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Glutamate [NMDA] receptor subunit epsilon 2 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
EliprodilKi13.0 [1]
4-(Trifluoromethoxy)-N'-[[2-(trifluoromethyl)phenyl]methyl]benzenecarboximidamideIC5047.0 [1]
4-(Trifluoromethoxy)-N'-[[2-(trifluoromethyl)phenyl]methyl]benzenecarboximidamideKi72.0 [1]
IfenprodilIC5020.0 [1]
IfenprodilKi10.0 [1]
3-Methoxy-N-(3-phenylpropyl)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-amineKi10.0 [1], 11.0 [2]
4-[(1S,2S)-2-(4-Benzyl-piperidin-1-yl)-1-hydroxy-propyl]-phenolKi10.0 [1]
N-BenzylbenzamidineKi10000.0 [1], 15000.0 [2]
(E)-N-Benzyl-3-phenyl-acrylamidineKi9.0 [1]
N-(4-(Benzyloxy)phenethyl)pyridin-4-amineIC50102.0 [1]
N-(4-(Benzyloxy)phenethyl)pyridin-4-amineKi93.0 [1]
N-(2-Methoxy-benzyl)-4-trifluoromethoxy-benzamidineIC504.1 [1]
N-(2-Methoxy-benzyl)-4-trifluoromethoxy-benzamidineKi5.7 [1]
N-(4-Phenylcyclohexyl)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-amineKi2.3 [1], 5.7 [2]
3,4-Dichloro-N-(3-chloro-benzyl)-benzamidineIC50110.0 [1]
3,4-Dichloro-N-(3-chloro-benzyl)-benzamidineKi16.0 [1]
3-Chloro-N-(3-chloro-benzyl)-benzamidineIC50420.0 [1]
3-Chloro-N-(3-chloro-benzyl)-benzamidineKi800.0 [1]
4-Chloro-N-(3-chloro-benzyl)-benzamidineIC50160.0 [1]
4-Chloro-N-(3-chloro-benzyl)-benzamidineKi63.0 [1]
N-(3-Chloro-benzyl)-4-fluoro-benzamidineIC50450.0 [1]
N-(3-Chloro-benzyl)-4-fluoro-benzamidineKi600.0 [1]
2-(3-Chloro-benzyl)-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineIC5049.0 [1]
2-(3-Chloro-benzyl)-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineKi8.0 [1]
N-Benzyl-4-chloro-benzamidineIC50720.0 [1]
N-Benzyl-4-chloro-benzamidineKi970.0 [1]
N-(3,5-Dimethyl-benzyl)-4-trifluoromethyl-benzamidineIC508.7 [1]
N-(3,5-Dimethyl-benzyl)-4-trifluoromethyl-benzamidineKi3.9 [1]
4-Trifluoromethyl-N-(3-trifluoromethyl-benzyl)-benzamidineIC50660.0 [1]
4-Trifluoromethyl-N-(3-trifluoromethyl-benzyl)-benzamidineKi700.0 [1]
N-(3-Chloro-benzyl)-4-trifluoromethyl-benzamidineIC5032.0 [1]
N-(3-Chloro-benzyl)-4-trifluoromethyl-benzamidineKi20.0 [1]
N-(2-Chloro-benzyl)-4-trifluoromethyl-benzamidineIC5048.0 [1]
N-(2-Chloro-benzyl)-4-trifluoromethyl-benzamidineKi56.0 [1]
N-Benzyl-4-trifluoromethyl-benzamidineIC50360.0 [1]
N-Benzyl-4-trifluoromethyl-benzamidineKi480.0 [1]
5-(3-Chlorophenyl)-2-(4-(trifluoromethoxy)phenyl)-4,5-dihydro-1H-imidazoleIC501976.0 [1]
5-(3-Chlorophenyl)-2-(4-(trifluoromethoxy)phenyl)-4,5-dihydro-1H-imidazoleKi296.0 [1]
5-(3-Chlorophenyl)-2-[3-chloro-4-(trifluoromethoxy)phenyl]-4,5-dihydro-1H-imidazoleIC50266.0 [1]
5-(3-Chlorophenyl)-2-[3-chloro-4-(trifluoromethoxy)phenyl]-4,5-dihydro-1H-imidazoleKi66.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-(3,5-dichlorophenyl)-4,5-dihydro-1H-imidazoleIC503670.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-(3,5-dichlorophenyl)-4,5-dihydro-1H-imidazoleKi223.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-(2-methoxyphenyl)-4,5-dihydro-1H-imidazoleIC50108.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-(2-methoxyphenyl)-4,5-dihydro-1H-imidazoleKi75.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-[2-(trifluoromethyl)phenyl]-4,5-dihydro-1H-imidazoleIC501270.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-[2-(trifluoromethyl)phenyl]-4,5-dihydro-1H-imidazoleKi353.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-[2-(trifluoromethoxy)phenyl]-4,5-dihydro-1H-imidazoleIC503480.0 [1]
2-[3-Chloro-4-(trifluoromethoxy)phenyl]-5-[2-(trifluoromethoxy)phenyl]-4,5-dihydro-1H-imidazoleKi505.0 [1]
2-Benzofuran-7-ylmethyl-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineIC5012.0 [1]
2-Benzofuran-7-ylmethyl-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineKi2.2 [1]
(3R)-3-[(3S,4S)-3-Fluoro-4-(4-hydroxyphenyl)piperidin-1-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-oneIC5024.0 [1]
(3R)-3-[(3S,4S)-3-Fluoro-4-(4-hydroxyphenyl)piperidin-1-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-oneKi6.3 [1]
3,4-Dichloro-N-(2-trifluoromethoxy-benzyl)-benzamidineIC5057.0 [1]
3,4-Dichloro-N-(2-trifluoromethoxy-benzyl)-benzamidineKi12.0 [1]
N-(3-Methoxy-benzyl)-4-trifluoromethoxy-benzamidineIC509.7 [1]
N-(3-Methoxy-benzyl)-4-trifluoromethoxy-benzamidineKi23.0 [1]
2-(2-Methoxy-benzyl)-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineIC505.9 [1]
2-(2-Methoxy-benzyl)-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineKi3.6 [1]
N-Benzyl-4-trifluoromethoxy-benzamidineIC5046.0 [1]
N-Benzyl-4-trifluoromethoxy-benzamidineKi120.0 [1]
N-(3,5-Dimethyl-benzyl)-4-trifluoromethoxy-benzamidineIC504.2 [1]
N-(3,5-Dimethyl-benzyl)-4-trifluoromethoxy-benzamidineKi1.2 [1]
2-(3,5-Dimethyl-benzyl)-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineIC5039.0 [1]
2-(3,5-Dimethyl-benzyl)-5-trifluoromethoxy-2,3-dihydro-isoindol-1-ylideneamineKi2.0 [1]
N-(3,5-Dichloro-benzyl)-4-trifluoromethoxy-benzamidineIC5024.0 [1]
N-(3,5-Dichloro-benzyl)-4-trifluoromethoxy-benzamidineKi0.6 [1]
(5S,7S)-2-Methoxy-7-(3-phenylpropylamino)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-5-olIC5012.0 [1]
(5S,7S)-2-Methoxy-7-(3-phenylpropylamino)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-5-olKi16.0 [1]
2-Methyl-6-(phenylethynyl)pyridineIC5018000.0 [1]
2-Methyl-4-(pyridin-3-ylethynyl)thiazoleIC50300000.0 [1]
4-[(1R,2S)-3-(4-Benzylpiperidin-1-yl)-1-hydroxy-2-methylpropyl]phenolKi173.0 [1]
TraxoprodilIC5074.0 [1]
BesonprodilKi30.0 [1]
4-[4-(4-Benzylpiperidino)-1-butynyl]phenolIC50100.0 [1]
N-(2-Methoxybenzyl)cinnamamidineKi0.7 [1]
7-(3-Phenylpropylamino)-6,7,8,9-tetrahydro-5H-benzocyclohepteneKi16.0 [1]
7-Methoxy-3-(4-phenylbutyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-1-olKi5.4 [1]
2-(4-Benzylpiperidin-1-yl)-1-(1H-indol-3-yl)ethanoneIC50769.0 [1]
2-Methoxy-7-(3-phenylpropylamino)-6,7,8,9-tetrahydro-5H-benzo[7]annulen-5-olKi16.0 [1]
2-Methyl-5-[3-(4-benzylpiperidino)propylthio]-1,3,4-thiadiazoleIC506400.0 [1]
2-Hydroxy-5-phenyl-7-azatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaene-12-carbonitrileIC509.0 [1]
Benzyl 4-[(1,3-thiazol-2-ylamino)methyl]piperidine-1-carboxylateKi122.0 [1]
7-(Phenethylamino)-6,7,8,9-tetrahydro-5H-benzocyclohepteneKi20.0 [1]
7-(4-Phenylbutylamino)-6,7,8,9-tetrahydro-5H-benzocyclohepteneKi17.0 [1]
7-(4-Phenylpiperazine-1-yl)-6,7,8,9-tetrahydro-5H-benzocyclohepteneKi12.0 [1]
7-(4-Benzylpiperidine-1-yl)-6,7,8,9-tetrahydro-5H-benzocyclohepteneKi2.9 [1]
Benzyl 4-[(pyridin-2-ylamino)methyl]piperidine-1-carboxylateKi37.0 [1]
Benzyl 4-[(pyrimidin-4-ylamino)methyl]piperidine-1-carboxylateKi75.0 [1]
4-Fluorobenzyl 4-[(2-pyrimidinylamino)methyl]-1-piperidinecarboxylateKi18.0 [1]
2-Hydroxy-5-piperidin-1-yl-7-azatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaene-12-carbonitrileIC5027.0 [1]
5-[2-(4-Benzylpiperidino)ethylthio]-1H-1,2,4-triazole-3-amineIC5035.0 [1]
(3R)-1-[(4-Fluorophenyl)methyl]-3-[4-(4-hydroxyphenyl)piperidin-1-yl]pyrrolidin-2-oneIC504.2 [1]
4-[4-Chloro-3-(difluoromethoxy)phenyl]-1-[(5-ethyl-1H-pyrazol-4-yl)methyl]pyrazoleIC503700.0 [1]
3-[[4-[4-Chloro-3-(difluoromethoxy)phenyl]pyrazol-1-yl]methyl]-1-methylpyrazoleIC502460.0 [1]
4-[4-Chloro-3-(difluoromethyl)phenyl]-1-(1H-pyrazol-5-ylmethyl)pyrazoleIC50890.0 [1]
4-[3-(Difluoromethoxy)-4-fluorophenyl]-1-(1H-pyrazol-5-ylmethyl)pyrazoleIC50370.0 [1]
4-[4-Chloro-3-(difluoromethoxy)phenyl]-1-(1H-pyrazol-5-ylmethyl)pyrazoleIC50230.0 [1]
4-[4-Chloro-3-(difluoromethoxy)phenyl]-1-[(1-methylpyrazol-4-yl)methyl]pyrazoleIC501750.0 [1]
4-[4-Chloro-3-(difluoromethoxy)phenyl]-1-(1H-pyrazol-4-ylmethyl)pyrazoleIC50350.0 [1]
1-[3-(Phenylthio)propyl]-4-benzylpiperidineIC504300.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Glutamate [NMDA] receptor subunit epsilon 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/glutamate-nmda-receptor-subunit-epsilon-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Glutamate [NMDA] receptor subunit epsilon 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-nmda-receptor-subunit-epsilon-2-inhibitors-ic50-ki.
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