![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_81661d366f997deb965803fe664d33ae.svg) | beta-Alanine | IC50 | 100000.0 [1], 209000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_3b2e1267f539475c4be5cce73d16727c.svg) | (S)-Snap 5114 | IC50 | 11900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_617b2d21d944db453a88b080bb0ecb89.svg) | Nipecotic acid | IC50 | 66000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_93514df6b1af1be3dbc80f2afaaffe22.svg) | Guvacine | IC50 | 66000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_ce543d9dd4ac190af2c0df148708156a.svg) | 1-[3-(9H-Carbazol-9-yl)propyl]-4-(2-methoxyphenyl)piperidin-4-ol | IC50 | 6200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_f1aef2d17d67a9ff6cf3d9275aa95c73.svg) | N-(1-Benzylpiperidin-4-yl)-2,4-dichlorobenzamide | Ki | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_e8251b94fa3f2e780d246eaf85d05072.svg) | N-(1-Benzylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_706ffcada7a7c5aaeb03a2f8c4a21d90.svg) | 2-Ethoxy-N-[1-(phenylmethyl)-4-piperidinyl]benzamide | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_80cadb7f2ce8258495cbd9fd0e3168b1.svg) | N-(1-Benzylpiperidin-4-yl)-2,3-dimethoxybenzamide | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_b8dbc59ca89a3d7778ba527532b42036.svg) | N-(1-Benzylpiperidine-4-yl)-2-naphthamide | Ki | 23000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_2abcc273fdc69eb067635205adf3325b.svg) | N-(1-Benzylpiperidin-4-yl)-4-fluorobenzamide | IC50 | 300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_67633a5ead9d76af4bdd96e03377ce91.svg) | CID 118711599 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_e1a97dfd1e2b3ca5b0a39fd1c9ca26b4.svg) | N-(1-Benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide | IC50 | 479000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_a6e4ff11d511dedef7e9d88dad948944.svg) | 2,4-Dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_000cda5f1e3af1ca4589a1a67fea1782.svg) | 2,4-Dichloro-N-[1-[(4-nitrophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_684f7e44cd92c36f4c32485f7246b936.svg) | 2,4-Dichloro-N-(1-phenacylpiperidin-4-yl)benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_86db192d08c4afc699a58491b98205c4.svg) | 2,4-Dichloro-N-[1-[(E)-3-phenylprop-2-enyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_d4b354a9d573270af5ae59f2f2a694bb.svg) | 2,4-Dichloro-N-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_a7642a62a99ec0e92844ccdad0de0875.svg) | 2,4-Dichloro-N-[1-[(4-iodophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_e605e6fe1589b4ae045a6dbab2390642.svg) | 2,4-Dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_f7626027ada922444c935ac2198af92c.svg) | Methyl 4-[[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]methyl]benzoate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_ea8dc82cd3905db788dd0a1fa88a2dc1.svg) | 2,4-Dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_8f4e08550de3792d3a6c5a42f0a20de3.svg) | 2,4-Dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_34326d8ad65a6f28879da289bd79145f.svg) | Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_e43a6528578f9528bdbcb03b9713889d.svg) | 2,4-Dichloro-N-(1-prop-2-ynylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_53ac528552cd24172839d51be9b810b1.svg) | 2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_a4b883447e5f5c42253b42fc1cfc283e.svg) | 2,4-Dichloro-N-[1-[(2-cyanophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_d75a4a0115727fab3a83b4a499332a38.svg) | 2,4-Dichloro-N-[1-[(2-nitrophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_bb5973db39c8b9268b3140773d5f12b9.svg) | 2,4-Dichloro-N-[1-[(4-cyanophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_586af14b8186c6d852228989577e7e15.svg) | 2,4-Dichloro-N-[1-(quinolin-2-ylmethyl)piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_6b57995e3d7c88b836bc3311ab556d3a.svg) | N-(1-Benzylpiperidin-4-yl)-2-methylpropanamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_d528db6bd84ff4945f10f4c1a6619acc.svg) | 2,4-Dichloro-N-(1-propylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_f78547cee860e8fabfa3022ac16fe7cb.svg) | 2,4-Dichloro-N-(1-ethylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_bdc67cffced46c5b38cbd53c3daed336.svg) | N-(1-Benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide | IC50 | 500000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_9347c611f243c2e2442bd866d4551baa.svg) | CID 43345728 | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_c9859040707bbdecc1071b160a34b78d.svg) | 2,4-Dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_cbfff684ee2ec11b94079a060657f854.svg) | (3R)-1-[(E)-4-(2-Fluorophenyl)-4-(2-methylphenyl)but-3-enyl]piperidine-3-carboxylic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_1eece05b4c84ffa7a153a8f4a3abbd4f.svg) | 2-[(1S,2S)-2-Aminocyclopropyl]acetic acid | IC50 | 36900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_889e33839e3bd8def9b5ce7c058bbc78.svg) | 2,4-Dichloro-N-(1-methylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_21030f65fe977febbf7bad2ab24ee0a0.svg) | 2-[(1S,2R)-2-Aminocyclopropyl]acetic acid;hydrochloride | IC50 | 36900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/gaba-transporter-2_a423b58ca59daab4d6e8c6b0655af299.svg) | N-(1-Benzyl-4-piperidinyl)-1,3-benzodioxole-5-carboxamide | Ki | 63000.0 [1] |