![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 198.8 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_6724fa0e470bbc3197fba3b69ba792aa.svg) | Hematoxyline | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_b96c95589239aa5fc9b995c3e9055da0.svg) | 4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazole | IC50 | 7800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_986db0437f20070dfb14143a9f1b018d.svg) | Dasatinib | IC50 | 4.4 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_cc44f1f60583450bd176b7ecb852e3dc.svg) | 1-Tert-butyl-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 52000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_b5f9e60dc2b2b7e76e07307c1d8f7888.svg) | Bosutinib | IC50 | 8.5 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_ad465c21dbd002c135a4fe93dc9f7695.svg) | N-(3-Bromophenyl)-6,7-dimethoxyquinazolin-4-amine | IC50 | 10200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_00972cb4f918648725e1458fd9644446.svg) | 6,7-Dimethoxy-2-phenylquinoxaline | IC50 | 110000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_ae3c621c3ca0049e7a4045efa2e650e7.svg) | Tivozanib | IC50 | 17.5 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_86e23d55fdceb70174cbbe43cedcb982.svg) | 4-[3-Hydroxyanilino]-6,7-dimethoxyquinazoline | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_6925afc0497f067aee8668b4ed241d61.svg) | N-(4-Chloro-2-fluorophenyl)-6,7-dimethoxyquinazolin-4-amine | IC50 | 8500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_9cf1a487e0964a270ab59f7c8543fcd7.svg) | Src Kinase Inhibitor I | IC50 | 86000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_e64a68a1b916eb172c739c821d2bf15c.svg) | N-{4-[(3-Bromophenyl)amino]quinazolin-6-Yl}propanamide | IC50 | 180000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_ce8ad170b9daf725c7ab1a506e8363d6.svg) | 3-(4-Dimethylaminobenzylidenyl)-2-indolinone | IC50 | 27500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_39086cf2e214e5f323b181cb6ff08cf7.svg) | 2-(4-Hydroxyanilino)naphthalene-1,4-dione | IC50 | 38000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_5f06bd92f0ce452686a8455d54879f47.svg) | N-(3-Bromophenyl)-1H-imidazo[4,5-g]quinazolin-8-amine | IC50 | 22000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_96eefe9147840094954db89e1a18c4c0.svg) | N-(3-Imidazol-1-ylpropyl)-7H-purin-6-amine | IC50 | 5200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_71a9e423238295190551f437438116b2.svg) | 5-[1-Furan-2-yl-meth-(Z)-ylidene]-2-(4-methoxy-phenylamino)-thiazol-4-one | IC50 | 230000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_8f7dbca03dee2628925e79313cd5633a.svg) | N-(Pyridin-2-ylmethyl)-9H-purin-6-amine | IC50 | 106000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_c5eae2d9c2706750b2d1af999006528b.svg) | CID 44478401 | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_b7afca5bd685218d3ea22d105a1b0822.svg) | 4-N-(3-Bromophenyl)-7-N-methylquinazoline-4,7-diamine | IC50 | 34000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_2c43102721ec7ed2d36759ac8811216e.svg) | N'-(5-Chloro-1,3-benzodioxol-4-yl)-N-(3-methylsulfonylphenyl)pyrimidine-2,4-diamine | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_1acb9af54a0300732fbc15732fce477a.svg) | 4-[(2-Morpholin-4-yl-7H-purin-6-yl)amino]benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_dccd273262f72ca8a6b5928832f6e716.svg) | 5-[(Z)-1-(3,4-Dimethoxyphenyl)methylidene]-2-(4-hydroxyanilino)-1,3-thiazol-4-one | IC50 | 220000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_eea21e29768ccbc2e2a76f9f5c79fb41.svg) | N-(2-Methoxyphenyl)-2-[(5-methyl-5H-[1,2,4]triazino[5,6-b]indol-3-yl)sulfanyl]acetamide | IC50 | 136000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_0b87bdde2207195191bc2845f16c59ba.svg) | 2-[3-[3-Tert-butyl-5-[(2,3-dichlorophenyl)carbamoylamino]pyrazol-1-yl]phenyl]acetamide | IC50 | 82.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_fcca6043b08d60b7934c389a846b207f.svg) | 3-(4-Acetylpiperazin-1-yl)-5-(3-nitrobenzylamino)-7-(trifluoromethyl)quinoline | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_f212d574e725b6e4990a2dd9b43bcebe.svg) | 5-Fluoro-2-[[(1S)-1-(5-fluoropyridin-2-yl)ethyl]amino]-6-[(5-methyl-1H-pyrazol-3-yl)amino]pyridine-3-carbonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_b47eb0b10c004af2684a6d610b4c991d.svg) | Ethyl 8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carboxylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_f83aeef223e4cffa787f7bf871c66dc3.svg) | 1-(4-Fluorophenyl)-N-[3-fluoro-4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)oxyphenyl]-2-oxopyridine-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 7200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_eda1570f6e608eea37da447234534ac5.svg) | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 2158.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_be9a3af1440a45c943620056d9f96910.svg) | CID 71718651 | IC50 | 3800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_91a153dbf6ba57c0b9f24811cb69daf6.svg) | 4-Chloro-N-(2-phenylimidazo[1,2-a]pyrimidin-3-yl)benzamide | IC50 | 88000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_398e1f1b8c9cb4c69d665efa9d71c685.svg) | 1-[3-[6-(4-Fluorophenyl)pyrazine-2-yloxy]phenyl]-3-(5-tert-butylisoxazole-3-yl)urea | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_3ba30d11460b1bc0f3b0022a589906f6.svg) | 1-[3-[6-(p-Anisyl)pyrazine-2-yloxy]phenyl]-3-(5-tert-butylisoxazole-3-yl)urea | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_188035063362160fba24e588a355c671.svg) | 1-[3-[6-(3-Thienyl)pyrazine-2-yloxy]phenyl]-3-(5-tert-butylisoxazole-3-yl)urea | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_3f31224bc6b47209efd1735e3e979dbd.svg) | 1-[3-[6-(1-Methyl-1H-pyrazole-4-yl)pyrazine-2-yloxy]phenyl]-3-(5-tert-butylisoxazole-3-yl)urea | IC50 | 880.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_3ebf43d9522220430ffaa4df39a5e52d.svg) | 2-[3-[5-[(2,3-Dichlorophenyl)carbamoylamino]-3-thiophen-2-ylpyrazol-1-yl]phenyl]acetamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_082faee0fa74cca054c7a52b9562ae77.svg) | 3-[2-(4-Amino-1-ethylpyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-4-methyl-N-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]benzamide | IC50 | 26.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_cb768783449d0b92ba3d637351784fb5.svg) | 1-[4-[6,7-Bis(trideuteriomethoxy)quinolin-4-yl]oxy-2-chlorophenyl]-3-(5-methyl-1,2-oxazol-3-yl)urea | IC50 | 26.8 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_04ebf89eb58a644099e78fe3d1da5112.svg) | 1-(5-Tert-butyl-1,2-oxazol-3-yl)-3-[3-[6-(4-methylsulfonylphenyl)pyrazin-2-yl]oxyphenyl]urea | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_d1fe5152a21eb5c45e8f8a146f4dc5fc.svg) | 1-(3-Tert-butyl-1,2-oxazol-5-yl)-3-[4-[6-(1-methylpyrazol-4-yl)pyrazin-2-yl]phenyl]urea | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_f12411c8798fb008e72ad160d3e18336.svg) | 1-(5-Tert-butyl-2-methylpyrazol-3-yl)-3-[4-[6-(1-methylpyrazol-4-yl)pyrazin-2-yl]phenyl]urea | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_dc5ff7b87d06ec962585df9a614f5950.svg) | 6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_c4b2bbc8da3445973fd48f1caf9c3c0a.svg) | c-Met-IN-2 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_f5f70c2153651394c9fda3e5554e93b5.svg) | 3-(4-Methoxy-phenyl)-1-[2-(2-methyl-1H-indol-3-yl)-ethyl]-1-pyridin-4-ylmethyl-thiourea | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_4967be45bbbbed4f5b1d07e080ba10dc.svg) | 3-(4-Fluoro-phenyl)-1-[2-(2-methyl-1H-indol-3-yl)-ethyl]-1-pyridin-4-ylmethyl-thiourea | IC50 | 104000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_dbefe622a2a18ff750504a05bec3c0ba.svg) | 3-(4-Chloro-phenyl)-1-[2-(5-fluoro-2-methyl-1H-indol-3-yl)-ethyl]-1-pyridin-4-ylmethyl-thiourea | IC50 | 65000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_0bfec4b60134fd28951b12d14a56d72e.svg) | 3-[3-(2-Fluoro-phenyl)-[1,2,4]oxadiazol-5-yl]-N-(3-isopropoxy-propyl)-propionamide | IC50 | 201000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_03e0d1a2e88126708ed3a73e7e36755b.svg) | N-[5-[6-(Methylamino)pyrazin-2-yl]-2-oxo-1H-pyridin-3-yl]-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]benzamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_aa4ae17562dce9cc41b6870887651f84.svg) | 3-[(1R)-1-(2,6-Dichloro-3-fluorophenyl)ethyl]sulfanyl-5-(1-piperidin-4-ylpyrazol-4-yl)pyridin-2-amine | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_ad946fa32618a037eb1c316583993f21.svg) | 9-[[8-Fluoro-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]sulfanyl]-4-methyl-[1,4]oxazino[3,2-c]quinolin-3-one | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ephrin-type-b-receptor-2_d12f5b53170ebcdbe640da62f40a49bf.svg) | N-[(E)-1-(2-Amino-4-methyl-1,3-thiazol-5-yl)ethylideneamino]-2-(benzenesulfonamido)-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 94000.0 [1] |