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GABA receptor alpha-3 subunit Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
Ethyl (7S)-15-methoxy-12-oxo-2,4,11-triazatetracyclo[11.4.0.02,6.07,11]heptadeca-1(17),3,5,13,15-pentaene-5-carboxylateKi25.0 [1]
L-838417Ki0.7 [1]
Ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi25.8 [1]
3-[3-Tert-butyl-2-[(2-methyl-1,2,4-triazol-3-yl)methoxy]pyrazolo[1,5-d][1,2,4]triazin-7-yl]-5-methyl-1,2-oxazoleKi0.8 [1]
CID 9971547Ki300.0 [1]
Tert-butyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi18.7 [1]
Ethyl 8-ethynyl-6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi96.0 [1]
CID 5255267Ki858.0 [1]
13-(4-Methyl-1,3-thiazol-2-yl)-15-pyridin-4-yl-4,11-diazatricyclo[9.4.0.02,7]pentadeca-1(15),2(7),3,5,13-pentaen-12-oneKi0.5 [1]
3-(8-Ethyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxypropyl 8-ethyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi8545.0 [1]
3-(8-Ethynyl-6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxypropyl 8-ethynyl-6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi272.0 [1]
5-(8-Ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxypentyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi2666.0 [1]
(8-Ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxymethoxymethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi1864.0 [1]
Tert-butyl 5-methyl-6-oxo-8-(2-trimethylsilylethynyl)-3a,4-dihydro-1H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylateKi255.0 [1]
Ethyl 7-ethynyl-4-methyl-5-oxoimidazo[1,5-a]quinazoline-3-carboxylateKi198.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ GABA receptor alpha-3 subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc.21 Dec2024https://www.aatbio.com/data-sets/gaba-receptor-alpha-3-subunit-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024December 21). Quest Database™ GABA receptor alpha-3 subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-receptor-alpha-3-subunit-inhibitors-ic50-ki.
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