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G protein-coupled receptor kinase 6 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
3-Methyl-8-(3-morpholin-4-ylpropyliminomethyl)-5-propan-2-yl-2-[1,6,7-trihydroxy-3-methyl-8-(3-morpholin-4-ylpropyliminomethyl)-5-propan-2-ylnaphthalen-2-yl]naphthalene-1,6,7-triolIC5010120.0 [1], 16890.0 [2]
StaurosporineIC5034000.0 [1]
BaicaleinIC508700.0 [1]
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamideIC507000000.0 [1]
Bisindolylmaleimide IXIC50350000.0 [1]
ScutellareinIC506610.0 [1]
DoramapimodIC5030000.0 [1]
BalanolIC50490.0 [1]
PerimidineIC5012540.0 [1]
CID 11677079IC5030000.0 [1]
N-{4-[4-(4-Hydroxy-phenyl)-phthalazin-1-ylamino]-phenyl}-acetamideIC5060000.0 [1]
2,7-Diamino-4-(4-methylphenyl)-4H-chromene-3-carbonitrileIC5025960.0 [1]
3-Ethyl-1-(2-hydroxy-ethyl)-1-(6-oxo-5,6-dihydro-[1,3]dioxolo[4,5-g]quinolin-7-ylmethyl)-thioureaIC5060000.0 [1]
7,8-Dihydroxy-4-(4-methoxyphenyl)-2H-chromen-2-oneIC507160.0 [1]
5-(Diethylamino)-2-(2,3-dihydro-1H-perimidin-2-yl)phenolIC508440.0 [1]
4-(2,3-Dihydro-1H-benzo[f]cyclopenta[c]quinolin-4-yl)benzene-1,2-diolIC5028420.0 [1]
Ethyl 5-[2-oxo-2-(2,3,4-trihydroxyphenyl)ethyl]furan-2-carboxylateIC507050.0 [1]
3-Amino-5-(2-diethylamino-ethyl)-5H-pyrido[4,3-b]indole-4-carbonitrileIC5018750.0 [1]
2-Amino-1-butyl-1H-pyrrolo[2,3-b]quinoxaline-3-carbonitrileIC501560.0 [1]
2-[(5-Thiophen-2-yl-1H-1,2,4-triazol-3-yl)sulfanyl]acetic acidIC504600.0 [1]
7-((Pyridin-2-ylamino)(pyridin-3-yl)methyl)quinolin-8-olIC506750.0 [1]
N1-(4-(2-Methylimidazo[1,2-a]pyridin-3-yl)IC5060000.0 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-oneIC5010000.0 [1]
N-Benzyl-3-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methylamino]benzamideIC5030000.0 [1]
N-Benzyl-3-[(4-methyl-3-pyridin-4-yl-1H-pyrazol-5-yl)methylamino]benzamideIC5030000.0 [1]
3-(9-Oxa-3,4,6,12-tetrazatricyclo[8.4.0.02,6]tetradeca-1(10),2,4,11,13-pentaen-5-ylmethylamino)-N-[[2-(trifluoromethyl)phenyl]methyl]benzamideIC5030000.0 [1]
N-Benzyl-3-[(4-ethyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)methylamino]benzamideIC5030000.0 [1]
N-Methyl-3-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methylamino]benzamideIC5030000.0 [1]
Methyl 2-amino-1-hexyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylateIC501430.0 [1]
2,7-Diamino-4-(thiophen-2-yl)-4H-chromene-3-carbonitrileIC5011770.0 [1]
7-(((4-Ethoxyphenyl)amino)(pyridin-2-yl)methyl)quinolin-8-olIC504480.0 [1]
Pyridine, 3-(5-(p-methoxyphenyl)-2-oxazolyl)-IC5060000.0 [1]
1-[[5-(3-Methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propan-2-oneIC50100000.0 [1]
N,N-Dimethyl-2-[[5-(3-methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamideIC50100000.0 [1]
4-(Azepan-1-ylsulfonyl)-N-[2-(4-methylfuran-2-yl)phenyl]benzenesulfonamideIC5060000.0 [1]
(5Z)-5-(3,4-Dihydroxybenzylidene)-2-[(2,3-dimethylphenyl)amino]-1,3-thiazol-4(5H)-oneIC507110.0 [1]
4-[2-(5-Bromo-2-oxo-1,2-dihydro-3H-indol-3-yliden)hydrazino]-N~1~-(2-ethylhexyl)benzamideIC5060000.0 [1]
2-[[5-(2-Hydroxy-5-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC504550.0 [1]
2-[[5-(2-Hydroxy-5-methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC502710.0 [1]
2-[[5-(3-Formyl-2-hydroxy-5-methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5045300.0 [1]
3-[3-(Carboxymethylsulfanyl)-1H-1,2,4-triazol-5-yl]-4-hydroxybenzoic acidIC50100000.0 [1]
2-[[5-(4-Hydroxy-2,6-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50100000.0 [1]
2-[[5-(2-Hydroxy-6-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50100000.0 [1]
4-[5-(2-Phenylethylamino)-1,3,4-thiadiazol-2-yl]phenolIC5060000.0 [1]
2-[[5-(5-Bromo-2-hydroxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC501050.0 [1]
2-[[5-(3-Fluoro-4-hydroxy-5-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC503300.0 [1]
2-[[5-(2-Hydroxy-4-methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC506880.0 [1]
2-[[5-(2,4-Dihydroxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5011600.0 [1]
2-[[5-(4-Hydroxy-3-methoxy-5-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5015900.0 [1]
2-[[5-[4-(Diethylamino)-2-hydroxyphenyl]-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5025800.0 [1]
2-[[5-(2-Hydroxy-3-methoxy-5-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5034800.0 [1]
2-[[5-(3-Fluoro-4-hydroxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC507300.0 [1]
2-[[5-(2,5-Dihydroxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC506160.0 [1]
2-[[5-(4-Hydroxy-3-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC506800.0 [1]
2-[[5-(3-Fluoro-2-hydroxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC508750.0 [1]
2-[[5-(2-Hydroxy-4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5020900.0 [1]
N-(Furan-2-ylmethyl)-5-(4-phenylphenyl)-3,6-dihydro-1,3,4-thiadiazin-2-imineIC5010440.0 [1]
2-[[5-(2-Hydroxy-5-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5014100.0 [1]
2-[[5-(3,4-Dihydroxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC505020.0 [1]
2-[[5-(2-Hydroxy-3-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5070000.0 [1]
2-[[5-(4-Hydroxy-3,5-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC508830.0 [1]
5-(4-Chloro-3-nitrophenyl)-N-(furan-2-ylmethyl)-3,6-dihydro-1,3,4-thiadiazin-2-imineIC506620.0 [1]
(5E)-5-(4-Hydroxy-3-methoxybenzylidene)-3-(pyridin-3-yl)-2-thioxo-1,3-thiazolidin-4-oneIC5040620.0 [1]
4-(Azepan-1-ylsulfonyl)-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamideIC5060000.0 [1]
Methyl 2-amino-1-pentyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylateIC501030.0 [1]
4-[(3As,4R,9bR)-8-iodo-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-4-yl]benzoic acidIC506660.0 [1]
2-[[5-(3-Methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC501440.0 [1]
2-[[5-(4-Methyl-3-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50751.0 [1]
2-[[5-(3-Fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC504700.0 [1]
4,4'-{[4-(Diethylamino)phenyl]methanediyl}bis(3-methyl-1H-pyrazol-5-ol)IC509930.0 [1]
Acetic acid, ((5-(3,4,5-trimethoxyphenyl)-1H-1,2,4-triazol-3-yl)thio)-IC508230.0 [1]
1,4-Diamino-9,10-dioxoanthracene-2-carboxamideIC5012650.0 [1]
2,7-Diamino-4-(6-chloro-[1,3]dioxolo[4,5-g]quinolin-7-yl)-4H-chromene-3-carbonitrileIC506480.0 [1]
7-{[(5-Methyl-1,2-oxazol-3-yl)amino](pyridin-2-yl)methyl}quinolin-8-olIC506450.0 [1]
7-{[(4-Methoxyphenyl)amino](pyridin-2-yl)methyl}quinolin-8-olIC5010260.0 [1]
N-(6-Methyl-1,3-benzothiazol-2-yl)formamideIC5060000.0 [1]
4-Amino-5-N-[2-(2-methoxyethylamino)-2-oxoethyl]-5-N-phenyl-1,2-thiazole-3,5-dicarboxamideIC5060000.0 [1]
{[5-(3-Methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acidIC505850.0 [1]
2-[[5-[3-(Trifluoromethyl)phenyl]-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC503020.0 [1]
2-[[5-(3-Nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC501400.0 [1]
2-[[5-[4-(Dimethylamino)phenyl]-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50100000.0 [1]
2-[[5-(2,3-Dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50100000.0 [1]
2-[[5-(3,4-Difluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC503360.0 [1]
2-[[5-(4-Methoxy-3-nitrophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC501050.0 [1]
2-[[5-(3-Cyanophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC502310.0 [1]
2-[[5-(3,5-Dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC506100.0 [1]
2-[[5-(3-Methylsulfonylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC506360.0 [1]
2-[[5-(2,6-Dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50100000.0 [1]
2-[[4-Methyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoic acidIC50100000.0 [1]
(4S,12Ar)-4,7-bis(dimethylamino)-1,10,11,12a-tetrahydroxy-3,12-dioxo-4a,5,5a,6-tetrahydro-4H-tetracene-2-carboxamideIC501370.0 [1]
2-[[5-(2,3-Difluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5010700.0 [1]
2-[[5-(2,5-Dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC50100000.0 [1]
2-[[5-[4-(Trifluoromethoxy)phenyl]-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC505920.0 [1]
Methyl 2-amino-1-(prop-2-en-1-yl)-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylateIC50973.0 [1]
Ethyl 2-amino-1-cyclopropyl-1H-pyrrolo(2,3-B)quinoxaline-3-carboxylateIC502830.0 [1]
6-(3,4-Dihydroxy-phenyl)-8-ethoxy-1,3-dimethyl-cyclohepta[c]furan-4-oneIC504410.0 [1]
2-[[5-(3-Piperidin-1-ylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetic acidIC5051800.0 [1]
3-[3-(Carboxymethylsulfanyl)-1H-1,2,4-triazol-5-yl]-4-fluorobenzoic acidIC5081700.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ G protein-coupled receptor kinase 6 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/g-protein-coupled-receptor-kinase-6-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ G protein-coupled receptor kinase 6 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/g-protein-coupled-receptor-kinase-6-inhibitors-ic50-ki.
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