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Glutamate receptor ionotropic kainate 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
▲
▼
2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxalineIC5037000.0 [1], 50000.0 [2]
2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxalineKi11730.0 [1]
(2S,4R)-2-Amino-4-[(E)-3-naphthalen-2-ylprop-2-enyl]pentanedioic acidKi14.0 [1], 14.8 [2], 15.0 [3], 10000.0 [4]
4-Chloro-2-(3-(naphthalen-2-yl)ureido)benzoic acidIC501200.0 [1], 30000.0 [2], 69000.0 [3]
2-(3-(3-Bromophenyl)ureido)-4-chlorobenzoic acidIC504800.0 [1], 30000.0 [2]
TezampanelIC50500.0 [1]
TezampanelKi4160.0 [1], 4200.0 [2]
Glutamic acidKi701.0 [1]
Kainic acidKi177.0 [1]
Apoptosis Inhibitor II, NS3694IC505000.0 [1]
(3S,4As,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenoxy]-decahydro-isoquinoline-3-carboxylic acidKi1200.0 [1], 1690.0 [2]
(3S,4Ar,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenylamino]-decahydro-isoquinoline-3-carboxylic acidKi800.0 [1], 1550.0 [2]
(3S,4Ar,6S,8aR)-6-[(4-carboxyphenyl)methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochlorideKi3600.0 [1]
1-(3-Bromophenyl)-3-[5-chloro-2-(2H-tetrazol-5-yl)phenyl]ureaIC502000.0 [1], 30000.0 [2]
2-[3-(3-Bromophenyl)ureido]-4-chlorobenzenesulfonic acidIC501500.0 [1], 30000.0 [2]
1-(3-Bromophenyl)-3-[5-chloro-2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]ureaIC504600.0 [1], 30000.0 [2]
(2S,4R)-2-Amino-4-[(E)-3-(4-chlorophenyl)prop-2-enyl]pentanedioic acidKi8.0 [1]
{2-[3-(3-Bromophenyl)ureido]-4-chlorophenyl}acetic acidIC503600.0 [1], 30000.0 [2]
alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACIDKi740.0 [1]
(S)-AmpaKi1150.0 [1]
2S,4R-4-MethylglutamateKi3.0 [1]
DysiherbaineKi0.74 [1]
LY382884Ki17130.0 [1]
N-(3-(Trifluoromethyl)phenyl)-N'-(2-hydroxy-5-chlorophenyl)ureaIC5030000.0 [1]
Benzoic acid, 2-((((3-(trifluoromethyl)phenyl)amino)carbonyl)amino)-IC5072000.0 [1]
2-Amino-3-(4-bromo-3-hydroxyisoxazol-5-YL)propanoic acidKi4800.0 [1]
4-Methylene-L-glutamic acidKi270.0 [1]
Cl-HIBOKi6800.0 [1]
5-Carboxy-2,4-dibenzamidobenzoic acidIC501600.0 [1]
(3S,4Ar,6S,8aR)-6-[[(2S)-2-carboxy-4,4-difluoropyrrolidin-1-yl]methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acidKi50.0 [1]
(RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acidKi5450.0 [1]
2-Amino-3-(5-(2-ethyl-2H-tetrazol-5-yl)-3-hydroxyisoxazol-4-yl)propanoic acidKi2920.0 [1]
(2S,4R)-4-Propylglutamic acidKi123.0 [1]
2-Amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acidKi34200.0 [1]
2-[(Anilinocarbonyl)amino]benzoic acidIC50100000.0 [1]
(S)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-YL)isoxazol-4-YL]propionic acidKi81.0 [1]
(2R,4S)-2-Allyl-4-aminopentanedioic acidKi56.0 [1]
(4R)-4-(3-Phenylpropyl)-L-glutamic acidKi1190.0 [1]
(2S,4R)-4-Pentylglutamic acidKi267.0 [1]
(S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxythiophene-3-ylmethyl)pyrimidine-2,4-dioneIC50680.0 [1]
(2S)-2-Amino-3-(2,4-dioxo-5,7-dihydrothieno[3,4-d]pyrimidin-1-yl)propanoic acidIC503.8 [1]
(2S)-2-Amino-3-(2,4-dioxothieno[3,2-d]pyrimidin-1-yl)propanoic acidIC501.9 [1]
(2R,3S)-1-(9-Iodophenanthrene-3-carbonyl)piperazine-2,3-dicarboxylic acidIC50650.0 [1]
4-Chloro-2-[(3-iodophenyl)carbamoylamino]benzoic AcidIC502200.0 [1]
2-(3-Benzo[1,3]dioxol-5-yl-ureido)-4-chloro-benzoic acidIC503600.0 [1]
4-Chloro-2-[3-(4-fluoro-phenyl)-ureido]-benzoic acidIC5014000.0 [1]
4-Chloro-2-[3-(4-chloro-phenyl)-ureido]-benzoic acidIC503100.0 [1]
2-[3-(4-Bromo-phenyl)-ureido]-4-chloro-benzoic acidIC502200.0 [1]
2-Methyl-6-[3-(3-trifluoromethyl-phenyl)-ureido]-benzoic acidIC50100000.0 [1]
3-[3-(3-Trifluoromethyl-phenyl)-ureido]-naphthalene-2-carboxylic acidIC5060000.0 [1]
(2S)-2-Amino-4-cyclopentylidenepentanedioic acidKi32.6 [1]
4-Trifluoromethyl-2-[3-(3-trifluoromethyl-phenyl)-ureido]-benzoic acidIC5021000.0 [1]
4-Chloro-2-[3-(2-hydroxy-phenyl)-ureido]-benzoic acidIC5021000.0 [1]
5-Methyl-2-[3-(3-trifluoromethyl-phenyl)-ureido]-benzoic acidIC50100000.0 [1]
3-Methyl-2-[3-(3-trifluoromethyl-phenyl)-ureido]-benzoic acidIC50100000.0 [1]
4-Bromo-2-[3-(3-trifluoromethyl-phenyl)-ureido]-benzoic acidIC506100.0 [1]
4-Chloro-2-[3-(2-trifluoromethyl-phenyl)-ureido]-benzoic acidIC504500.0 [1]
4-Chloro-2-[3-(4-iodo-phenyl)-ureido]-benzoic acidIC504700.0 [1]
CID 10330442Ki54.4 [1]
4-[(E)-2,2-Dimethylpropylidene]-L-glutamic acidKi85.7 [1]
4-Chloro-2-(3-phenyl-ureido)-benzoic acidIC5010000.0 [1]
4-Chloro-2-(3-cyclohexyl-ureido)-benzoic acidIC50100000.0 [1]
2-[3-(2-Bromo-phenyl)-ureido]-4-chloro-benzoic acidIC504500.0 [1]
(2s)-2-Amino-3-(4-Hydroxy-1,2,5-Thiadiazol-3-Yl)propanoic AcidKi18500.0 [1]
4-Chloro-2-[3-(2-methoxy-phenyl)-ureido]-benzoic acidIC5012000.0 [1]
4-Chloro-2-[3-(3-chloro-phenyl)-ureido]-benzoic acidIC501300.0 [1]
2-(3-Biphenyl-2-yl-ureido)-4-chloro-benzoic acidIC5010000.0 [1]
4-Chloro-2-(3-thiophen-2-yl-ureido)-benzoic acidIC5018000.0 [1]
(2S)-2-Amino-4-pentan-3-ylidenepentanedioic acidKi241.0 [1]
4-Chloro-2-(3-pyridin-2-yl-ureido)-benzoic acidIC5031000.0 [1]
4-Chloro-2-(3-pyridin-4-yl-ureido)-benzoic acidIC5088000.0 [1]
4-Chloro-2-[3-(2-iodo-phenyl)-ureido]-benzoic acidIC505000.0 [1]
(2r)-2-Amino-3-(4-Hydroxy-1,2,5-Thiadiazol-3-Yl)propanoic AcidKi10000.0 [1]
2-(3-Biphenyl-4-yl-ureido)-4-chloro-benzoic acidIC5029000.0 [1]
2-[7-[3-[[(4-Nitrophenyl)carbamoylamino]methyl]pyrrol-1-yl]-2,3-dioxo-6-(trifluoromethyl)-4H-quinoxalin-1-yl]acetic acidKi100.0 [1]
4-Chloro-2-[3-(4-methoxy-phenyl)-ureido]-benzoic acidIC5010000.0 [1]
2-(3-Biphenyl-3-yl-ureido)-4-chloro-benzoic acidIC5012000.0 [1]
E-2-Amino-4-[3-(2-chloro-phenyl)-allyl]-pentanedioic acidKi254.0 [1]
E-2-Amino-4-[3-(4-carboxy-phenyl)-allyl]-pentanedioic acidKi3590.0 [1]
E-2-Amino-4-[3-(4-isopropyl-phenyl)-allyl]-pentanedioic acidKi58.0 [1]
E-2-Amino-4-[3-(2,6-dichloro-phenyl)-allyl]-pentanedioic acidKi131.0 [1]
(2S,4R)-2-Amino-4-[(Z)-pent-2-enyl]pentanedioic acidKi160.0 [1]
(2S,4R)-2-Amino-4-[(E)-3-(2-methoxyphenyl)prop-2-enyl]pentanedioic acidKi26.0 [1]
2-Amino-4-but-2-enyl-pentanedioic acidKi577.0 [1]
2-Amino-4-hex-2-ynyl-pentanedioic acidKi3606.0 [1]
2-Amino-4-(2-methyl-3-phenyl-allyl)-pentanedioic acidKi670.0 [1]
E-2-Amino-4-[3-(4-fluoro-phenyl)-allyl]-pentanedioic acidKi78.0 [1]
E-2-Amino-4-[3-(4-methoxy-phenyl)-allyl]-pentanedioic acidKi284.0 [1]
E-2-Amino-4-[3-(4-trifluoromethyl-phenyl)-allyl]-pentanedioic acidKi52.0 [1]
2-Amino-4-pent-2-ynyl-pentanedioic acidKi831.0 [1]
2-Amino-4-pent-2-enyl-pentanedioic acidKi161.0 [1]
E-2-Amino-4-[3-(4-methylsulfanyl-phenyl)-allyl]-pentanedioic acidKi32.0 [1]
E-2-Amino-4-[3-(4-cyano-phenyl)-allyl]-pentanedioic acidKi367.0 [1]
E-2-Amino-4-[3-(3-chloro-phenyl)-allyl]-pentanedioic acidKi60.0 [1]
E-2-Amino-4-[3-(4-nitro-phenyl)-allyl]-pentanedioic acidKi59.0 [1]
2-Amino-4-hexyl-pentanedioic acidKi2376.0 [1]
E-2-Amino-4-[3-(3,4-dimethoxy-phenyl)-allyl]-pentanedioic acidKi540.0 [1]
(2S,4S)-2-Amino-4-prop-2-ynylpentanedioic acidKi307.0 [1]
(2S,4R)-2-Amino-4-[(E)-but-2-enyl]pentanedioic acidKi21.0 [1]
2-Amino-4-(3-chloro-allyl)-pentanedioic acidKi41.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Glutamate receptor ionotropic kainate 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-kainate-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Glutamate receptor ionotropic kainate 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-kainate-1-inhibitors-ic50-ki.
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