![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_103cf7391970afed8a6564df558b4de5.svg) | Perampanel | IC50 | 243.0 [1], 485.0 [2], 623.0 [3], 1180.0 [4], 6510.0 [5] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_aaf3f0b5d17cdfff9ee677abf92678c0.svg) | 4-[Methyl-(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]phenol | IC50 | 2970.0 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_bfc819183f2cf277c891caeebe90b592.svg) | Glutamic acid | Ki | 1360.0 [1], 1362.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_533dec12a2edd4e5a4a8bf0f4f3f0d48.svg) | Kainic acid | Ki | 7449.0 [1], 7450.0 [2], 7500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_a1fa4b88669eb85bf6a9ac3e3b1528b3.svg) | Argiotoxin 636 | IC50 | 350.0 [1], 3400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_354794f6916c5f993912257ec454ff83.svg) | 6-((1S)-1-(1-(5-(2-Hydroxyethoxy)-2-pyridinyl)-1H-pyrazol-3-yl)ethyl)-2(3H)-benzothiazolone | IC50 | 65.3 [1], 68500.0 [2], 83300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f0d496cde22081b203e16e33fa37d7a8.svg) | 6-[(1S)-1-[1-[5-(3-Hydroxy-3-methylbutyl)pyridin-2-yl]pyrazol-3-yl]ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 160.0 [1], 9260.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_16cce4d7ae4bc4acaea555677920d8c5.svg) | 6-[(1S)-1-[1-[5-(2-Hydroxyethyl)pyridin-2-yl]pyrazol-3-yl]ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 61.6 [1], 25700.0 [2], 83300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_4fdfc07140b0fd21e5b89a58d3698bb6.svg) | 6-[(1R)-1-(1-Pyridin-2-ylpyrazol-3-yl)ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 615.0 [1], 9260.0 [2], 83300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_143d82ec99ef5f74e36f304c0aa7ea1d.svg) | 6-[(1S)-1-(1-Pyridin-2-ylpyrazol-3-yl)ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 50.9 [1], 9260.0 [2], 83300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f26a41fedeb563ccf571096ea8255ebb.svg) | N-(1H-Indazol-5-yl)-N-[(1-methylpyrazol-3-yl)methyl]-4-pyridin-2-yl-1,3-thiazol-2-amine | IC50 | 53.9 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_86b5973cec95ced5ca196965b7522538.svg) | 6-[(1R)-1-[1-[5-(2-Hydroxyethyl)pyridin-2-yl]pyrazol-3-yl]ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 2820.0 [1], 9260.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_53abf530875921ee223ae83b64712a15.svg) | 6-[Methyl-(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]-3H-1,3-benzothiazol-2-one | IC50 | 70.0 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_26f0376762ba64a64844771d42161ba3.svg) | 6-[(1S)-1-[1-(5-Fluoropyridin-2-yl)pyrazol-3-yl]ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 53.6 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_3d0feab51a46cc12fe29a3f82564df94.svg) | N-(1H-Indazol-5-yl)-N-methyl-4-pyridin-2-yl-1,3-thiazol-2-amine | IC50 | 147.0 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f4e20f445ff628f40bc4da591244d0e1.svg) | N-Methyl-N-(1-pyridin-2-ylpyrazol-3-yl)-1H-indazol-5-amine | IC50 | 353.0 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_432bcfc90155021c7a569f96f2fb6563.svg) | 6-[1-(1-Pyridin-2-ylpyrazol-3-yl)ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 122.0 [1], 83300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_45165330e651a199e8a52b8fa1499743.svg) | 6-[(1R)-1-[1-[5-(2-Hydroxyethoxy)pyridin-2-yl]pyrazol-3-yl]ethyl]-3H-1,3-benzothiazol-2-one | IC50 | 1790.0 [1], 9260.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_9aa811db64317f7611351f7066ca80d6.svg) | (S)-Ampa | Ki | 21.9 [1], 103.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_6830c471230bebcdb0e2186e8c2b9e4c.svg) | 2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_6830c471230bebcdb0e2186e8c2b9e4c.svg) | 2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline | Ki | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_098f149a9418cb8ddb08d5ebe901a713.svg) | Tezampanel | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_b02deac1433d560f422b172c2a18c17a.svg) | N-[1-{3-[4-(3-Amino-propylamino)-butylamino]-propylcarbamoyl}-2-(4-hydroxy-phenyl)-ethyl]-butyramide | Ki | 22000.0 [1], 170000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_25990dc834192c4d96b909a9dd81f2d4.svg) | N-[1-[8-(3-Amino-propylamino)-octylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl]-butyramide | Ki | 65.0 [1], 8000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_bce24e213c4ecca82f704c2b2bb91d5a.svg) | 6-(4-Amino-3,5-dimethylphenyl)-8-[(3-bromo-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3,10-dihydro-2H-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one | Ki | 6400.0 [1], 13200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_a295e9af31da270f98461c20a01a598d.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]cyclohexanecarboxamide | Ki | 78.0 [1], 240.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_4e2a421f9c0acd721845241dd50f7b11.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]pyridine-4-carboxamide | Ki | 64.0 [1], 330.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_ccf191765c49f9ba4aa3022528a2df57.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]pyridine-3-carboxamide | Ki | 88.0 [1], 210.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_9657737ca59e88a0eef88aa0a2491673.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]hexanamide | Ki | 68.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_41cfdea6866c918597c8b231b4978914.svg) | N-[8-(3-Aminopropylamino)octyl]-3-(4-hydroxyphenyl)-2-(propanoylamino)propanamide | Ki | 100.0 [1], 280.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_d0a4ad09398a88de9e19910a93561bcb.svg) | N-[1-[3-(8-Aminooctylamino)propylamino]-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]butanamide | Ki | 350.0 [1], 8100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_87ddfa857d9c8fb4b1e413452eea17fd.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-2,2-dimethylpropanamide | Ki | 90.0 [1], 140.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_4e508ed98a359c482ad09b1980212d40.svg) | N-[1-[4-(7-Aminoheptylamino)butylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]butanamide | Ki | 38.0 [1], 135.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_acf58e4458867c2741c0d670f0d78460.svg) | N-[8-(3-Aminopropylamino)octyl]-3-(4-hydroxyphenyl)-2-[(2-phenylacetyl)amino]propanamide | Ki | 110.0 [1], 250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_7e3ab546cb008e0b5c3a3f8a8bd8b9a7.svg) | 2-Acetamido-N-[8-(3-aminopropylamino)octyl]-3-(4-hydroxyphenyl)propanamide | Ki | 220.0 [1], 300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_b63128bb1092d77261984e37c4673b24.svg) | N-[8-(3-Aminopropylamino)octyl]-3-(4-hydroxyphenyl)-2-[[(E)-3-phenylprop-2-enoyl]amino]propanamide | Ki | 110.0 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_78111f8693063443c8ea56af1a9caeed.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]pyridine-2-carboxamide | Ki | 130.0 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_2047bfda71633831cdbf164b69755892.svg) | N-[8-(3-Aminopropylamino)octyl]-3-(4-hydroxyphenyl)-2-(3-phenylpropanoylamino)propanamide | Ki | 250.0 [1], 254.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_82ebae4e28181dedde8b979e4543616b.svg) | N-[1-[5-(6-Aminohexylamino)pentylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]butanamide | Ki | 3.3 [1], 287.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f8d28602d3b748544462537d172e66c3.svg) | N-[1-[8-(3-Aminopropylamino)octylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]benzamide | Ki | 130.0 [1], 250.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_d106b359f537e3cd99341d3ed4e1d1b3.svg) | N-[1-[7-(4-Amino-butylamino)-heptylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl]-butyramide | Ki | 168.0 [1], 3000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_568ac1714ca5ee034b4c8bfa62b6eaa2.svg) | N-[1-[9-(2-Aminoethylamino)nonylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]butanamide | Ki | 410.0 [1], 6200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_fe7abec5f058c49707a44fb144107a06.svg) | N-[1-[6-(5-Aminopentylamino)hexylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]butanamide | Ki | 468.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_3a609542ef6028c5380d15d307592e09.svg) | alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID | Ki | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_d3960c986f122a12885ab0a72b117926.svg) | Joro spider toxin | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_103616395dd66f26f921fab1aa97fc55.svg) | Willardiine | Ki | 386.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_dacbbff0c89e46e344ee5d75618a287d.svg) | 2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-YL)-propionic acid | Ki | 14.7 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_46ee62ea2faae64339874a9aa414b95b.svg) | Iodo-willardiine | Ki | 163.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_93214b41b9a1ac2e981cecade6180721.svg) | Bromo-willardiine | Ki | 92.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_10e30f1c1bbd2d12a799df5bbf2ceb72.svg) | 2-Amino-3-(4-bromo-3-hydroxyisoxazol-5-YL)propanoic acid | Ki | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f4bb5330d6171f1a9d21b58944a3ffb9.svg) | Cl-HIBO | Ki | 130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_906db03a68fc7dcd81d002840aba74ec.svg) | (2S,4R)-2-Amino-4-[(E)-3-naphthalen-2-ylprop-2-enyl]pentanedioic acid | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_4f39a6958b195f30072f4d350a8d34ba.svg) | 3-(5-Chloro-2,4-Dioxo-3,4-Dihydropyrimidin-1(2h)-Yl)-L-Alanine | Ki | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_d68e7ef12c4d63bdcef0ac5d2a673e7c.svg) | 3-(5-Nitro-2,4-Dioxo-3,4-Dihydropyrimidin-1(2h)-Yl)-L-Alanine | Ki | 279.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_499ac462ab0a9bdddb90333e6aacd797.svg) | (RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid | Ki | 5150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_093f2cb59e4907ba19b8fe6ee09768b7.svg) | 2-Amino-3-(5-(2-ethyl-2H-tetrazol-5-yl)-3-hydroxyisoxazol-4-yl)propanoic acid | Ki | 145.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_0326e286ffb0bc633f9efa4027124c32.svg) | 2-Amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acid | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_dd43aca9eeb7e287bb617d57cb5fc7a7.svg) | (S)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-YL)isoxazol-4-YL]propionic acid | Ki | 5.22 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_20f86ba77dbb851a656e282b9965e97e.svg) | Philanthotoxin-74 | Ki | 168.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_5077a6d3391dcb32208e1d43a73d4a7d.svg) | 4-Chloro-2-(3-(naphthalen-2-yl)ureido)benzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_26203dd39c2214a5aa4cea9297a4b80b.svg) | (2S)-2-Amino-3-(2,4-dioxothieno[3,2-d]pyrimidin-1-yl)propanoic acid | IC50 | 374.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_897915006e04f9e2bc2fea83dbc3d147.svg) | 2-(3-(3-Bromophenyl)ureido)-4-chlorobenzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_54d7b7763ceedb579a21870a525b4883.svg) | (2S)-2-Amino-4-cyclopentylidenepentanedioic acid | Ki | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f82710b3951f52c05d620c67e547348e.svg) | CID 10330442 | Ki | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_eb7b4abb504f722de5d1b09e809f87d2.svg) | (2s)-2-Amino-3-(4-Hydroxy-1,2,5-Thiadiazol-3-Yl)propanoic Acid | Ki | 185.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_a543be41acc510fc78c6d273762269c9.svg) | (2S)-2-Amino-4-pentan-3-ylidenepentanedioic acid | Ki | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_70efa62ad5cd789e44e92bbdf61b7629.svg) | (2r)-2-Amino-3-(4-Hydroxy-1,2,5-Thiadiazol-3-Yl)propanoic Acid | Ki | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_e3ee201fe0cb9e332b32b2d8590711c9.svg) | (2S,4R)-2-Amino-4-[(E)-3-(2-methoxyphenyl)prop-2-enyl]pentanedioic acid | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f3d7cd048eeab2c43751a9c6bf90742d.svg) | (2S,4Z)-2-Amino-4-(2-methylpropylidene)pentanedioic Acid | Ki | 113400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f2c80fa1ed513a02bbcf0cb0324b4ff8.svg) | 6-[2-Ethoxyethyl-(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]-3H-1,3-benzothiazol-2-one | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_6b1268589b81c8dd5afe061f5dd75a9a.svg) | (S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid | Ki | 7.1 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_5b09bf3e80863da4762fc1ce46d346d2.svg) | (2S)-2-Amino-3-(6-methyl-3,5-dioxo-1,2,4-triazin-2-yl)propanoic acid | Ki | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_5e19f45b556506f8bc8d08908e62f3dc.svg) | (S)-2-Amino-3-(3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid | Ki | 163.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_f257b7c28b4890bf6e5562309dd067c4.svg) | (2S)-2-Amino-3-(6-iodo-3,5-dioxo-1,2,4-triazin-2-yl)propanoic acid | Ki | 73.9 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_5663921d8853062aa29da52ffb8a740a.svg) | (3S,4Ar,6S,8aR)-6-[(4-carboxyimidazol-1-yl)methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;dihydrochloride | Ki | 134000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_68b167d8a544dccede4c4eedb8897793.svg) | (S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid | Ki | 29.0 [1] |
![](https://images.aatbio.com/dataset/ic50/glutamate-receptor-ionotropic-ampa-1_e38626a232554611fbd926c061ab29ff.svg) | (2S,4R)-2-Amino-4-[(E)-3-(4-chlorophenyl)prop-2-enyl]pentanedioic acid | Ki | 10000.0 [1] |