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Excitatory amino acid transporter 2 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
(3s)-3-(Benzyloxy)-L-Aspartic AcidIC50954.99 [1], 1905.46 [2], 3800.0 [3], 164000.0 [4]
N-[4-(2-Bromo-4,5-difluorophenoxy)phenyl]-L-asparagineIC5070.79 [1], 80.0 [2], 130.0 [3]
(2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic AcidIC50300000.0 [1], 3162277.66 [2]
(2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic AcidKi3162277.66 [1]
Glutamic acidIC5052480.75 [1]
Glutamic acidKi63095.73 [1]
Tfb-tboaIC5010.0 [1], 17.0 [2]
2-Amino-3-phenylmethoxybutanedioic acidIC501995.26 [1], 7000.0 [2]
(1R,4S,5R,6S)-3-Azabicyclo[3.3.0]octane-4,6-dicarboxylic acidKi52000.0 [1]
(2S,4R)-4-(3-Amino-3-oxopropyl)glutamic acidIC501000000.0 [1]
(2S,4R)-4-(3-Amino-3-oxopropyl)glutamic acidKi316227.77 [1]
(4r)-4-[3-(Methylamino)-3-Oxopropyl]-L-Glutamic AcidIC501000000.0 [1]
(4r)-4-[3-(Methylamino)-3-Oxopropyl]-L-Glutamic AcidKi630957.34 [1]
1,2,4-Butanetricarboxylic acid, 4-amino-, (2S,4S)-IC503162277.66 [1]
1,2,4-Butanetricarboxylic acid, 4-amino-, (2S,4S)-Ki3162277.66 [1]
(2s,4r)-4-(3-Methoxy-3-Oxopropyl) Glutamic AcidIC50316227.77 [1]
(2s,4r)-4-(3-Methoxy-3-Oxopropyl) Glutamic AcidKi158489.32 [1]
(2S,4R)-4-(3-Benzylamino-3-oxopropyl)glutamic acidIC50316227.77 [1]
(2S,4R)-4-(3-Benzylamino-3-oxopropyl)glutamic acidKi398107.17 [1]
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acidIC5079432.82 [1]
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acidKi100000.0 [1]
(2S,4S)-4-(Hydroxymethyl)glutamic AcidIC50316227.77 [1]
(2S,4S)-4-(Hydroxymethyl)glutamic AcidKi125892.54 [1]
(2S,4S)-4-(Benzyloxymethyl)glutamic AcidIC50316227.77 [1]
(2S,4S)-4-(Benzyloxymethyl)glutamic AcidKi316227.77 [1]
(1R,2S)-2-[(S)-Amino(carboxy)methyl]-2-methylcyclobutane-1-carboxylic acidKi6600.0 [1], 125892.54 [2]
(2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acidIC503162277.66 [1]
(2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acidKi3162277.66 [1]
(2S)-2-Amino-4-oxo-4-[4-[3-(trifluoromethyl)phenyl]anilino]butanoic acidIC5010.0 [1], 60.0 [2]
Aspartic acidIC5033113.11 [1]
alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACIDIC501000000.0 [1]
Dihydrokainic acidIC5079432.82 [1]
DL-Threo-beta-Hydroxyaspartic acidIC509549.93 [1]
HinokininIC50100000.0 [1]
2S,4R-4-MethylglutamateKi11748.98 [1]
2-Amino-5,6,7,8-tetrahydro-4-(4-methoxyphenyl)-7-(naphthalen-1-YL)-5-oxo-4H-chromene-3-carbonitrileIC50316227.77 [1]
L-beta-Threo-benzyl-aspartateIC5042657.95 [1]
2-Amino-4-methyl-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50300000.0 [1]
2-Amino-4-(1,3-benzodioxol-5-yl)-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50316227.77 [1]
2-Amino-5-oxo-7-phenyl-4-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50316227.77 [1]
2-Amino-3-(2,5-dihydro-5-oxo-4-isoxazolyl)propanoic acidIC50240000.0 [1]
(2S)-2-Amino-4-(9H-fluoren-2-ylamino)-4-oxobutanoic acidIC50700.0 [1]
(2S,4R)-4-Propylglutamic acidKi20892.96 [1]
2-Amino-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50316227.77 [1]
2-Amino-4-(2-fluorophenyl)-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromen-3-yl cyanideIC50100000.0 [1]
(1s,2r)-2-[(S)-Amino(Carboxy)methyl]cyclobutanecarboxylic AcidKi6309.57 [1]
(1R,2S)-2-((S)-Amino(carboxy)methyl)cyclopropanecarboxylic acidIC504000.0 [1]
2-Amino-4-(2-fluorophenyl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50316227.77 [1]
(RS)-2-amino-3-(1-hydroxy-1,2,3-triazol-5-yl)propionateIC50300000.0 [1]
(2S,4R)-4-Pentylglutamic acidKi67608.3 [1]
(3S)-3-(1-Naphthylmethoxy)-L-aspartic acidIC501300.0 [1]
(3S)-3-(2-Naphthylmethoxy)-L-aspartic acidIC502200.0 [1]
2-Amino-4-(4-methoxyphenyl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-4-[4-(methylsulfanyl)phenyl]-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50100000.0 [1]
2-Amino-4-(4-nitrophenyl)-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromen-3-yl cyanideIC50100000.0 [1]
2-Amino-4-(1H-indol-3-yl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-5-oxo-7-phenyl-4-thiophen-2-yl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-5-oxo-7-phenyl-4-(4-phenylphenyl)-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-4-(4-bromothiophen-2-yl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-4-(2,3-dimethoxyphenyl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-7-(2-chlorophenyl)-4-(4-methoxyphenyl)-5-oxo-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50316227.77 [1]
2-Amino-4-(1,3-benzodioxol-5-yl)-7-methyl-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50316227.77 [1]
(4r)-4-{3-[Hydroxy(Methyl)amino]-3-Oxopropyl}-L-Glutamic AcidIC501000000.0 [1]
(2S,4R)-2-Amino-4-(2-cyanoethyl)pentanedioic acidIC5024000.0 [1]
(2S,4R)-2-Amino-4-[3-(hydroxyamino)-3-oxopropyl]pentanedioic acidIC50700000.0 [1]
(2S,4R)-2-Amino-4-(2-aminoethyl)pentanedioic acidIC501000000.0 [1]
(2S,4R)-2-Amino-4-(3-aminopropyl)pentanedioic acidIC501000000.0 [1]
(2S,4R)-4-Ethylglutamic acidKi10715.19 [1]
5-Methyl-3-hydroxy-alpha-amino-3H-1,2,3-triazole-4-propionic acidIC50490000.0 [1]
(3S,5S)-2-Aza-bicyclo[2.2.1]heptane-3,5-dicarboxylic acidKi400000.0 [1]
(2S,3S)-Pyrrolidine-2,3-dicarboxylic acidKi12000.0 [1]
5-Methyl-1-hydroxy-alpha-amino-1H-imidazole-2-propionic acidIC501000000.0 [1]
4-Methyl-2-hydroxy-alpha-amino-2H-pyrazole-3-propionic acidIC501000000.0 [1]
2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic acidIC50430000.0 [1]
2-Methyl-3-hydroxy-alpha-amino-3H-imidazole-4-propionic acidIC501000000.0 [1]
2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic acidIC501000000.0 [1]
2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic acidIC501000000.0 [1]
5-Methyl-3-hydroxy-alpha-amino-3H-imidazole-4-propionic acidIC501000000.0 [1]
(2S,4R)-4-Isobutylglutamic acidKi21877.62 [1]
(2S)-2-Amino-4-[4-(2-methylphenyl)anilino]-4-oxobutanoic acidIC50100.0 [1]
(2S,4R)-4-Isopentylglutamic acidKi21877.62 [1]
(2S,4R)-4-Butylglutamic acidKi38018.94 [1]
(2S)-2-Amino-4-oxo-4-[[7-(trifluoromethyl)-9H-fluoren-2-yl]amino]butanoic acidIC50100.0 [1]
(3S)-3-Methoxyaspartic acidIC502000.0 [1]
(1R,2S)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(1S,2S)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(1R,2R)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(1S,2R)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(2S,3S)-2-Amino-3-[[3-[[2-(trifluoromethyl)benzoyl]amino]phenyl]methoxy]butanedioic acidIC5085.11 [1]
(2S)-2-Amino-3-[[4-(trifluoromethyl)phenyl]sulfonylamino]butanedioic acidIC5050118.72 [1]
(2S)-2-Amino-3-[(3,4-difluorophenyl)sulfonylamino]butanedioic acidIC501096.48 [1]
(2S,3R)-2-Amino-3-(benzenesulfonamido)butanedioic acidIC50300000.0 [1]
(2S)-2-Amino-3-(thiophen-2-ylsulfonylamino)butanedioic acidIC507244.36 [1]
(2S)-2-Amino-3-(phenoxycarbonylamino)butanedioic acidIC50316227.77 [1]
(2S)-2-Amino-3-[(4-methoxyphenyl)sulfonylamino]butanedioic acidIC5031622.78 [1]
(2S)-2-Amino-3-[(4-tert-butylphenyl)sulfonylamino]butanedioic acidIC5050118.72 [1]
(2S)-2-Amino-3-(benzylsulfonylamino)butanedioic acidIC5060255.96 [1]
(2S)-2-Amino-3-[[3-(trifluoromethyl)phenyl]sulfonylamino]butanedioic acidIC502800.0 [1]
(2S)-2-Amino-3-[(4-nitrophenyl)sulfonylamino]butanedioic acidIC5050118.72 [1]
(2S)-2-Amino-3-[(2-chlorophenyl)sulfonylamino]butanedioic acidIC503300.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Excitatory amino acid transporter 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/excitatory-amino-acid-transporter-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Excitatory amino acid transporter 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/excitatory-amino-acid-transporter-2-inhibitors-ic50-ki.
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