Gamma-glutamyltranspeptidase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Aspirin	IC50	36000.0 [1]
	N-[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]-4-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxybutanamide	IC50	3300.0 [1]
	(2S)-N-[3-[2-(3,4-Dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-2-(methanesulfonamido)-3-phenylpropanamide	IC50	31900.0 [1]
	(2S)-2-Acetamido-N-[3-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-3-(4-fluorophenyl)propanamide	IC50	26300.0 [1]
	(2S)-N-[3-[2-(3,4-Dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-3-(4-fluorophenyl)-2-(methanesulfonamido)propanamide	IC50	19700.0 [1]
	(2S)-2-Acetamido-N-[3-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-3-(4-methoxyphenyl)propanamide	IC50	34800.0 [1]
	(2S)-2-Acetamido-N-[3-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-3-phenylpropanamide	IC50	22900.0 [1]
	(2S)-N-[3-[2-(3,4-Dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-2-(methanesulfonamido)-3-(4-methoxyphenyl)propanamide	IC50	9900.0 [1]
	(2S)-N-[3-[2-(3,4-Dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-2-(methanesulfonamido)-3-pyridin-4-ylpropanamide	IC50	19000.0 [1]
	Tert-butyl N-[(2S)-1-[3-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropylamino]-3-(4-methoxyphenyl)-1-oxopropan-2-yl]carbamate	IC50	50000.0 [1]
	(2S)-2-Acetamido-N-[3-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-3-pyridin-3-ylpropanamide	IC50	50000.0 [1]
	(2S)-N-[3-[2-(3,4-Dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-2-(methanesulfonamido)-3-pyridin-3-ylpropanamide	IC50	50000.0 [1]
	(2S)-2-Acetamido-N-[3-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxypropyl]-3-pyridin-4-ylpropanamide	IC50	26900.0 [1]
	N-[(2S)-1-Amino-3-(4-methoxyphenyl)-1-oxopropan-2-yl]-4-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxybutanamide	IC50	3100.0 [1]
	N-[(2S)-1-Amino-3-(4-fluorophenyl)-1-oxopropan-2-yl]-4-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxybutanamide	IC50	2400.0 [1]
	N-[(2S)-1-Amino-1-oxo-3-pyridin-3-ylpropan-2-yl]-4-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxybutanamide	IC50	11600.0 [1]
	N-[(2S)-1-Amino-1-oxo-3-pyridin-4-ylpropan-2-yl]-4-[2-(3,4-dichlorophenyl)-4-(2-methylsulfanylethyl)-5-pyridin-3-ylpyrazol-3-yl]oxybutanamide	IC50	7800.0 [1]
	1-N,3-N,4-Trimethyl-2-phenyl-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	20000.0 [1]
	1-N,3-N,4-Trimethyl-2-(2-methylphenyl)-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	22000.0 [1]
	2-(4-Chlorophenyl)-1-N,3-N,4-trimethyl-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	35000.0 [1]
	1-N,3-N,4-Trimethyl-2-(4-nitrophenyl)-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	36000.0 [1]
	2-(4-Methoxyphenyl)-1-N,3-N,4-trimethyl-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	25000.0 [1]
	1-N,3-N,4-Trimethyl-2-(2-methylphenyl)-10H-phenothiazine-1,3-dicarboxamide	IC50	25000.0 [1]
	2-(4-Chlorophenyl)-1-N,3-N,4-trimethyl-10H-phenothiazine-1,3-dicarboxamide	IC50	20000.0 [1]
	2-(4-Methoxyphenyl)-1-N,3-N,4-trimethyl-10H-phenothiazine-1,3-dicarboxamide	IC50	21000.0 [1]
	1-N,3-N,4-Trimethyl-2-phenyl-10H-phenothiazine-1,3-dicarboxamide	IC50	20000.0 [1]
	2-(2-Chlorophenyl)-1-N,3-N,4-trimethyl-10H-phenothiazine-1,3-dicarboxamide	IC50	18000.0 [1]
	2-(2-Methoxyphenyl)-1-N,3-N,4-trimethyl-10H-phenothiazine-1,3-dicarboxamide	IC50	28000.0 [1]
	2-(2-Chlorophenyl)-1-N,3-N,4-trimethyl-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	19000.0 [1]
	2-(2-Methoxyphenyl)-1-N,3-N,4-trimethyl-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	30000.0 [1]
	2-(1,3-Benzodioxol-5-yl)-1-N,3-N,4-trimethyl-2,10-dihydro-1H-phenothiazine-1,3-dicarboxamide	IC50	30000.0 [1]
	3-Acetyl-2-(1,3-benzodioxol-5-yl)-N,4-dimethyl-10H-phenothiazine-1-carboxamide	IC50	18000.0 [1]
	3-Acetyl-N,4-dimethyl-2-(4-nitrophenyl)-10H-phenothiazine-1-carboxamide	IC50	22000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 33 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Gamma-glutamyltranspeptidase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/gamma-glutamyltranspeptidase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Gamma-glutamyltranspeptidase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gamma-glutamyltranspeptidase-1-inhibitors-ic50-ki.
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