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Enteropeptidase Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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4-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]cyclohexane-1-carboxylic acidKi1.11 [1], 1.53 [2]
(4-Carbamimidoyl-2-fluorophenyl) 5-[2,2-dimethyl-3-oxo-3-[(2-oxo-1H-pyridin-3-yl)amino]propyl]thiophene-2-carboxylateKi6.66 [1]
(3S)-1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]pyrrolidine-3-carboxylic acidKi0.9 [1], 1.02 [2]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-2-(4-hydroxyphenyl)acetic acidKi0.67 [1], 0.72 [2]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]butanedioic acidKi0.26 [1]
(2S)-2-[[1-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]cyclobutanecarbonyl]amino]butanedioic acidKi0.14 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]acetic acidKi0.29 [1]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-3-hydroxypropanoic acidKi0.46 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-prop-2-enylamino]acetic acidKi0.24 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-2-methylpropanoic acidKi0.69 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-propylamino]acetic acidKi0.49 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-3-hydroxypropanoic acidKi0.94 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-3-methylbutanoic acidKi1.56 [1]
3-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]propanoic acidKi0.99 [1]
2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoic acidKi1.24 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]butanoic acidKi0.65 [1]
2-[(2S)-1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]pyrrolidin-2-yl]acetic acidKi1.58 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]pentanedioic acidKi0.42 [1]
(2S)-4-Amino-2-[[2-[[5-(4-carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-4-oxobutanoic acidKi0.67 [1]
5-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-2-hydroxybenzoic acidKi0.53 [1]
1-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]cyclobutane-1-carboxylic acidKi0.51 [1]
4-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-4-(2-carboxyethyl)heptanedioic acidKi0.71 [1]
5-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]benzene-1,3-dicarboxylic acidKi0.31 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[2,2-dimethyl-3-oxo-3-[2-(2H-tetrazol-5-yl)ethylamino]propyl]thiophene-2-carboxylateKi0.53 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[2,2-dimethyl-3-oxo-3-(2H-tetrazol-5-ylmethylamino)propyl]thiophene-2-carboxylateKi0.53 [1]
5-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]benzene-1,3-dicarboxylic acidKi0.71 [1]
4-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]phthalic acidKi0.24 [1]
1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]azetidine-3-carboxylic acidKi0.63 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-prop-2-enylamino]ethanesulfonic acidKi1.81 [1]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-3-methylbutanoic acidKi0.79 [1]
2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]-methylamino]acetic acidKi0.88 [1]
(2S)-2-[[1-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]cyclopentanecarbonyl]amino]butanedioic acidKi0.73 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[2-ethyl-2-(2H-tetrazol-5-ylmethylcarbamoyl)butyl]thiophene-2-carboxylateKi1.2 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-methylamino]acetic acidKi0.41 [1]
(2S)-1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]pyrrolidine-2-carboxylic acidKi0.87 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-3-hydroxybutanoic acidKi0.84 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-3-phenylpropanoic acidKi1.1 [1]
(2S)-1-[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]pyrrolidine-2-carboxylic acidKi1.0 [1]
2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]-propylamino]acetic acidKi2.61 [1]
1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]piperidine-4-carboxylic acidKi1.33 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]propanoic acidKi0.73 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]pentanoic acidKi1.18 [1]
4-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]butanoic acidKi0.94 [1]
4-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]benzoic acidKi1.08 [1]
3-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]benzoic acidKi1.43 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[2-ethyl-2-[[(3S)-5-oxooxolan-3-yl]carbamoyl]butyl]thiophene-2-carboxylateKi2.56 [1]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-2-cyclohexylacetic acidKi4.7 [1]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-2-phenylacetic acidKi0.97 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[2,2-dimethyl-3-oxo-3-(pyridin-3-ylamino)propyl]thiophene-2-carboxylateKi7.56 [1]
(2S)-5-Amino-2-[[2-[[5-(4-carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-5-oxopentanoic acidKi1.69 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[3-[(6-methoxypyridin-3-yl)amino]-2,2-dimethyl-3-oxopropyl]thiophene-2-carboxylateKi4.13 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[3-(3,3-difluoroazetidin-1-yl)-2,2-dimethyl-3-oxopropyl]thiophene-2-carboxylateKi5.27 [1]
2-[4-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]phenyl]acetic acidKi2.41 [1]
2-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-3,4-dihydro-1H-isoquinoline-7-carboxylic acidKi3.46 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[3-[(2-methoxypyridin-3-yl)amino]-2,2-dimethyl-3-oxopropyl]thiophene-2-carboxylateKi3.75 [1]
(2S)-2-Amino-5-[[2-[[5-(4-carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]pentanoic acidKi5.53 [1]
4-[[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]methyl]benzoic acidKi2.69 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[3-[(6-fluoropyridin-3-yl)amino]-2,2-dimethyl-3-oxopropyl]thiophene-2-carboxylateKi2.51 [1]
1-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]cyclopropane-1-carboxylic acidKi0.67 [1]
Dimethyl 5-[[3-[5-(4-carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]benzene-1,3-dicarboxylateKi1.22 [1]
(2S)-1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]aziridine-2-carboxylic acidKi1.13 [1]
5-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]pentanoic acidKi0.98 [1]
(4-Carbamimidoyl-2-fluorophenyl) 5-[3-(2-cyanoethylamino)-2,2-dimethyl-3-oxopropyl]thiophene-2-carboxylateKi2.9 [1]
3-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-5-methoxycarbonylbenzoic acidKi3.73 [1]
6-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]hexanoic acidKi4.97 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]benzoic acidKi2.41 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]terephthalic acidKi0.39 [1]
2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-(cyclopropylmethyl)amino]acetic acidKi0.67 [1]
2-[[2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]acetyl]amino]acetic acidKi0.69 [1]
1-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]cyclopropane-1-carboxylic acidKi1.12 [1]
1-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]cyclobutane-1-carboxylic acidKi1.33 [1]
3-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]-5-hydroxybenzoic acidKi0.58 [1]
5-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-2-hydroxybenzoic acidKi3.52 [1]
(1R,3S)-3-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]cyclohexane-1-carboxylic acidKi0.81 [1]
2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]acetic acidKi0.72 [1]
(2S)-2-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-3-(2H-tetrazol-5-yl)propanoic acidKi0.24 [1]
1-[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]azetidine-3-carboxylic acidKi1.0 [1]
3-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]benzenesulfonic acidKi0.84 [1]
4-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]phthalic acidKi0.55 [1]
(2S,4R)-1-[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]-4-hydroxypyrrolidine-2-carboxylic acidKi0.3 [1]
(1R,6S)-6-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2,2-dimethylpropanoyl]amino]cyclohex-3-ene-1-carboxylic acidKi1.3 [1]
(4S)-4-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-4-(2H-tetrazol-5-yl)butanoic acidKi0.43 [1]
(3S)-3-[[2-[[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]methyl]-2-ethylbutanoyl]amino]-4-methylhexanoic acidKi3.26 [1]
(2S)-2-[[3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]pentanedioic acidKi1.63 [1]
(2S)-2-[[3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.61 [1]
(2R)-2-[[3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.42 [1]
(2R)-2-[[3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]pentanedioic acidKi0.57 [1]
(2R)-2-[2-[[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]methyl]butanoylamino]butanedioic acidKi0.5 [1]
(2R)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.25 [1]
(2S)-2-[3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]propanoylamino]butanedioic acidKi0.57 [1]
(2S)-2-[[2-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]acetyl]amino]butanedioic acidKi0.67 [1]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2-methylpropanoyl]amino]pentanedioic acidKi0.56 [1]
(2R)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.5 [1]
(2R)-2-[[3-[5-(4-Carbamimidoylphenoxy)carbonylthiophen-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi1.47 [1]
(2S)-2-[[(2S)-3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.4 [1]
(2S)-2-[[(2R)-3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.33 [1]
(2R)-2-[[(2S)-3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.46 [1]
(2S)-2-[[3-[5-(4-Carbamimidoyl-2-fluorophenoxy)carbonylthiophen-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.28 [1]
(2R)-2-[[(2R)-3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]-2-methylpropanoyl]amino]butanedioic acidKi0.35 [1]
3-[3-[5-(4-Carbamimidoylphenoxy)carbonylfuran-2-yl]propanoyl-(carboxymethyl)amino]propanoic acidKi0.6 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Enteropeptidase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/enteropeptidase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Enteropeptidase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/enteropeptidase-inhibitors-ic50-ki.
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