GABA receptor alpha-3 subunit Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Ethyl (7S)-15-methoxy-12-oxo-2,4,11-triazatetracyclo[11.4.0.02,6.07,11]heptadeca-1(17),3,5,13,15-pentaene-5-carboxylate	Ki	25.0 [1]
	L-838417	Ki	0.7 [1]
	Ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	25.8 [1]
	3-[3-Tert-butyl-2-[(2-methyl-1,2,4-triazol-3-yl)methoxy]pyrazolo[1,5-d][1,2,4]triazin-7-yl]-5-methyl-1,2-oxazole	Ki	0.8 [1]
	CID 9971547	Ki	300.0 [1]
	Tert-butyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	18.7 [1]
	Ethyl 8-ethynyl-6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	96.0 [1]
	CID 5255267	Ki	858.0 [1]
	13-(4-Methyl-1,3-thiazol-2-yl)-15-pyridin-4-yl-4,11-diazatricyclo[9.4.0.02,7]pentadeca-1(15),2(7),3,5,13-pentaen-12-one	Ki	0.5 [1]
	3-(8-Ethyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxypropyl 8-ethyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	8545.0 [1]
	3-(8-Ethynyl-6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxypropyl 8-ethynyl-6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	272.0 [1]
	5-(8-Ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxypentyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	2666.0 [1]
	(8-Ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carbonyl)oxymethoxymethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	1864.0 [1]
	Tert-butyl 5-methyl-6-oxo-8-(2-trimethylsilylethynyl)-3a,4-dihydro-1H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	255.0 [1]
	Ethyl 7-ethynyl-4-methyl-5-oxoimidazo[1,5-a]quinazoline-3-carboxylate	Ki	198.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 15 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ GABA receptor alpha-3 subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/gaba-receptor-alpha-3-subunit-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 20). Quest Database™ GABA receptor alpha-3 subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-receptor-alpha-3-subunit-inhibitors-ic50-ki.
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