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Endoplasmic reticulum aminopeptidase 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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[(2S)-2-[[(2S)-1-Amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC5033.0 [1], 48.0 [2]
[(2S)-2-[[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC503694.0 [1]
[(2S)-2-[[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidKi3500.0 [1]
Leucine Phosphonic AcidKi5080.0 [1]
Phosphonic acid, (1-amino-3-phenylpropyl)-Ki26900.0 [1]
2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi19100.0 [1]
2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-(4-hydroxyphenyl)propanoic acidKi6470.0 [1]
CID 118720630Ki530.0 [1]
CID 127052870Ki250000.0 [1]
[(1S)-1-Amino-3-methylbutyl]phosphonic acidKi249000.0 [1]
[1-Amino-2-(cyclohexylamino)ethyl]phosphonic acidKi250000.0 [1]
2-[[[1-Amino-3-(3,5-dimethylphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi31600.0 [1]
2-[[[1-Amino-3-(3-hydroxyphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi87100.0 [1]
2-[[[1-Amino-3-(4-hydroxyphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi11300.0 [1]
2-[[[1-Amino-3-[4-(hydroxymethyl)phenyl]propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi991.0 [1]
2-[[(1-Amino-3-pyridin-3-ylpropyl)-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi12300.0 [1]
2-[[(1-Amino-3-pyridin-4-ylpropyl)-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi2540.0 [1]
2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-(3,5-dimethylphenyl)propanoic acidKi250000.0 [1]
2-[[3-(Aminomethyl)phenyl]methyl]-3-[(1-amino-3-phenylpropyl)-hydroxyphosphoryl]propanoic acidKi18600.0 [1]
2-[[4-(Aminomethyl)phenyl]methyl]-3-[(1-amino-3-phenylpropyl)-hydroxyphosphoryl]propanoic acidKi3730.0 [1]
Methyl N-[4-Amino-3-(L-Arginylamino)benzene-1-Carbonyl]-L-TyrosinateIC509600.0 [1]
(1-Amino-2-morpholin-4-ylethyl)phosphonic acidKi250000.0 [1]
2-[[[1-Amino-2-(2-methylpropylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi250000.0 [1]
2-[[[1-Amino-2-(cyclohexylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi250000.0 [1]
[1-Amino-2-(oxolan-2-ylmethylamino)ethyl]phosphonic acidKi250000.0 [1]
(1-Amino-2-piperidin-1-ylethyl)phosphonic acidKi250000.0 [1]
[1-Amino-2-[(2-aminocyclohexyl)amino]ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-(1-phenylethylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-[2-(dimethylamino)ethylamino]ethyl]phosphonic acidKi250000.0 [1]
2-Benzyl-3-[1,2-diaminoethyl(hydroxy)phosphoryl]propanoic acidKi250000.0 [1]
[1-Amino-2-(cycloheptylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-(2-phenylethylamino)ethyl]phosphonic acidKi250000.0 [1]
2-[[[1-Amino-2-(propylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi250000.0 [1]
[1-Amino-2-(2-piperazin-1-ylethylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-[(4-tert-butylphenyl)methylamino]ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-[(4-aminophenyl)methylamino]ethyl]phosphonic acidKi250000.0 [1]
2-[[[1-Amino-2-(cycloheptylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi250000.0 [1]
[1-Amino-2-[(4-methoxyphenyl)methylamino]ethyl]phosphonic acidKi250000.0 [1]
2-[[[1-Amino-2-[2-(4-methoxyphenyl)ethylamino]ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acidKi250000.0 [1]
[1-Amino-2-(hexylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-[[4-(aminomethyl)phenyl]methylamino]ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-(piperidin-4-ylmethylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-(benzylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-(methylamino)ethyl]phosphonic acidKi250000.0 [1]
(1,2-Diaminoethyl)phosphonic acidKi250000.0 [1]
(2s)-3-[(S)-[(1r)-1-Amino-3-Phenylpropyl](Hydroxy)phosphoryl]-2-Benzylpropanoic AcidKi6270.0 [1]
Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]hexanoateIC502000.0 [1]
CID 71817810IC502600.0 [1]
[(1r)-1-Amino-3-Phenylpropyl]phosphonic AcidKi5550.0 [1]
[1-Amino-2-(propylamino)ethyl]phosphonic acidKi250000.0 [1]
[1-Amino-2-(2-aminoethylamino)ethyl]phosphonic acidKi250000.0 [1]
4-Amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoic acidIC50100000.0 [1]
Methyl 4-amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoateIC50100000.0 [1]
Methyl 4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoateIC50100000.0 [1]
Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoyl]amino]hexanoateIC50100000.0 [1]
Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-(4-phenylmethoxyphenyl)butanoyl]amino]benzoyl]amino]hexanoateIC50100000.0 [1]
(2S)-6-Amino-2-[[4-amino-3-[[(2S)-2-amino-4-methylpentanoyl]amino]benzoyl]amino]hexanoic acidIC506800.0 [1]
Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]hexanoateIC5018300.0 [1]
Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]hexanoateIC5042000.0 [1]
Methyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoateIC50110000.0 [1]
Methyl (2S,3R)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-hydroxybutanoateIC50100000.0 [1]
Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC509800.0 [1]
(2S)-2-[[4-Amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC5012100.0 [1]
Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-(4-phenylmethoxyphenyl)butanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC50100000.0 [1]
(2S)-2-[[4-Amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC5038400.0 [1]
Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoateIC50100000.0 [1]
Methyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoateIC50100000.0 [1]
Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC50920.0 [1]
(2S)-2-[[4-Amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC503600.0 [1]
Methyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-5-(diaminomethylideneamino)pentanoateIC5010700.0 [1]
(2S)-2-[[4-Amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC501200.0 [1]
Methyl 3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoateIC50100000.0 [1]
Methyl (2S)-6-amino-2-[(3,4-diaminobenzoyl)amino]hexanoateIC50100000.0 [1]
(2S)-2-[(3,4-Diaminobenzoyl)amino]-3-(1H-indol-3-yl)propanoic acidIC50100000.0 [1]
Methyl (2S)-2-[(3,4-diaminobenzoyl)amino]-5-(diaminomethylideneamino)pentanoateIC5035000.0 [1]
Methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoateIC509400.0 [1]
Benzyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC5013400.0 [1]
Methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-5-(diaminomethylideneamino)pentanoateIC5012000.0 [1]
Methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoateIC5016700.0 [1]
Benzyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-3-(4-phenylmethoxyphenyl)propanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC501100.0 [1]
(2S)-2-[[3-Amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC5019500.0 [1]
Methyl (2S)-6-amino-2-[[3-amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]hexanoateIC50100000.0 [1]
(2S)-2-[[3-Amino-4-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC50800.0 [1]
Benzyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-methylpentanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC508900.0 [1]
Benzyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoateIC50100000.0 [1]
Methyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoateIC50100000.0 [1]
Benzyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoateIC502500.0 [1]
(2S)-2-[[3-Amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC502800.0 [1]
Methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoateIC502600.0 [1]
(2S)-2-[[3-Amino-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acidIC5038200.0 [1]
[(1R)-1-Amino-3-phenylpropyl]-[(2S)-2-carbamoyl-4-methylpentyl]phosphinic acidIC50520.0 [1]
2-[[4-(Aminomethyl)phenyl]methyl]-3-[(1-amino-3-pyridin-4-ylpropyl)-hydroxyphosphoryl]propanoic acidKi1520.0 [1]
2-[[3-(Aminomethyl)phenyl]methyl]-3-[(1-amino-3-pyridin-3-ylpropyl)-hydroxyphosphoryl]propanoic acidKi4940.0 [1]
[(2S)-2-[[(2S)-1-Amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC501969.0 [1]
[(2S)-3-[[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]amino]-3-oxo-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]propyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC50126.0 [1]
[(2S)-3-[[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]amino]-2-[[3,5-bis(3-chlorophenyl)phenyl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC5025111.0 [1]
[(2S)-2-[[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC5031212.0 [1]
[(2S)-2-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC507473.0 [1]
[(2R)-3-[[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[(3,5-diphenylphenyl)methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC50100000.0 [1]
[(2S)-2-(1-Adamantylmethyl)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acidIC50726.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Endoplasmic reticulum aminopeptidase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/endoplasmic-reticulum-aminopeptidase-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Endoplasmic reticulum aminopeptidase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/endoplasmic-reticulum-aminopeptidase-1-inhibitors-ic50-ki.
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