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Glucokinase/Glucokinase regulatory protein Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-[6-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-methoxypyridin-3-yl]-1,1,1,3,3,3-hexafluoropropan-2-olIC504506.0 [1]
2-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)pyridine-3-carbonitrileIC50796.0 [1]
(2S)-4-[2-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)pyridin-3-yl]but-3-yn-2-olIC5042.0 [1]
4-[2-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)pyridin-3-yl]-2-methylbut-3-yn-2-olIC50211.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(methylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50140.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(ethylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50152.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(propan-2-ylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50288.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(cyclopropylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50238.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(cyclohexylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC5099.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-anilinopyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC507.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(benzylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50233.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-phenoxypyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC506021.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(pyridin-4-ylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC5015.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(pyridin-3-ylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC5038.0 [1]
2-[6-[6-(6-Aminopyridin-3-yl)sulfonyl-2-(pyridin-2-ylamino)pyridin-3-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50120.0 [1]
2-[2-[5-(6-Aminopyridin-3-yl)sulfonylthiophen-2-yl]pyrimidin-5-yl]-1,1,1-trifluoropropan-2-olIC50480.0 [1]
2-[4-[5-(6-Aminopyridin-3-yl)sulfonylthiophen-2-yl]phenyl]-1,1,1-trifluoropropan-2-olIC501930.0 [1]
2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]phenyl]-1,1,1,3,3,3-hexafluoropropan-2-olIC50534.0 [1]
2-[4-[4-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]phenyl]-1,1,1,3,3,3-hexafluoropropan-2-olIC5033000.0 [1]
2-[4-[4-(6-Aminopyridin-3-yl)sulfonyl-1-methylimidazol-2-yl]phenyl]-1,1,1,3,3,3-hexafluoropropan-2-olIC5033000.0 [1]
2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1-methylimidazol-2-yl]phenyl]-1,1,1-trifluoropropan-2-olIC5033000.0 [1]
2-[6-[5-(6-Aminopyridin-3-yl)sulfonylthiophen-2-yl]-5-chloropyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50129.0 [1]
2-[6-[5-(6-Aminopyridin-3-yl)sulfonylthiophen-2-yl]-5-prop-1-ynylpyridin-3-yl]-1,1,1-trifluoropropan-2-olIC5051.0 [1]
2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]-1,1,1-trifluoropropan-2-olIC5023.0 [1]
(2R)-2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]-1,1,1-trifluoropropan-2-olIC5037.0 [1]
(2S)-2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]-1,1,1-trifluoropropan-2-olIC5018.0 [1]
2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]propan-2-olIC5015.0 [1]
4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorobenzenesulfonamideIC50257.0 [1]
2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]propane-1,2-diolIC5010.0 [1]
(2R)-2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]propane-1,2-diolIC506.0 [1]
(2S)-2-[4-[5-(6-Aminopyridin-3-yl)sulfonyl-1,3-thiazol-2-yl]-3-chlorophenyl]propane-1,2-diolIC5061.0 [1]
2-(6-(4-((6-Amino-3-pyridinyl)sulfonyl)phenyl)-3-pyridinyl)-1,1,1,3,3,3-hexafluoro-2-propanolIC50358.0 [1]
2-(4-(4-((6-Amino-3-pyridinyl)sulfonyl)-1-piperazinyl)phenyl)-1,1,1-trifluoro-2-propanolIC50454.0 [1]
2-(4'-((6-Amino-3-pyridinyl)sulfonyl)-4-biphenylyl)-1,1,1-trifluoro-2-propanolIC501010.0 [1]
2-[6-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-chloropyridin-3-yl]-1,1,1,3,3,3-hexafluoropropan-2-olIC501885.0 [1]
2-[6-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-prop-1-ynylpyridin-3-yl]-1,1,1,3,3,3-hexafluoropropan-2-olIC5084.0 [1]
2-[6-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-(3-methoxyprop-1-ynyl)pyridin-3-yl]-1,1,1,3,3,3-hexafluoropropan-2-olIC5021.0 [1]
2-[6-[4-(6-Aminopyridin-3-yl)sulfonylphenyl]-5-(3-hydroxyprop-1-ynyl)pyridin-3-yl]-1,1,1,3,3,3-hexafluoropropan-2-olIC5065.0 [1]
2-[6-[5-(6-Aminopyridin-3-yl)sulfonylpyridin-2-yl]pyridin-3-yl]-1,1,1-trifluoropropan-2-olIC50434.0 [1]
2-(2-(4-((6-Amino-3-pyridinyl)sulfonyl)phenyl)-5-pyrimidinyl)-1,1,1,3,3,3-hexafluoro-2-propanolIC50104.0 [1]
Items per page: 1 - 10 of 40
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References

This online tool may be cited as follows

MLA

"Quest Database™ Glucokinase/Glucokinase regulatory protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/glucokinase-glucokinase-regulatory-protein-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Glucokinase/Glucokinase regulatory protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glucokinase-glucokinase-regulatory-protein-inhibitors-ic50-ki.
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