![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_c410e5af606a08989ab48be584c73f68.svg) | Azd4547 | IC50 | 103.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_0a82b2fcefb5f2b85b04ee97b06eb370.svg) | N-[2-[[6-(2,6-Dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_5f74e8a3c9ec10c4178077a648e31819.svg) | Infigratinib | IC50 | 0.82 [1], 60.0 [2], 62.0 [3], 64.0 [4], 71.0 [5] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_161fa5ee586e171acaf4cea810b3ba31.svg) | 2-Formyl-N-[5-(trifluoromethyl)pyridin-2-yl]quinoline-8-carboxamide | IC50 | 57.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_63f9b5c12b3ac2bfdf0fdcf2c3e35759.svg) | (1S,2S,3R,4R)-3-[[5-Cyano-2-[4-[4-(dimethylamino)piperidin-1-yl]-2-(2-methylpropoxy)anilino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | IC50 | 6.9 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ee8ec81232d884fb37ff6e0ad87d9764.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-2-(prop-2-enoylamino)benzamide | IC50 | 0.8 [1], 1.5 [2], 3.6 [3], 443.0 [4] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_069b2003931b5f9a3b881486ba535953.svg) | 6-Chloro-N-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-3-nitropyridin-2-amine | IC50 | 21.0 [1], 32.0 [2], 53.0 [3], 10000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_c38cbdee4404993837adfc282c860ec1.svg) | Nvp-tae 684 | IC50 | 16.0 [1], 20.0 [2], 1920.0 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ebc51d09388d6e683e7e3843fa6ae230.svg) | N-[3-[[3-(2,6-Dichloro-3,5-dimethoxyphenyl)-7-[4-(diethylamino)butylamino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-1-yl]methyl]phenyl]prop-2-enamide | IC50 | 189.0 [1], 261.0 [2], 261.3 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_83192c16ea9732c64a10a3847fed4688.svg) | N-(5-Cyano-4-methoxypyridin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 6.3 [1], 72.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_af5aa4e11fdf3187b051977296dc225a.svg) | N-[5-Cyano-4-(2-methoxyethoxy)pyridin-2-yl]-2-formyl-5,6,7,8-tetrahydropyrido[2,3-b]azepine-9-carboxamide | IC50 | 175.0 [1], 741.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b0c33e8ef03d48b2f99875ae25bdd3ac.svg) | N-(5-Chloropyridin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 21.0 [1], 916.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_622da44f7119f937578463a45a70d0f7.svg) | N-[5-Cyano-4-[2-(dimethylamino)ethoxy]pyridin-2-yl]-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 10.6 [1], 11.0 [2], 588.0 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_8bf159aeb520a318ef5bb9c146d4fabb.svg) | N-(5-Cyanopyrimidin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 45.0 [1], 131.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_67e40f118c2dc2fc4dc8b22808459952.svg) | N-(5-Cyanopyridin-2-yl)-2-formyl-5,6,7,8-tetrahydropyrido[2,3-b]azepine-9-carboxamide | IC50 | 660.0 [1], 3000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_6a50b4a93b791d791e549eb68ddb0fd4.svg) | 6-Formyl-N-[5-(trifluoromethyl)pyridin-2-yl]-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide | IC50 | 42.0 [1], 531.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b53497488e0d1c1952ccf2e6abd1afa9.svg) | N-(5-Cyano-4-morpholin-4-ylpyridin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 27.0 [1], 224.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_531215c25402ac03b4fd91e3d59960ed.svg) | N-[5-Cyano-4-(4-hydroxy-4-methylpiperidin-1-yl)pyridin-2-yl]-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 1.2 [1], 24.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_75d414250c4e749bccb9c68540fe0ace.svg) | N-[5-Cyano-4-(2-methoxyethoxy)pyridin-2-yl]-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 1.3 [1], 18.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_6340ee23fe9adb335f0852cd192603f4.svg) | N-(5-Cyano-4-propan-2-yloxypyridin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 0.7 [1], 29.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_1b704d9514dbbfedc5ab0df0c05e85c4.svg) | N-(5-Cyanopyridin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 15.8 [1], 16.0 [2], 108.0 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_8654c6eb3c2bfa955fb6160cd7b2b3af.svg) | 7-Formyl-N-(6-methoxypyrimidin-4-yl)-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 140.0 [1], 3000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_39e6576513d4347b357b1d026a235c75.svg) | N-(5-Cyano-4-propan-2-yloxypyridin-2-yl)-6-formyl-2,3-dihydropyrrolo[2,3-b]pyridine-1-carboxamide | IC50 | 1.1 [1], 55.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_4dcca4531c39c71fff87844557464327.svg) | N-[5-Cyano-4-(oxan-4-yl)pyridin-2-yl]-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 17.0 [1], 150.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_e22fc87037ea084867175ea4dcf8a3c1.svg) | B-Cell Immunosuppressant | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_7506e10d7aa3bbea9276cbad94a43d9f.svg) | 8-[[5-(Trifluoromethyl)pyridin-2-yl]carbamoyl]quinoline-2-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_9f49ffe67c9ea45b9cde7fbaf218eda8.svg) | 2-(Hydroxymethyl)-N-[5-(trifluoromethyl)pyridin-2-yl]quinoline-8-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ad4052b60c84d4e49f62045bc162d72e.svg) | 2-Formyl-N-[4-(trifluoromethyl)phenyl]quinoline-8-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_2637c1097c5b51648932c96eac45b5b7.svg) | Debio-1347 | IC50 | 290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_c6a654ab2a80479be435287d3d61f1cc.svg) | H3B-6527 | IC50 | 0.2 [1], 1.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_fe488f1f0ab2c047ee8c00c265c5ee26.svg) | N-[2-[[5-[(2,6-Dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 4.0 [1], 11.1 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_31800f62ec3d5e2408262b35fd2ea602.svg) | 7-Formyl-N-[5-(trifluoromethyl)pyridin-2-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 13.0 [1], 13.3 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_989e7465a61b9888b32717cdd9777ffc.svg) | 7-Formyl-N-pyridin-2-yl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_8d5910fbfb81fd6a5bd566106045c10a.svg) | N-(5-Cyanopyrazin-2-yl)-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 33.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_50496bbf8200ff768a58b4c6c452584d.svg) | 2-[4-[6-Chloro-2-[4-(4-methylpiperazin-1-yl)phenyl]-1H-imidazo[4,5-b]pyridin-7-yl]piperazin-1-yl]-N-(1,3-thiazol-2-yl)acetamide | IC50 | 20.0 [1], 130.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_6cd963385a14d30f0462a301beda2c5c.svg) | 3-[5-Cyano-4-(2-methoxyethylamino)pyridin-2-yl]-1-(6-formylpyridin-2-yl)-1-methylurea | IC50 | 6.5 [1], 41.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_82e23a669958487729fd4a59d8989f39.svg) | 3-[5-Cyano-4-(2-methoxyethylamino)pyridin-2-yl]-1-(6-formylpyridin-2-yl)-1-(2-methoxyethyl)urea | IC50 | 7.4 [1], 91.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_dbf08bacbdaff28e6a58834f6a8461b1.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-formyl-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 23.0 [1], 2800.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_3b277bdffa206c61242ae6053e448ed3.svg) | 7-Formyl-N-(5-methyl-1H-pyrazol-3-yl)-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide | IC50 | 790.0 [1], 3000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_e42013f06b4ed63631c6521cddbef788.svg) | N-(5-Cyano-4-propan-2-yloxypyridin-2-yl)-6-formylpyrrolo[2,3-b]pyridine-1-carboxamide | IC50 | 3.2 [1], 750.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_a840767d7ddb2c27c40164419a996160.svg) | Infigratinib phosphate | IC50 | 60.0 [1], 168.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_d82fab1028f4e0de22d7e5370ed8f8b9.svg) | 4-N-(3,5-Dimethoxyphenyl)-4-N-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-1-N-propan-2-ylcyclohexane-1,4-diamine | IC50 | 6.76 [1], 25.12 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 148.3 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ee0e7cfe47cadc1651c09b051ac07ddd.svg) | Acrylamide | IC50 | 938.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_8edb893ba88c5700603edef201da4265.svg) | Nintedanib | IC50 | 610.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_12fa190f2d2e4b2561e24185e6a9c597.svg) | Nintedanib esylate | IC50 | 610.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_4e9df3bd1ea0920231ce5d4b41666b94.svg) | Ponatinib | IC50 | 7.1 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_295456cbf7462dfb1eaccb88d6610904.svg) | Ceritinib | IC50 | 950.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_a257c791d1de1df5d4a1fa04612f9c76.svg) | Nvp-aew541 | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_2cf324237228e1f753214eb9a2ce619a.svg) | Erdafitinib | IC50 | 6.61 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b63a2565bd4d512206a1c9679cacee61.svg) | 3-((4-Bromo-2,6-difluorobenzyl)oxy)-5-(3-(4-(pyrrolidin-1-yl)butyl)ureido)isothiazole-4-carboxamide | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_10b979513d2e855fbc4454fcc705914e.svg) | 1-[2-Amino-6-(2,6-dichlorophenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylurea | IC50 | 560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_f8dea142aa4a3f574f20a24329144dbd.svg) | CID 118295624 | IC50 | 19.3 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_977881cff21801cb818f36d79a4f4834.svg) | Roblitinib | IC50 | 1.9 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_cc5bc7310bc863c88072f5adeababc04.svg) | 6H-Purin-6-one, 2-amino-1,7-dihydro-8-phenyl- | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b43f9b172387f2a84cebdafc2497da4c.svg) | cis-3-[4-Amino-7-(3-azetidin-1-ylmethyl-cyclobutyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]-phenol | IC50 | 2800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_101f274fa0d894c601461fd7747171a3.svg) | 7-[3-(Azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2S)-oxolan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_c89eb280cebe7a1be770abaa2c58bf54.svg) | N-[4-[[3-(3,5-Dimethoxyphenyl)-7-[4-(4-methylpiperazin-1-yl)anilino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-1-yl]methyl]phenyl]prop-2-enamide | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_507966d387462fd7ae0b3ec2dded03f4.svg) | 6-[2-[(E)-2-[4-(Morpholin-4-ylmethyl)phenyl]ethenyl]pyridin-4-yl]-3,7-dihydropyrrolo[2,3-d]pyrimidin-4-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_9869d4afb98ef2c3ccd6540bb969cfa4.svg) | CID 46864270 | IC50 | 34.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b47eb0b10c004af2684a6d610b4c991d.svg) | Ethyl 8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_bd7ab61fd74e87578c2dfefbcc47d031.svg) | 7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_871d853c2ba64c7dea86f43b9412ef22.svg) | N-(3-Imidazo[1,2-b]pyridazin-6-yloxyphenyl)-3-(trifluoromethyl)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_e8f80e84b0622638790c204b1bf7bcce.svg) | 2-[3-[[4-[(2,2-Difluoro-3-oxo-4H-1,4-benzoxazin-6-yl)amino]-5-fluoropyrimidin-2-yl]amino]phenoxy]-N-methylacetamide | Ki | 217.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_49267c7ecf3b71293f5fe75dcbbc5c0d.svg) | 1-[3-[8-(Pyridin-4-ylmethylamino)imidazo[1,2-a]pyrazin-6-yl]phenyl]-3-[3-(trifluoromethyl)phenyl]urea | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b6faf72dfa81ac6f5cbbee7518dcb7f6.svg) | 4-[6-(Benzylamino)imidazo[1,2-B]pyridazin-3-Yl]benzonitrile | IC50 | 5900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_5d7901f03aa52a959c119b7fc87d0b0c.svg) | 6-[(2r)-2-(3-Fluorophenyl)pyrrolidin-1-Yl]-3-(Pyridin-2-Yl)imidazo[1,2-B]pyridazine | IC50 | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_07f245678e6fcc2d52455f8c1a6544d0.svg) | 2-[4-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperazin-1-yl]acetic acid | IC50 | 5300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_cadcfe40c75731fb4d071e8664de359c.svg) | 1-[4-[6-[(2R)-2-(3-Fluorophenyl)pyrrolidin-1-yl]imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl]piperidin-4-ol | IC50 | 4400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ffe03ecf7e6e5217b6f4d31768d4e4fa.svg) | N-[(3R,4S)-4-[[5-[(2,6-Difluoro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]oxolan-3-yl]prop-2-enamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_fefa37c9055748854606b692d516ebaa.svg) | N-[2-[[5-[(2,6-Difluoro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_6a366a757bce9e5065ca192708f3947b.svg) | N-[2-[[5-[(2,6-Difluoro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-5-(4-ethylpiperazin-1-yl)-3-methylphenyl]prop-2-enamide | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_c1c23c26ef96fb9ec2be798b78caf509.svg) | N-[2-[[5-[(2,6-Difluoro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]phenyl]prop-2-enamide | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_48fa1a833d11c0d8458d67a252a238e5.svg) | 4-Chloro-N-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[2-(5-morpholin-4-ylpyridin-3-yl)ethynyl]benzamide | IC50 | 5.5 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_1e49aaca4633a76158513beb3216d092.svg) | 7-(1,3,4,6,7,8,9,9a-Octahydropyrido[1,2-a]pyrazin-2-yl)-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amine | IC50 | 52.7 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_17d903b0da529a78ce24ad01131e046a.svg) | Clk1-IN-1 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ed54b1f4442847f3529ef0ad5ea76c81.svg) | [5-Amino-1-(2-chloro-5-hydroxyphenyl)pyrazol-4-yl]-(3-methylphenyl)methanone | IC50 | 4100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_9bb803b67830b84f79d2523ea1aed043.svg) | 5-[5-Amino-4-(1H-indole-2-carbonyl)pyrazol-1-yl]-1,3-dihydrobenzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_407fb30385e454d199873d40d39563d4.svg) | [5-Amino-1-(2-chlorophenyl)pyrazol-4-yl]-(1H-indol-2-yl)methanone | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_775e368ae27a9f287a41bda6dbc30947.svg) | [5-Amino-1-(1H-indol-5-yl)pyrazol-4-yl]-(1H-indol-2-yl)methanone | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_ab4c2cb5c7548808e4662bf9ea927177.svg) | [5-Amino-1-(2-chloro-5-hydroxyphenyl)pyrazol-4-yl]-quinolin-6-ylmethanone | IC50 | 740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_4c6e740269e5ce22fa9e9af192d6e72c.svg) | [5-Amino-1-(2-chloro-5-hydroxyphenyl)pyrazol-4-yl]-(1H-indol-2-yl)methanone | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_fac30547e036967a52ef6fac02bca233.svg) | [5-Amino-1-(2-methyl-1H-indol-5-yl)pyrazol-4-yl]-(1H-indol-2-yl)methanone | IC50 | 85.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_43f788d96ec0ff7e5665a2cc0c477be7.svg) | [5-Amino-1-(2-chloro-5-hydroxyphenyl)pyrazol-4-yl]-[5-(morpholin-4-ylmethyl)-1H-indol-2-yl]methanone | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_5ea54bf25909fbc198769649d71ae0de.svg) | [5-Amino-1-(2-chloro-5-hydroxyphenyl)pyrazol-4-yl]-(1-benzofuran-2-yl)methanone | IC50 | 730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_d787529a69209223ef1585f4eb620655.svg) | N-[2-[[5-[(3,5-Dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 188.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_d226e4a41089877b3ea212647fba3e00.svg) | N-[3-Chloro-2-[[5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]phenyl]prop-2-enamide | IC50 | 3.8 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_d30b9911bce6232783745cf461116717.svg) | N-[2-[[5-[(2,6-Dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-(trifluoromethyl)phenyl]prop-2-enamide | IC50 | 24.9 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_47d9fc0b02919a6ce19da72d3faff87b.svg) | N-[2-[[5-[(2,6-Dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-methoxyphenyl]prop-2-enamide | IC50 | 4.8 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_2af594e0b6f36d9ce98c5d1a69b0d498.svg) | N-[3,5-Dichloro-2-[[5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]phenyl]prop-2-enamide | IC50 | 8.5 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_974d84c7f7bc5201046272be284d22ee.svg) | N-[3-Chloro-2-[[5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-5-fluorophenyl]prop-2-enamide | IC50 | 2.6 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_b568fcdb2660d06f7006b9df5b666215.svg) | N-[2-[[5-[(2,6-Dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-fluorophenyl]prop-2-enamide | IC50 | 5.3 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-4_62fa363a3f0d521561c9256da42f8cae.svg) | N-[2-[[5-[1-(2,6-Dichloro-3,5-dimethoxyphenyl)ethoxy]pyrimidin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 10000.0 [1] |