![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_1cc257bab28d3e85f276bcae9f111347.svg) | Methotrexate | IC50 | 106.0 [1], 211.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_567a3300d143a91f2e91ad015695c1c3.svg) | Pemetrexed | IC50 | 60.0 [1], 254.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_3f53ada1766cdeccc391487c0352c435.svg) | Raltitrexed | IC50 | 22.0 [1], 746.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_2aa8bc65b75d01f4497d054f8de7ec3e.svg) | (2S)-2-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]pentanedioic acid | IC50 | 0.17 [1], 126.0 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_984013162eda994b64c9057c12d4a205.svg) | N-{4-[4-(2-Amino-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)butyl]benzoyl}-L-glutamic Acid | IC50 | 5.6 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_15eb4c59f69915adea286192e9521740.svg) | (2S)-2-[[4-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]pentanedioic acid | IC50 | 0.34 [1], 557.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_51c43dab8d68e6716d3c1851aa62c4b6.svg) | (2S)-2-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-3-carbonyl]amino]pentanedioic acid | IC50 | 0.1 [1], 654.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_97d0f873ba4318ccaa31c8f07b949622.svg) | (2S)-2-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]hexanedioic acid | IC50 | 3.6 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_3ae9b8c764e0b775ea3ecdb05e8a68e6.svg) | (2S)-2-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]pentanoic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_1f908e05f00329f6781cfc6813713c25.svg) | 4-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]butanoic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_e98557eb119eca07920c20a2739acd94.svg) | (2S)-2-[[5-[3-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]butanedioic acid | IC50 | 347.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_2fe55254ecbe887ed2fb1f228101cfcc.svg) | 5-[3-(2-Amino-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-6-yl)-propyl]-thiophene-2-carboxylic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_e28f4c81a27d1bae7f882d0739b35fc8.svg) | (2S)-2-[[5-[4-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)butyl]pyridine-2-carbonyl]amino]pentanedioic acid | IC50 | 0.58 [1], 471.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_e2a1ce84d6069ebb05ff4e5197370490.svg) | (2S)-2-[[6-[4-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)butyl]pyridine-3-carbonyl]amino]pentanedioic acid | IC50 | 37.41 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_f8f3b1fd2481a8bdc74707f6b45c2b34.svg) | (2S)-2-[[6-[4-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)but-1-ynyl]pyridine-2-carbonyl]amino]pentanedioic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_8f48010b90ed739c033be08d0545f93f.svg) | (2S)-2-[[6-[4-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)butyl]pyridine-2-carbonyl]amino]pentanedioic acid | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_a2047cae009b1b180c5615dfdf260069.svg) | (2S)-2-[[6-[4-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)but-1-ynyl]pyridine-3-carbonyl]amino]pentanedioic acid | IC50 | 839.1 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_a1e7ae63e79cdcf5694ce552cb0dbdf6.svg) | (2S)-2-[[5-[4-(2-Amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)but-1-ynyl]pyridine-2-carbonyl]amino]pentanedioic acid | IC50 | 18.8 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_59b02b5a493c0d753bd88304339de09f.svg) | (S)-2-(4-(3-(2,4-Diaminofuro[2,3-d]pyrimidine-5-yl)propyl)-2-thienylcarbonylamino)glutaric acid | IC50 | 17.5 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/folate-receptor-beta_c635692ab9f03ce2483f9e392cfc7eb2.svg) | (S)-2-(2-(3-(2,4-Diaminofuro[2,3-d]pyrimidine-5-yl)propyl)-4-thienylcarbonylamino)glutaric acid | IC50 | 54.3 [1], 1000.0 [2] |