![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_bfc819183f2cf277c891caeebe90b592.svg) | Glutamic acid | Ki | 868.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_533dec12a2edd4e5a4a8bf0f4f3f0d48.svg) | Kainic acid | Ki | 1710.0 [1], 1714.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_9aa811db64317f7611351f7066ca80d6.svg) | (S)-Ampa | Ki | 40.0 [1], 155.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_6830c471230bebcdb0e2186e8c2b9e4c.svg) | 2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_6830c471230bebcdb0e2186e8c2b9e4c.svg) | 2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline | Ki | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_098f149a9418cb8ddb08d5ebe901a713.svg) | Tezampanel | Ki | 50000.0 [1], 50500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_906db03a68fc7dcd81d002840aba74ec.svg) | (2S,4R)-2-Amino-4-[(E)-3-naphthalen-2-ylprop-2-enyl]pentanedioic acid | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_bce24e213c4ecca82f704c2b2bb91d5a.svg) | 6-(4-Amino-3,5-dimethylphenyl)-8-[(3-bromo-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3,10-dihydro-2H-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one | Ki | 7400.0 [1], 11400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_3a609542ef6028c5380d15d307592e09.svg) | alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID | Ki | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_103616395dd66f26f921fab1aa97fc55.svg) | Willardiine | Ki | 8850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_a1fa4b88669eb85bf6a9ac3e3b1528b3.svg) | Argiotoxin 636 | IC50 | 430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_dacbbff0c89e46e344ee5d75618a287d.svg) | 2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-YL)-propionic acid | Ki | 305.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_46ee62ea2faae64339874a9aa414b95b.svg) | Iodo-willardiine | Ki | 972.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_93214b41b9a1ac2e981cecade6180721.svg) | Bromo-willardiine | Ki | 457.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_10e30f1c1bbd2d12a799df5bbf2ceb72.svg) | 2-Amino-3-(4-bromo-3-hydroxyisoxazol-5-YL)propanoic acid | Ki | 11700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_f4bb5330d6171f1a9d21b58944a3ffb9.svg) | Cl-HIBO | Ki | 11900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_7996bbf076fca5004472ed7837c972f2.svg) | 2-[(3-Bromophenyl)methyl]-6,8-dichloro-1,1-dioxo-3,4-dihydro-1lambda6,2,4-benzothiadiazine-3-carboxylic acid | IC50 | 38000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_4f39a6958b195f30072f4d350a8d34ba.svg) | 3-(5-Chloro-2,4-Dioxo-3,4-Dihydropyrimidin-1(2h)-Yl)-L-Alanine | Ki | 451.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_d68e7ef12c4d63bdcef0ac5d2a673e7c.svg) | 3-(5-Nitro-2,4-Dioxo-3,4-Dihydropyrimidin-1(2h)-Yl)-L-Alanine | Ki | 207.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_499ac462ab0a9bdddb90333e6aacd797.svg) | (RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid | Ki | 732.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_093f2cb59e4907ba19b8fe6ee09768b7.svg) | 2-Amino-3-(5-(2-ethyl-2H-tetrazol-5-yl)-3-hydroxyisoxazol-4-yl)propanoic acid | Ki | 44.4 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_0326e286ffb0bc633f9efa4027124c32.svg) | 2-Amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acid | Ki | 2350.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_dd43aca9eeb7e287bb617d57cb5fc7a7.svg) | (S)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-YL)isoxazol-4-YL]propionic acid | Ki | 2.7 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_5077a6d3391dcb32208e1d43a73d4a7d.svg) | 4-Chloro-2-(3-(naphthalen-2-yl)ureido)benzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_897915006e04f9e2bc2fea83dbc3d147.svg) | 2-(3-(3-Bromophenyl)ureido)-4-chlorobenzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_54d7b7763ceedb579a21870a525b4883.svg) | (2S)-2-Amino-4-cyclopentylidenepentanedioic acid | Ki | 533.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_f82710b3951f52c05d620c67e547348e.svg) | CID 10330442 | Ki | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_eb7b4abb504f722de5d1b09e809f87d2.svg) | (2s)-2-Amino-3-(4-Hydroxy-1,2,5-Thiadiazol-3-Yl)propanoic Acid | Ki | 182.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_a543be41acc510fc78c6d273762269c9.svg) | (2S)-2-Amino-4-pentan-3-ylidenepentanedioic acid | Ki | 4710.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_70efa62ad5cd789e44e92bbdf61b7629.svg) | (2r)-2-Amino-3-(4-Hydroxy-1,2,5-Thiadiazol-3-Yl)propanoic Acid | Ki | 1055.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_e3ee201fe0cb9e332b32b2d8590711c9.svg) | (2S,4R)-2-Amino-4-[(E)-3-(2-methoxyphenyl)prop-2-enyl]pentanedioic acid | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_f3d7cd048eeab2c43751a9c6bf90742d.svg) | (2S,4Z)-2-Amino-4-(2-methylpropylidene)pentanedioic Acid | Ki | 10300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_6b1268589b81c8dd5afe061f5dd75a9a.svg) | (S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid | Ki | 3.6 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_5b09bf3e80863da4762fc1ce46d346d2.svg) | (2S)-2-Amino-3-(6-methyl-3,5-dioxo-1,2,4-triazin-2-yl)propanoic acid | Ki | 89.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_5e19f45b556506f8bc8d08908e62f3dc.svg) | (S)-2-Amino-3-(3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid | Ki | 189.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_f257b7c28b4890bf6e5562309dd067c4.svg) | (2S)-2-Amino-3-(6-iodo-3,5-dioxo-1,2,4-triazin-2-yl)propanoic acid | Ki | 19.9 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_5663921d8853062aa29da52ffb8a740a.svg) | (3S,4Ar,6S,8aR)-6-[(4-carboxyimidazol-1-yl)methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;dihydrochloride | Ki | 262000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-4_68b167d8a544dccede4c4eedb8897793.svg) | (S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid | Ki | 7.9 [1] |