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Estrogen receptor beta Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
EstradiolIC503.6 [1]
EstradiolKi0.01 [1]
RaloxifeneIC5012.0 [1]
GenisteinIC509.7 [1], 10.0 [2], 83.0 [3], 395.0 [4]
GenisteinKi0.59 [1], 24.0 [2]
TamoxifenIC501000.0 [1], 1660.0 [2]
TamoxifenKi0.51 [1]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-(2-piperidin-1-ylethoxy)phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5043.0 [1], 45.0 [2]
(Z)-4-(1-(4-(2-(Dimethylamino)ethoxy)-phenyl)-2-phenylbut-1-en-1-yl)phenolIC501.0 [1], 20.0 [2], 26.1 [3], 100.0 [4]
(Z)-4-(1-(4-(2-(Dimethylamino)ethoxy)-phenyl)-2-phenylbut-1-en-1-yl)phenolKi0.01 [1], 1.7 [2], 3.16 [3]
DaidzeinIC50303.0 [1], 1100.0 [2], 1200.0 [3], 2800.0 [4]
DaidzeinKi300.0 [1]
FulvestrantIC503.8 [1], 7.0 [2], 8.4 [3], 21.0 [4], 44.1 [5]
FulvestrantKi1.39 [1]
2-Phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-1,2,3,4-tetrahydroisoquinolin-6-olIC50289.07 [1]
2-Phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1,2,3,4-tetrahydroisoquinolin-6-olIC5022.2 [1], 165.96 [2], 166.0 [3], 291.0 [4], 291.07 [5]
AfimoxifeneIC5021.0 [1], 32.0 [2]
AfimoxifeneKi0.16 [1], 0.5 [2]
LasofoxifeneIC501.8 [1], 13.0 [2], 24.0 [3]
ErteberelKi0.17 [1], 0.19 [2]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5064.0 [1]
2-(4-Fluorophenyl)-1-methyl-1-[4-(2-piperidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC5092.0 [1], 92.04 [2], 316.96 [3], 317.0 [4]
2-(4-Fluorophenyl)-1-methyl-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC5082.0 [1], 82.04 [2], 204.0 [3], 204.17 [4]
1-Methyl-1-[4-(2-piperidin-1-ylethoxy)phenyl]-2-(3-propan-2-ylphenyl)-3,4-dihydroisoquinolin-6-olIC50492.0 [1], 492.04 [2], 1104.08 [3], 1105.0 [4]
1-Methyl-2-(4-methylphenyl)-1-[4-(2-piperidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50420.73 [1], 421.0 [2], 486.0 [3], 486.41 [4]
2-(4-Chlorophenyl)-1-methyl-1-[4-(2-piperidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50396.0 [1], 396.28 [2], 552.0 [3], 552.08 [4]
2-(3-Hydroxyphenyl)-1-methyl-1-[4-(2-piperidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC5046.99 [1], 47.0 [2], 304.0 [3], 304.09 [4]
2-(3-Chlorophenyl)-1-methyl-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50105.93 [1], 106.0 [2], 272.0 [3], 272.27 [4]
2-(3-Chlorophenyl)-1-methyl-1-[4-(2-piperidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50158.85 [1], 159.0 [2], 283.79 [3], 284.0 [4]
1-Methyl-2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-1,2,3,4-tetrahydroisoquinolin-6-olIC5082.99 [1], 83.0 [2], 103.99 [3], 104.0 [4]
2-(3-Fluorophenyl)-1-methyl-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50123.0 [1], 123.03 [2], 198.0 [3], 198.15 [4]
2-(3-Hydroxyphenyl)-1-methyl-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC5033.0 [1], 33.04 [2], 190.0 [3], 190.11 [4]
1-Methyl-2-(4-methylphenyl)-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50354.0 [1], 447.71 [2], 448.0 [3]
2-(4-Chlorophenyl)-1-methyl-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC50302.0 [1], 530.88 [2], 531.0 [3]
1-{4-[2-(Azepan-1-yl)ethoxy]phenyl}-1-methyl-2-phenyl-1,2,3,4-tetrahydroisoquinolin-6-olIC5079.98 [1], 80.0 [2], 199.99 [3], 200.0 [4]
1-Methyl-2-(4-propan-2-ylphenyl)-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC501972.42 [1], 1974.0 [2], 4974.0 [3], 4977.37 [4]
1-Methyl-1-[4-(2-piperidin-1-ylethoxy)phenyl]-2-(4-propan-2-ylphenyl)-3,4-dihydroisoquinolin-6-olIC503687.0 [1], 3689.78 [2], 4775.29 [3], 4776.0 [4]
1-Methyl-2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1,2,3,4-tetrahydroisoquinolin-6-olIC5082.99 [1], 83.0 [2], 226.99 [3], 227.0 [4]
2-[3-(Dimethylamino)phenyl]-1-methyl-1-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-3,4-dihydroisoquinolin-6-olIC502202.93 [1], 2205.0 [2], 2971.67 [3], 2974.0 [4]
(2R,3S)-3-(4-Hydroxyphenyl)-2-[4-(2-piperidin-1-ylethoxy)phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5052.0 [1], 287.0 [2], 3876.0 [3]
TestosteroneIC5010000.0 [1]
DiethylstilbestrolIC504.0 [1], 610.0 [2]
DiethylstilbestrolKi0.63 [1]
MifepristoneIC50812.0 [1]
MifepristoneKi750.0 [1], 2876.0 [2]
Raloxifene hydrochlorideIC5043.0 [1], 260.0 [2], 341.0 [3]
CoumestrolIC502.0 [1], 18.6 [2]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-[2-[(3R)-3-methylpyrrolidin-1-yl]ethoxy]phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5087.0 [1], 161.0 [2]
2-(5-Hydroxy-naphthalen-1-YL)-1,3-benzooxazol-6-OLIC505.0 [1]
3-(6-Hydroxy-naphthalen-2-YL)-benzo[D]isooxazol-6-OLIC501.0 [1], 1.4 [2]
(2S,3R)-3-(3-Hydroxyphenyl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5037.0 [1], 38.0 [2], 40.1 [3]
(3Ar,4S,9bS)-4-(4-hydroxyphenyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-8-olKi0.47 [1], 1.54 [2]
2,4-Diisobutylamino-6-isopentylpyrimidineIC501000000.0 [1]
2,4-Diisobutylamino-6-isopentylpyrimidineKi2800.0 [1], 1000000.0 [2]
(2S,3R)-3-(3-Hydroxyphenyl)-2-[4-(2-piperidin-1-ylethoxy)phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC50115.0 [1], 157.4 [2]
(2R,3S)-3-(4-Hydroxyphenyl)-2-[4-(2-piperidin-1-ylethoxy)phenyl]-2,3-dihydro-1,4-benzoxathiin-7-olIC5044.4 [1], 45.0 [2], 238.8 [3]
4-(4-((2,4-Dioxothiazolidin-5-ylidene)methyl)-2-methoxyphenoxy)-3-(trifluoromethyl)benzonitrileIC50550.0 [1], 6300.0 [2], 15000.0 [3]
(E)-3-[2-(4-Hydroxyphenyl)-3-[4-(2-piperidin-1-ylethoxy)benzoyl]-1-benzothiophen-6-yl]prop-2-enoic acidIC50104.0 [1], 10000.0 [2]
PrednisoloneIC5010000.0 [1], 100000.0 [2]
EstroneIC5031.0 [1], 540.0 [2]
Ethinyl estradiolIC508.1 [1], 17.78 [2]
SpironolactoneIC5020000.0 [1]
EmodinIC505200.0 [1]
EmodinKi1500.0 [1]
AndrostenediolIC509.9 [1], 10.0 [2]
BazedoxifeneIC503.8 [1], 85.0 [2]
ArzoxifeneIC5066.3 [1], 240.0 [2]
EstetrolKi19.0 [1]
Lasofoxifene hydrochlorideIC5013.0 [1], 24.0 [2]
PrinaberelIC505.0 [1]
2,6-DihydroxyanthraquinoneIC502400.0 [1]
2,6-DihydroxyanthraquinoneKi690.0 [1]
7-Bromo-2-(4-hydroxyphenyl)-1,3-benzoxazol-5-OLIC502.0 [1]
(3As,4R,9bR)-2,2-difluoro-4-(4-hydroxyphenyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-8-olKi0.44 [1]
Emodin-8-glucosideIC5062000.0 [1]
Emodin-8-glucosideKi18000.0 [1]
6-(4-Hydroxyphenyl)-2-naphtholIC5016.0 [1], 16.3 [2]
(E)-3-[4-[(E)-1-(4-Hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]prop-2-enoic acidIC503.0 [1]
(E)-3-[4-[(E)-1-(4-Hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]prop-2-enoic acidKi10.0 [1]
3-(4-Hydroxy-phenyl)-4H-chromen-7-olIC50680.0 [1]
6-(2-Hydroxyphenyl)-2-naphtholIC502000.0 [1]
4-Bromo-6-(6-hydroxy-1,2-benzisoxazol-3-yl)benzene-1,3-diolIC501.8 [1]
2-(4-Hydroxy-phenyl)benzofuran-5-OLIC506.0 [1]
4-Bromo-9a-butyl-7-hydroxy-1,2,9,9a-tetrahydro-fluoren-3-oneIC501.8 [1]
4-Chloro-6-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-1,3-diolIC502.0 [1]
5-Hydroxy-2-(4-hydroxy-phenyl)-benzooxazole-7-carbonitrileIC506.0 [1]
4,4'-(5,7-Bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2,3-diyl)diphenolIC50600.0 [1]
4,4'-(5,7-Bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2,3-diyl)diphenolKi48.0 [1]
2-(4-Hydroxyphenyl)benzo[d]oxazol-6-olIC5050.0 [1]
2-(4-Hydroxy-phenyl)-7-vinyl-benzooxazol-5-olIC503.5 [1]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-[(2S)-2-pyrrolidin-1-ylpropoxy]phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5045.0 [1]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-[(2R)-2-pyrrolidin-1-ylpropoxy]phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5071.0 [1]
2-(6-Hydroxynaphthalen-1-yl)benzo[d]oxazol-6-olIC503.0 [1]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-[2-[(3S)-3-methylpyrrolidin-1-yl]ethoxy]phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5050.0 [1]
2-Naphthalen-1-yl-benzooxazol-6-olIC501050.0 [1]
(2S,3R)-3-(4-Hydroxyphenyl)-2-[4-[(2S)-2-[(3R)-3-methylpyrrolidin-1-yl]propoxy]phenyl]-2,3-dihydro-1,4-benzoxathiin-6-olIC5052.0 [1]
2-(5-Bromo-6-hydroxynaphthalen-1-yl)benzo[d]oxazol-6-olIC50134.0 [1]
6-Butyl-2,4-dipropylaminopyrimidineKi16000.0 [1], 1000000.0 [2]
5-Fluoro-2-(6-hydroxynaphthalen-1-yl)benzo[d]oxazol-6-olIC5046.0 [1]
Items per page: 1 - 10 of 99
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References

This online tool may be cited as follows

MLA

"Quest Database™ Estrogen receptor beta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/estrogen-receptor-beta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Estrogen receptor beta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/estrogen-receptor-beta-inhibitors-ic50-ki.
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