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Glutamate (NMDA) receptor subunit zeta 1 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
5-[3-(4-Benzylpiperidin-1-yl)prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC505.3 [1], 35000.0 [2], 100000.0 [3]
5-[3-[4-[(4-Fluorophenyl)methyl]piperidin-1-yl]prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC508.2 [1], 38000.0 [2], 100000.0 [3]
5-(3-(4-Benzylpiperidin-1-yl)prop-1-ynyl)-1-methyl-1H-benzo[d]imidazol-2(3H)-oneIC5062000.0 [1], 89000.0 [2], 100000.0 [3]
5-[3-[4-[(3-Fluorophenyl)methyl]piperidin-1-yl]prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC506.1 [1], 100000.0 [2]
5-[4-(4-Benzylpiperidin-1-yl)but-1-ynyl]-1,3-dihydroindol-2-oneIC50320.0 [1], 52000.0 [2], 100000.0 [3]
5-[3-(4-Benzylpiperidin-1-yl)prop-1-ynyl]-1,3-dihydroindol-2-oneIC50110.0 [1], 100000.0 [2]
5-[3-(4-Benzyl-4-hydroxypiperidin-1-yl)prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC5019.0 [1], 100000.0 [2]
5-[3-(4-Benzylpiperidin-1-yl)prop-1-ynyl]-1,3-dihydrobenzimidazole-2-thioneIC5016.0 [1], 25000.0 [2], 100000.0 [3]
5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1H-indoleIC5015000.0 [1], 100000.0 [2]
5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1H-benzotriazoleIC50420.0 [1], 100000.0 [2]
5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1H-indazoleIC50250.0 [1], 95000.0 [2], 100000.0 [3]
5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1H-benzotriazoleIC50220.0 [1], 100000.0 [2]
5-[4-(4-Benzylpiperidin-1-yl)but-1-ynyl]-1,3-dihydrobenzimidazole-2-thioneIC50180.0 [1], 75000.0 [2], 100000.0 [3]
5-[3-(4-Benzyl-piperidin-1-yl)-prop-1-ynyl]-1H-indazoleIC50380.0 [1], 100000.0 [2]
5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1,3-dihydro-benzoimidazol-2-oneIC5089.0 [1], 39000.0 [2], 100000.0 [3]
7-[4-(4-Benzylpiperidin-1-yl)but-1-ynyl]-4H-1,4-benzoxazin-3-oneIC501100.0 [1], 100000.0 [2]
5-[3-[4-[(4-Methoxyphenyl)methyl]piperidin-1-yl]prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC5026.0 [1], 100000.0 [2]
6-[4-(4-Benzylpiperidin-1-yl)but-1-ynyl]-3H-1,3-benzoxazol-2-oneIC50120.0 [1], 39000.0 [2], 100000.0 [3]
5-[4-(4-Benzyl-piperidin-1-yl)-but-1-ynyl]-1H-indole-2,3-dioneIC501800.0 [1], 57000.0 [2]
4,6-Dichloro-1H-indole-2-carboxylic acidKi2900.0 [1]
[(1S)-1-{[(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl)methyl]amino}ethyl]phosphonic acidIC505.0 [1]
[(1S)-1-[(7-Nitro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acidIC5032.0 [1]
[(1S)-1-[[2,3-Dioxo-7-(trifluoromethyl)-1,4-dihydroquinoxalin-5-yl]methylamino]ethyl]phosphonic acidIC508.0 [1]
CID 9863759IC501.0 [1]
4,6-Dichloro-3-[(2,4-dioxo-3-phenylimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi22.0 [1]
[(1S)-1-[(7-Iodo-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acidIC508.0 [1]
4,6-Dichloro-3-[(2,4-dioxo-3-phenyl-5-propan-2-ylimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi1100.0 [1]
5-[3-[4-[(4-Chlorophenyl)methyl]piperidin-1-yl]prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC5019.0 [1]
5-[3-[4-[(4-Methylphenyl)methyl]piperidin-1-yl]prop-1-ynyl]-1,3-dihydrobenzimidazol-2-oneIC5017.0 [1]
5-[3-(4-Benzylpiperidin-1-yl)prop-1-ynyl]-3-methyl-1H-benzimidazol-2-oneIC50100000.0 [1]
6-[3-(4-Benzylpiperidin-1-yl)prop-1-ynyl]-3H-1,3-benzoxazol-2-oneIC5049.0 [1]
4,6-Dichloro-3-[[3-(3-methylphenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi45.0 [1]
4,6-Dichloro-3-[[3-(3,5-dichlorophenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi80.0 [1]
4,6-Dichloro-3-[(3-cyclohexyl-2,4-dioxoimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi130.0 [1]
4,6-Dichloro-3-[[3-(4-methoxyphenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi100.0 [1]
3-(Benzenesulfonylamino-methyl)-4,6-dichloro-1H-indole-2-carboxylic acidKi990.0 [1]
3-[[3-(3-Acetylphenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-4,6-dichloro-1H-indole-2-carboxylic acidKi57.0 [1]
4,6-Dichloro-3-[[3-(4-methylphenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi36.0 [1]
4,6-Dichloro-3-[(4-oxo-3-phenyl-2-sulfanylideneimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi580.0 [1]
4,6-Dichloro-3-[[3-(4-chlorophenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi120.0 [1]
4,6-Dichloro-3-[(5-methyl-2,4-dioxo-3-phenylimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi310.0 [1]
4,6-Dichloro-3-[(3-phenyl-ureido)-methyl]-1H-indole-2-carboxylic acidKi14.0 [1]
4,6-Dichloro-3-[[3-(3-chlorophenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi85.0 [1]
3-(Benzylamino-methyl)-4,6-dichloro-1H-indole-2-carboxylic acidKi92000.0 [1]
3-(Benzoylamino-methyl)-4,6-dichloro-1H-indole-2-carboxylic acidKi120.0 [1]
4,6-Dichloro-3-[(3-ethyl-2,4-dioxoimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi1000.0 [1]
4,6-Dichloro-3-(2-oxo-3-phenyl-imidazolidin-1-ylmethyl)-1H-indole-2-carboxylic acidKi58.0 [1]
3-[(Benzenesulfonylcarbamoylamino)methyl]-4,6-dichloro-1H-indole-2-carboxylic acidKi72.0 [1]
4,6-Dichloro-3-[[3-(4-fluorophenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-1H-indole-2-carboxylic acidKi53.0 [1]
4,6-Dichloro-3-[(2,4-dioxo-3-propan-2-ylimidazolidin-1-yl)methyl]-1H-indole-2-carboxylic acidKi1050.0 [1]
3-[[3-(4-Acetylphenyl)-2,4-dioxoimidazolidin-1-yl]methyl]-4,6-dichloro-1H-indole-2-carboxylic acidKi150.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl)-N-(2-hydroxypropyl)methanesulfonamideIC5040.0 [1]
2-[(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-methylsulfonylamino]acetic acidIC502.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3,3,3-trifluoropropyl)ethanesulfonamideIC5027.0 [1]
[(1S)-1-[(7-Cyano-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acidIC5076.0 [1]
[(1S)-1-[(7-Fluoro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acidIC509.0 [1]
[(1S)-1-[(7-Chloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acidIC506.0 [1]
N-(7-Chloro-6-methyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-hydroxyethyl)methanesulfonamideIC5014.0 [1]
N-(6-Chloro-7-methyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-hydroxyethyl)methanesulfonamideIC504.0 [1]
N-(7-Chloro-6-ethyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-hydroxyethyl)methanesulfonamideIC5058.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3-hydroxypropyl)methanesulfonamideIC5041.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-[(3-methoxyphenyl)methyl]methanesulfonamideIC5012.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-[(3-fluorophenyl)methyl]methanesulfonamideIC5045.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(oxan-2-ylmethyl)methanesulfonamideIC5039.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(oxolan-2-ylmethyl)methanesulfonamideIC5059.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-[2-(2-ethoxyethoxy)ethyl]methanesulfonamideIC50166.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-methoxyethyl)methanesulfonamideIC5038.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3-methoxypropyl)methanesulfonamideIC5024.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-ethoxyethyl)methanesulfonamideIC50209.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3-ethoxypropyl)methanesulfonamideIC5019.0 [1]
N-(6,7-Dichloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3,3,3-trifluoropropyl)methanesulfonamideIC5018.0 [1]
N-(7-Chloro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3-methoxypropyl)methanesulfonamideIC50728.0 [1]
N-(6-Chloro-7-methyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-methoxyethyl)methanesulfonamideIC5077.0 [1]
N-(7-Chloro-6-methyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(2-methoxyethyl)methanesulfonamideIC5074.0 [1]
N-(6-Chloro-7-ethyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-N-(3-methoxypropyl)methanesulfonamideIC5049.0 [1]
2-[(7-Chloro-6-methyl-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-methylsulfonylamino]acetic acidIC502.0 [1]
Items per page: 1 - 10 of 76
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References

This online tool may be cited as follows

MLA

"Quest Database™ Glutamate (NMDA) receptor subunit zeta 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/glutamate-nmda-receptor-subunit-zeta-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Glutamate (NMDA) receptor subunit zeta 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-nmda-receptor-subunit-zeta-1-inhibitors-ic50-ki.
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