 | Palmitic acid | IC50 | 1200.0 [1] |
 | Palmitic acid | Ki | 802.0 [1] |
 | (2S,4S)-3-(6-Acetamidonaphthalen-1-yl)oxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 970.0 [1], 7080.0 [2] |
 | (2R,4R)-2,4-Diphenyl-3-[[4-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3-thiazol-2-yl]carbamoyl]cyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | 3-(Naphthyloxycarbonyl)-2,4-diphenylcyclobutanecarboxylic acid | Ki | 810.0 [1], 900.0 [2] |
 | Oleic acid | Ki | 248.0 [1] |
 | 2-((2'-(5-Ethyl-3,4-diphenyl-1H-pyrazol-1-yl)-[1,1'-biphenyl]-3-yl)oxy)acetic acid | Ki | 350.0 [1] |
 | Truxillic acid | Ki | 10000.0 [1] |
 | 2,4,6-Triisopropylbenzoic acid | IC50 | 50000.0 [1] |
 | (E)-4-[(2-Methoxycarbonyl-5-thiophen-2-ylthiophen-3-yl)amino]-4-oxobut-2-enoic acid | Ki | 3400.0 [1] |
 | 3-Carbazol-9-yl-propionic acid | IC50 | 30000.0 [1] |
 | 5-(2-(4,5-Diphenyloxazol-2-yl)phenoxy)pentanoic acid | Ki | 2000.0 [1] |
 | 6-Chloro-4-Phenyl-2-(Piperidin-1-Yl)-3-(1h-Tetrazol-5-Yl)quinoline | Ki | 86.0 [1] |
 | [[2'-(4,5-Diphenyl-2-oxazolyl)-1,1'-biphenyl-3-yl]oxy]acetic acid | Ki | 2000.0 [1] |
 | (2R,4R)-3-Naphthalen-1-yloxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 710.0 [1] |
 | (1s,2s,3s,4s)-3-{[(Naphthalen-1-Yl)oxy]carbonyl}-2,4-Diphenylcyclobutane-1-Carboxylic Acid | Ki | 790.0 [1] |
 | 2,4,6-Triisopropylbenzenesulfonic acid | IC50 | 16000.0 [1] |
 | 2-(2,3-Bis(2-chlorobenzyloxy)phenyl)acetic acid | Ki | 3.0 [1] |
 | 1,3-Cyclobutanedicarboxylic acid, 2,4-bis(4-hydroxy-3-methoxyphenyl)- | Ki | 10000.0 [1] |
 | 2-((2'-(1-Ethyl-4,5-diphenyl-1H-imidazol-2-yl)(1,1'-biphenyl)-3-yl)oxy)-acetic acid | Ki | 830.0 [1] |
 | 2-[3-[2-(1-Ethyl-4,5-diphenylimidazol-2-yl)phenyl]anilino]acetic acid | Ki | 2000.0 [1] |
 | (2S,4S)-3-[(4-Methoxyphenyl)methoxycarbonyl]-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 2150.0 [1] |
 | (2S,4S)-3-(9H-Fluoren-9-ylmethoxycarbonyl)-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 2560.0 [1] |
 | (2S,4S)-3-[3-[1-[2-[2-(2-Ethoxyethoxy)ethoxy]ethyl]triazol-4-yl]phenoxy]carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | (2S,4S)-3-[2-(2-Hydroxyphenyl)phenoxy]carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 1590.0 [1] |
 | (2S,4S)-3-(3-Ethynylphenoxy)carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 890.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-(2-phenylphenoxy)carbonylcyclobutane-1-carboxylic acid | Ki | 770.0 [1] |
 | (2S,4S)-3-(2-Iodophenoxy)carbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 1340.0 [1] |
 | (2S,4S)-3-(5-Ethynylnaphthalen-1-yl)oxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 3920.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-(4-phenylphenoxy)carbonylcyclobutane-1-carboxylic acid | Ki | 2520.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-(3-phenylphenoxy)carbonylcyclobutane-1-carboxylic acid | Ki | 850.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 180.0 [1] |
 | (2S,4S)-3-Naphthalen-1-yloxycarbonyl-2,4-bis(2-nitrophenyl)cyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | (2S,4S)-2,4-Bis(2-chlorophenyl)-3-(9H-fluoren-9-ylmethoxycarbonyl)cyclobutane-1-carboxylic acid | Ki | 890.0 [1] |
 | (2S,4S)-2,4-Bis(2-methoxyphenyl)-3-quinolin-5-yloxycarbonylcyclobutane-1-carboxylic acid | Ki | 3930.0 [1] |
 | Fabp-IN-1 | Ki | 550.0 [1] |
 | (2S,4S)-2,4-Bis(2-chlorophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 1700.0 [1] |
 | (2S,4S)-2,4-Bis(2-methoxyphenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 680.0 [1] |
 | Fabp5-IN-1 | Ki | 1720.0 [1] |
 | (2S,4S)-2,4-Bis(4-hydroxy-3-methoxyphenyl)-3-naphthalen-1-yloxycarbonylcyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | (2S,4S)-3-[(4-Fluorophenyl)methoxycarbonyl]-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 2420.0 [1] |
 | (2S,4S)-3-(2,3-Dihydro-1H-inden-2-yloxycarbonyl)-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 1570.0 [1] |
 | (2S,4S)-3-[(4-Bromophenyl)methoxycarbonyl]-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 1580.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-[(1S,2R)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 200.0 [1] |
 | Bis(oxan-4-ylmethyl) 2,4-diphenylcyclobutane-1,3-dicarboxylate | Ki | 10000.0 [1] |
 | (2S,4S)-2,4-Bis(4-hydroxyphenyl)-3-naphthalen-1-yloxycarbonylcyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | Bis[(4-methoxyphenyl)methyl] 2,4-diphenylcyclobutane-1,3-dicarboxylate | Ki | 10000.0 [1] |
 | (2S,4S)-2,4-Bis(2-nitrophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-(2,2,2-trifluoroethoxycarbonyl)cyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | (2S,4S)-2,4-Bis(2-bromophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 2760.0 [1] |
 | Dibenzyl 2,4-diphenylcyclobutane-1,3-dicarboxylate | Ki | 10000.0 [1] |
 | Bis[(4-fluorophenyl)methyl] 2,4-diphenylcyclobutane-1,3-dicarboxylate | Ki | 10000.0 [1] |
 | (2R,4R)-2,4-Diphenyl-3-[(3-phenylphenyl)carbamoyl]cyclobutane-1-carboxylic acid | Ki | 10000.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-(2,4,5-trichlorophenoxy)carbonylcyclobutane-1-carboxylic acid | Ki | 800.0 [1] |
 | (2S,4S)-2,4-Bis(2,6-dichlorophenyl)-3-[(1R,2S)-2-phenylcyclohexyl]oxycarbonylcyclobutane-1-carboxylic acid | Ki | 1230.0 [1] |
 | 2,4-Bis(3,4-dimethoxyphenyl)cyclobutane-1,3-dicarboxylic acid | Ki | 10000.0 [1] |
 | Benzeneacetic acid, 2,3-bis((2-chlorophenyl)methoxy)-alpha-hydroxy-, (alphaS)- | Ki | 33.0 [1] |
 | 2-[3-[2-(1-Methyl-4,5-diphenylimidazol-2-yl)phenyl]phenoxy]acetic acid | Ki | 830.0 [1] |
 | 2-[3-[2-[1-(2-Fluoroethyl)-4,5-diphenylimidazol-2-yl]phenyl]phenoxy]acetic acid | Ki | 2000.0 [1] |
 | 2-[3-[2-[1-(Carboxymethyl)-4,5-diphenylimidazol-2-yl]phenyl]anilino]acetic acid | Ki | 2000.0 [1] |
 | 2-[3-[2-[1-(2-Methylpropyl)-4,5-diphenylimidazol-2-yl]phenyl]anilino]acetic acid | Ki | 2000.0 [1] |
 | 2-[3-[2-(1-Methyl-4,5-diphenylimidazol-2-yl)phenyl]anilino]acetic acid | Ki | 2000.0 [1] |
 | 2-[3-[2-(3-Ethyl-4,5-diphenylfuran-2-yl)phenyl]phenoxy]acetic acid | Ki | 290.0 [1] |
 | 2-[3-[2-(4,5-Diphenyl-1H-imidazol-2-yl)phenyl]phenoxy]acetic acid | Ki | 2000.0 [1] |
 | 2-[3-[2-(4,5-Diphenyl-1H-imidazol-2-yl)phenyl]anilino]acetic acid | Ki | 2000.0 [1] |
 | 2-[3-[2-(4,5-Diphenylfuran-2-yl)phenyl]phenoxy]acetic acid | Ki | 2000.0 [1] |
 | 2-(2,3-Bis(2-chlorobenzyloxy)phenyl)-2-methoxyacetic acid | Ki | 9.0 [1] |
 | 2-[2,3-Bis[(2-chlorophenyl)methoxy]phenyl]-2-oxoacetic acid | Ki | 2.0 [1] |
 | (2S,4S)-2,4-Diphenyl-3-phenylmethoxycarbonylcyclobutane-1-carboxylic acid | Ki | 3810.0 [1] |
 | 5-Carbazol-9-yl-pentanoic acid | IC50 | 3000.0 [1] |
 | 3-(5-Bromo-indole-1-sulfonyl)-thiophene-2-carboxylic acid | IC50 | 14000.0 [1] |
 | 2-(Carbazole-9-sulfonyl)-benzoic acid | IC50 | 17000.0 [1] |
 | 3-(Carbazole-9-sulfonyl)-thiophene-2-carboxylic acid | IC50 | 9100.0 [1] |
 | 1-(2,3-Bis(2-chlorobenzyloxy)phenyl)ethane-1,2-diol | Ki | 2000.0 [1] |
 | 2-[3-[2-(5-Ethyl-3,4-diphenylpyrazol-1-yl)phenyl]phenyl]-2-hydroxyacetic acid | Ki | 550.0 [1] |
 | 3-[2-(5-Ethyl-3,4-diphenylpyrazol-1-yl)phenyl]benzoic acid | Ki | 240.0 [1] |
 | 2,3-Bis[(2,4-dichloro-3-tritiophenyl)methoxy]benzoic acid | Ki | 2.0 [1] |
 | Carbazole butanoic acid | IC50 | 6700.0 [1] |
 | (2S,4S)-3-Cyclohexyloxycarbonyl-2,4-diphenylcyclobutane-1-carboxylic acid | Ki | 2170.0 [1] |
 | 6-Chloranyl-2-Methyl-4-Phenyl-Quinoline-3-Carboxylic Acid | Ki | 23200.0 [1] |
 | 5-(6-Chloro-4-phenyl-2-piperidin-1-yl-quinolin-3-yl)-3H-[1,3,4]oxadiazole-2-thione | Ki | 133.0 [1] |
 | 6-Chloro-4-phenyl-2-propan-2-ylquinoline-3-carboxylic acid | Ki | 1200.0 [1] |
 | 6-Chloranyl-4-Phenyl-2-Piperidin-1-Yl-Quinoline-3-Carboxylic Acid | Ki | 500.0 [1] |
 | 6,8-Dichloro-4-Phenyl-2-(Piperidin-1-Yl)quinoline-3-Carboxylic Acid | Ki | 120.0 [1] |
 | 6-Chloro-8-methyl-4-phenyl-2-piperidin-1-yl-quinoline-3-carboxylic acid | Ki | 100.0 [1] |
 | 5-(6-Chloro-4-phenyl-2-piperidin-1-yl-quinolin-3-yl)-3H-[1,3,4]oxadiazol-2-one | Ki | 167.0 [1] |
 | 6-Chloro-2-dimethylamino-4-(3-isopropyl-phenyl)-quinoline-3-carboxylic acid | Ki | 4300.0 [1] |
 | 2-[3-[2-(4,5-Diphenyl-1H-pyrrol-2-yl)phenyl]phenoxy]acetic acid | Ki | 2000.0 [1] |
 | 2-[[5-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-4-methylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 30.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-4,5-dimethylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 30.0 [1] |
 | 2-[[4-Cyclopropyl-5-methyl-3-[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 30.0 [1] |
 | 3-[[4-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-5-methylthiophen-2-yl]carbamoyl]bicyclo[2.2.2]oct-2-ene-2-carboxylic acid | IC50 | 40.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 890.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-4-methyl-5-(oxetan-3-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 60.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-4-methyl-5-(oxetan-3-yl)thiophen-2-yl]carbamoyl]cyclohexene-1-carboxylic acid | IC50 | 227.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-5-methyl-4-(trifluoromethyl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 60.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-5-ethoxycarbonyl-4-methylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 130.0 [1] |
 | 2-[[3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-5-(dimethylcarbamoyl)-4-methylthiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 2709.7 [1] |
 | 2-[[5-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 125.8 [1] |
 | 2-[[4-Cyclopropyl-3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]carbamoyl]cyclopentene-1-carboxylic acid | IC50 | 38.8 [1] |