![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_0ccfbdb7949682b5c076b91dfa58d29f.svg) | Ramatroban | IC50 | 28.0 [1], 29.0 [2], 169.0 [3], 461.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_0ccfbdb7949682b5c076b91dfa58d29f.svg) | Ramatroban | Ki | 4.3 [1], 290.0 [2], 340.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_7f90212ca8691232ca4fae2f43101f78.svg) | Nvp-qav680 | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_7f90212ca8691232ca4fae2f43101f78.svg) | Nvp-qav680 | Ki | 29.0 [1], 36.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_db82db5a868b600f41cbf41bb039e06d.svg) | MK-7246 | IC50 | 2.2 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_db82db5a868b600f41cbf41bb039e06d.svg) | MK-7246 | Ki | 2.5 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_a2ee89f5b9df63e6e9252a355dfe5fbd.svg) | 2-[3-[[2-(Benzenesulfonyl)phenyl]methyl]-2-methyl-4-oxo-6,7-dihydro-5H-pyrrolo[3,2-c]pyridin-1-yl]acetic acid | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_230afff0a01f7d70042640f7d82fe383.svg) | 2-(1-(3,4-Difluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | IC50 | 9.0 [1], 60.0 [2], 150.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_230afff0a01f7d70042640f7d82fe383.svg) | 2-(1-(3,4-Difluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | Ki | 31.0 [1], 33.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_00e3c01e14439ab09f82499d0730f244.svg) | 2-(2-Benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid | IC50 | 110.0 [1], 170.0 [2], 190.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_d7ee970807058c97259ca7da2362b816.svg) | Fevipiprant | IC50 | 1.4 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_d7ee970807058c97259ca7da2362b816.svg) | Fevipiprant | Ki | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_68c8109e931ed886c392cff9314d7ece.svg) | 2-(5-Fluoro-2-methyl-3-(quinolin-2-ylmethyl)-1H-indol-1-yl)acetic acid | IC50 | 19.0 [1], 28.0 [2], 35.0 [3], 100.0 [4], 130.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_68c8109e931ed886c392cff9314d7ece.svg) | 2-(5-Fluoro-2-methyl-3-(quinolin-2-ylmethyl)-1H-indol-1-yl)acetic acid | Ki | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_c61a95f397b5ad881f39dc013a3df222.svg) | Amg-009 | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_96ebf23979f9914c63b4670633763911.svg) | [5-Fluoro-1-(4-methanesulfonyl-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid | IC50 | 67.0 [1], 74.0 [2], 106.0 [3], 158.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_96ebf23979f9914c63b4670633763911.svg) | [5-Fluoro-1-(4-methanesulfonyl-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid | Ki | 68.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_717455ea21aea29c266632270650797a.svg) | 2-[2-Benzoyl-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 50.0 [1], 130.0 [2], 160.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_2773f4bdb605ab3fea1c5489433eca89.svg) | 2-(1-(3-Cyano-4-fluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | IC50 | 8.0 [1], 40.0 [2], 101.0 [3], 168.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_2773f4bdb605ab3fea1c5489433eca89.svg) | 2-(1-(3-Cyano-4-fluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | Ki | 36.0 [1], 37.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_adec659617a828b7d72c3b61f653d432.svg) | [1-(4-Fluoro-3-methoxy-benzenesulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | IC50 | 18.0 [1], 91.0 [2], 156.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_adec659617a828b7d72c3b61f653d432.svg) | [1-(4-Fluoro-3-methoxy-benzenesulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | Ki | 56.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_4802b18c66258ab891ad340ab765f1a3.svg) | 2-(1-(4-Chloro-3-cyanophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | IC50 | 6.0 [1], 41.0 [2], 56.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_4802b18c66258ab891ad340ab765f1a3.svg) | 2-(1-(4-Chloro-3-cyanophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | Ki | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_8ee001d6cc11856ad1101dea6db0208f.svg) | {4-Chloro-2-[(3-chlorophenyl)ethynyl]phenoxy}acetic acid | IC50 | 29.0 [1], 104.0 [2], 114.0 [3], 1200.0 [4], 6900.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_8ee001d6cc11856ad1101dea6db0208f.svg) | {4-Chloro-2-[(3-chlorophenyl)ethynyl]phenoxy}acetic acid | Ki | 29.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1726fb62075414b31f6badae81f4cc0b.svg) | Setipiprant | IC50 | 6.0 [1], 30.0 [2], 80.0 [3], 235.0 [4], 340.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e3ce6611855e9f67908169aea6525094.svg) | AM-156 free acid | IC50 | 6.5 [1], 13.0 [2], 14.0 [3], 16.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e3ce6611855e9f67908169aea6525094.svg) | AM-156 free acid | Ki | 13.5 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_d38de8837806400f6d87cd71d29214db.svg) | 2-(4-Chloro-2-cycloheptylphenoxy)acetic acid | IC50 | 148.0 [1], 248.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_d38de8837806400f6d87cd71d29214db.svg) | 2-(4-Chloro-2-cycloheptylphenoxy)acetic acid | Ki | 59.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_917cd3b3382403539276a2062075d1a5.svg) | 2-(1-(4-Chlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | IC50 | 108.0 [1], 565.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_917cd3b3382403539276a2062075d1a5.svg) | 2-(1-(4-Chlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | Ki | 103.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1739350a9d2d7441e7b77456f885c7a7.svg) | 2-[1-[4-[(3,4-Dichlorobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid | IC50 | 13.0 [1], 19.0 [2], 23.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_a226fe9cacbc2869e82ce280cef7a834.svg) | 2-[4-[[2-(Benzenesulfonyl)phenyl]methyl]-5-methyl-3-phenylpyrazol-1-yl]acetic acid | IC50 | 40.0 [1], 50.0 [2], 85.0 [3], 240.0 [4], 520.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_96a09f23739a00eb8b22c8ddac09bc1c.svg) | 2-[2-(3-Chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 9.0 [1], 40.0 [2], 60.0 [3], 95.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_0e28f5466535639a173121ca50b0971d.svg) | 2-[2-[4-(4-Ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 4.0 [1], 7.0 [2], 190.0 [3], 240.0 [4], 320.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_91e9b943cd05ea29048f0f88b27257da.svg) | [1-(4-Methanesulfonyl-3-trifluoromethyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | IC50 | 4.0 [1], 11.0 [2], 40.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_91e9b943cd05ea29048f0f88b27257da.svg) | [1-(4-Methanesulfonyl-3-trifluoromethyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | Ki | 22.0 [1], 31.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_5bf2d0e15b6ca3033e3c7742851e20b8.svg) | 2-[2-(3-Chlorobenzoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 10.0 [1], 30.0 [2], 40.0 [3], 50.0 [4], 70.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_d517ac9e5b89536996cbf398d26589bf.svg) | [1-(2-Chloro-4-methanesulfonyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | IC50 | 1.7 [1], 14.0 [2], 47.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_d517ac9e5b89536996cbf398d26589bf.svg) | [1-(2-Chloro-4-methanesulfonyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | Ki | 3.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_f3987e82e81290fae256397508b6f83c.svg) | 2-[8-Fluoro-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 4.0 [1], 12.0 [2], 34.0 [3], 40.0 [4], 70.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_13bab1227d167d07b81fdb61ab02d03f.svg) | [2-(Naphthalene-1-carbonyl)-1,2,3,4-tetrahydro-pyrido[4,3-b]indol-5-yl]-acetic acid | IC50 | 9.0 [1], 30.0 [2], 140.0 [3], 420.0 [4], 1120.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_f82aa84d4718d29e5c311c5eb9623b84.svg) | [1-(4-Ethanesulfonyl-2-trifluoromethyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | IC50 | 0.8 [1], 4.0 [2], 22.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_f82aa84d4718d29e5c311c5eb9623b84.svg) | [1-(4-Ethanesulfonyl-2-trifluoromethyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | Ki | 7.0 [1], 8.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_32aae38c3aeec0fa123890cd21984369.svg) | [1-(2-Chloro-4-ethanesulfonyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | IC50 | 1.3 [1], 7.0 [2], 16.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_32aae38c3aeec0fa123890cd21984369.svg) | [1-(2-Chloro-4-ethanesulfonyl-benzyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | Ki | 6.0 [1], 7.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_77851834016d7034c5ee1c6586c8ca32.svg) | 2-(1-(4-Cyano-3-ethoxyphenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | IC50 | 5.0 [1], 31.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_77851834016d7034c5ee1c6586c8ca32.svg) | 2-(1-(4-Cyano-3-ethoxyphenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | Ki | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e2b53f13305e67ddae1a41c05a613f7a.svg) | [2-Methyl-1-(4-nitro-benzyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | IC50 | 24.0 [1], 143.0 [2], 144.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e2b53f13305e67ddae1a41c05a613f7a.svg) | [2-Methyl-1-(4-nitro-benzyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-acetic acid | Ki | 147.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1c5343431b9c913e0b1e829ed52479bf.svg) | 2-[2-Methyl-1-[(2-methyl-4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid | IC50 | 4.0 [1], 26.0 [2], 32.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1c5343431b9c913e0b1e829ed52479bf.svg) | 2-[2-Methyl-1-[(2-methyl-4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid | Ki | 31.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_200b139cb1771efb7af132e4a8c633c9.svg) | 2-[8-Fluoro-2-(2-naphthalen-1-ylacetyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 4.0 [1], 70.0 [2], 160.0 [3], 180.0 [4], 275.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_b1fb8cfc258a501d538574b9b5f90c19.svg) | 2-[8-Chloro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 4.0 [1], 30.0 [2], 65.0 [3], 100.0 [4], 110.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_ad7e04a3317d10c942521743f3345fe9.svg) | 2-[2-(Naphthalene-1-carbonyl)-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 11.0 [1], 20.0 [2], 70.0 [3], 180.0 [4], 380.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_c83b5cfc3171b970f9699f28bf844ebf.svg) | 2-[8-Fluoro-2-[2-(1H-indol-3-yl)acetyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 5.0 [1], 15.0 [2], 35.0 [3], 40.0 [4], 50.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_a29e4087daaa697fbf97a15a0d833f2d.svg) | 2-[8-Fluoro-2-(3-naphthalen-1-ylpropanoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid | IC50 | 10.0 [1], 30.0 [2], 65.0 [3], 160.0 [4], 210.0 [5] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_72ea362236a06ea655539d5c59aa3212.svg) | 2-[1-[[2,4-Bis(trifluoromethyl)phenyl]methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid | IC50 | 14.0 [1], 64.0 [2], 214.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_72ea362236a06ea655539d5c59aa3212.svg) | 2-[1-[[2,4-Bis(trifluoromethyl)phenyl]methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid | Ki | 29.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_4e580f477286fcc416c29dd8fbd694de.svg) | Fentiazac | IC50 | 550.0 [1], 960.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_a574090a3670262d315c9b04d5574485.svg) | 5-Thiazoleacetic acid, 4-(4-chlorophenyl)-2-(phenylamino)- | IC50 | 100.0 [1], 1300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_9d87b59319d568b327f6d8aaa63c861f.svg) | [3-(2-Benzenesulfonylbenzyl)-5-fluoro-2-methylindol-1-yl]acetic acid | IC50 | 5.0 [1], 14.0 [2], 16.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_59f791f2b3efc80640b14e5bf0af9291.svg) | 2-[5-Chloro-1'-[(3-methyl-5-phenyl-1,2-oxazol-4-yl)methyl]-2,2'-dioxospiro[indole-3,4'-pyrrolidine]-1-yl]acetic acid | IC50 | 0.23 [1], 19.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_59f791f2b3efc80640b14e5bf0af9291.svg) | 2-[5-Chloro-1'-[(3-methyl-5-phenyl-1,2-oxazol-4-yl)methyl]-2,2'-dioxospiro[indole-3,4'-pyrrolidine]-1-yl]acetic acid | Ki | 3.8 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_3a07314da20a7f91961e1c25c49a10fd.svg) | 2-[(3S)-5-Chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-2,2'-dioxospiro[indole-3,4'-pyrrolidine]-1-yl]acetic acid | IC50 | 62.0 [1], 1800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_3a07314da20a7f91961e1c25c49a10fd.svg) | 2-[(3S)-5-Chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-2,2'-dioxospiro[indole-3,4'-pyrrolidine]-1-yl]acetic acid | Ki | 13.0 [1], 683.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_b0ba3a44743bf6f15512f8ff17a14ed9.svg) | 2-[(3R)-3-[(4-Fluorophenyl)sulfonyl-methylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]acetic acid | IC50 | 1.2 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_b0ba3a44743bf6f15512f8ff17a14ed9.svg) | 2-[(3R)-3-[(4-Fluorophenyl)sulfonyl-methylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]acetic acid | Ki | 0.6 [1], 1.5 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_fa75e652e93b6fce45922f2e8b509bd5.svg) | 2-(2-(Biphenyl-2-ylmethyl)-4-(4-chlorophenyl)thiazol-5-yl)acetic acid | IC50 | 41.0 [1], 510.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e5412596e4d0a821211cb871e8a700d5.svg) | 2-(2-Benzyl-4-(4-chlorophenyl)thiazol-5-yl)acetic acid | IC50 | 180.0 [1], 4100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_ae8d2e572abe5f258c834cd2ae4ae2aa.svg) | 2-(4-(4-Chlorophenyl)-2-(4-phenoxyphenyl)thiazol-5-yl)acetic acid | IC50 | 93.0 [1], 1300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_b49b281a399bc0753e92ba85f4769a5a.svg) | 2-[4-Chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid | IC50 | 7.0 [1], 32.0 [2], 81.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_b49b281a399bc0753e92ba85f4769a5a.svg) | 2-[4-Chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_57007f1d8b6301db6b19d26e31cecf52.svg) | 4-(N-[(2S,4R)-1-Benzoyl-2-methyl-3,4-dihydro-2H-quinolin-4-yl]anilino)-4-oxobutanoic acid | IC50 | 0.77 [1], 3.0 [2], 130.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_dd87a7186226dd8de27adf4d486ec77a.svg) | 2-[3-[[1-[(2,4-Difluorophenyl)methyl]-6-oxopyridazin-3-yl]methyl]-5-fluoro-2-methylindol-1-yl]acetic acid | IC50 | 0.8 [1], 1.2 [2], 2.0 [3], 3.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1314623ee7bf97d97176c877e120eea7.svg) | 2-[4-Chloro-2-[2-(2-fluoro-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid | IC50 | 8.0 [1], 23.0 [2], 28.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1314623ee7bf97d97176c877e120eea7.svg) | 2-[4-Chloro-2-[2-(2-fluoro-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid | Ki | 3.4 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_f0a1db222f2d694cc187793b4a650b0e.svg) | 2-[1-[4-[(3,4-Dichlorophenyl)methoxy]benzoyl]isoquinolin-4-yl]acetic acid | IC50 | 38.0 [1], 180.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_500b77a06b6a37ad171bc955f50442ef.svg) | 2-[1-[4-[[(E)-3-(3,4-Dichlorophenyl)prop-2-enoyl]amino]benzoyl]isoquinolin-4-yl]acetic acid | IC50 | 4.0 [1], 17.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_370f32f90d8f9a3f2dc89d5667b74555.svg) | 2-[1-(4-Benzamidobenzoyl)isoquinolin-4-yl]acetic acid | IC50 | 7.9 [1], 42.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_0d2b455d17afbf3dc109a5ca9154708e.svg) | 2-[1-[4-[[4-(Trifluoromethyl)benzoyl]amino]benzoyl]isoquinolin-4-yl]acetic acid | IC50 | 4.9 [1], 15.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_1b18e946c8d96224ad5d9d413fcefb62.svg) | 2-[1-[4-(Pyrimidine-2-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid | IC50 | 290.0 [1], 550.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_211819ac596c63f9b8dad3a1f2bfd0d0.svg) | 2-[1-[2-[[Cyclopropanecarbonyl(ethyl)amino]methyl]-4-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid | IC50 | 9.0 [1], 20.0 [2], 34.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_665b68a7f082c78ac4fbbaec560ccd5b.svg) | 2-[8-[2-[[Cyclopropanecarbonyl(ethyl)amino]methyl]-4-(trifluoromethyl)phenyl]pyrrolo[1,2-a]pyrimidin-6-yl]acetic acid | IC50 | 1.4 [1], 13.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_ac5fb51f1637d6db9f589cfbe73572fe.svg) | 2-[3-[2-[[Cyclopropanecarbonyl(ethyl)amino]methyl]-4-(trifluoromethyl)phenyl]pyrrolo[3,2-b]pyridin-1-yl]acetic acid | IC50 | 14.0 [1], 15.0 [2], 20.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_11864a4fa2c02dbcb2c58d79e72a65b3.svg) | 2-[3-[2-[[Cyclopropanecarbonyl(ethyl)amino]methyl]-4-(trifluoromethyl)phenyl]indazol-1-yl]acetic acid | IC50 | 19.0 [1], 47.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_0eefae632f99c63fb675adab905a859b.svg) | 2-[1-[2-[[Cyclopropanecarbonyl(ethyl)amino]methyl]-4-(trifluoromethyl)phenyl]indol-3-yl]acetic acid | IC50 | 37.0 [1], 84.0 [2] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_7d7c721b2c807e40f2d40ec35ad8580b.svg) | 2-[3-[(E)-2-Cyano-3-(3,4-dihydro-2H-quinolin-1-yl)-3-oxoprop-1-enyl]indol-1-yl]acetic acid | IC50 | 10.0 [1], 14.0 [2], 54.0 [3], 160.0 [4] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e1fb94224112958dc79231fd105da219.svg) | 2-(1-(3,4-Dichlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | IC50 | 112.0 [1], 354.0 [2], 629.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_e1fb94224112958dc79231fd105da219.svg) | 2-(1-(3,4-Dichlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid | Ki | 52.0 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_ece94e696adcd4b5cc94dd93bdd7e34d.svg) | 2-[[(2As,8R,8aR)-3-(3-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylcarbamoyl]oxyacetic acid | IC50 | 0.8 [1], 1.1 [2], 13.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_ece94e696adcd4b5cc94dd93bdd7e34d.svg) | 2-[[(2As,8R,8aR)-3-(3-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylcarbamoyl]oxyacetic acid | Ki | 4.1 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_8cd77d29e87e5f53bc909ff4704afb81.svg) | 4-[[(2As,8R,8aR)-3-(4-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylamino]-4-oxobutanoic acid | IC50 | 8.9 [1], 12.0 [2], 20.0 [3] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_8cd77d29e87e5f53bc909ff4704afb81.svg) | 4-[[(2As,8R,8aR)-3-(4-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylamino]-4-oxobutanoic acid | Ki | 7.3 [1] |
![](https://images.aatbio.com/dataset/ic50/g-protein-coupled-receptor-44_9531eabe43dba481f8f19246fdf9928e.svg) | 2-[[(2As,8R,8aR)-3-(4-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylcarbamoyl]oxyacetic acid | IC50 | 1.4 [1], 2.0 [2], 3.6 [3] |