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EML4-ALK Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
CrizotinibIC50605.0 [1]
LorlatinibIC509.0 [1]
(16R)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,8,20-triaza-5-azoniatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2,5,10(15),11,13,18,20-octaen-9-oneIC500.7 [1], 14.0 [2]
AlectinibIC502.0 [1]
CeritinibIC5041.0 [1]
Alk-IN-1IC505.0 [1]
EntrectinibIC5028.0 [1]
JH-VIII-157-02IC502.0 [1]
9-Ethyl-6,6-dimethyl-8-[1-(oxan-4-yl)pyrazol-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC5078.0 [1]
9-Ethyl-6,6-dimethyl-11-oxo-8-(1-piperidin-4-ylpyrazol-4-yl)-5H-benzo[b]carbazole-3-carbonitrileIC5040.0 [1]
8-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]-9-ethyl-6,6-dimethyl-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC502.0 [1]
8-[1-[3-(Dimethylamino)propyl]pyrazol-4-yl]-9-ethyl-6,6-dimethyl-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC5014.0 [1]
2-[4-(3-Cyano-9-ethyl-6,6-dimethyl-11-oxo-5H-benzo[b]carbazol-8-yl)pyrazol-1-yl]-N,N,2-trimethylpropanamideIC506.0 [1]
4-(3-Cyano-9-ethyl-6,6-dimethyl-11-oxo-5H-benzo[b]carbazol-8-yl)-N,N-dimethylpyrazole-1-carboxamideIC5056.0 [1]
9-Ethyl-6,6-dimethyl-11-oxo-8-(2H-triazol-4-yl)-5H-benzo[b]carbazole-3-carbonitrileIC50115.0 [1]
8-[4-(Dimethylamino)piperidin-1-yl]-9-ethyl-6,6-dimethyl-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC502.0 [1]
9-Ethyl-6,6-dimethyl-11-oxo-8-(1H-pyrazol-5-yl)-5H-benzo[b]carbazole-3-carbonitrileIC5050.0 [1]
9-Ethyl-6,6-dimethyl-8-(1-methylpyrazol-4-yl)-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC5061.0 [1]
9-Ethyl-6,6-dimethyl-11-oxo-8-(1H-pyrazol-4-yl)-5H-benzo[b]carbazole-3-carbonitrileIC5064.0 [1]
9-Ethyl-6,6-dimethyl-8-(1,2-oxazol-4-yl)-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC5059.0 [1]
9-Ethyl-6,6-dimethyl-8-(4-methylpiperazin-1-yl)-11-oxo-5H-benzo[b]carbazole-3-carbonitrileIC502.0 [1]
Items per page: 1 - 10 of 21
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References

This online tool may be cited as follows

MLA

"Quest Database™ EML4-ALK Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/eml4-alk-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ EML4-ALK Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/eml4-alk-inhibitors-ic50-ki.
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