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Excitatory amino acid transporter 1 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
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▼
2-Amino-5,6,7,8-tetrahydro-4-(4-methoxyphenyl)-7-(naphthalen-1-YL)-5-oxo-4H-chromene-3-carbonitrileIC50123.03 [1], 660.0 [2], 660.69 [3]
(3s)-3-(Benzyloxy)-L-Aspartic AcidIC501621.81 [1], 2089.3 [2], 817000.0 [3]
2-Amino-4-methyl-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC509120.11 [1], 9200.0 [2]
(2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic AcidIC50300000.0 [1], 3162277.66 [2]
(2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic AcidKi3162277.66 [1]
2-Amino-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50300000.0 [1], 316227.77 [2]
Glutamic acidIC5011481.54 [1]
Glutamic acidKi31622.78 [1]
N-[4-(2-Bromo-4,5-difluorophenoxy)phenyl]-L-asparagineIC50851.14 [1], 5000.0 [2]
2-Amino-3-phenylmethoxybutanedioic acidIC503162.28 [1], 48000.0 [2]
(2S,4R)-4-(3-Amino-3-oxopropyl)glutamic acidIC503162277.66 [1]
(2S,4R)-4-(3-Amino-3-oxopropyl)glutamic acidKi3162277.66 [1]
(4r)-4-[3-(Methylamino)-3-Oxopropyl]-L-Glutamic AcidIC501000000.0 [1]
(4r)-4-[3-(Methylamino)-3-Oxopropyl]-L-Glutamic AcidKi3162277.66 [1]
1,2,4-Butanetricarboxylic acid, 4-amino-, (2S,4S)-IC503162277.66 [1]
1,2,4-Butanetricarboxylic acid, 4-amino-, (2S,4S)-Ki3162277.66 [1]
(2s,4r)-4-(3-Methoxy-3-Oxopropyl) Glutamic AcidIC501000000.0 [1]
(2s,4r)-4-(3-Methoxy-3-Oxopropyl) Glutamic AcidKi3162277.66 [1]
2-Amino-4-(2-fluorophenyl)-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromen-3-yl cyanideIC504786.3 [1]
2-Amino-4-(2-fluorophenyl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50316227.77 [1]
(RS)-2-amino-3-(1-hydroxy-1,2,3-triazol-5-yl)propionateIC50100000.0 [1]
2-Amino-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC503900.0 [1], 6309.57 [2]
(2S,4R)-4-(3-Benzylamino-3-oxopropyl)glutamic acidIC501000000.0 [1]
(2S,4R)-4-(3-Benzylamino-3-oxopropyl)glutamic acidKi1000000.0 [1]
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acidIC501000000.0 [1]
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acidKi3162277.66 [1]
(2S,4S)-4-(Hydroxymethyl)glutamic AcidIC503162277.66 [1]
(2S,4S)-4-(Hydroxymethyl)glutamic AcidKi3162277.66 [1]
(2S,4S)-4-(Benzyloxymethyl)glutamic AcidIC501000000.0 [1]
(2S,4S)-4-(Benzyloxymethyl)glutamic AcidKi501187.23 [1]
2-Amino-4-methyl-7-naphthalen-1-yl-5-oxo-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50338.84 [1], 420.0 [2]
2-Amino-4-(1,3-benzodioxol-5-yl)-7-methyl-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC50316227.77 [1]
2-Amino-7-benzyl-4-(4-methoxyphenyl)-5-oxo-4,6,7,8-tetrahydrochromene-3-carbonitrileIC504786.3 [1], 5100.0 [2]
(2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acidIC503162277.66 [1]
(2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acidKi3162277.66 [1]
Aspartic acidIC509332.54 [1]
alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACIDIC501000000.0 [1]
Dihydrokainic acidIC503162277.66 [1]
DL-Threo-beta-Hydroxyaspartic acidIC503890.45 [1]
HinokininIC50500000.0 [1]
L-Serine O-sulfateIC50100000.0 [1]
Tfb-tboaIC503.55 [1]
L-beta-Threo-benzyl-aspartateIC5051286.14 [1]
2-Amino-4-(1,3-benzodioxol-5-yl)-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC503981.07 [1]
2-Amino-5-oxo-7-phenyl-4-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC5031622.78 [1]
2-Amino-3-(2,5-dihydro-5-oxo-4-isoxazolyl)propanoic acidIC50270000.0 [1]
(2S)-2-Amino-4-(9H-fluoren-2-ylamino)-4-oxobutanoic acidIC50300.0 [1]
(1R,4S,5R,6S)-3-Azabicyclo[3.3.0]octane-4,6-dicarboxylic acidKi127000.0 [1]
(2S,4R)-4-Propylglutamic acidKi10232.93 [1]
(1s,2r)-2-[(S)-Amino(Carboxy)methyl]cyclobutanecarboxylic AcidKi200000.0 [1]
(2S,4R)-4-Pentylglutamic acidKi117489.76 [1]
(3S)-3-(1-Naphthylmethoxy)-L-aspartic acidIC5015000.0 [1]
(3S)-3-(2-Naphthylmethoxy)-L-aspartic acidIC5016000.0 [1]
2-Amino-4-(4-methoxyphenyl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC502290.87 [1]
2-Amino-4-[4-(methylsulfanyl)phenyl]-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrileIC502754.23 [1]
2-Amino-4-(4-nitrophenyl)-5-oxo-7-phenyl-5,6,7,8-tetrahydro-4H-chromen-3-yl cyanideIC503630.78 [1]
2-Amino-4-(1H-indol-3-yl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC50100000.0 [1]
2-Amino-5-oxo-7-phenyl-4-thiophen-2-yl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC5014125.38 [1]
2-Amino-5-oxo-7-phenyl-4-(4-phenylphenyl)-4,6,7,8-tetrahydrochromene-3-carbonitrileIC502137.96 [1]
2-Amino-4-(4-bromothiophen-2-yl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC504677.35 [1]
2-Amino-4-(2,3-dimethoxyphenyl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrileIC5050118.72 [1]
2-Amino-7-(2-chlorophenyl)-4-(4-methoxyphenyl)-5-oxo-4,6,7,8-tetrahydrochromene-3-carbonitrileIC503235.94 [1]
(4r)-4-{3-[Hydroxy(Methyl)amino]-3-Oxopropyl}-L-Glutamic AcidIC503000000.0 [1]
(2S,4R)-2-Amino-4-(2-cyanoethyl)pentanedioic acidIC50200000.0 [1]
(2S,4R)-2-Amino-4-[3-(hydroxyamino)-3-oxopropyl]pentanedioic acidIC501000000.0 [1]
(2S,4R)-2-Amino-4-(2-aminoethyl)pentanedioic acidIC501000000.0 [1]
(2S,4R)-2-Amino-4-(3-aminopropyl)pentanedioic acidIC501000000.0 [1]
(1R,2S)-2-[(S)-Amino(carboxy)methyl]-2-methylcyclobutane-1-carboxylic acidKi200000.0 [1]
(2S,4R)-4-Ethylglutamic acidKi22908.68 [1]
5-Methyl-3-hydroxy-alpha-amino-3H-1,2,3-triazole-4-propionic acidIC501000000.0 [1]
(3S,5S)-2-Aza-bicyclo[2.2.1]heptane-3,5-dicarboxylic acidKi400000.0 [1]
5-Methyl-1-hydroxy-alpha-amino-1H-imidazole-2-propionic acidIC501000000.0 [1]
4-Methyl-2-hydroxy-alpha-amino-2H-pyrazole-3-propionic acidIC501000000.0 [1]
2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic acidIC501000000.0 [1]
2-Methyl-3-hydroxy-alpha-amino-3H-imidazole-4-propionic acidIC501000000.0 [1]
2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic acidIC501000000.0 [1]
2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic acidIC501000000.0 [1]
5-Methyl-3-hydroxy-alpha-amino-3H-imidazole-4-propionic acidIC501000000.0 [1]
(2S,4R)-4-Isobutylglutamic acidKi55000.0 [1]
(2S)-2-Amino-4-[4-(2-methylphenyl)anilino]-4-oxobutanoic acidIC502000.0 [1]
(2S,4R)-4-Isopentylglutamic acidKi28840.32 [1]
(2S,4R)-4-Butylglutamic acidKi50000.0 [1]
(2S)-2-Amino-4-oxo-4-[[7-(trifluoromethyl)-9H-fluoren-2-yl]amino]butanoic acidIC503800.0 [1]
(3S)-3-Methoxyaspartic acidIC5069000.0 [1]
(1R,2S)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(1S,2S)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(1R,2R)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(1S,2R)-1-[(2S)-2-Amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acidIC50300000.0 [1]
(2S,3S)-2-Amino-3-[[3-[[2-(trifluoromethyl)benzoyl]amino]phenyl]methoxy]butanedioic acidIC5030.9 [1]
(2S)-2-Amino-3-[[4-(trifluoromethyl)phenyl]sulfonylamino]butanedioic acidIC5031622.78 [1]
(2S)-2-Amino-3-[(3,4-difluorophenyl)sulfonylamino]butanedioic acidIC50794.33 [1]
(2S,3R)-2-Amino-3-(benzenesulfonamido)butanedioic acidIC50200000.0 [1]
(2S)-2-Amino-3-(thiophen-2-ylsulfonylamino)butanedioic acidIC509332.54 [1]
(2S)-2-Amino-3-(phenoxycarbonylamino)butanedioic acidIC5079432.82 [1]
(2S)-2-Amino-3-[(4-methoxyphenyl)sulfonylamino]butanedioic acidIC504073.8 [1]
(2S)-2-Amino-3-[(4-tert-butylphenyl)sulfonylamino]butanedioic acidIC50300000.0 [1]
(2S)-2-Amino-3-(benzylsulfonylamino)butanedioic acidIC5048977.88 [1]
(2S)-2-Amino-3-[[3-(trifluoromethyl)phenyl]sulfonylamino]butanedioic acidIC50100000.0 [1]
(2S)-2-Amino-3-[(4-nitrophenyl)sulfonylamino]butanedioic acidIC5012882.5 [1]
(2S)-2-Amino-3-[(2-chlorophenyl)sulfonylamino]butanedioic acidIC501700.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Excitatory amino acid transporter 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/excitatory-amino-acid-transporter-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Excitatory amino acid transporter 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/excitatory-amino-acid-transporter-1-inhibitors-ic50-ki.
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