GABA A receptor alpha-6/beta-2/gamma-2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Ethyl-8-azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo-1,4-benzodiazepine-3-carboxylate	Ki	3.8 [1], 5.1 [2], 5.4 [3]
	Diazepam	Ki	7000.0 [1]
	Zolpidem	Ki	15000.0 [1]
	Eszopiclone	Ki	15000.0 [1]
	Panadiplon	Ki	603.0 [1]
	Ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	28.8 [1]
	Tert-butyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	5.1 [1]
	Tert-butyl 5-methyl-6-oxo-8-(2-trimethylsilylethynyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	58.6 [1]
	Ethyl 5-methyl-6-oxo-8-(2-trimethylsilylethynyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	113.7 [1]
	Tert-butyl 8-bromo-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	9.4 [1]
	Ethyl 8-ethyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	176.0 [1]
	CID 10519948	Ki	44.3 [1]
	Tert-butyl 8-ethyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	22.9 [1]
	Ethyl 5-methyl-6-oxo-8-(3-trimethylsilylprop-1-ynyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	300.0 [1]
	Ethyl 5-methyl-6-oxo-8-prop-1-ynyl-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate	Ki	100.0 [1]
	4,5-Dihydro-3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-acetylimidazo[1,5-a]quinoxaline	Ki	124.0 [1]
	Unii-82MI0GT75Z	Ki	10000.0 [1]
	4,5-Dihydro-3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-benzoylimidazo[1,5-a]quinoxaline	Ki	1140.0 [1]
	[3-(5-Cyclopropyl-1,2,4-oxadiazol-3-yl)-6-fluoro-4H-imidazo[1,5-a]quinoxalin-5-yl]-morpholin-4-ylmethanone	Ki	13.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 19 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ GABA A receptor alpha-6/beta-2/gamma-2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-6-beta-2-gamma-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ GABA A receptor alpha-6/beta-2/gamma-2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-a-receptor-alpha-6-beta-2-gamma-2-inhibitors-ic50-ki.
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