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Endothelial PAS domain-containing protein 1 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
3-[[(1S)-2,2-Difluoro-1-hydroxy-7-methylsulfonyl-1,3-dihydroinden-4-yl]oxy]-5-fluorobenzonitrileIC5012.0 [1]
3-[[(1S)-7-(Difluoromethylsulfonyl)-2,2-difluoro-1-hydroxy-1,3-dihydroinden-4-yl]oxy]-5-fluorobenzonitrileIC505.0 [1]
N-(3-Chloro-5-Fluorophenyl)-4-Nitro-2,1,3-Benzoxadiazol-5-AmineIC50490.0 [1]
2-(3-Chloro-5-fluorophenoxy)-5-(trifluoromethylsulfonyl)benzoic acidIC5044400.0 [1]
2-Bromo-1-(3-chloro-5-fluorophenoxy)-4-methylsulfonylbenzeneIC504400.0 [1]
2-Bromo-1-(3-chloro-5-fluorophenoxy)-4-(trifluoromethylsulfonyl)benzeneIC50170.0 [1]
2-Chloro-1-(3-chloro-5-fluorophenoxy)-4-(difluoromethylsulfonyl)-3-(methoxymethyl)benzeneIC504200.0 [1]
4-(3-Chloro-5-fluorophenoxy)-7-(difluoromethylsulfonyl)-2,3-dihydro-1H-inden-1-olIC505.0 [1]
N-[[2-Bromo-3-(3-chloro-5-fluorophenoxy)-6-(difluoromethylsulfonyl)phenyl]methyl]acetamideIC5018200.0 [1]
[2-(3-Chloro-5-fluorophenoxy)-5-(trifluoromethylsulfonyl)phenyl]methanolIC501200.0 [1]
Methyl 2-(3-chloro-5-fluorophenoxy)-5-(trifluoromethylsulfonyl)benzoateIC5052900.0 [1]
[2-Bromo-3-(3-chloro-5-fluorophenoxy)-6-(difluoromethylsulfonyl)phenyl]methanamineIC50700.0 [1]
2-Bromo-1-(3-chloro-5-fluorophenoxy)-4-(difluoromethylsulfonyl)benzeneIC50180.0 [1]
3-[[(1S)-7-Ethylsulfonyl-2,2-difluoro-1-hydroxy-1,3-dihydroinden-4-yl]oxy]-5-fluorobenzonitrileIC5031.0 [1]
[2-Chloro-3-(3-chloro-5-fluorophenoxy)-6-(difluoromethylsulfonyl)phenyl]methanolIC5046.0 [1]
2-(3-Chloro-5-fluorophenoxy)-5-(trifluoromethylsulfonyl)benzamideIC5022600.0 [1]
2-Chloro-1-(3-chloro-5-fluorophenoxy)-4-(trifluoromethylsulfonyl)benzeneIC50140.0 [1]
(1S)-4-(5-Chloropyridin-3-yl)oxy-7-(difluoromethylsulfonyl)-2,2-difluoro-1,3-dihydroinden-1-olIC5060.0 [1]
3-Fluoro-5-[[(1S,2S)-2-fluoro-1-hydroxy-7-methylsulfonyl-2,3-dihydro-1H-inden-4-yl]oxy]benzonitrileIC50350.0 [1]
3-[[(1S)-2,2-Difluoro-7-(fluoromethylsulfonyl)-1-hydroxy-1,3-dihydroinden-4-yl]oxy]-5-fluorobenzonitrileIC505.0 [1]
3-[(6,6-Difluoro-5-hydroxy-4-methylsulfonyl-7,8-dihydro-5H-naphthalen-1-yl)oxy]-5-fluorobenzonitrileIC503600.0 [1]
(Rac)-PT2399IC5010.0 [1]
3-[[(1S)-2,2-Difluoro-1-hydroxy-7-(trifluoromethylsulfonyl)-1,3-dihydroinden-4-yl]oxy]-5-fluorobenzonitrileIC505.0 [1]
4-(3-Chloro-5-fluorophenoxy)-7-(difluoromethylsulfonyl)-2,2-difluoro-1,3-dihydroinden-1-olIC505.0 [1]
2-(3-Chloro-5-fluorophenoxy)-5-(trifluoromethylsulfonyl)benzonitrileIC5034.0 [1]
3-Fluoro-5-[[(1S,2R)-2-fluoro-1-hydroxy-7-methylsulfonyl-2,3-dihydro-1H-inden-4-yl]oxy]benzonitrileIC5041.0 [1]
4-(Difluoromethyl)-5-(3,5-difluorophenoxy)-2,2-difluoro-1,1-dioxo-3H-1-benzothiophen-3-olIC5011.0 [1]
5-(3-Chloro-5-fluorophenoxy)-2,2-difluoro-4-methyl-1,1-dioxo-3H-1-benzothiophen-3-olIC5020.0 [1]
5-(3-Chloro-5-fluorophenoxy)-4-(difluoromethyl)-2,2-difluoro-1,1-dioxo-3H-1-benzothiophen-3-olIC505.0 [1]
4-Bromo-5-(3-chloro-5-fluorophenoxy)-1,1-dioxo-2,3-dihydro-1-benzothiophen-3-olIC502400.0 [1]
5-(5-Chloropyridin-3-yl)oxy-4-(difluoromethyl)-2,2-difluoro-1,1-dioxo-3H-1-benzothiophen-3-olIC50350.0 [1]
4-Bromo-5-(3-chloro-5-fluorophenoxy)-2,2-difluoro-1,1-dioxo-3H-1-benzothiophen-3-olIC505.0 [1]
5-(3-Chloro-5-fluorophenoxy)-2,2-difluoro-1,1-dioxo-3H-1-benzothiophen-3-olIC501100.0 [1]
5-(3-Chloro-5-fluorophenoxy)-2,2-difluoro-3-hydroxy-1,1-dioxo-3H-1-benzothiophene-4-carbonitrileIC5049.0 [1]
5-[[4-(Difluoromethyl)-2,2-difluoro-3-hydroxy-1,1-dioxo-3H-1-benzothiophen-5-yl]oxy]pyridine-3-carbonitrileIC50140.0 [1]
3-[[4-(Difluoromethyl)-2,2-difluoro-3-hydroxy-1,1-dioxo-3H-1-benzothiophen-5-yl]oxy]-5-fluorobenzonitrileIC5014.0 [1]
4-Bromo-5-(3-chloro-5-fluorophenoxy)-2,2-dimethyl-1,1-dioxo-3H-1-benzothiophen-3-olIC5019600.0 [1]
4-Chloro-5-(3-chloro-5-fluorophenoxy)-2,2-difluoro-1,1-dioxo-3H-1-benzothiophen-3-olIC5020.0 [1]
5-(3-Chloro-5-fluorophenoxy)-2,2-difluoro-1,1-dioxo-4-(trifluoromethyl)-3H-1-benzothiophen-3-olIC505.0 [1]
3-[[(3S)-4-(Difluoromethyl)-2,2-difluoro-3-hydroxy-1,1-dioxo-3H-1-benzothiophen-5-yl]oxy]-5-fluorobenzonitrileIC501700.0 [1]
5-(Difluoromethyl)-6-(3,5-difluorophenoxy)-1,1-dioxo-3,4-dihydro-2H-thiochromen-4-olIC503200.0 [1]
(1R)-4-(3-Chloro-5-fluorophenoxy)-7-(difluoromethylsulfonyl)-2,3-dihydro-1H-inden-1-olIC505.0 [1]
{2-Bromo-3-(3-chloro-5-fluorophenoxy)-6-[(difluoromethyl)sulfonyl]phenyl}methanolIC5055.0 [1]
1-(3-Chloro-5-fluorophenoxy)-2-(difluoromethyl)-4-(trifluoromethylsulfonyl)benzeneIC50220.0 [1]
(1S)-4-(3-Chloro-5-fluorophenoxy)-7-(difluoromethylsulfonyl)-2,3-dihydro-1H-inden-1-olIC50460.0 [1]
(5S,7R)-5-(3-Bromophenyl)-7-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC50248.0 [1]
(5R,7S)-5-(3-Bromophenyl)-7-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
N-(3-Chloro-5-fluorophenyl)-2-nitro-4-[(trifluoromethyl)sulfonyl]anilineIC505.0 [1]
(5s,7r)-5,7-Bis(3-Bromophenyl)-4,5,6,7-Tetrahydrotetrazolo[1,5-A]pyrimidineIC50112.0 [1]
(5S,7R)-5-(3-Bromo-5-fluorophenyl)-7-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5043.0 [1]
CID 136268871IC50195.0 [1]
(5S,7R)-7-(2-Bromophenyl)-5-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC50314.0 [1]
(5S,7R)-5-(3-Bromo-5-fluorophenyl)-7-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5097.0 [1]
(5S,7R)-7-(5-Bromo-2-chlorophenyl)-5-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5087.0 [1]
(5S,7R)-7-(3-Bromo-2,6-difluorophenyl)-5-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5032.0 [1]
CID 137036807IC501000.0 [1]
(5R,7S)-5-(3-Iodophenyl)-7-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
(5R,7S)-7-(2-Bromophenyl)-5-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5028300.0 [1]
(5R,7S)-5-(3-Bromophenyl)-7-(2-chlorophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
(5R,7S)-5,7-Bis(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
CID 137036812IC50108.0 [1]
(5R,7S)-5-(3-Bromophenyl)-7-(3-iodophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
(5R,7S)-7-(5-Bromo-2-chlorophenyl)-5-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
(5R,7S)-7-(3-Bromo-2,6-difluorophenyl)-5-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5022300.0 [1]
(5R,7S)-5-(3-Bromo-5-fluorophenyl)-7-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
(5R,7S)-5-(3-Bromo-5-fluorophenyl)-7-(3-bromophenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidineIC5030000.0 [1]
N-(3-Chloro-5-fluorophenyl)-2-nitro-4-(trifluoromethyl)anilineIC50280.0 [1]
N-(3-Chloro-5-fluorophenyl)-4-(fluoromethylsulfonyl)-2-nitroanilineIC50280.0 [1]
1-(3-Chloro-5-fluorophenoxy)-2-nitro-4-(trifluoromethylsulfonyl)benzeneIC5032.0 [1]
1-[4-(3-Chloro-5-fluoroanilino)-3-nitrophenyl]ethanolIC5012700.0 [1]
3-(3-Cyano-5-fluorophenoxy)-2-(difluoromethyl)-6-(difluoromethylsulfonyl)benzoic acidIC50100000.0 [1]
4-(3-Chloro-5-fluoroanilino)-N-methyl-3-nitrobenzenesulfonamideIC504200.0 [1]
N-(3-Chloro-5-fluorophenyl)-4-(difluoromethylsulfonyl)-2-nitroanilineIC5016.0 [1]
Hif-2|A-IN-1IC505.0 [1]
Items per page: 1 - 10 of 74
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References

This online tool may be cited as follows

MLA

"Quest Database™ Endothelial PAS domain-containing protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/endothelial-pas-domain-containing-protein-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Endothelial PAS domain-containing protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/endothelial-pas-domain-containing-protein-1-inhibitors-ic50-ki.
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