 | Genistein | Ki | 7000.0 [1] |
 | 2-[2-(4-Chlorophenyl)-3-[[4-(3-fluorobenzoyl)piperazin-1-yl]methyl]imidazo[1,2-a]pyridin-6-yl]benzonitrile | IC50 | 25.7 [1], 77.62 [2], 398.11 [3] |
 | Ethyl (3S,3aR,9E)-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]-1-(naphthalen-1-ylmethyl)-2-oxo-3,4,5,6,7,8-hexahydrocycloocta[b]pyrrole-3a-carboxylate | IC50 | 2000.0 [1], 10000.0 [2] |
 | Ethyl (3S,3aR,9E)-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]-1-(naphthalen-1-ylmethyl)-2-oxo-3,4,5,6,7,8-hexahydrocycloocta[b]pyrrole-3a-carboxylate | Ki | 1200.0 [1] |
 | 5-O-Tert-butyl 3a-O-ethyl (3S,3aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-3-[2-(naphthalen-1-ylmethylamino)-2-oxoethyl]-2-oxo-4,6-dihydro-3H-pyrrolo[3,2-c]pyridine-3a,5-dicarboxylate | IC50 | 1000.0 [1], 3000.0 [2] |
 | 5-O-Tert-butyl 3a-O-ethyl (3S,3aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-3-[2-(naphthalen-1-ylmethylamino)-2-oxoethyl]-2-oxo-4,6-dihydro-3H-pyrrolo[3,2-c]pyridine-3a,5-dicarboxylate | Ki | 800.0 [1] |
 | N-[[3-[2-(4-Fluorophenyl)ethoxy]phenyl]methyl]-2-(4-methoxyphenyl)-N-(pyridin-4-ylmethyl)acetamide | IC50 | 21800.0 [1], 100000.0 [2] |
 | 4-Methoxy-N-[[3-[(3-methoxyphenyl)methoxy]phenyl]methyl]-N-(pyridin-4-ylmethyl)benzamide | IC50 | 28500.0 [1], 100000.0 [2] |
 | Cycloheximide | IC50 | 228.0 [1] |
 | Cytidine | IC50 | 12000.0 [1] |
 | Kaempferol | IC50 | 4000.0 [1] |
 | Emetine | IC50 | 108.0 [1] |
 | Gossypol | Ki | 20000.0 [1] |
 | Phloretin | IC50 | 21400.0 [1] |
 | Anisomycin | IC50 | 321.0 [1] |
 | Imidocarb | IC50 | 12000.0 [1] |
 | Berbamine hydrochloride | IC50 | 12000.0 [1] |
 | Hesperadin | IC50 | 1434.0 [1] |
 | 6-(2,6-Dichlorophenyl)-2-[4-[2-(diethylamino)ethoxy]anilino]-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 9992.0 [1] |
 | Polysulfide rubber | IC50 | 12000.0 [1] |
 | N-(4-(4-Methyl-1-piperazinyl)phenyl)-9-acridinamine | IC50 | 5816.0 [1] |
 | CID 46830365 | IC50 | 10900.0 [1] |
 | 9-((3-Dimethylaminopropyl)amino)acridine | IC50 | 1558.0 [1] |
 | 6-(2,6-Dichlorophenyl)-8-methyl-2-(4-morpholin-4-ylanilino)pyrido[2,3-d]pyrimidin-7-one | IC50 | 5387.0 [1] |
 | N'-(7-Chloroquinolin-4-yl)-N,N-diethylethane-1,2-diamine | IC50 | 12000.0 [1] |
 | 5-Methyl-n-(naphthalen-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | IC50 | 12000.0 [1] |
 | 3-(4-Methylphenyl)-5H-indeno[1,2-c]pyridazin-5-one | IC50 | 12000.0 [1] |
 | 2-Amino-6,7-dimethoxy-N-phenylquinoline-3-carboxamide | IC50 | 12000.0 [1] |
 | 1,3-Bis(3,4-dichlorophenyl)urea | IC50 | 12000.0 [1] |
 | 9(2H)-Acridinone, 1,3,4,10-tetrahydro- | IC50 | 12000.0 [1] |
 | 1-(2,4-Dichlorophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid | IC50 | 12000.0 [1] |
 | 3-(4-Methoxyphenyl)-5H-indeno[1,2-c]pyridazin-5-one | IC50 | 12000.0 [1] |
 | 5-Chloro-2-hydroxy-N-[3-(trifluoromethyl)phenyl]benzamide | IC50 | 6594.0 [1] |
 | 2-(1,3-Benzodioxol-5-yl)-1,3-dimethyl-2,3-dihydro-1H-benzimidazole | IC50 | 12000.0 [1] |
 | N-[3-[[3-(1H-Benzimidazol-2-yl)phenyl]carbamoyl]phenyl]furan-2-carboxamide | IC50 | 12000.0 [1] |
 | Glucopiericidin A | IC50 | 4.9 [1] |
 | 1-(4-Ethoxyphenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-triazine-2,4-diamine | IC50 | 12000.0 [1] |
 | 8-Chloro-N-[3-(morpholin-4-yl)propyl]-5H-pyrimido[5,4-b]indol-4-amine | IC50 | 12000.0 [1] |
 | 7-Chloro-4-(1-pyrrolidinyl)quinoline | IC50 | 12000.0 [1] |
 | (3-Methyl-pyridin-2-yl)-(4-pyridin-2-yl-thiazol-2-yl)-amine | IC50 | 2254.0 [1] |
 | 2-[2-(3-Methoxy-phenylamino)-quinazolin-4-ylamino]-ethanol | IC50 | 12000.0 [1] |
 | Ethyl 6-methoxy-4-[4-(4-methylpiperazin-1-yl)anilino]quinoline-3-carboxylate | IC50 | 6745.0 [1] |
 | N-[4-(Trifluoromethyl)phenyl]-1,2,3-benzotriazin-4-amine | IC50 | 12000.0 [1] |
 | N-(3-Methoxyphenyl)-4-{[3-(4-methylpiperidin-1-yl)propyl]amino}-3-nitrobenzamide | IC50 | 2395.0 [1] |
 | 2-Bromo-N-(4-(pyridin-2-yl)thiazol-2-yl)benzamide | IC50 | 9858.0 [1] |
 | 4-[[4-(4-Methylpiperazin-1-yl)quinazolin-2-yl]amino]phenol;hydrochloride | IC50 | 12000.0 [1] |
 | 2-(Sec-butylamino)-1,1-bis(4-chlorophenyl)-1-ethanol | IC50 | 12000.0 [1] |
 | 4-(Pyridin-2-yl)-N-p-tolylthiazol-2-amine | IC50 | 12000.0 [1] |
 | Bisphenol C | IC50 | 12000.0 [1] |
 | N-[2-(4-Ethylpiperazin-1-yl)-4-methylquinolin-6-yl]-3,4-dimethoxybenzamide | IC50 | 12000.0 [1] |
 | N-[4-(4-Methylpiperazin-1-yl)-3-(trifluoromethyl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amine | IC50 | 580.0 [1] |
 | 3,4-Dimethoxy-N-(4-methyl-2-piperidin-1-ylquinolin-6-yl)benzamide | IC50 | 12000.0 [1] |
 | 2-(2-Methoxyanilino)-3-piperidin-1-ylnaphthalene-1,4-dione | IC50 | 12000.0 [1] |
 | 3-(3-(Trifluoromethyl)phenyl)-1,2,3-benzotriazin-4(3H)-imine | IC50 | 12000.0 [1] |
 | 3-(3,4-Dimethoxyphenyl)-N-[3-(dipropylamino)propyl]-1-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide | IC50 | 12000.0 [1] |
 | 2-[(4-Benzhydrylpiperazin-1-yl)methyl]phenol;oxalic acid | IC50 | 12000.0 [1] |
 | {4-[1-(1-Cyclohexyl-1H-tetrazol-5-yl)-butyl]-piperazin-1-yl}-furan-2-yl-methanone | IC50 | 12000.0 [1] |
 | 11-(3-Fluorophenyl)-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one | IC50 | 11560.0 [1] |
 | 1-(3-Bromophenyl)-2-[2-imino-3-(2-piperidin-1-ylethyl)benzimidazol-1-yl]ethanol;hydrochloride | IC50 | 12000.0 [1] |
 | N-[2-(1H-Indol-3-yl)ethyl]acridin-9-amine | IC50 | 6745.0 [1] |
 | 7-Amino-3-(3,4-dimethoxyphenyl)-2-methylpyrazolo[1,5-a]pyrimidine-6-carbonitrile | IC50 | 12000.0 [1] |
 | 2,7-Bis(4-Hydroxybutyl)benzo[lmn][3,8]phenanthroline-1,3,6,8(2H,7H)-tetrone | IC50 | 12000.0 [1] |
 | 2-(Butylamino)-1,1-bis(4-chlorophenyl)-1-ethanol | IC50 | 12000.0 [1] |
 | N-Cyclopropyl-5-[(4-methylphenyl)methylsulfanylmethyl]furan-2-carboxamide | IC50 | 12000.0 [1] |
 | 1,2-Ethanediamine, N,N-dimethyl-N'-(2-phenyl-4-quinolinyl)- | IC50 | 7118.0 [1] |
 | N-(4-Ethylphenyl)-2,5-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | IC50 | 12000.0 [1] |
 | N-(7-Chloroquinolin-4-yl)-N'-methylpropane-1,3-diamine | IC50 | 12000.0 [1] |
 | Ethyl 1-ethyl-6-fluoro-4-oxo-7-(piperidin-1-yl)-1,4-dihydroquinoline-3-carboxylate | IC50 | 12000.0 [1] |
 | 1-(4-Cyclopentylpiperazin-1-yl)-3-methylpyrido[1,2-a]benzimidazole-4-carbonitrile | IC50 | 12000.0 [1] |
 | (4,6-Dimethoxy-[1,3,5]triazin-2-yl)-(4-isopropyl-phenyl)-amine | IC50 | 12000.0 [1] |
 | N~2~-Benzyl-N~4~-(3-fluorophenyl)-6-methylpyrimidine-2,4-diamine | IC50 | 4398.0 [1] |
 | 7-Chloro-N-(4-ethoxyphenyl)quinolin-4-amine | IC50 | 12000.0 [1] |
 | N-[2-(3,4-Diethoxyphenyl)ethyl]thiophene-2-carboxamide | IC50 | 12000.0 [1] |
 | (4-(4-Chlorobenzo[d]thiazol-2-yl)piperazin-1-yl)(5-nitrofuran-2-yl)methanone | IC50 | 6853.0 [1] |
 | 2-Methyl-3-propylquinolin-4-ol | IC50 | 12000.0 [1] |
 | 1,4,8-Trimethyl-12-quinolino[2,3-b]quinolinamine | IC50 | 12000.0 [1] |
 | 2-Butyl-1-methyl-3-propyl-1H-quinolin-4-ylideneamine | IC50 | 9012.0 [1] |
 | 5-(4-Bromophenyl)-N-[4-(morpholin-4-ylmethyl)phenyl]furan-2-carboxamide | IC50 | 12000.0 [1] |
 | N~4~-Benzyl-N~2~-(4-methoxyphenyl)quinazoline-2,4-diamine | IC50 | 4477.0 [1] |
 | 6-Methyl-2-{3-methyl-5-[(4-methylphenyl)amino]-1H-pyrazol-1-yl}-1,4-dihydropyrimidin-4-one | IC50 | 15859.0 [1] |
 | Ethyl 4-benzyl-1-(2-hydroxy-3-methoxybenzyl)piperidine-4-carboxylate | IC50 | 12000.0 [1] |
 | 4-Octyl-2,3,5,6,7,8-hexahydro-1H-cyclopenta[b]quinolin-9-imine;hydrobromide | IC50 | 612.0 [1] |
 | CID 16192765 | IC50 | 604.0 [1] |
 | 2-((((3r,5r,7r)-Adamantan-1-ylmethyl)amino)methyl)phenol hydrochloride | IC50 | 12000.0 [1] |
 | 4-Ethyl-1,2,3,4,5,6,7,8-octahydro-cyclopenta[b]quinolin-9-ylideneamine | IC50 | 12000.0 [1] |
 | 1,3-Diamino-7-(1-ethylpropyl)-8-methyl-7H-pyrrolo(3,2-f)quinazoline | IC50 | 2022.0 [1] |
 | N-[2-(1,3-Benzodioxol-5-yl)-2-[4-(4-methoxyphenyl)piperazin-1-yl]ethyl]-3,3-dimethylbutanamide | IC50 | 12000.0 [1] |
 | 5-(2,5-Dichlorophenyl)-N-[4-(morpholin-4-ylmethyl)phenyl]furan-2-carboxamide | IC50 | 12000.0 [1] |
 | N-(5-Chloro-2,4-dimethoxyphenyl)-N-methyl-5,5-dioxo-4H-thieno[3,2-c]thiochromene-2-carboxamide | IC50 | 12000.0 [1] |
 | 2-(4-Chlorophenyl)-3-(4-methoxyphenyl)-6-methyl-1-morpholin-4-ylheptan-3-ol | IC50 | 12000.0 [1] |
 | 2-[2-Methoxyethyl-(2-thiophen-2-ylacetyl)amino]-N-[(4-methoxyphenyl)methyl]-2-(4-propan-2-ylphenyl)acetamide | IC50 | 12000.0 [1] |
 | 3-(2,4-Dioxo-1,4-dihydrothieno[3,2-d]pyrimidin-3(2H)-yl)-N-(2-methoxybenzyl)propanamide | IC50 | 12000.0 [1] |
 | N-Cyclohexyl-3-[(4-fluorobenzoyl)amino]-2-thiophenecarboxamide | IC50 | 12000.0 [1] |
 | N-Cyclohexyl-6-phenyl-3-(2-pyridinyl)-1,2,4-triazin-5-amine | IC50 | 2158.0 [1] |
 | 2-Hexyl-2-azatricyclo[7.3.0.03,7]dodeca-1(9),3(7)-dien-8-imine;hydrobromide | IC50 | 251.0 [1] |
 | Ethyl 4-(benzylamino)-6-methoxyquinoline-3-carboxylate | IC50 | 12000.0 [1] |
 | 2-Methyl-N-(2-(piperidin-1-yl)ethyl)benzo[h]quinolin-4-amine | IC50 | 12000.0 [1] |
 | [4-(4-Ethyl-1,3-benzothiazol-2-yl)piperazin-1-yl]-(5-nitrofuran-2-yl)methanone | IC50 | 3050.0 [1] |
 | (4-(4,5-Dimethylbenzo[d]thiazol-2-yl)piperazin-1-yl)(5-nitrofuran-2-yl)methanone | IC50 | 2960.0 [1] |
 | 3-Allyl-2-methylquinolin-4(1H)-one | IC50 | 12000.0 [1] |