 | Acetic acid | IC50 | 120000.0 [1] |
 | Propionic acid | IC50 | 130000.0 [1] |
 | CID 57520598 | IC50 | 9.0 [1] |
 | 2-(4-Chlorophenyl)-3-methyl-N-(thiazol-2-yl)butanamide | IC50 | 800.0 [1] |
 | 2-(4-Chlorophenyl)-3-methylbutanoic acid | IC50 | 100000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(thiazol-2-yl)butanamide | IC50 | 700.0 [1] |
 | (S)-4-Cmtb | IC50 | 500.0 [1] |
 | 4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide | IC50 | 39810.72 [1] |
 | (3R)-3-Benzyl-4-[cyclopropyl-[4-(2,5-dichlorophenyl)-1,3-thiazol-2-yl]amino]-4-oxobutanoic acid | Ki | 199.53 [1] |
 | (3R)-3-[Cyclopropyl-[4-[2-(6-methoxypyridin-3-yl)phenyl]-1,3-thiazol-2-yl]carbamoyl]-5-methylhexanoic acid | Ki | 251.19 [1] |
 | (3R)-3-[Cyclopropyl-[4-[2-(6-pyrazol-1-ylpyridin-3-yl)phenyl]-1,3-thiazol-2-yl]carbamoyl]-5-methylhexanoic acid | Ki | 158.49 [1] |
 | (3R)-3-(Cyclopentylmethyl)-4-[cyclopropyl-[4-[2-(6-pyrazol-1-ylpyridin-3-yl)phenyl]-1,3-thiazol-2-yl]amino]-4-oxobutanoic acid | Ki | 63.1 [1] |
 | N-[(4-Chlorophenyl)methyl]-1-[2-(3,5-dimethylphenyl)acetyl]-2-methylazetidine-2-carboxamide | IC50 | 10000.0 [1] |
 | N-[(4-Chlorophenyl)methyl]-1-[2-(3,5-dimethylphenyl)acetyl]-2-methyl-N-[2-(methylcarbamoylamino)ethyl]azetidine-2-carboxamide | IC50 | 10000.0 [1] |
 | N-(2-Acetamidoethyl)-1-[2-(1-benzothiophen-3-yl)acetyl]-N-[(4-chlorophenyl)methyl]-2-methylazetidine-2-carboxamide | IC50 | 337.0 [1] |
 | N-[(4-Chlorophenyl)methyl]-N,2-dimethyl-1-[2-(3-thiophen-3-ylphenyl)acetyl]azetidine-2-carboxamide | IC50 | 5800.0 [1] |
 | N-[(4-Chlorophenyl)methyl]-N,2-dimethyl-1-(naphthalene-1-carbonyl)azetidine-2-carboxamide | IC50 | 3350.0 [1] |
 | 1-(5-Chloro-4-methoxythiophene-3-carbonyl)-N-[(4-chlorophenyl)methyl]-N,2-dimethylazetidine-2-carboxamide | IC50 | 3350.0 [1] |
 | N-[(4-Chlorophenyl)methyl]-1-(2-imidazo[1,2-a]pyridin-3-ylacetyl)-N,2-dimethylazetidine-2-carboxamide | IC50 | 10000.0 [1] |
 | 1-(1-Benzofuran-3-carbonyl)-N-[(4-chlorophenyl)methyl]-N,2-dimethylazetidine-2-carboxamide | IC50 | 10000.0 [1] |
 | 1-[2-(1-Benzothiophen-7-yl)acetyl]-N-[(4-chlorophenyl)methyl]-N,2-dimethylazetidine-2-carboxamide | IC50 | 10000.0 [1] |
 | 1-(1-Benzothiophene-2-carbonyl)-N-[(4-chlorophenyl)methyl]-N,2-dimethylazetidine-2-carboxamide | IC50 | 10000.0 [1] |
 | 1-(5-Chloro-1-benzothiophene-3-carbonyl)-N-[(4-chlorophenyl)methyl]-N,2-dimethylazetidine-2-carboxamide | IC50 | 3350.0 [1] |
 | 1-[3-(1-Benzothiophen-3-yl)propanoyl]-N-[(4-chlorophenyl)methyl]-N,2-dimethylazetidine-2-carboxamide | IC50 | 20000.0 [1] |
 | 2-[[1-[2-(Benzimidazol-1-yl)acetyl]-2-methylazetidine-2-carbonyl]-[(4-chlorophenyl)methyl]amino]acetic acid | IC50 | 10000.0 [1] |
 | 4-[[1-(1-Benzothiophene-3-carbonyl)-2-methylazetidine-2-carbonyl]-methylamino]butanoic acid | IC50 | 10000.0 [1] |
 | 4-[[1-(1-Benzothiophene-3-carbonyl)-2-methylazetidine-2-carbonyl]-butylamino]butanoic acid | IC50 | 10000.0 [1] |
 | 4-[[1-(1-Benzothiophene-3-carbonyl)-2-methylazetidine-2-carbonyl]-cyclohexylamino]butanoic acid | IC50 | 10000.0 [1] |
 | 4-[[1-[2-(1-Benzofuran-3-yl)acetyl]-2-methylazetidine-2-carbonyl]-[(3-chlorophenyl)methyl]amino]butanoic acid | IC50 | 10000.0 [1] |
 | 2-(4-Chlorophenyl)-3-methylbutanamide | IC50 | 100000.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3-methyl-N-(4-oxo-1,3-thiazolidin-2-ylidene)butanamide | IC50 | 20000.0 [1] |
 | (2R,4R)-2-(2-Chlorophenyl)-3-[4-(3,5-dimethyl-1,2-oxazol-4-yl)benzoyl]-1,3-thiazolidine-4-carboxylic acid | Ki | 204.17 [1] |
 | (3S)-3-Benzyl-4-[[4-(2-chlorophenyl)-1,3-thiazol-2-yl]-methylamino]-4-oxobutanoic acid | Ki | 10000.0 [1] |
 | (3R)-4-[[4-[5-Chloro-2-(6-methoxypyridin-3-yl)phenyl]-1,3-thiazol-2-yl]-cyclopropylamino]-3-(furan-2-ylmethyl)-4-oxobutanoic acid | Ki | 100.0 [1] |
 | (2R,4R)-2-(2-Chlorophenyl)-3-[4-(2-methoxyphenyl)benzoyl]-1,3-thiazolidine-4-carboxylic acid | Ki | 338.84 [1] |
 | (2R,4R)-2-(2-Chlorophenyl)-3-(4-phenylbenzoyl)-1,3-thiazolidine-4-carboxylic acid | Ki | 977.24 [1] |
 | (2S,5R)-5-(2-Chlorophenyl)-1-[4-(3,5-dimethyl-1,2-oxazol-4-yl)benzoyl]pyrrolidine-2-carboxylic acid | Ki | 398.11 [1] |
 | (2R,4R)-3-[4-(2-Methoxyphenyl)benzoyl]-2-phenyl-1,3-thiazolidine-4-carboxylic acid | Ki | 1202.26 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(5-methylthiazol-2-yl)butanamide | IC50 | 800.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(4,5-dihydrothiazol-2-yl)-3-methylbutanamide | IC50 | 2100.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(pyridin-4-yl)butanamide | IC50 | 56000.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3-methyl-N-(1,3,4-thiadiazol-2-yl)butanamide | IC50 | 12000.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3-methyl-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]butanamide | IC50 | 1900.0 [1] |
 | (S)-Methyl 2-(2-(4-chlorophenyl)-3-methylbutanamido)thiazole-5-carboxylate | IC50 | 2000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N,3-dimethyl-N-(thiazol-2-yl)butanamide | IC50 | 84000.0 [1] |
 | (S)-N-(1-(4-Chlorophenyl)-2-methylpropyl)thiazole-2-carboxamide | IC50 | 100000.0 [1] |
 | (S)-N-(2-(4-Chlorophenyl)-3-methylbutyl)thiazol-2-amine | IC50 | 100000.0 [1] |
 | Rac-1-(4-chlorophenyl)-2-methyl-N-(thiazol-2-yl)propane-1-sulfonamide | IC50 | 100000.0 [1] |
 | (S)-N-(1-(4-Chlorophenyl)-2-methylpropyl)thiazole-2-sulfonamide | IC50 | 100000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N,3-dimethylbutanamide | IC50 | 11000.0 [1] |
 | (S)-N-Tert-butyl-2-(4-chlorophenyl)-3-methylbutanamide | IC50 | 100000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-phenylbutanamide | IC50 | 100000.0 [1] |
 | Rac-2-(4-chlorophenyl)-3-methyl-N-(pyridin-3-yl)butanamide | IC50 | 49000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(pyridin-2-yl)butanamide | IC50 | 1400.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(6-fluoropyridin-2-yl)-3-methylbutanamide | IC50 | 1100.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(5-fluoropyridin-2-yl)-3-methylbutanamide | IC50 | 1300.0 [1] |
 | Rac-2-(4-chlorophenyl)-3-methyl-N-(pyrimidin-2-yl)butanamide | IC50 | 53000.0 [1] |
 | Rac-2-(4-chlorophenyl)-3-methyl-N-(pyrazin-2-yl)butanamide | IC50 | 5700.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(pyridazin-3-yl)butanamide | IC50 | 2300.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(oxazol-2-yl)butanamide | IC50 | 25000.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3-methyl-N-(1,2,4-thiadiazol-5-yl)butanamide | IC50 | 2000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(1H-imidazol-2-yl)-3-methylbutanamide | IC50 | 20000.0 [1] |
 | Rac-2-(4-chlorophenyl)-3-methyl-N-(1H-tetrazol-5-yl)butanamide | IC50 | 100000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(1H-pyrazol-3-yl)butanamide | IC50 | 100000.0 [1] |
 | Rac-(S)-2-(4-chlorophenyl)-N-(isoxazol-3-yl)-3-methylbutanamide | IC50 | 36000.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3-methyl-N-(thiadiazol-5-yl)butanamide | IC50 | 57000.0 [1] |
 | Rac-N-(benzo[d]thiazol-2-yl)-2-(4-chlorophenyl)-3-methylbutanamide | IC50 | 3000.0 [1] |
 | (S)-N-(5-Chlorobenzo[d]oxazol-2-yl)-2-(4-chlorophenyl)-3-methylbutanamide | IC50 | 4300.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(4-(trifluoromethyl)thiazol-2-yl)butanamide | IC50 | 17000.0 [1] |
 | (S)-N-(4-Tert-butylthiazol-2-yl)-2-(4-chlorophenyl)-3-methylbutanamide | IC50 | 7900.0 [1] |
 | 2-(4-Chlorophenyl)-3-methyl-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)butanamide | IC50 | 100000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(4,5-dimethylthiazol-2-yl)-3-methylbutanamide | IC50 | 1800.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(5-chlorothiazol-2-yl)-3-methylbutanamide | IC50 | 700.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-methyl-N-(5-(trifluoromethyl)thiazol-2-yl)butanamide | IC50 | 1500.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(5-cyanothiazol-2-yl)-3-methylbutanamide | IC50 | 2000.0 [1] |
 | (S)-2-(2-(4-Chlorophenyl)-3-methylbutanamido)thiazole-5-carboxylic acid | IC50 | 79000.0 [1] |
 | (S)-2-(2-(4-Chlorophenyl)-3-methylbutanamido)thiazole-5-carboxamide | IC50 | 71000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(5-fluorothiazol-2-yl)-3,3-dimethylbutanamide | IC50 | 700.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(5-chlorothiazol-2-yl)-3,3-dimethylbutanamide | IC50 | 1000.0 [1] |
 | (S)-N-(5-Bromothiazol-2-yl)-2-(4-chlorophenyl)-3,3-dimethylbutanamide | IC50 | 700.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(5-cyanothiazol-2-yl)-3,3-dimethylbutanamide | IC50 | 1500.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3,3-dimethyl-N-[5-(trifluoromethyl)-1,3-thiazol-2-yl]butanamide | IC50 | 1500.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3,3-dimethyl-N-(5-methylsulfanyl-1,3-thiazol-2-yl)butanamide | IC50 | 500.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3,3-dimethyl-N-(5-methylsulfonyl-1,3-thiazol-2-yl)butanamide | IC50 | 3400.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3,3-dimethyl-N-(5-phenylthiazol-2-yl)butanamide | IC50 | 700.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-N-[5-[(4-chlorophenyl)methyl]-1,3-thiazol-2-yl]-3,3-dimethylbutanamide | IC50 | 25000.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-N-[5-(dimethylamino)-1,3-thiazol-2-yl]-3,3-dimethylbutanamide | IC50 | 1600.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3,3-dimethyl-N-(5-morpholinothiazol-2-yl)butanamide | IC50 | 1600.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-3,3-dimethyl-N-[5-(4-methylpiperazin-1-yl)-1,3-thiazol-2-yl]butanamide | IC50 | 3800.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-N-[5-(1,1-dioxo-1,4-thiazinan-4-yl)-1,3-thiazol-2-yl]-3,3-dimethylbutanamide | IC50 | 2400.0 [1] |
 | (2S)-2-(4-Chlorophenyl)-N-[5-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-1,3-thiazol-2-yl]-3,3-dimethylbutanamide | IC50 | 1200.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(thiazol-2-yl)propanamide | IC50 | 46000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(thiazol-2-yl)butanamide | IC50 | 5000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(thiazol-2-yl)pentanamide | IC50 | 5500.0 [1] |
 | (S)-2-(4-Chlorophenyl)-2-cyclopropyl-N-(5-fluorothiazol-2-yl)acetamide | IC50 | 1200.0 [1] |
 | (S)-2-(4-Chlorophenyl)-4-methyl-N-(thiazol-2-yl)pentanamide | IC50 | 600.0 [1] |
 | (S)-2-(4-Chlorophenyl)-3-cyclopropyl-N-(thiazol-2-yl)propanamide | IC50 | 8800.0 [1] |
 | (S)-2-(4-Chlorophenyl)-4-methoxy-N-(thiazol-2-yl)butanamide | IC50 | 170000.0 [1] |
 | (S)-2-(4-Chlorophenyl)-N-(thiazol-2-yl)pent-4-enamide | IC50 | 1100.0 [1] |
 | 2,2-Bis(4-chlorophenyl)-N-(thiazol-2-yl)acetamide | IC50 | 100000.0 [1] |