 | Doramapimod | IC50 | 9400.0 [1] |
 | (5e)-5-(Quinolin-6-Ylmethylidene)-2-[(Thiophen-2-Ylmethyl)amino]-1,3-Thiazol-4(5h)-One | Ki | 2000.0 [1] |
 | (5Z)-5-(Quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5H)-one | Ki | 2000.0 [1] |
 | CID 6918852 | Ki | 5000.0 [1] |
 | CID 44478401 | IC50 | 15.0 [1] |
 | N-(2-Chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 1000.0 [1] |
 | Ldn-211904 oxalate | IC50 | 79.0 [1] |
 | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
 | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
 | CID 71718651 | IC50 | 4400.0 [1] |
 | 7-(4-Fluoroanilino)-1-[(1R,3R)-3-hydroxycyclopentyl]-3-(4-methoxyphenyl)-4H-pyrimido[4,5-d]pyrimidin-2-one | IC50 | 1250.0 [1] |
 | 11,13-Dimethyl-12-prop-2-enyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-amine | Ki | 5000.0 [1] |
 | (Z)-2-((1R,2S)-2-Phenylcyclopropylamino)-5-(quinolin-6-ylmethylene)thiazol-4(5H)-one | Ki | 2000.0 [1] |
 | (5Z)-2-Imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-one | Ki | 2000.0 [1] |
 | N-(2-Chlorophenyl)-6-(4-hydroxypiperidin-4-yl)imidazo[1,2-a]pyridine-3-carboxamide | IC50 | 228.0 [1] |
 | N-(2-Chlorophenyl)-6-(piperidin-1-yl)imidazo[1,2-a]pyridine-3-carboxamide | IC50 | 87.0 [1] |
 | N-(2-Fluorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2,3-Dichlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-(Trifluoromethyl)phenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-Cyanophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | 2-Chloro-N-(pyrazolo[1,5-a]pyridin-3-yl)benzamide | IC50 | 20000.0 [1] |
 | 2-Chloro-N-(pyrazolo[1,5-a]pyridin-3-ylmethyl)aniline | IC50 | 20000.0 [1] |
 | N-(2-Chlorophenyl)-4-methylpyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 15000.0 [1] |
 | N-(2-Chlorophenyl)-5-methylpyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 260.0 [1] |
 | N-(2-Chlorophenyl)-6-methylpyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 15000.0 [1] |
 | 4-Chloro-N-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | 5-Chloro-N-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 2000.0 [1] |
 | 6-Chloro-N-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-Chlorophenyl)-5-methoxypyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 190.0 [1] |
 | N-(2-Chlorophenyl)-5-phenylpyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 66.0 [1] |
 | N-(2-Chlorophenyl)-5-(dimethylamino)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 77.0 [1] |
 | N-(2-Chlorophenyl)-5-pyrrol-1-ylpyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 200.0 [1] |
 | N-(2-Chlorophenyl)-5-morpholinopyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 240.0 [1] |
 | N-(2-Chlorophenyl)-5-(piperidin-1-yl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 63.0 [1] |
 | 5-(Benzyloxy)-N-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-Chlorophenyl)-1H-indazole-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-Chlorophenyl)-[1,2,3]triazolo[1,5-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-Chlorophenyl)pyrazolo[1,5-a]pyrazine-3-carboxamide | IC50 | 15000.0 [1] |
 | N-(2-Chlorophenyl)imidazo[1,2-a]pyridine-3-carboxamide | IC50 | 460.0 [1] |
 | N-(2-Chlorophenyl)-6-phenylimidazo[1,2-a]pyridine-3-carboxamide | IC50 | 60.0 [1] |
 | N-(2-Methoxyphenyl)-6-phenylimidazo[1,2-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | N-(2-Chlorophenyl)-2-methyl-6-phenylimidazo[1,2-a]pyridine-3-carboxamide | IC50 | 20000.0 [1] |
 | 6-Bromo-N-(2-chlorophenyl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide | IC50 | 173.0 [1] |
 | 7-Anilino-1-[(1R,3R)-3-hydroxycyclopentyl]-3-(4-methoxyphenyl)-4H-pyrimido[4,5-d]pyrimidin-2-one | IC50 | 1090.0 [1] |