 | 2-((2'-(5-Ethyl-3,4-diphenyl-1H-pyrazol-1-yl)-[1,1'-biphenyl]-3-yl)oxy)acetic acid | IC50 | 221.0 [1] |
 | 2-((2'-(5-Ethyl-3,4-diphenyl-1H-pyrazol-1-yl)-[1,1'-biphenyl]-3-yl)oxy)acetic acid | Ki | 2.0 [1], 7.4 [2], 15.0 [3], 160.0 [4], 220.0 [5] |
 | Linoleic acid | IC50 | 1000.0 [1], 13600.0 [2], 17700.0 [3] |
 | Linoleic acid | Ki | 6800.0 [1] |
 | Oleic acid | IC50 | 26100.0 [1] |
 | Oleic acid | Ki | 185.0 [1], 1500.0 [2] |
 | 2-(2-(3,5-Dichlorophenylamino)-2-oxoethylthio)acetic acid | IC50 | 1000.0 [1], 13500.0 [2] |
 | 2-(2-(3,5-Dichlorophenylamino)-2-oxoethylthio)acetic acid | Ki | 1660.0 [1] |
 | Palmitic acid | IC50 | 930.0 [1] |
 | Palmitic acid | Ki | 336.0 [1] |
 | 2-(2-(2-Chloro-6-phenoxybenzylamino)-2-oxoethylthio)acetic acid | IC50 | 3100.0 [1], 42200.0 [2] |
 | 2-[3-[2-(1,5-Diphenylpyrazol-3-yl)phenyl]phenoxy]acetic acid | IC50 | 987.0 [1] |
 | 2-[3-[2-(1,5-Diphenylpyrazol-3-yl)phenyl]phenoxy]acetic acid | Ki | 32.0 [1] |
 | 6-Chloro-4-Phenyl-2-(Piperidin-1-Yl)-3-(1h-Tetrazol-5-Yl)quinoline | Ki | 11.0 [1], 87.0 [2] |
 | [[2'-(4,5-Diphenyl-2-oxazolyl)-1,1'-biphenyl-3-yl]oxy]acetic acid | Ki | 6.0 [1], 95.0 [2] |
 | 2-((2'-(1-Ethyl-4,5-diphenyl-1H-imidazol-2-yl)(1,1'-biphenyl)-3-yl)oxy)-acetic acid | Ki | 2.0 [1], 3.3 [2] |
 | 2-[3-[2-(1-Ethyl-4,5-diphenylimidazol-2-yl)phenyl]anilino]acetic acid | Ki | 3.4 [1], 13.0 [2] |
 | 2-[3-[2-(1-Methyl-4,5-diphenylimidazol-2-yl)phenyl]phenoxy]acetic acid | Ki | 2.0 [1], 13.0 [2] |
 | 2-[3-[2-[1-(2-Fluoroethyl)-4,5-diphenylimidazol-2-yl]phenyl]phenoxy]acetic acid | Ki | 2.0 [1], 8.7 [2] |
 | 2-[3-[2-(1-Methyl-4,5-diphenylimidazol-2-yl)phenyl]anilino]acetic acid | Ki | 2.7 [1], 48.0 [2] |
 | 2-[3-[2-(3-Ethyl-4,5-diphenylfuran-2-yl)phenyl]phenoxy]acetic acid | Ki | 3.5 [1], 32.0 [2] |
 | 2-[3-[2-(4,5-Diphenyl-1H-imidazol-2-yl)phenyl]anilino]acetic acid | Ki | 18.0 [1], 300.0 [2] |
 | 9-Propyl-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 670.0 [1], 730.0 [2] |
 | 5-(2-Carbamoylbenzyl)-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-4-carboxylic acid | IC50 | 98.0 [1], 400.0 [2] |
 | 2-[2-Oxo-2-[(2-piperidin-1-ylphenyl)methylamino]ethyl]sulfanylacetic acid | IC50 | 4100.0 [1], 56300.0 [2] |
 | 2-(2-(3-Chloro-4-fluorophenylamino)-2-oxoethylthio)acetic acid | IC50 | 4400.0 [1], 59500.0 [2] |
 | 5-(3-Carbamoylbenzyl)-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-4-carboxylic acid | IC50 | 69.0 [1], 450.0 [2] |
 | 5-(2-(Trifluoromethyl)benzyl)-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-4-carboxylic acid | IC50 | 49.0 [1], 650.0 [2] |
 | 5-Propyl-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-4-carboxylic acid | IC50 | 430.0 [1], 580.0 [2] |
 | 5-Benzyl-5,6,7,8,9,10-hexahydrocyclohepta[b]indole-4-carboxylic acid | IC50 | 96.0 [1], 590.0 [2] |
 | 8-Anilino-1-naphthalenesulfonic acid | Ki | 1000.0 [1] |
 | 2,4,6-Triisopropylbenzoic acid | IC50 | 4000.0 [1] |
 | [(4-{[(4-Chlorophenyl)sulfonyl]amino}-1-hydroxy-2-naphthyl)thio]acetic acid | Ki | 2300.0 [1] |
 | Carbazol-9-yl-acetic acid | IC50 | 100000.0 [1] |
 | 4-(4-Methylphenyl)-2-[(4-methylphenyl)sulfanyl]-4-oxobutanoic acid | IC50 | 100000.0 [1] |
 | (E)-4-[(2-Methoxycarbonyl-5-thiophen-2-ylthiophen-3-yl)amino]-4-oxobut-2-enoic acid | Ki | 670.0 [1] |
 | 3-(2-Phenyl-1H-indol-1-yl)propanoic acid | Ki | 1400.0 [1] |
 | 2-[(4-Chlorobenzyl)amino]-6-methylpyrimidin-4(3H)-one | IC50 | 100000.0 [1] |
 | 2-[2-[[4-(4-Methoxyphenyl)-2-methyl-5-(trifluoromethyl)pyrazol-3-yl]amino]-2-oxoethyl]sulfanylacetic acid | IC50 | 100000.0 [1] |
 | 3-Carbazol-9-yl-propionic acid | IC50 | 9400.0 [1] |
 | 5-(2-(4,5-Diphenyloxazol-2-yl)phenoxy)pentanoic acid | Ki | 58.0 [1] |
 | 10-Chloro-1-azapentacyclo[10.6.1.03,7.08,19.013,17]nonadeca-5,8,10,12(19),14-pentaene-2-carboxylic acid | Ki | 690.0 [1] |
 | 9,11-Dimethyl-1-azapentacyclo[10.6.1.03,7.08,19.013,17]nonadeca-5,8,10,12(19),14-pentaene-2-carboxylic acid | Ki | 610.0 [1] |
 | 1-((2,4,6-Triisopropylphenyl)sulfonyl)-1H-imidazole | IC50 | 16800.0 [1] |
 | CID 49872404 | Ki | 1.0 [1] |
 | 4-[2-[1-(4-Bromophenyl)-5-phenyl-1H-pyrazole-3-yl]phenoxy]butyric acid | IC50 | 5640.0 [1] |
 | 2,6-Bis((1H-benzo[d]imidazol-2-ylthio)methyl)pyridine | IC50 | 100000.0 [1] |
 | 9-Benzyl-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 590.0 [1] |
 | 9-(3-Fluorobenzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 400.0 [1] |
 | 9-[2-(Trifluoromethyl)benzyl]-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 400.0 [1] |
 | 2,4,6-Triisopropylbenzenesulfonic acid | IC50 | 7900.0 [1] |
 | 9-(4-Fluorobenzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 830.0 [1] |
 | 9-(3-Methoxybenzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 550.0 [1] |
 | 9-(4-Methoxybenzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 2680.0 [1] |
 | 2-(2,3-Bis(2-chlorobenzyloxy)phenyl)acetic acid | Ki | 16.0 [1] |
 | 9-(2-Methoxybenzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 600.0 [1] |
 | 9-(4-(Trifluoromethyl)benzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 2390.0 [1] |
 | 9-(3-(Trifluoromethyl)benzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 1660.0 [1] |
 | 9-(2-Methylbenzyl)-8-(prop-1-en-2-yl)-2,3,4,9-tetrahydro-1H-fluorene | IC50 | 400.0 [1] |
 | 9-(4-Methylbenzyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxylic acid | IC50 | 1090.0 [1] |
 | 2-Methyl-1-[2,4,6-tri(propan-2-yl)phenyl]sulfonylbenzimidazole | IC50 | 100000.0 [1] |
 | 9-Benzyl-2,3,4,9-tetrahydro-1H-carbazole-7-carboxylic acid | IC50 | 750.0 [1] |
 | 3-[(5E)-5-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoic acid | Ki | 2500.0 [1] |
 | 3-[5-Cyclopropyl-3-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(3-propan-2-yloxyphenyl)indol-1-yl]propanoic acid | Ki | 30.0 [1] |
 | 6-Chloro-5-(2-nitrophenyl)sulfanyl-1-azapentacyclo[10.6.1.03,7.08,19.013,17]nonadeca-8,10,12(19),14-tetraene-2-carboxylic acid | Ki | 3100.0 [1] |
 | 2-Fluoranyl-5-[(4-methoxynaphthalen-1-yl)sulfonylamino]benzoic acid | Ki | 210.0 [1] |
 | 4-Fluoranyl-3-[(4-methoxynaphthalen-1-yl)sulfonylamino]benzoic acid | Ki | 200.0 [1] |
 | 2-Fluoranyl-3-[(4-methoxynaphthalen-1-yl)sulfonylamino]benzoic acid | Ki | 7750.0 [1] |
 | 5-[(4-Methoxynaphthalen-1-yl)sulfonylamino]pentanoic acid | Ki | 590.0 [1] |
 | 5-[(4-Bromanylnaphthalen-1-yl)sulfonylamino]pentanoic acid | Ki | 1160.0 [1] |
 | 2-(4-Chloro-benzylamino)-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 2900.0 [1] |
 | 2-[(2-Oxo-2-piperidin-1-ylethyl)thio]-6-(trifluoromethyl)pyrimidin-4(1H)-one | IC50 | 1000.0 [1] |
 | 2-[[(E)-3-(2,5-Dichloroanilino)-1-hydroxy-3-oxo-1-phenylprop-1-en-2-yl]diazenyl]benzoic acid | Ki | 10300.0 [1] |
 | 3-[2-[(Z)-[2-(3,4-Dimethylphenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]pyrrol-1-yl]benzoic acid | Ki | 3600.0 [1] |
 | 2-(4-Chloro-benzylamino)-6-ethyl-pyrimidin-4-ol | IC50 | 47000.0 [1] |
 | 2-Phenylamino-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 6-Trifluoromethyl-2-(4-methoxy-phenylmethyl)thio-4-pyrimidinol | IC50 | 600.0 [1] |
 | 2-(4-Chloro-benzylamino)-6-phenyl-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 2-(Benzyl-methyl-amino)-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 24000.0 [1] |
 | 2-(4-Methoxy-benzylamino)-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 3900.0 [1] |
 | 2-(3-Chloro-benzylamino)-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 33000.0 [1] |
 | 2-(4-Chloro-benzylamino)-6-(2-fluoro-phenyl)-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 2-[(Biphenyl-4-ylmethyl)-amino]-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 2-Benzylamino-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 33000.0 [1] |
 | 2-[(4-Chloro-benzyl)-methyl-amino]-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 4000.0 [1] |
 | 2-(2-Chloro-benzylamino)-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 23000.0 [1] |
 | 2-(4-Methyl-benzylamino)-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 33000.0 [1] |
 | 2-[2-(4-Methoxy-phenyl)-ethyl]-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 25000.0 [1] |
 | 2-(4-Hydroxy-6-trifluoromethyl-pyrimidin-2-ylamino)-1-piperidin-1-yl-ethanone | IC50 | 37000.0 [1] |
 | 2-Phenethyl-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 2-[(Pyridin-4-ylmethyl)-amino]-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 2-Phenethylamino-6-trifluoromethyl-pyrimidin-4-ol | IC50 | 100000.0 [1] |
 | 5-(1-Phenyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazol-3-yl)pent-4-enoic acid | IC50 | 1100.0 [1] |
 | 4-[[(4-Methoxynaphthalen-1-yl)sulfonylamino]methyl]benzoic acid | Ki | 760.0 [1] |
 | 2,4-Difluoro-5-[(4-methoxynaphthalen-1-yl)sulfonylamino]benzoic acid | Ki | 230.0 [1] |
 | 5-[(2,3,4,5,6-Pentamethylphenyl)sulfonylamino]pentanoic acid | Ki | 910.0 [1] |
 | 3-[[(4-Methoxynaphthalen-1-yl)sulfonylamino]methyl]benzoic acid | Ki | 2120.0 [1] |
 | 4-Methoxy-3-[(4-methoxynaphthalen-1-yl)sulfonylamino]benzoic acid | Ki | 6140.0 [1] |
 | 4-Chloro-3-[(4-methoxynaphthalen-1-yl)sulfonylamino]benzoic acid | Ki | 930.0 [1] |
 | 3-[3-[(4-Methoxynaphthalen-1-yl)sulfonylamino]phenyl]propanoic acid | Ki | 580.0 [1] |