![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_c410e5af606a08989ab48be584c73f68.svg) | Azd4547 | IC50 | 2.5 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 1.77 [1], 3.36 [2], 5.8 [3], 34.0 [4] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_2637c1097c5b51648932c96eac45b5b7.svg) | Debio-1347 | IC50 | 7.6 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_ebc51d09388d6e683e7e3843fa6ae230.svg) | N-[3-[[3-(2,6-Dichloro-3,5-dimethoxyphenyl)-7-[4-(diethylamino)butylamino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-1-yl]methyl]phenyl]prop-2-enamide | IC50 | 2.29 [1], 2.3 [2], 6.2 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_1e49aaca4633a76158513beb3216d092.svg) | 7-(1,3,4,6,7,8,9,9a-Octahydropyrido[1,2-a]pyrazin-2-yl)-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amine | IC50 | 0.2 [1], 0.4 [2], 0.8 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_68cbe63d62204863632720dd1e248b65.svg) | 4-Fluoro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 1.6 [1], 24.8 [2], 155.7 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_a840767d7ddb2c27c40164419a996160.svg) | Infigratinib phosphate | IC50 | 1.4 [1], 2.0 [2], 4.9 [3] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5f74e8a3c9ec10c4178077a648e31819.svg) | Infigratinib | IC50 | 1.0 [1], 1.2 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_fa37ae125bcd4e6df1af4be57fbea491.svg) | 1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)urea | IC50 | 1.0 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_2f15fb478c8045b6bf5d450f1eb5924b.svg) | Lucitanib | IC50 | 82.5 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_b63a2565bd4d512206a1c9679cacee61.svg) | 3-((4-Bromo-2,6-difluorobenzyl)oxy)-5-(3-(4-(pyrrolidin-1-yl)butyl)ureido)isothiazole-4-carboxamide | IC50 | 3.08 [1], 8.79 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_0a82b2fcefb5f2b85b04ee97b06eb370.svg) | N-[2-[[6-(2,6-Dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 246.9 [1], 1700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5f02b655eda2ba8c931019b391ac0d51.svg) | 2-[2-[4-[4-(4-Tert-butylanilino)phenoxy]-6-methoxyquinolin-7-yl]oxyethylamino]ethanol | IC50 | 69.0 [1], 88.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5b10441bbfcd2a7880fba7127c6144c0.svg) | 3-[[5-[6-[(3-Chlorophenyl)amino]pyrazinyl]-3-pyridinyl]amino]-1-propanol | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_c89eb280cebe7a1be770abaa2c58bf54.svg) | N-[4-[[3-(3,5-Dimethoxyphenyl)-7-[4-(4-methylpiperazin-1-yl)anilino]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-1-yl]methyl]phenyl]prop-2-enamide | IC50 | 4.0 [1], 58.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_fb822231eed670f8c91ff43b84a344f6.svg) | 6,6-Dimethyl-8-[1-(oxetan-3-yl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_50496bbf8200ff768a58b4c6c452584d.svg) | 2-[4-[6-Chloro-2-[4-(4-methylpiperazin-1-yl)phenyl]-1H-imidazo[4,5-b]pyridin-7-yl]piperazin-1-yl]-N-(1,3-thiazol-2-yl)acetamide | IC50 | 20.0 [1], 63.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_899121b30cafe1d5047ff767ae93b9df.svg) | 4-N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-ethylpiperazin-1-yl)-2-N-[(3-methyl-1,2-oxazol-5-yl)methyl]quinazoline-2,4-diamine | IC50 | 10.0 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_d7c2ffe13b78a31283362b058c34b3bf.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-5-methoxyquinazolin-4-amine | IC50 | 100.9 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_b2b717a51217c1838151753de834a07e.svg) | 8-Chloro-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amine | IC50 | 4.8 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_fe691a412c2c2c55ec025949adbc2d7e.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-8-methoxyquinazolin-4-amine | IC50 | 3.9 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_7111ff6e484768209d33dc320f51949f.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-8-(4-ethylpiperazin-1-yl)quinazolin-4-amine | IC50 | 4.3 [1], 13.8 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_4642c830fa93aacd0334f55f8ebf7e9d.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-ethylpiperazin-1-yl)quinazolin-4-amine | IC50 | 0.8 [1], 1.2 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5bfea7cf7caf87ed1a89a7c0c00f8d36.svg) | N-[5-[2-(2,6-Dichloro-3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-ethylpiperazin-1-yl)quinazolin-4-amine | IC50 | 0.3 [1], 1.4 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_d3818a5c4efff618066916ab918a337e.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-methylpiperazin-1-yl)quinazolin-4-amine | IC50 | 0.7 [1], 1.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_d3baeadbf79835e8366d18f7ac76a7b5.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-propan-2-ylpiperazin-1-yl)quinazolin-4-amine | IC50 | 0.1 [1], 0.6 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_a504cdcf7ca2995e00ed32fc69e1fa9e.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-[3-(dimethylamino)pyrrolidin-1-yl]quinazolin-4-amine | IC50 | 0.4 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_df68a4faa5259a58cdaae4ca083739e4.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-[(3S,5R)-3,4,5-trimethylpiperazin-1-yl]quinazolin-4-amine | IC50 | 0.1 [1], 0.2 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_fd0dda512c995a585eeb251e3274903b.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-methyl-1,4-diazepan-1-yl)quinazolin-4-amine | IC50 | 0.7 [1], 10.8 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_079813eab3ac91e8764c879180b36f55.svg) | 2-Chloro-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-ethylpiperazin-1-yl)quinazolin-4-amine | IC50 | 0.6 [1], 108.2 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_41d35f9bb7a616845c27948e2bc77dc5.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-6-(4-ethylpiperazin-1-yl)isoquinolin-1-amine | IC50 | 1.2 [1], 1.8 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_c907e855ff19f7b8259891e0d8950242.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-[4-(dimethylamino)piperidin-1-yl]quinazolin-4-amine | IC50 | 0.3 [1], 17.5 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_d8c32d5402d53831d07387ab323869bf.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(1-methylpiperidin-4-yl)quinazolin-4-amine | IC50 | 0.8 [1], 9.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_9e6a84d20b0698e09c0bd50e1d68c86d.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amine | IC50 | 3.2 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_903cf2d12aae9544456fa5515b9812fb.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-morpholin-4-ylquinazolin-4-amine | IC50 | 0.4 [1], 3.9 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_9dc34c38c52d2276307242c103f32756.svg) | 4-N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-N-(2-morpholin-4-ylethyl)quinazoline-4,7-diamine | IC50 | 1.3 [1], 13.2 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_0869723359f568d555d94f9a1486cd3a.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-ethylpiperazin-1-yl)-2-methylquinazolin-4-amine | IC50 | 0.6 [1], 105.7 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_de0e0054e522c7e64853b688387e417a.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-2-ethyl-7-(4-ethylpiperazin-1-yl)quinazolin-4-amine | IC50 | 0.5 [1], 24.7 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_ec35f12d725a9fa4c0a85cbdb4427721.svg) | N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-(4-ethylpiperazin-1-yl)-2-propylquinazolin-4-amine | IC50 | 0.7 [1], 90.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_7a0d7dafda8e14cc74d256a65fb61560.svg) | 5-Chloro-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amine | IC50 | 16.9 [1], 200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_7604f9e80df6b3be83b86758d161e072.svg) | 4-N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-7-N-(2-methoxyethyl)quinazoline-4,7-diamine | IC50 | 2.7 [1], 10.3 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_2d3b1e23940088d265d5b435c7a748b9.svg) | 7-(4-Cyclobutylpiperazin-1-yl)-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]quinazolin-4-amine | IC50 | 0.1 [1], 0.6 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_25be3fc7aeabe3f032b08a388602acce.svg) | 4-Chloro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-isoquinolin-6-ylpyridin-2-yl]phenol | IC50 | 2.0 [1], 249.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_58e0053da379fa3464b86e2ae4113ca2.svg) | 4,5-Difluoro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 2.8 [1], 288.6 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_7166dacdfe33c4cd0eb621cf8bc8afb0.svg) | 2-[5-[[(1R)-2-Hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 3.0 [1], 57.5 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_0e15332c5c37f694c83d6081e570c1e0.svg) | (2R)-2-[[5-(3-Methyl-2H-indazol-5-yl)-6-phenylpyridin-3-yl]amino]-2-phenylethanol | IC50 | 26.3 [1], 677.7 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_da819cf8d2b7e86f40ccc2e5e950528e.svg) | 4-Chloro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-pyrazolo[3,4-b]pyridin-5-yl)pyridin-2-yl]phenol | IC50 | 6.6 [1], 2281.3 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_c23da44159559bbaf40af86512dea73f.svg) | 2,4-Difluoro-6-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 3.4 [1], 280.1 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5dfd7bf06ab62aaaef4955ebb4ab716c.svg) | 5-Fluoro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 4.7 [1], 313.3 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_917aa43334b03f7833efe05134efdcdc.svg) | 2-Fluoro-6-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 2.5 [1], 293.5 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_bfd6b87cf089aa6a697f222ce580e253.svg) | 4-Chloro-2-[5-[[(1R)-2-hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 8.6 [1], 24.8 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5dba392838508516cefbc5456e5a7d21.svg) | 3-[5-[[(1R)-2-Hydroxy-1-phenylethyl]amino]-3-(3-methyl-2H-indazol-5-yl)pyridin-2-yl]phenol | IC50 | 21.4 [1], 36.2 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_0bd521817a78d41ea847a2a17686d577.svg) | [5-Amino-1-(2-ethyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-(1H-indol-2-yl)methanone | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_098abef22f402fcca475171b05f02d82.svg) | [5-Amino-1-(2-methyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-(6-bromo-1H-indol-2-yl)methanone | IC50 | 8.9 [1], 19.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_e6e997064ff5307b81b74bec6ae90f8c.svg) | [5-Amino-1-(2-methyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-[6-(morpholin-4-ylmethyl)-1H-indol-2-yl]methanone | IC50 | 3.4 [1], 3.6 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_f52a1359ba743d23e8550a3204284dc1.svg) | [5-Amino-1-(2-methyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-(6-phenyl-1H-indol-2-yl)methanone | IC50 | 26.0 [1], 41.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_e23244040ac1c6dadcf3004ac57cfba3.svg) | [5-Amino-1-(2-methyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-(6-methylsulfonyl-1H-indol-2-yl)methanone | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_650245f33e4eaadd52fcd32b9b1fe044.svg) | [5-Amino-1-(2-methyl-3H-benzimidazol-5-yl)pyrazol-4-yl]-[6-[(4,4-difluoropiperidin-1-yl)methyl]-1H-indol-2-yl]methanone | IC50 | 9.4 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_a83aeaea70fa861211ce633587a8a7c8.svg) | N-[4-[[(2,6-Dichloro-3,5-dimethoxyphenyl)carbamoyl-[6-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide | IC50 | 1.0 [1], 64.0 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_d82fab1028f4e0de22d7e5370ed8f8b9.svg) | 4-N-(3,5-Dimethoxyphenyl)-4-N-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-1-N-propan-2-ylcyclohexane-1,4-diamine | IC50 | 1.78 [1], 2.4 [2] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_01384179eb1c1c1ef001bfbf31bfa500.svg) | Ibrutinib | IC50 | 280.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_8edb893ba88c5700603edef201da4265.svg) | Nintedanib | IC50 | 37.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_12fa190f2d2e4b2561e24185e6a9c597.svg) | Nintedanib esylate | IC50 | 37.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_4e9df3bd1ea0920231ce5d4b41666b94.svg) | Ponatinib | IC50 | 1.3 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_295456cbf7462dfb1eaccb88d6610904.svg) | Ceritinib | IC50 | 260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_a59db47f5f7aa063c6007dcf79b51cfe.svg) | PD173074 | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 24000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_a257c791d1de1df5d4a1fa04612f9c76.svg) | Nvp-aew541 | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_94feb385cecaa610e1d68d9fb9d55ef3.svg) | Pyridone 6 | IC50 | 940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_1e4105883592759a0b68e5545a24288d.svg) | 4-({5-Amino-1-[(2,6-Difluorophenyl)carbonyl]-1h-1,2,4-Triazol-3-Yl}amino)benzenesulfonamide | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_2cf324237228e1f753214eb9a2ce619a.svg) | Erdafitinib | IC50 | 4.47 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_bcc8f093556dc854edb8b08f9766cee0.svg) | Cudc-101 | IC50 | 3430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_f3d0fcadcce0816240114937491b30f7.svg) | 1-(2,4-Difluorophenyl)-3-(4-(6,7-dimethoxyquinolin-4-yloxy)-2-fluorophenyl)urea | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_179888a64edb35ddee0be2a16e245b3a.svg) | MK-2461 | IC50 | 39.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_6365365977462e08c2ff13fed8625161.svg) | 7-(2,6-Dichlorophenyl)-5-methyl-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-1,2,4-benzotriazin-3-amine | Ki | 493.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_a97274caafef70d6423d3784397e9e54.svg) | Pyrimidone, 22 | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_9b758bfffd41ecd8dbc5fd96a1378a28.svg) | CID 53246941 | IC50 | 320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_64f69317c84e5d1efc4211ef1e986fd2.svg) | 2-(4-Fluoroanilino)-5-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]-3-methylpyrimidin-4-one | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_969493da19549693a0acb94f703a8630.svg) | N-(4-Chlorophenyl)-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide | IC50 | 55.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_10b979513d2e855fbc4454fcc705914e.svg) | 1-[2-Amino-6-(2,6-dichlorophenyl)pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butylurea | IC50 | 130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_c6a654ab2a80479be435287d3d61f1cc.svg) | H3B-6527 | IC50 | 1980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_f8dea142aa4a3f574f20a24329144dbd.svg) | CID 118295624 | IC50 | 1.3 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5337373476537f777db31ec6dc31dd28.svg) | CID 91827382 | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_cc5bc7310bc863c88072f5adeababc04.svg) | 6H-Purin-6-one, 2-amino-1,7-dihydro-8-phenyl- | IC50 | 13460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_1acb9af54a0300732fbc15732fce477a.svg) | 4-[(2-Morpholin-4-yl-7H-purin-6-yl)amino]benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_dc2725d937b73506c3d7d4792b6e31ea.svg) | 9-Ethyl-6,6-dimethyl-8-[4-(oxetan-3-yl)piperazin-1-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_b00071ca0e36ca4f06fafeca8a36c1b6.svg) | (4-t-Butylphenyl){4-[(6,7-dimethoxy-4-quinolyl)oxy]phenyl}methanone | IC50 | 190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_fe488f1f0ab2c047ee8c00c265c5ee26.svg) | N-[2-[[5-[(2,6-Dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl]amino]-3-methylphenyl]prop-2-enamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_67b666e57b1ced47c841c60c0b226bfb.svg) | 4-(1H-Indazol-6-yl)phenol | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_482caccce5577424472b4f30ef45663d.svg) | [6-Chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_9869d4afb98ef2c3ccd6540bb969cfa4.svg) | CID 46864270 | IC50 | 1.5 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_937815501a4377d32f1ec2930f9de533.svg) | (6s)-6-Phenyl-5,6-Dihydrobenzo[h]quinazolin-2-Amine | IC50 | 1230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_b47eb0b10c004af2684a6d610b4c991d.svg) | Ethyl 8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_f4b4713d56837446ccc856142c96542c.svg) | Pyrazine-Pyridine Biheteroaryl 39 | IC50 | 2360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_5bfce131505d259ec77e7ee0501dc544.svg) | Pyrazine-Pyridine Biheteroaryl 41 | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/fibroblast-growth-factor-receptor-2_bd7ab61fd74e87578c2dfefbcc47d031.svg) | 7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | IC50 | 10000.0 [1] |