| 1-Acetyl-4-phenyl-6-(4-phenylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 4.0 [1], 10.0 [2] |
| 1-Acetyl-4-(4-hydroxyphenyl)-6-(4-phenylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 240.0 [1] |
| 1-[2,2,4-Trimethyl-4-phenyl-6-[(4-phenylphenyl)methoxy]-3H-quinolin-1-yl]ethanone | IC50 | 166.0 [1] |
| 1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(4-[trifluoromethyl]benzoyl)amino-2,2,4-trimethylquinoline | IC50 | 7.0 [1] |
| 1-Acetyl-6-(4-phenylbenzoyl)amino-8-methoxy-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 30.0 [1] |
| 1-Acetyl-6-(4-chlorobenzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 31.0 [1] |
| 1-[6-[(4-Tert-butylphenyl)methylamino]-2,2,4-trimethyl-4-phenyl-3H-quinolin-1-yl]ethanone | IC50 | 930.0 [1] |
| 1-Acetyl-6-(2-furoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 27.0 [1] |
| N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-phenylbenzamide | IC50 | 9.0 [1] |
| 1-Acetyl-6-(4-phenylbenzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4,7-tetramethylquinoline | IC50 | 5.0 [1] |
| N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-2-phenylbenzamide | IC50 | 25.0 [1] |
| N-[1-Acetyl-4-(2-methoxyphenyl)-2,2,4-trimethyl-3H-quinolin-6-yl]-4-phenylbenzamide | IC50 | 170.0 [1] |
| N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-2-[(2-methylpropan-2-yl)oxy]acetamide | IC50 | 76.0 [1] |
| N-[1-Acetyl-2,2,4-trimethyl-4-(4-methylphenyl)-3H-quinolin-6-yl]-4-phenylbenzamide | IC50 | 50.0 [1] |
| N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-4-propylbenzamide | IC50 | 5.0 [1] |
| 1-Acetyl-4-phenyl-6-(phenylaminocarbonyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 580.0 [1] |
| N-(1-Acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-1-phenylmethanesulfonamide | IC50 | 2800.0 [1] |
| 1-Acetyl-N-[2-(4-methoxyphenyl)ethyl]-2,2,4-trimethyl-4-phenyl-3H-quinoline-6-carboxamide | IC50 | 1880.0 [1] |
| 1-Acetyl-4-phenyl-6-(4-phenylbenzoyl)oxy-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline | IC50 | 54.0 [1] |
| N-[(4R)-1-Acetyl-2,2,4-trimethyl-4-(4-prop-2-ynoxyphenyl)-3H-quinolin-6-yl]-4-phenylbenzamide | IC50 | 39.0 [1] |
| 4-[3-[[2-[[1-[2-[2-[2-[4-[[4-[(4R)-1-Acetyl-2,2,4-trimethyl-6-[(4-phenylbenzoyl)amino]-3H-quinolin-4-yl]phenoxy]methyl]triazol-1-yl]ethoxy]ethoxy]ethyl]triazol-4-yl]methylamino]-2-oxoethyl]amino]phenyl]-5-amino-N-tert-butyl-2-methylsulfanylthieno[2,3-d]pyrimidine-6-carboxamide | IC50 | 920.0 [1] |
| 4-[3-[[2-[[1-[2-[2-[2-[2-[4-[[4-[(4R)-1-Acetyl-2,2,4-trimethyl-6-[(4-phenylbenzoyl)amino]-3H-quinolin-4-yl]phenoxy]methyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]methylamino]-2-oxoethyl]amino]phenyl]-5-amino-N-tert-butyl-2-methylsulfanylthieno[2,3-d]pyrimidine-6-carboxamide | IC50 | 1662.0 [1] |
| 4-[3-[[2-[[1-[2-[2-[2-[2-[2-[4-[[4-[(4R)-1-Acetyl-2,2,4-trimethyl-6-[(4-phenylbenzoyl)amino]-3H-quinolin-4-yl]phenoxy]methyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]methylamino]-2-oxoethyl]amino]phenyl]-5-amino-N-tert-butyl-2-methylsulfanylthieno[2,3-d]pyrimidine-6-carboxamide | IC50 | 1023.0 [1] |
| N-[(4R)-1-Acetyl-4-[4-[[1-[2-[2-(2-azidoethoxy)ethoxy]ethyl]triazol-4-yl]methoxy]phenyl]-2,2,4-trimethyl-3H-quinolin-6-yl]-4-phenylbenzamide | IC50 | 324.0 [1] |