0 [1]
	(2S,4R)-2-Amino-4-[(E)-3-naphthalen-2-ylprop-2-enyl]pentanedioic acid	Ki	617.0 [1]
	2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline	Ki	18000.0 [1]
	Tezampanel	Ki	100000.0 [1]
	(S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxybenzyl)pyrimidine-2,4-dione	IC50	4000.0 [1]
	2-[[3-(2-Amino-2-carboxyethyl)-2,6-dioxo-1-pyrimidinyl]methyl]benzoic acid	Ki	374000.0 [1]
	(3S,4Ar,6S,8aR)-6-[[(2S)-2-carboxy-4,4-difluoropyrrolidin-1-yl]methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid	Ki	8900.0 [1]
	(S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxythiophene-3-ylmethyl)pyrimidine-2,4-dione	Ki	111000.0 [1]
	(2R,3S)-1-(9-Iodophenanthrene-3-carbonyl)piperazine-2,3-dicarboxylic acid	IC50	81300.0 [1]
	(2S)-2-Amino-4-cyclopentylidenepentanedioic acid	Ki	5730.0 [1]
	CID 10330442	Ki	518.0 [1]
	(2S)-2-Amino-4-pentan-3-ylidenepentanedioic acid	Ki	12400.0 [1]
	2-[7-[3-[[(4-Nitrophenyl)carbamoylamino]methyl]pyrrol-1-yl]-2,3-dioxo-6-(trifluoromethyl)-4H-quinoxalin-1-yl]acetic acid	Ki	46.0 [1]
	(2S,4R)-2-Amino-4-[(E)-3-(2-methoxyphenyl)prop-2-enyl]pentanedioic acid	Ki	42.0 [1]
	(2S,4Z)-2-Amino-4-(2-methylpropylidene)pentanedioic Acid	Ki	10500.0 [1]
	2-[6-Nitro-2,3-dioxo-7-[3-(piperidin-1-ylmethyl)pyrrol-1-yl]-4H-quinoxalin-1-yl]acetic acid	Ki	5700.0 [1]
	2-[6-Nitro-2,3-dioxo-7-[3-[(4-phenylpiperidin-1-yl)methyl]pyrrol-1-yl]-4H-quinoxalin-1-yl]acetic acid	Ki	530.0 [1]
	2,3-Dioxo-6-nitro-7-(3-carboxy-1H-pyrrole-1-yl)-1,2,3,4-tetrahydroquinoxaline-1-acetic acid	Ki	4100.0 [1]
	2-[6-Nitro-2,3-dioxo-7-[3-[(3-phenylpropylamino)methyl]pyrrol-1-yl]-4H-quinoxalin-1-yl]acetic acid	Ki	1400.0 [1]
	3-(6-Nitro-2,3-dioxo-7-pyrrol-1-yl-4H-quinoxalin-1-yl)propanoic acid	Ki	2500.0 [1]
	2-[6-Nitro-2,3-dioxo-7-[3-[[4-(2-phenylethyl)piperazin-1-yl]methyl]pyrrol-1-yl]-4H-quinoxalin-1-yl]acetic acid	Ki	1400.0 [1]
	(2S,4R)-2-Amino-4-[(E)-3-(4-chlorophenyl)prop-2-enyl]pentanedioic acid	Ki	423.0 [1]
	2-[7-[3-[(4-Benzylpiperazin-1-yl)methyl]pyrrol-1-yl]-6-nitro-2,3-dioxo-4H-quinoxalin-1-yl]acetic acid	Ki	680.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ Glutamate receptor ionotropic kainate 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-kainate-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Glutamate receptor ionotropic kainate 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-kainate-3-inhibitors-ic50-ki.
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