Eukaryotic initiation factor 4A-I Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(1R,2R,3S,3Ar,8bS)-1,8b-dihydroxy-N,6,8-trimethoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxamide	IC50	0.5 [1], 20.0 [2]
	Hippuristanol	IC50	3100.0 [1]
	Eif4A3-IN-2	IC50	100000.0 [1]
	4-Chloro-7-fluoro-6-propan-2-yl-1H-indole-2-carboxylic acid	IC50	100000.0 [1]
	6-Benzyl-3-[3-(1,3-thiazol-5-ylmethoxy)phenyl]-1,4-dihydropyrido[4,3-d]pyrimidine-2,7-dione	IC50	100000.0 [1]
	(3S,3'R,5'S)-5-Fluoro-3'-methyl-1'-(1-methylimidazole-4-carbonyl)-5'-(2-methylpropyl)spiro[1H-indole-3,2'-pyrrolidine]-2-one	IC50	100000.0 [1]
	(3S,3'R,5'S)-1'-(1-Benzylimidazole-4-carbonyl)-5-fluoro-3'-methyl-5'-(2-methylpropyl)spiro[1H-indole-3,2'-pyrrolidine]-2-one	IC50	100000.0 [1]
	6-Benzyl-3-(3-phenylmethoxyphenyl)-1,4-dihydropyrido[4,3-d]pyrimidine-2,7-dione	IC50	100000.0 [1]
	7-Fluoro-6-propan-2-yl-1H-indole-2-carboxylic acid	IC50	100000.0 [1]
	Eif4A3-IN-1	IC50	100000.0 [1]
	(3R,3'S,5'R)-1'-(1-Benzylimidazole-4-carbonyl)-5-fluoro-3'-methyl-5'-(2-methylpropyl)spiro[1H-indole-3,2'-pyrrolidine]-2-one	IC50	100000.0 [1]
	6-Benzyl-3-[2-(3-fluoropyridin-2-yl)-6-methyl-3,4-dihydro-2H-chromen-7-yl]-1,4-dihydropyrido[4,3-d]pyrimidine-2,7-dione	IC50	100000.0 [1]
	4-Chloro-6-propan-2-yl-1H-indole-2-carboxylic acid	IC50	100000.0 [1]
	(3R,3'S,5'R)-5-Fluoro-3'-methyl-1'-(1-methylimidazole-4-carbonyl)-5'-(2-methylpropyl)spiro[1H-indole-3,2'-pyrrolidine]-2-one	IC50	100000.0 [1]
	6-Benzyl-3-[3-(pyridin-3-ylmethoxy)phenyl]-1,4-dihydropyrido[4,3-d]pyrimidine-2,7-dione	IC50	100000.0 [1]
	5-[(3S)-4-(5-Bromopyridine-2-carbonyl)-3-(4-chlorophenyl)piperazine-1-carbonyl]-1-phenyl-3-[3-(trifluoromethyl)phenyl]pyridin-2-one	IC50	100000.0 [1]
	3-[5-[(3S)-4-(5-Bromopyridine-2-carbonyl)-3-(4-chlorophenyl)piperazine-1-carbonyl]-1-methyl-2-oxopyridin-3-yl]benzonitrile	IC50	100000.0 [1]
	3-[5-[(Z)-(2-Cyclohexyl-5-imino-7-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-6-ylidene)methyl]furan-2-yl]benzoic acid	IC50	57000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 18 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Eukaryotic initiation factor 4A-I Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/eukaryotic-initiation-factor-4a-i-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Eukaryotic initiation factor 4A-I Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/eukaryotic-initiation-factor-4a-i-inhibitors-ic50-ki.
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