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Glutamate NMDA receptor; GRIN1/GRIN2A Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
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▼
MemantineIC500.95 [1], 911.0 [2], 4360.0 [3], 4400.0 [4], 5600.0 [5]
KetamineIC503310.0 [1], 6100.0 [2]
TacrineIC504900.0 [1]
DexoxadrolIC509.7 [1]
DexoxadrolKi19.0 [1]
2-Methyl-9-[9-(2-methylpyrido[3,4-b]indol-2-ium-9-yl)nonyl]pyrido[3,4-b]indol-2-iumIC501400.0 [1]
PhencyclidineIC5011.8 [1]
AmantadineKi10000.0 [1]
PentamidineIC50720.0 [1]
DextrorphanIC501300.0 [1]
MethoctramineIC50138.0 [1]
LatrepirdineIC5013900.0 [1]
EsketamineIC5011.4 [1]
Philanthotoxin 343IC502739.0 [1]
EtoxadrolKi22.0 [1]
PeaqxIC50270.0 [1]
N,N'-Bis[6-(2,2-diphenylethylamino)hexyl]octane-1,8-diamineIC5011.0 [1]
N,N'-Bis[6-(2,2-diphenylethylamino)hexyl]dodecane-1,12-diamineIC504.2 [1]
[(2R,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methanamineIC5071.2 [1]
[(2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methanamineIC5017.7 [1]
(6,6-Diphenyl-1,4-dioxan-2-yl)methanamineIC5024.2 [1]
N'-[(2-Methoxyphenyl)methyl]-N-[6-[8-[(2-methoxyphenyl)methylamino]octylamino]hexyl]octane-1,8-diamineIC50256.7 [1]
N-[4-[4-(4-Aminobutylamino)butylamino]butyl]-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamideIC5072.0 [1]
N-[4-[3-(4-Aminobutylamino)propylamino]butyl]carbazole-9-carboxamideIC50211.0 [1]
N-[4-[3-(4-Aminobutylamino)propylamino]butyl]benzo[b][1]benzazepine-11-carboxamideIC50198.0 [1]
N-[4-[3-(4-Aminobutylamino)propylamino]butyl]-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamideIC50117.0 [1]
1-(4-Hydroxyphenyl)-2-[4-[(4-isothiocyanatophenyl)methyl]piperidin-1-yl]ethanoneIC5016000.0 [1]
N,N'-Bis[5-[(2-methoxyphenyl)methylamino]pentyl]decane-1,10-diamineIC5089.3 [1]
[(2,3-Dioxo-1,4-dihydroquinoxalin-5-yl)-[[(1S)-1-naphthalen-1-ylethyl]amino]methyl]phosphonic acidIC501700.0 [1]
[Anilino-(2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acidIC50490.0 [1]
[7-(4-Chlorophenyl)-2,3-dioxo-1,4-dihydroquinoxalin-5-yl]methylphosphonic acidIC500.2 [1]
[(Benzhydrylamino)-(2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acidIC50170.0 [1]
[(2,3-Dioxo-1,4-dihydroquinoxalin-5-yl)-(2-phenylethylamino)methyl]phosphonic acidIC5040.0 [1]
[[Acetyl(methyl)amino]-(2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acidIC502800.0 [1]
[(2,3-Dioxo-1,4-dihydroquinoxalin-5-yl)-(methylamino)methyl]phosphonic acidIC50790.0 [1]
[(Methoxycarbonylamino)-(7-nitro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acidIC50110.0 [1]
[[[(1S)-2,3-Dihydro-1H-inden-1-yl]amino]-(2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acidIC5060.0 [1]
[(2,3-Dioxo-1,4-dihydroquinoxalin-5-yl)-[[(1R)-1-phenylethyl]amino]methyl]phosphonic acidIC5050.0 [1]
[[Benzyl(methyl)amino]-(2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acidIC50600.0 [1]
Hydroxy(2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-5-yl)methylphosphonic acidIC501.1 [1]
[(2,3-Dioxo-1,4-dihydroquinoxalin-5-yl)-[[(1S)-1-phenylethyl]amino]methyl]phosphonic acidIC5018.0 [1]
N-[3-[4-(3-Aminopropylamino)butylamino]propyl]-9,10-dioxoanthracene-2-carboxamideIC50392.0 [1]
N-[3-[4-(3-Aminopropylamino)butylamino]propyl]benzo[b][1]benzazepine-11-carboxamideIC50203.0 [1]
N-[4-[4-(4-Aminobutylamino)butylamino]butyl]benzo[b][1]benzazepine-11-carboxamideIC50240.0 [1]
N-[3-[4-(3-Aminopropylamino)butylamino]propyl]-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamideIC50958.0 [1]
N-[3-[4-(3-Aminopropylamino)butylamino]propyl]phenothiazine-10-carboxamideIC50215.0 [1]
N-[4-[3-(4-Aminobutylamino)propylamino]butyl]phenothiazine-10-carboxamideIC5078.0 [1]
N-[4-[4-(4-Aminobutylamino)butylamino]butyl]phenothiazine-10-carboxamideIC50127.0 [1]
N-[3-[4-(3-Aminopropylamino)butylamino]propyl]carbazole-9-carboxamideIC50145.0 [1]
N-[4-[4-(4-Aminobutylamino)butylamino]butyl]carbazole-9-carboxamideIC50111.0 [1]
[(7-Nitro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)-(propylamino)methyl]phosphonic acid;hydrochlorideIC5090.0 [1]
Benzyl-[(benzylamino)-(7-nitro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphinic acid;hydrobromideIC5050.0 [1]
[(Benzylamino)-(7-nitro-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]-methylphosphinic acid;hydrobromideIC50200.0 [1]
[(Benzylamino)-(2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methyl]phosphonic acid;hydrobromideIC504.2 [1]
2-[3-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)propyl]-9H-pyrido[3,4-b]indol-2-ium;dibromideIC5024800.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-3-cyclohexyl-1-oxopropan-2-yl]cyclopropanecarboxamideIC502567.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-3-cyclohexyl-1-oxopropan-2-yl]cyclohexanecarboxamideIC50656.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-3-cyclohexyl-1-oxopropan-2-yl]-4-phenylbenzamideIC501446.0 [1]
(2S)-N-[3-[4-(3-Aminopropylamino)butylamino]propyl]-3-cyclohexyl-2-[(2-naphthalen-1-ylacetyl)amino]propanamideIC5047.0 [1]
(2S)-2-[[2-(1-Adamantyl)acetyl]amino]-N-[3-[4-(3-aminopropylamino)butylamino]propyl]-3-cyclohexylpropanamideIC50794.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-1-oxo-3-[(2-phenylacetyl)amino]propan-2-yl]cyclohexanecarboxamideIC502805.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-1-oxo-5-[(2-phenylacetyl)amino]pentan-2-yl]cyclohexanecarboxamideIC501026.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-3-cyclohexyl-1-oxopropan-2-yl]butanamideIC504383.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-1-oxo-4-[(2-phenylacetyl)amino]butan-2-yl]benzamideIC50106.0 [1]
N-[(2S)-1-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-1-oxo-6-[(2-phenylacetyl)amino]hexan-2-yl]benzamideIC501349.0 [1]
N,N'-Bis[5-[(2-methoxyphenyl)methylamino]pentyl]hexane-1,6-diamineIC50315.0 [1]
[(3R,5R,8S,9S,10S,13R,14S,17S)-10,13,17-Trimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl] hydrogen sulfateIC50600.0 [1]
2-Methyl-5-[6-(2-methylpyrido[4,3-b]indol-2-ium-5-yl)hexyl]pyrido[4,3-b]indol-2-iumIC5013800.0 [1]
2-Methyl-5-[7-(2-methylpyrido[4,3-b]indol-2-ium-5-yl)heptyl]pyrido[4,3-b]indol-2-iumIC503800.0 [1]
2-Methyl-5-[8-(2-methylpyrido[4,3-b]indol-2-ium-5-yl)octyl]pyrido[4,3-b]indol-2-iumIC50570.0 [1]
2-Methyl-5-[9-(2-methylpyrido[4,3-b]indol-2-ium-5-yl)nonyl]pyrido[4,3-b]indol-2-iumIC50400.0 [1]
8-Methoxy-5-[9-(8-methoxy-2-methylpyrido[4,3-b]indol-2-ium-5-yl)nonyl]-2-methylpyrido[4,3-b]indol-2-iumIC502400.0 [1]
2-Ethyl-5-[9-(2-ethylpyrido[4,3-b]indol-2-ium-5-yl)nonyl]pyrido[4,3-b]indol-2-iumIC50590.0 [1]
2-[5-[9-[2-(2-Hydroxyethyl)pyrido[4,3-b]indol-2-ium-5-yl]nonyl]pyrido[4,3-b]indol-2-ium-2-yl]ethanolIC50740.0 [1]
2-Propyl-5-[9-(2-propylpyrido[4,3-b]indol-2-ium-5-yl)nonyl]pyrido[4,3-b]indol-2-iumIC501000.0 [1]
2-[2-[2-[2-[2-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)ethoxy]ethoxy]ethoxy]ethyl]-9H-pyrido[3,4-b]indol-2-iumIC5060900.0 [1]
2-[5-(6-Hydroxy-9H-pyrido[3,4-b]indol-2-ium-2-yl)pentyl]-9H-pyrido[3,4-b]indol-2-ium-6-olIC5022700.0 [1]
6-Methoxy-2-[5-(6-methoxy-9H-pyrido[3,4-b]indol-2-ium-2-yl)pentyl]-9H-pyrido[3,4-b]indol-2-iumIC5029400.0 [1]
2-[5-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)pentyl]-9H-pyrido[3,4-b]indol-2-iumIC5020500.0 [1]
2-[6-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)hexyl]-9H-pyrido[3,4-b]indol-2-iumIC502200.0 [1]
2-[7-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)heptyl]-9H-pyrido[3,4-b]indol-2-iumIC506100.0 [1]
2-[9-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)nonyl]-9H-pyrido[3,4-b]indol-2-iumIC5013500.0 [1]
2-[10-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)decyl]-9H-pyrido[3,4-b]indol-2-iumIC509100.0 [1]
2-[11-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)undecyl]-9H-pyrido[3,4-b]indol-2-iumIC505100.0 [1]
2-[12-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)dodecyl]-9H-pyrido[3,4-b]indol-2-iumIC502600.0 [1]
2-[8-(9H-Pyrido[3,4-b]indol-2-ium-2-yl)octyl]-9H-pyrido[3,4-b]indol-2-iumIC503500.0 [1]
2-Methyl-9-[12-(2-methylpyrido[3,4-b]indol-2-ium-9-yl)dodecyl]pyrido[3,4-b]indol-2-iumIC504400.0 [1]
8-Methyl-2-[6-(8-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)hexyl]-1,3,4,5-tetrahydropyrido[4,3-b]indoleIC5011000.0 [1]
8-Methyl-2-[7-(8-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)heptyl]-1,3,4,5-tetrahydropyrido[4,3-b]indoleIC5012600.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Glutamate NMDA receptor; GRIN1/GRIN2A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/glutamate-nmda-receptor-grin1-grin2a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Glutamate NMDA receptor; GRIN1/GRIN2A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-nmda-receptor-grin1-grin2a-inhibitors-ic50-ki.
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